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Published April 29, 2022 | Version v1

Modulation of Multidrug Resistance Protein 1-mediated transport processes by the antiretroviral drug ritonavir

  • 1. Hybrid Materials Interfaces Group, University of Bremen
  • 1. Centre for Biomolecular Interactions Bremen, University of Bremen
  • 2. Hybrid Materials Interfaces Group, University of Bremen

Description

We here provide the structure files, trajectories and topology files for analyzing and reproducing simulations performed in the publication: "Modulation of Multidrug Resistance Protein 1-mediated transport processes by the antiretroviral drug ritonavir".

Classical molecular dynamics simulation of rat Mrp1 have been performed in complex with native substrates like GSH and GSSG  or drug molecules like ritonavir, to study binding modes of different combinations. 

Structure and trajectory files (all 1 µs long) are provided for the following simulation systems:

1. GSH bound to rat Mrp1

2. GSSG bound to rat Mrp1

3. Ritonavir bound to rat Mrp1

4. GSH + Ritonavir bound to rat Mrp1

5. GSSG + Ritonavir bound to rat Mrp1

Additionally itp files (GROMACS format) containing parameter information about the ligands GSH, GSSG and Ritonavir are provided for the force field CHARMM36m. 

Raw data of the homology modeling of rat Mrp1 by I-Tasser as well as Docking results produced via AutoDock4 are uploaded as zip directories. 

Files

Autodock_results.zip

Files (9.3 GB)

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