brd	smi	cid	dataset
BRD-K00036326	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccccc1F	CID:60184829	phase I
BRD-K00233837	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3cncnc3)C[C@@H]1N2	CID:60185108	phase I
BRD-K00403046	Cc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1ccccc1F	CID:60185252	phase I
BRD-K00585841	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Cc1ccccc1	CID:60184986	phase I
BRD-K00845702	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)CN1CCOCC1	CID:60185201	phase I
BRD-K01214267	CCCNC(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccccc1C	CID:60185000	phase I
BRD-K01425431	N#Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3ccccc3)C[C@@H]1N2	CID:60185110	phase I
BRD-K01448700	COc1cc(CN2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2ccncc2)cc(OC)c1	CID:60185468	phase I
BRD-K01658702	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3cccc(F)c3)C[C@@H]1N2	CID:60185148	phase I
BRD-K01855742	O=S(=O)(N1C[C@@H]2N[C@H](C1)[C@@H]2c1ccc(cc1)-c1ccncc1)c1ccc(cc1)-c1ccccc1	CID:60184990	phase I
BRD-K02098967	Fc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3cncnc3)C[C@@H]1N2	CID:60185256	phase I
BRD-K02796109	COc1cccc(CN2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2ccccc2C)c1	CID:60185203	phase I
BRD-K03522229	COc1cccc(NC(=O)N2[C@H]3CNC[C@@H]2[C@@H]3c2ccc(cc2)-c2ccncc2)c1	CID:60184914	phase I
BRD-K03701362	COc1ccccc1S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccccc1C	CID:60184979	phase I
BRD-K04021565	O=C(NC1CCCCC1)N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60185357	phase I
BRD-K04266880	C\C=C\c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CCC1	CID:60184959	phase I
BRD-K04362735	O=C(NC1CCCC1)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1cccnc1	CID:60184879	phase I
BRD-K04364654	COc1ccccc1S(=O)(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccncc1	CID:60184989	phase I
BRD-K04561891	O=C(CN1CCOCC1)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccncc1	CID:60185106	phase I
BRD-K04562016	COc1ccccc1CN1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1cccc(c1)C#N	CID:60184860	phase I
BRD-K04803823	COc1ccccc1CN1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cccc(c1)C#N	CID:60185154	phase I
BRD-K04887706	O=c1[nH]c2ccccc2n1C3CCN(Cc4ccc(cc4)c5nc6cc7[nH]cnc7cc6nc5c8ccccc8)CC3	CID:135398501	phase I
BRD-K04923131	O\N=C1/C(Nc2ccccc12)=C1/C(=O)Nc2cc(Br)ccc12	CID:448949	phase I
BRD-K05004643	Cn1cnc(c1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccccc1F	CID:60184958	phase I
BRD-K05335890	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3cocn3)C[C@@H]1N2	CID:60185055	phase I
BRD-K05572312	COc1cccc(c1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccccc1F	CID:60185058	phase I
BRD-K06212126	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3cncnc3)C[C@@H]1N2	CID:60184909	phase I
BRD-K06436793	C\C=C\c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc2OCOc2c1	CID:60184805	phase I
BRD-K06725890	C\C=C\c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3cncnc3)C[C@@H]1N2	CID:60185103	phase I
BRD-K06902185	Nc1cc(nc(N)[n+]1[O-])N1CCCCC1	CID:4201	phase I
BRD-K07667918	C[C@@]1(O)CC(C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12	CID:11640390	phase I
BRD-K08725381	Fc1ccc(cc1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60184834	phase I
BRD-K09333299	COc1cc(CN2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2cncnc2)cc(OC)c1	CID:60185156	phase I
BRD-K09487323	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Nc1ccc2OCOc2c1	CID:60185174	phase I
BRD-K09964916	Cc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3ccccc3F)C[C@@H]1N2	CID:60185009	phase I
BRD-K10064333	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccc2OCOc2c1	CID:60184974	phase I
BRD-K10177585	CC[C@@H]1CN2C(=N1)c1[nH]c(nc1N(C)C2=O)-c1ccccc1	CID:135433658	phase I
BRD-K10749532	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1cccnc1	CID:60184830	phase I
BRD-K10860596	CN1[C@H]2CCC[C@@H]1C[C@@H](C2)NC(=O)c3nn(C)c4ccccc34	CID:5284566	phase I
BRD-K11293573	COc1cccc(c1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(\C=C\C)cc1	CID:60185277	phase I
BRD-K11555344	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)NC1CCCCC1	CID:60184857	phase I
BRD-K11677408	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1cccc(Cl)c1	CID:60184960	phase I
BRD-K11679888	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Nc1ccccc1	CID:60185124	phase I
BRD-K11840410	C\C=C\c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc(cc1)C(F)(F)F	CID:60184825	phase I
BRD-K12027235	Fc1cccc(CN2C[C@H]3N[C@@H](C2)[C@@H]3c2ccc(\C=C\c3ccccc3)cc2)c1	CID:60185138	phase I
BRD-K12309761	N#Cc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccc2OCOc2c1	CID:60184875	phase I
BRD-K12604570	FC(F)(F)c1ccc(NC(=O)N2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2cccc(c2)C#N)cc1	CID:60184988	phase I
BRD-K12676148	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1ccccc1C(F)(F)F	CID:60184963	phase I
BRD-K12744550	O=C(Cc1ccncc1)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60184985	phase I
BRD-K14031425	Cc1ccc(cc1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cccc(C)c1	CID:60185127	phase I
BRD-K14074563	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Nc1ccc(F)cc1	CID:60184934	phase I
BRD-K14086402	C(N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1cccnc1)c1ccc2OCOc2c1	CID:60185273	phase I
BRD-K14172822	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CCCCC1	CID:60185007	phase I
BRD-K14310250	Cc1ccccc1S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cccc(c1)C#N	CID:60185080	phase I
BRD-K14356875	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2N[C@@H]1CN(C2)S(=O)(=O)c1cccc(Cl)c1	CID:60185013	phase I
BRD-K14611588	COc1cccc(NC(=O)N2[C@H]3CNC[C@@H]2[C@@H]3c2ccc(\C=C\C)cc2)c1	CID:60184854	phase I
BRD-K15014948	NC[C@H]1CC[C@@H](CC1)C(O)=O	CID:5526	phase I
BRD-K15042749	C\C=C\c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1cn(C)cn1	CID:60184874	phase I
BRD-K15111910	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CCOCC1	CID:60184913	phase I
BRD-K15531302	Fc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccccc1	CID:60185126	phase I
BRD-K15600710	COC1=CC(=N\C\1=C/c1[nH]c(C)cc1C)c1cc2ccccc2[nH]1	CID:66751253	phase I
BRD-K16149111	C\C=C\c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)NC1CCCCC1	CID:60185027	phase I
BRD-K16274875	O=C(C1CC1)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cncnc1	CID:60185283	phase I
BRD-K16329066	Fc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3ccccn3)C[C@@H]1N2	CID:60185130	phase I
BRD-K16425675	COc1ccccc1NC(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60185248	phase I
BRD-K16798053	O=C/1NC(=S)N(C(=O)\C1=C\c2c[nH]c3ccccc23)c4cccc5ccccc45	CID:1104457	phase I
BRD-K16971439	CS(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccccc1	CID:60185024	phase I
BRD-K17070436	COc1ccccc1CN1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60185168	phase I
BRD-K17203693	Fc1cccc(F)c1S(=O)(=O)N[C@H]2CC[C@H](CNS(=O)(=O)c3ccc4OCCOc4c3)CC2	CID:44142072	phase I
BRD-K17349619	CN(C)CCCNc1c2ccccc2n(C)c2nc(=O)n(C)c(=O)c12	CID:135403620	phase I
BRD-K18359792	Fc1ccccc1S(=O)(=O)N1C[C@@H]2N[C@H](C1)[C@@H]2c1ccc(cc1)-c1cncnc1	CID:60185002	phase I
BRD-K18433151	C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(\C=C\c2ccccc2)cc1)c1cocn1	CID:60184831	phase I
BRD-K18598482	Fc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CC1	CID:60185081	phase I
BRD-K18772134	C\C=C\c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1ccccc1C(F)(F)F	CID:71759505	phase I
BRD-K19112099	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccccc1F	CID:60188251	phase I
BRD-K19873942	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3nccs3)C[C@@H]1N2	CID:60185005	phase I
BRD-K20351658	Fc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)NC1CCCCC1	CID:60185157	phase I
BRD-K20585111	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc(F)cc1	CID:60185030	phase I
BRD-K20898254	C\C=C\c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:60184862	phase I
BRD-K21154786	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccccc1F	CID:60184961	phase I
BRD-K21501851	CCCNC(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cccc(F)c1	CID:60184827	phase I
BRD-K21569926	C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cncnc1)c1ccc2OCOc2c1	CID:60185455	phase I
BRD-K22330909	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3ccccn3)C[C@@H]1N2	CID:60185012	phase I
BRD-K22649335	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc2OCOc2c1	CID:60184957	phase I
BRD-K22901619	CC[C@]12CC[C@H]3[C@@H](CCC4=CC(CC[C@H]34)=NO)[C@H]1CC[C@@]2(OC(C)=O)C#C	CID:73707471	phase I
BRD-K23172979	Fc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1cncnc1	CID:60182620	phase I
BRD-K24049756	CN(C)CC(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccccc1F	CID:60184910	phase I
BRD-K25082699	Fc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1ccc2OCOc2c1	CID:60185128	phase I
BRD-K25089649	O=C(Cc1ccccc1)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60184997	phase I
BRD-K25161260	CN(C)CC(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cccc(C)c1	CID:60185109	phase I
BRD-K25228014	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)Cc1ccccc1	CID:60184832	phase I
BRD-K25380480	Fc1ccc(cc1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60184850	phase I
BRD-K25510697	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1cn(C)cn1	CID:60185082	phase I
BRD-K25682970	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccccc1F	CID:60185272	phase I
BRD-K27304876	Fc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccc(Cl)cc1	CID:60185175	phase I
BRD-K27530838	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1cnccn1	CID:60184855	phase I
BRD-K27638907	COc1ccccc1CN1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60188256	phase I
BRD-K27760381	COc1cc(CN2[C@H]3CNC[C@@H]2[C@@H]3c2ccc(cc2)-c2ccc(C)cc2)cc(OC)c1	CID:60185010	phase I
BRD-K28029915	O=C(O[C@H]1C[C@H]2C[C@H]3C[C@@H](C1)N2CC3=O)c1c[nH]c2ccccc12	CID:3033818	phase I
BRD-K28162668	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1ccncc1	CID:60185149	phase I
BRD-K28563387	Fc1ccc(NC(=O)N2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(\C=C\c3ccccc3)cc2)cc1	CID:60185171	phase I
BRD-K28667196	COc1cc(ccc1O)C(=O)O[C@@H]2C[C@@H]3CC[C@H](C2)N3C	CID:933171	phase I
BRD-K29733039	CO[C@@H]1C[C@H](C[C@@H](C)[C@@H]2CC(=O)[C@H](C)\C=C(C)\[C@@H](O)[C@@H](OC)C(=O)[C@H](C)C[C@H](C)\C=C\C=C/C=C(C)/[C@H](C[C@@H]3CC[C@@H](C)[C@@](O)(O3)C(=O)C(=O)N3CCCC[C@H]3C(=O)O2)OC)CC[C@H]1OP(C)(C)=O	CID:74787553	phase I
BRD-K30015724	Fc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3ccccc3)C[C@@H]1N2	CID:60185229	phase I
BRD-K30160673	Fc1cccc(CN2C[C@H]3N[C@@H](C2)[C@@H]3c2ccc(cc2)-c2cncnc2)c1	CID:60185457	phase I
BRD-K30415102	C\C=C\c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1cccc(F)c1	CID:60184838	phase I
BRD-K30958256	COc1cc(CN2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(\C=C\c3ccccc3)cc2)cc(OC)c1	CID:60185096	phase I
BRD-K31274539	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(C)(=O)=O	CID:60185139	phase I
BRD-K31484631	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2C4=NC5(CCN(CC(C)C)CC5)NC4=C(NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)C(=O)c2c(O)c3C	CID:135398743	phase I
BRD-K31898736	COc1ccccc1NC(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:60185004	phase I
BRD-K32053286	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1cccnc1	CID:60184849	phase I
BRD-K32605960	O=C(N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(\C=C\c2ccccc2)cc1)c1cnccn1	CID:60185281	phase I
BRD-K33018174	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3ccc4OCOc4c3)C[C@@H]1N2	CID:60185029	phase I
BRD-K33453211	C[C@@H]1CN(CC[C@]1(C(O)=O)c1ccccc1)[C@H]1CC[C@](CC1)(C#N)c1ccc(F)cc1	CID:54385	phase I
BRD-K33462580	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc(Cl)cc1	CID:60184999	phase I
BRD-K33631051	CCCNC(=O)N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1ccc(C)cc1	CID:60185105	phase I
BRD-K34205220	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CCC1	CID:71760038	phase I
BRD-K34404444	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccccn1	CID:60185150	phase I
BRD-K34776109	CCC1=C(C)CN(C(=O)NCCc2ccc(cc2)S(=O)(=O)NC(=O)N[C@H]2CC[C@H](C)CC2)C1=O	CID:3476	phase I
BRD-K34812979	Fc1ccc(CN2[C@H]3CNC[C@@H]2[C@H]3c2ccc(cc2)-c2ccccc2)cc1	CID:60185254	phase I
BRD-K34816161	C(N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(\C=C\c2ccccc2)cc1)c1nccs1	CID:60185025	phase I
BRD-K35376105	O=C(N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cccc(c1)C#N)c1ccc2OCOc2c1	CID:60184852	phase I
BRD-K35410462	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3cocn3)C[C@@H]1N2	CID:60184835	phase I
BRD-K35862891	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Cc1ccncc1	CID:60185251	phase I
BRD-K36337571	COc1cccc(CN2[C@H]3CNC[C@@H]2[C@@H]3c2ccc(cc2)-c2ccccc2C)c1	CID:60184856	phase I
BRD-K37291743	O=C(C1CCCCC1)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60185279	phase I
BRD-K37306336	O=C(C1CCOCC1)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60185170	phase I
BRD-K37477851	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccccc1F	CID:60184949	phase I
BRD-K37584671	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccc(C)cc1	CID:60184881	phase I
BRD-K37795473	O=C(N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(\C=C\c2ccccc2)cc1)c1ccc2OCOc2c1	CID:60185158	phase I
BRD-K38181288	N#Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3cocn3)C[C@@H]1N2	CID:60185558	phase I
BRD-K38369496	C\C=C\c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1c(C)noc1C	CID:60184984	phase I
BRD-K38720323	NCCCn1c2cc(Cl)ccc2sc2cc(=O)c(=O)cc12	CID:125595	phase I
BRD-K39529907	Fc1ccc(cc1)C(=O)N1C[C@@H]2N[C@H](C1)[C@H]2c1ccc(cc1)-c1cccnc1	CID:60185169	phase I
BRD-K39658422	Fc1ccccc1NC(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccncc1	CID:60185107	phase I
BRD-K39812290	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccccc1Cl	CID:60184878	phase I
BRD-K40174747	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccc(C)cc1	CID:60185006	phase I
BRD-K40223625	Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc(F)cc1	CID:60185152	phase I
BRD-K40258090	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H]2CNC[C@@H]1N2	CID:60184962	phase I
BRD-K40530731	CN1[C@H]2CC[C@@H]1C[C@@H](C2)OC(=O)[C@H](CO)c3ccccc3	CID:154417	phase I
BRD-K40675267	FC(F)(F)c1ccccc1CN1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccncc1	CID:60185023	phase I
BRD-K41031205	Cc1ccccc1S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:71296075	phase I
BRD-K41824522	Clc1ccc2sc3c([nH]c2c1)c(=O)ccc3=O	CID:73707581	phase I
BRD-K41953699	COc1ccccc1NC(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cccc(c1)C#N	CID:60184908	phase I
BRD-K42843595	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccc(cc1)C(F)(F)F	CID:60185129	phase I
BRD-K42916718	COc1cccc(c1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:60184884	phase I
BRD-K43022624	C\C=C\c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)NC1CCCCC1	CID:60185228	phase I
BRD-K43379283	Clc1ccc(NC(=O)N2[C@H]3CNC[C@@H]2[C@H]3c2ccc(cc2)-c2ccc(cc2)C#N)cc1	CID:60184876	phase I
BRD-K43528099	O=C(C1CCOCC1)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccncc1	CID:60185176	phase I
BRD-K43571060	CC(=O)c1ccc(/N=N/C(=C\2/NC(C)(C)Cc3ccccc23)/C(=O)N)cc1	CID:3429861	phase I
BRD-K44289311	COc1cc(CN2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2ccc(cc2)C#N)cc(OC)c1	CID:60185135	phase I
BRD-K44353683	CC(C)[C@H]1CC[C@@H](CC1)C(=O)N[C@H](Cc1ccccc1)C(O)=O	CID:5311309	phase I
BRD-K45223163	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccccc1C	CID:60184880	phase I
BRD-K45347683	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1ccc(F)cc1	CID:60185054	phase I
BRD-K46378421	O=S(=O)(Cc1ccccc1)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60185001	phase I
BRD-K46808525	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3cccc(F)c3)C[C@@H]1N2	CID:60184833	phase I
BRD-K47342144	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3ccccc3F)C[C@@H]1N2	CID:60184882	phase I
BRD-K47692589	Cc1ccccc1S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60188272	phase I
BRD-K48528505	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2CC1CCCCC1	CID:60185132	phase I
BRD-K48545167	C(N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccccc1)c1cc(on1)-c1ccccc1	CID:60184981	phase I
BRD-K48774739	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccc2OCOc2c1	CID:60185136	phase I
BRD-K48932581	NC[C@H]1CC[C@@H](CC1)C(=O)Oc2ccc(CCC(=O)O)cc2	CID:2680	phase I
BRD-K49047603	Fc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CCOCC1	CID:60185104	phase I
BRD-K49066776	COc1ccc(NC(=O)N2C[C@H]3N[C@@H](C2)[C@@H]3c2ccc(cc2)-c2ccncc2)cc1	CID:60185253	phase I
BRD-K49075727	COC(=O)c1ccc2c(NC(=O)\C2=C(/Nc2ccc(cc2)N(C)C(=O)CN2CCN(C)CC2)c2ccccc2)c1	CID:135423438	phase I
BRD-K49849398	O=C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccc(cc1)C#N)c1ccncc1	CID:60185057	phase I
BRD-K49870009	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1ccccn1	CID:60185079	phase I
BRD-K49881099	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1ccncc1	CID:60185250	phase I
BRD-K49961249	C(N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1cccnc1)c1ccccn1	CID:60185155	phase I
BRD-K50281141	Fc1cccc(NC(=O)N2[C@H]3CNC[C@@H]2[C@H]3c2ccc(cc2)-c2cccc(c2)C#N)c1	CID:60191786	phase I
BRD-K50866992	CN1[C@H]2CC[C@@H]1C[C@@H](C2)OC(=O)c3c[nH]c4ccccc34	CID:656665	phase I
BRD-K51166678	C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cccnc1)c1ccc2OCOc2c1	CID:60184853	phase I
BRD-K51911655	C(C1CC1)N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1cccnc1	CID:60184987	phase I
BRD-K52136013	CN(C)CC(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60185205	phase I
BRD-K52468146	CCCNC(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccc(OC)cc1	CID:60185125	phase I
BRD-K52870470	Fc1ccc(cc1)C(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccccc1F	CID:60184976	phase I
BRD-K52882725	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1cnccn1	CID:60184977	phase I
BRD-K52913754	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1ccccc1F	CID:60185097	phase I
BRD-K53665955	OC(=O)[C@@]1(Cc2cccc(Nc3nccs3)n2)CC[C@@H](CC1)Oc1cccc(Cl)c1F	CID:24748204	phase I
BRD-K53955171	Cc1cccc(c1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cncnc1	CID:60185280	phase I
BRD-K54127914	COc1ccccc1CN1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccncc1	CID:60184964	phase I
BRD-K55216615	Fc1cccc(F)c1S(=O)(=O)[C@H]2CC[C@H](CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:44142158	phase I
BRD-K55996983	C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccncc1)c1nccs1	CID:60184859	phase I
BRD-K59899596	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccc(C)cc1	CID:60184841	phase I
BRD-K60260474	O=C(C1CCCC1)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cncnc1	CID:60186754	phase I
BRD-K60341033	Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CNC[C@@H]1N2	CID:60184980	phase I
BRD-K60393413	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H]2CN(Cc3cccc(OC)c3)C[C@@H]1N2	CID:60188214	phase I
BRD-K60474245	COc1cccc(CN2C[C@H]3N[C@@H](C2)[C@@H]3c2ccc(\C=C\C)cc2)c1	CID:60184937	phase I
BRD-K61847735	N#Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CNC[C@@H]1N2	CID:60184851	phase I
BRD-K62200616	Fc1cccc(NC(=O)N2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2cncnc2)c1	CID:60184983	phase I
BRD-K62695275	Fc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccccn1	CID:60185200	phase I
BRD-K62982419	COc1ccc(cc1OC1CCCC1)[C@@]1(CC[C@@H](CC1)C(O)=O)C#N	CID:151170	phase I
BRD-K63325940	C\C=C\c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2C(=O)Nc1ccccc1Cl	CID:60184861	phase I
BRD-K64517075	Cc1cc(O)c2C(=O)c3c(O)cc(O)c4C(=O)C(C)(C)c5cc(O)c1c2c5-c34	CID:135430323	phase I
BRD-K64639565	COc1ccccc1CN1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1cccnc1	CID:60185231	phase I
BRD-K65003634	COc1ccccc1NC(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccccc1C	CID:60185134	phase I
BRD-K65044501	Cc1cccc(c1)S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccccc1C	CID:60185153	phase I
BRD-K65395967	O=C(Nc1ccc2OCOc2c1)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccc(cc1)C#N	CID:60185133	phase I
BRD-K65402741	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)C1CCC1	CID:60185172	phase I
BRD-K65416438	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccccn1	CID:60184935	phase I
BRD-K65567503	COc1ccccc1CN1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cccnc1	CID:60185388	phase I
BRD-K65857447	Cc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccc(C)cc1	CID:60184717	phase I
BRD-K66968629	ONC(=O)c1ccc(cc1)\N=N\c1ccc(cc1)C(O)=O	CID:73707540	phase I
BRD-K67074672	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Nc1ccccc1F	CID:60185249	phase I
BRD-K68338581	O=C(N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1cccc(c1)C#N)c1cccnc1	CID:60185008	phase I
BRD-K68496959	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Nc1ccccc1F	CID:60184936	phase I
BRD-K68804560	CN1[C@H]2CC[C@@H]1C[C@@H](C2)OC(c1ccccc1)c1ccccc1	CID:1201549	phase I
BRD-K70165037	CN(C)CC(=O)N1C[C@@H]2N[C@H](C1)[C@H]2c1ccc(cc1)-c1ccncc1	CID:60184950	phase I
BRD-K70557564	O[C@@H](COc1cccc2ncccc12)CN1CCN(CC1)[C@@H]1c2ccccc2[C@@H]2[C@H](c3ccccc13)C2(F)F	CID:3036703	phase I
BRD-K71140693	Fc1cccc(F)c1S(=O)(=O)N[C@H]2CC[C@H](CC2)NS(=O)(=O)c3ccc4OCCOc4c3	CID:25243776	phase I
BRD-K71380401	CCc1ccc2NC(=O)/C(=C/3\NC(=S)NC3=O)/c2c1	CID:750586	phase I
BRD-K71515738	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccc(F)cc1	CID:60184982	phase I
BRD-K72567746	C(N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(\C=C\c2ccccc2)cc1)c1cncnc1	CID:60185282	phase I
BRD-K73368362	CN(C)Cc1cccc(N\C(c2ccccc2)=C2/C(=O)Nc3cc(ccc23)C(=O)N(C)C)c1	CID:135659062	phase I
BRD-K74133369	CC[C@H]1CC[C@@H]2O[C@]3(CC[C@@H](C)[C@@H](C[C@@H](C)O)O3)[C@H](C)[C@H](OC(=O)\C=C\[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@](C)(O)[C@H](O)[C@@H](C)C\C=C\C=C\1)[C@H]2C	CID:73707429	phase I
BRD-K74415279	C\C=C\c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccc(Cl)cc1	CID:60185026	phase I
BRD-K74663820	C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1ccccc1)c1cccnc1	CID:60185278	phase I
BRD-K74728819	O=C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cncnc1)c1ccc2OCOc2c1	CID:60184998	phase I
BRD-K75449859	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)Cc1ccccc1	CID:60184828	phase I
BRD-K75907833	C(C1CCCCC1)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccncc1	CID:60184978	phase I
BRD-K76211354	C(N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(\C=C\c2ccccc2)cc1)c1ccc2OCOc2c1	CID:60185056	phase I
BRD-K77403604	FC(F)(F)c1cccc(CN2[C@H]3CNC[C@@H]2[C@H]3c2ccc(cc2)-c2cccnc2)c1	CID:60184933	phase I
BRD-K77537540	Cc1ccccc1S(=O)(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1cccnc1	CID:60184826	phase I
BRD-K77790153	N#Cc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3cocn3)C[C@@H]1N2	CID:60185137	phase I
BRD-K78132017	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccc(F)cc1	CID:60185151	phase I
BRD-K78197930	FC(F)(F)c1ccc(NC(=O)N2C[C@H]3N[C@@H](C2)[C@H]3c2ccc(cc2)-c2cccnc2)cc1	CID:60185173	phase I
BRD-K79259704	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(Cc3ccccn3)C[C@@H]1N2	CID:60185255	phase I
BRD-K79500219	Fc1cccc(c1)S(=O)(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccccc1F	CID:60185022	phase I
BRD-K80021597	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)CN1CCOCC1	CID:60185028	phase I
BRD-K80674743	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Cc1ccncc1	CID:60185202	phase I
BRD-K81146569	Fc1ccc(NC(=O)N2[C@H]3CNC[C@@H]2[C@H]3c2ccc(cc2)-c2cccnc2)cc1	CID:60184839	phase I
BRD-K81210389	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2S(=O)(=O)c1ccccc1	CID:60184877	phase I
BRD-K81311598	CN(C)CC(=O)N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)C1=CCCCC1	CID:60185102	phase I
BRD-K81600610	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3nccs3)C[C@@H]1N2	CID:60185147	phase I
BRD-K81793693	C\C=C\c1ccc(cc1)[C@H]1[C@@H]2CNC[C@H]1N2Cc1ccccn1	CID:60185230	phase I
BRD-K82091397	COc1nccc(n1)-c1c(ncn1[C@H]1CC[C@H](O)CC1)-c1ccc(F)cc1	CID:5166	phase I
BRD-K82189384	ONC(=O)c1ccc(cc1)\N=N\c1ccccc1	CID:73707539	phase I
BRD-K82670191	CS(=O)(=O)N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1ccccc1	CID:60184840	phase I
BRD-K83048312	CCCN1[C@H]2CN(Cc3ccc(F)cc3)C[C@@H]1[C@H]2c1ccccc1	CID:71500439	phase I
BRD-K83216866	C(C1CCOCC1)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(\C=C\c2ccccc2)cc1	CID:60185204	phase I
BRD-K83860226	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(Cc3ccc4OCOc4c3)C[C@@H]1N2	CID:60184955	phase I
BRD-K84085265	O[C@H]1CC[C@H](CC1)Nc1ncc2nc(Nc3c(F)cc(F)cc3F)n([C@@H]3CCOC3)c2n1	CID:57394468	phase I
BRD-K84658672	CC(C)[C@H]1CC[C@@H](CC1)C(=O)N[C@@H](Cc1ccccc1)C(O)=O	CID:60026	phase I
BRD-K84679731	C(C1CC1)N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1ccncc1	CID:60188138	phase I
BRD-K84687999	Clc1cccc(c1)S(=O)(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1cccnc1	CID:60184863	phase I
BRD-K84792586	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)Cc1ccccc1	CID:60185011	phase I
BRD-K85275009	COC(=O)c1scc2c(O)cc(nc12)C(F)(F)F	CID:2775426	phase I
BRD-K86595100	CNC1=Nc2ccc(Cl)cc2C(=[N+]([O-])C1)c3ccccc3	CID:2712	phase I
BRD-K87927861	COc1ccccc1S(=O)(=O)N1C[C@H]2N[C@@H](C1)[C@@H]2c1ccc(cc1)-c1cccnc1	CID:60184956	phase I
BRD-K87939627	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccccc1C	CID:60185003	phase I
BRD-K88769248	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)C(=O)c1cnccn1	CID:60185131	phase I
BRD-K89793492	COc1cccc(CN2[C@H]3CNC[C@@H]2[C@H]3c2ccc(cc2)-c2ccc(cc2)C#N)c1	CID:60184912	phase I
BRD-K89843224	CC(=O)N1C(=N)S/C(=C/c2cc3ccc(C)cc3nc2O)/C1=O	CID:136848705	phase I
BRD-K89923877	CN1[C@H]2C[C@@H](C[C@@H]1[C@H]1O[C@@H]21)OC(=O)[C@H](CO)c1ccccc1	CID:3000322	phase I
BRD-K90041565	C\C=C\c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)c1ccccc1F	CID:60184883	phase I
BRD-K91454871	C(N1C[C@H]2N[C@@H](C1)[C@H]2c1ccc(cc1)-c1ccncc1)c1ccccc1	CID:60185512	phase I
BRD-K91938660	C[C@@]1(C[C@@H]2C[C@]3(C)C1)C[C@](N)(C2)C3	CID:1263681	phase I
BRD-K92543914	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H]2CN(C[C@@H]1N2)S(=O)(=O)Cc1ccccc1	CID:60184911	phase I
BRD-K92571446	CC(C)n1cnc2c(Nc3cccc(NC(=O)C=C)c3)nc(N[C@H]3CC[C@@H](CC3)N(C)C)nc12	CID:42628507	phase I
BRD-K92902323	COc1cccc(CN2[C@H]3CNC[C@@H]2[C@@H]3c2ccc(\C=C\c3ccccc3)cc2)c1	CID:60184837	phase I
BRD-K93386351	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1cccc(F)c1	CID:60184836	phase I
BRD-K94003664	Fc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H]2CN(C[C@@H]1N2)C(=O)Cc1ccncc1	CID:60184858	phase I
BRD-K94294671	COc1cccc2cc([nH]c12)-c1nc([C@@H]2CC[C@@H](CC2)C(O)=O)n2ncnc(N)c12	CID:135398516	phase I
BRD-K98333955	Nc1ncnc2n(cc(-c3ccc(OCc4ccccc4)cc3)c12)[C@H]1C[C@H](CN2CCC2)C1	CID:46881851	phase I
BRD-K98481427	COc1ccc(cc1)S(=O)(=O)N1[C@H]2CNC[C@@H]1[C@H]2c1ccc(cc1)-c1ccncc1	CID:60185206	phase I
BRD-K99185973	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H]2CNC[C@H]1N2Cc1cccnc1	CID:60184948	phase I
BRD-K99818283	COc1ccc2C3=NCCN3C(=Nc2c1OC)NC(=O)c4cccnc4	CID:135398491	phase I
BRD-K99875147	CCCNC(=O)N1[C@H]2CNC[C@@H]1[C@@H]2c1ccc(cc1)-c1ccccc1F	CID:60184975	phase I
BRD-K03319035	CNCCC[C@]1(CC[C@H]2c3ccccc31)c4ccccc24	CID:4011	phase I
BRD-K17894950	O=C1Nc2ccccc2\C1=C1\Nc2ccccc2C1=O	CID:10177	phase I
BRD-K19136521	O\N=C1c2ccccc2NC/1=C1\C(=O)Nc2ccccc12	CID:3707	phase I
BRD-K29673530	Cc1cc(O)c2c3c1c1c(C)cc(O)c4c1c1c3c3c(c(O)cc(O)c3c2=O)c2c(O)cc(O)c(c12)c4=O	CID:3663	phase I
BRD-K31633810	CN1[C@H]2CC[C@@H]1C[C@@H](C2)OC(=O)N1Cc2ccccc2NC1=O	CID:16759155	phase I
BRD-K44084986	C[C@@H](N)[C@H]1CC[C@@H](CC1)C(=O)Nc1ccncc1	CID:448042	phase I
BRD-K56558538	Nc1c(Br)cc(Br)cc1CN[C@H]1CC[C@H](O)CC1	CID:2132	phase I
BRD-K68103045	COc1ccc(cc1)-n1nc2c3CCCCCc3[nH]cc2c1=O	CID:163844	phase I
BRD-A00474148	Oc1ccc(cc1)N1CCN(CC1)[S+]([O-])(=O)c1ccc2NC(=O)Cc2c1	CID:44825297	phase I
BRD-A04756508	CC[C@]12CCC3C(CCC4=C\C(CCC34)=N\O)C1CC[C@@]2(OC(C)=O)C#C	CID:98042564	phase I
BRD-A07029265	CC(C)[N+]1(C)C2CC[C@@H]1C[C@H](C2)OC(=O)C(CO)c3ccccc3	CID:5702074	phase I
BRD-A09539288	CN1C2CC[C@H]1C[C@H](C2)OC(=O)C(O)c1ccccc1	CID:5702065	phase I
BRD-A12832192	CN([N+][O-])C(=O)NC1C(O)OC(CO)C(O)C1O	CID:73707368	phase I
BRD-A13711138	OCC=C1C[N@+]2(CC=C)CC[C@@]34[C@@H]2C[C@@H]1C1=CN2C5C(=CN(C31)c1ccccc41)[C@@H]1C[C@@H]3[C@@]5(CC[N@@+]3(CC=C)CC1=CCO)c1ccccc21	CID:73707450	phase I
BRD-A13946108	CC1=C(CC(O)=O)c2cc(F)ccc2C\1=C/c1ccc(cc1)S(C)=O	CID:1548887	phase I
BRD-A19248578	C[C@H]1CC[C@@H]2C[C@H](C[C@@](O)(O2)C2CSC(=O)N2)OC(=O)\C=C(C)/CC\C=C/1	CID:16760044	phase I
BRD-A21072306	O[Hg]c1c(O)c(Br)cc2c1Oc3cc(O)c(Br)cc3C42OC(=O)c5ccccc54	CID:4564401	phase I
BRD-A23801136	CCC(C)N1CCC2(CC1)NC3=C4NC(=O)C(=CC=C[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(=O)C)[C@H](C)[C@@H](OC)C=CO[C@@]5(C)Oc6c(C5=O)c(C3=N2)c(C4=O)c(O)c6C)C	CID:135899465	phase I
BRD-A24421185	CCCC[N+]1(C)[C@H]2C[C@@H](C[C@@H]1[C@@H]1O[C@@H]21)OC(=O)[C@H](CO)c1ccccc1	CID:73707491	phase I
BRD-A25576662	CN([N+][O-])C(=O)N[C@H]1C(O)O[C@H](CO)[C@@H](O)[C@@H]1O	CID:73707422	phase I
BRD-A31836915	C[C@H](CNC(=O)CC[C@]1(C)[C@@H](CC(N)=O)[C@@H]2N=C1C(C)=C1N=C(C=C3N=C(C(C)=C4[C@@H](CCC(N)=O)[C@](C)(CC(N)=O)[C@@]2(C)N4[Co+]C#N)[C@@](C)(CC(N)=O)[C@@H]3CCC(N)=O)C(C)(C)[C@@H]1CCC(N)=O)OP(O)(=O)O[C@@H]1[C@@H](CO)O[C@@H]([C@@H]1O)n1cnc2cc(C)c(C)cc12	CID:73707516	phase I
BRD-A32595718	CC(C)(C)c1ccc2OCC(Oc2c1)C(=O)N\N=C\c1ccc[nH]1	CID:135550902	phase I
BRD-A33973768	C[N+]1([O-])[C@H]2C[C@@H](C[C@@H]1[C@@H]1O[C@@H]21)OC(=O)[C@H](CO)c1ccccc1	CID:73707515	phase I
BRD-A35782587	COC(=O)CCc1c(C)c2cc3nc(cc4[nH]c(cc5nc(cc1[nH]2)c(CCC(O)=O)c5C)c(C=C)c4C)C1=CC=C(C(C(=O)OC)[C@@]31C)C(=O)OC	CID:11980942	phase I
BRD-A37432947	CC(C)[N+]1(C)[C@@H]2CC[C@@H]1C[C@H](C2)OC(=O)C(CO)c3ccccc3	CID:43232	phase I
BRD-A37444045	NN=C1N=NC=C2C=CC=CC12	CID:6852378	phase I
BRD-A38161572	Clc1ccc(cc1)[C@H]1CCC(CC1)C1C(=O)C(=O)c2ccccc2C1=O	CID:44483269	phase I
BRD-A48349196	CNCCCN1c2ccccc2S(=O)c2ccc(Cl)cc12	CID:11723560	phase I
BRD-A49906757	C[N+]1([O-])[C@H]2C[C@@H](C[C@@H]1[C@H]1O[C@@H]21)OC(=O)[C@H](CO)c1ccccc1	CID:3000667	phase I
BRD-A52627843	CCC(C)[C@@H]1N[C@@H]2C=Cc3c(cc(nc3[C@H]2O)C(=O)O[C@H](C)[C@@H]2NC(=O)c3csc(n3)[C@@H](NC(=O)[C@H]3CSC(=N3)C(NC(=O)[C@@H](NC(=O)c3csc(n3)[C@]3(CCC(=N[C@H]3c3csc2n3)c2nc(cs2)C(=O)NC(=C)C(=O)NC(=C)C(N)=O)NC(=O)[C@H](C)NC(=O)C(=C)NC(=O)[C@H](C)NC1=O)[C@@H](C)O)=CC)[C@@](C)(O)[C@@H](C)O)[C@H](C)O	CID:146170498	phase I
BRD-A52933579	CN1C2CC[C@@H]1C[C@H](C2)OC(c1ccc(Br)cc1)c1ccc(Br)cc1	CID:73707558	phase I
BRD-A56892734	COc1ccc2n([Mg]n3c(nc4cc(OC)ccc34)S(=O)Cc5ncc(C)c(OC)c5C)c(nc2c1)S(=O)Cc6ncc(C)c(OC)c6C	CID:5311083	phase I
BRD-A58564983	CO[C@H]1CC(O[C@H]2[C@@H](C)\C=C\C=C3/CO[C@@H]4C(=N/O)\C(C)=C[C@@H](C(=O)O[C@H]5C[C@@H](C\C=C2/C)O[C@@]2(CC[C@H](C)[C@H](O2)C2CCCCC2)C5)[C@]34O)O[C@@H](C)C1O	CID:98042561	phase I
BRD-A62035778	CN1C2C[C@@H](C[C@H]1[C@H]1OC21)OC(=O)[C@H](CO)c1ccccc1	CID:5702114	phase I
BRD-A65145453	CC(C)(C)c1onc(O)c1CC(N)C(O)=O	CID:2253	phase I
BRD-A65516924	OC(=O)c1ccc(cc1)N1CCN(CC1)[S+]([O-])(=O)c1ccc2NC(=O)Cc2c1	CID:44825310	phase I
BRD-A70541707	CN(C)CC(O)Cn1c2cc(Cl)ccc2sc2cc(=O)c(=O)cc12	CID:12321145	phase I
BRD-A73513677	CC(=N)C(C#N)C(=O)COC(=O)c1cc(C)n(c1C)c2ccc(F)cc2	CID:40619681	phase I
BRD-A74975734	CN1[C@H]2CC[C@@H]1C[C@@H](C2)OC(=O)C(O)c3ccccc3	CID:5282593	phase I
BRD-A78303415	CN1C2CC[C@@H]1C[C@H](C2)OC(=O)[C@H](CO)c1ccccc1	CID:5318386	phase I
BRD-A78360835	COc1c(O)c2c(=O)cc3OCOc4cc(O)c5c(=O)c(OC)c(CC(C)O)c6c(c1CC(C)O)c2c3c4c56	CID:2674	phase I
BRD-A79465854	CCP(CC)(CC)=[Au]SC1CC(OC(C)=O)C(OC(C)=O)C(OC(C)=O)C1OC(C)=O	CID:177748840	phase I
BRD-A79768653	COC1CC(CC(C)C2CC(=O)C(C)\C=C(C)\C(O)C(OC)C(=O)C(C)CC(C)\C=C\C=C\C=C(C)\C(CC3CCC(C)C(O)(O3)C(=O)C(=O)N3CCCCC3C(=O)O2)OC)CCC1O	CID:5374464	phase I
BRD-A81541225	CCC1CCC2OC3(CC[C@@H](C)C(C[C@H](C)O)O3)[C@H](C)C(OC(=O)\C=C\[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@H](C)C(=O)[C@@](C)(O)[C@H](O)[C@@H](C)C\C=C\C=C\1)[C@H]2C	CID:6364620	phase I
BRD-A82976242	O=Cc1ccc(cc1)N1CCN(CC1)[S+]([O-])(=O)c1ccc2NC(=O)Cc2c1	CID:44825307	phase I
BRD-A83892713	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c(O)c(\C=N\N4CCN(C)CC4)c(NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c(O)c2c(O)c3C	CID:135550179	phase I
BRD-A84282119	CC(N)[C@]12C[C@H]3C[C@H](C[C@@H](C3)C1)C2	CID:5071	phase I
BRD-A98175426	CC(=O)O[C@H]1C(OC=C(C)C(O)=O)C(C)(C)CC2C3=CCC4C5(C)CCC(OC6O[C@@H]([C@@H](O[C@@H]7O[C@H](CO)[C@@H](O)[C@H](O)[C@H]7O)[C@H](O)[C@H]6O[C@@H]6O[C@H](CO)[C@@H](O)[C@H](O)[C@H]6O)C(O)=O)[C@](C)(CO)C5CCC4(C)[C@]3(C)C[C@@H](O)C12CO	CID:73707521	phase I
BRD-A98838152	COc1cccc(C(=O)N[C@@H]2CC3CC[C@H](C2)N3Cc2ccccc2)c1OC	CID:73707589	phase I
BRD-K57631554	NCC(=O)CCC(O)=O	CID:137	phase I
BRD-K77914232	CC=O	CID:177	phase I
BRD-K87070823	CC(N)=O	CID:178	phase I
BRD-K82381502	CC(=O)OCC[N+](C)(C)C	CID:187	phase I
BRD-A67373739	NC(=O)c1ncn(C2OC(COP(O)(O)=O)C(O)C2O)c1N	CID:200	phase I
BRD-A96407378	NC(=O)NC1NC(=O)NC1=O	CID:204	phase I
BRD-A45889380	CCN(CC)CCCC(C)Nc1c2ccc(Cl)cc2nc2ccc(OC)cc12	CID:237	phase I
BRD-K53397409	OC(=O)c1ccccc1	CID:243	phase I
BRD-A51182606	OCC(NC(=O)C(Cl)Cl)C(O)c1ccc(cc1)[N+](=O)[O-]	CID:298	phase I
BRD-A68045637	ClC1(C(=O)C2(Cl)C3(Cl)C14Cl)C5(Cl)C2(Cl)C3(Cl)C(Cl)(Cl)C45Cl	CID:299	phase I
BRD-K23913458	O=c1ccc2ccccc2o1	CID:323	phase I
BRD-K77345217	OC(=O)c1cc(O)c(O)c(O)c1	CID:370	phase I
BRD-A24543851	C1CNC(C1)c1cccnc1	CID:412	phase I
BRD-A05186015	CC(NC(C)(C)C)C(=O)c1cccc(Cl)c1	CID:444	phase I
BRD-A60070924	CC12CCC3C(CCc4cc(O)ccc34)C1CCC2O	CID:450	phase I
BRD-A35258977	OCC(O)C(O)C(O)C(O)CO	CID:453	phase I
BRD-K96282009	COc1ccccc1O	CID:460	phase I
BRD-A77577770	CCCCCCCCCCCCCCCC(=O)OC(CC(O)=O)C[N+](C)(C)C	CID:462	phase I
BRD-A47441220	CC(O)(CCOP(O)(O)=O)CC(O)=O	CID:476	phase I
BRD-K64931368	NCCCCCC(O)=O	CID:564	phase I
BRD-A18929998	Nc1ccn(C2OC(CO)C(O)C2O)c(=O)n1	CID:596	phase I
BRD-K43887077	NCCc1ccc(O)c(O)c1	CID:681	phase I
BRD-K73866522	OCC(O)CO	CID:753	phase I
BRD-A07765530	CNCC(O)c1ccc(O)c(O)c1	CID:838	phase I
BRD-A74642112	NC(Cc1cc(I)c(Oc2ccc(O)c(I)c2)c(I)c1)C(=O)O	CID:861	phase I
BRD-K97530723	COc1ccc2[nH]cc(CCNC(C)=O)c2c1	CID:896	phase I
BRD-A79058669	CNCC(O)c1ccccc1	CID:913	phase I
BRD-A94669766	Oc1ccc(cc1)C2CC(=O)c3c(O)cc(O)cc3O2	CID:932	phase I
BRD-K28912512	NC(=O)c1cccnc1	CID:936	phase I
BRD-K60237333	OC(=O)c1cccnc1	CID:938	phase I
BRD-A91555231	NCC(O)c1ccc(O)c(O)c1	CID:951	phase I
BRD-K50711164	Oc1c(Cl)c(Cl)c(Cl)c(Cl)c1Cl	CID:992	phase I
BRD-A19232309	CC(O)CO	CID:1030	phase I
BRD-K28667793	NC(=O)c1cnccn1	CID:1046	phase I
BRD-K14349461	Cc1ncc(CO)c(CO)c1O	CID:1054	phase I
BRD-A64479082	COc1ccc2nccc(C(O)C3CC4CCN3CC4C=C)c2c1	CID:1065	phase I
BRD-K64634304	CC(=CCO)C=CC=C(C)C=CC1=C(C)CCCC1(C)C	CID:1071	phase I
BRD-K40438880	NCCCCNCCCN	CID:1102	phase I
BRD-K95785345	Cc1c(CCO)sc[n+]1Cc1cnc(C)nc1N	CID:1130	phase I
BRD-A07106394	NC(Cc1c[nH]c2ccccc12)C(=O)O	CID:1148	phase I
BRD-A61899133	OC1Cc2c(O)cc(O)cc2OC1c3ccc(O)c(O)c3	CID:1203	phase I
BRD-A39268308	Clc1ccc(cn1)C2CC3CCC2N3	CID:1204	phase I
BRD-A09828896	Oc1cc2C(CNCCc2c(Cl)c1O)c1ccccc1	CID:1218	phase I
BRD-A18795974	CCCN(CCC)C1CCc2ccc(O)cc2C1	CID:1219	phase I
BRD-A04438777	Oc1cc2C(CN(CC=C)CCc2c(Cl)c1O)c3ccccc3	CID:1225	phase I
BRD-A62336480	COC(=O)C1=C(C)NC(=C(C1c2cccc(c2)[N+](=O)[O-])C(=O)OCCCN3CCC(CC3)(c4ccccc4)c5ccccc5)C	CID:1236	phase I
BRD-A64227845	Oc1cc2CCN(CC=C)CC(c3ccccc3)c2cc1O	CID:1241	phase I
BRD-A52588987	CN1CCc2cc(Br)c(O)cc2C(C1)c1ccccc1	CID:1243	phase I
BRD-A85280935	CCCN1CCCC2Cc3n[nH]cc3CC21	CID:1257	phase I
BRD-A80383043	NC(C(O)=O)c1ccc(C(O)=O)c(O)c1	CID:1297	phase I
BRD-A87719232	COc1ccc2cc(ccc2c1)C(C)C(=O)O	CID:1302	phase I
BRD-K27305388	C[N+]1(C)CCN(CC1)c2ccccc2	CID:1316	phase I
BRD-A41451487	CCC(C)N(C)C(=O)c1cc2ccccc2c(n1)-c1ccccc1Cl	CID:1345	phase I
BRD-K90524085	Clc1cccc(Nc2nnc(-c3ccccc3)c3ccccc23)c1	CID:1348	phase I
BRD-K36965586	NC(=N)NC(=N)Nc1cccc(Cl)c1	CID:1354	phase I
BRD-K47598052	Cc1ccc(cc1)-c1nn(c2ncnc(N)c12)C(C)(C)C	CID:1400	phase I
BRD-K97764662	CCN(CC)CCCCNc1ncc2cc(-c3cc(OC)cc(OC)c3)c(NC(=O)NC(C)(C)C)nc2n1	CID:1401	phase I
BRD-K26015241	O=c1onc2cnc3ccccc3n12	CID:1456	phase I
BRD-K08554278	CCOc1ccc(cc1)c2nc3cc(ccc3[nH]2)c4nc5cc(ccc5[nH]4)N6CCN(C)CC6	CID:1464	phase I
BRD-A28318179	CC1CCN=C(N)S1	CID:1534	phase I
BRD-A94451536	CCCCCCCCCCCCCCC(F)C(=O)O	CID:1560	phase I
BRD-A27924917	NCC(O)(CS(O)(=O)=O)c1ccc(Cl)cc1	CID:1564	phase I
BRD-A64933752	Nc1nc(Nc2ccccc2)nc3n(cnc13)C4OC(CO)C(O)C4O	CID:1585	phase I
BRD-K32598858	Nc1nc[nH]n1	CID:1639	phase I
BRD-K08703257	NC(=O)c1cccc(N)c1	CID:1645	phase I
BRD-K61463582	Cc1ccc2cc3c(ccc4ccccc43)c5CCc1c52	CID:1674	phase I
BRD-A85587465	CN1C2CCC1CC(C2)OC(=O)c1cc(Cl)cc(Cl)c1	CID:1683	phase I
BRD-A76941896	COc1cccc2C(=O)c3c(O)c4CC(O)(CC(OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(=O)CO	CID:1691	phase I
BRD-K97118047	Brc1c(Br)c(Br)c2[nH]nnc2c1Br	CID:1694	phase I
BRD-K13087974	O=C1NC(=O)c2cc(Nc3ccccc3)c(Nc3ccccc3)cc12	CID:1697	phase I
BRD-K50214219	Nc1ccc2C(=O)NC(=O)c3cccc1c32	CID:1720	phase I
BRD-K28168037	CC(=CC=CC(=CC(=O)Nc1ccc(O)cc1)C)C=CC2=C(C)CCCC2(C)C	CID:1744	phase I
BRD-K55930204	O=C1NC(=O)C(N1)(c1ccccc1)c1ccccc1	CID:1775	phase I
BRD-K06080977	CCCCCC#CCC#CCC#CCC#CCCCC(=O)O	CID:1780	phase I
BRD-K40990712	NC(=N)NC(=O)c1nc(Cl)c(nc1N)N2CCCCCC2	CID:1794	phase I
BRD-K08219523	CCCCCCCCCOc1ccc2[nH]cc(CCN)c2c1	CID:1797	phase I
BRD-A18497530	Nc1ncnc2n(cc(I)c12)C3OC(CO)C(O)C3O	CID:1830	phase I
BRD-K30197592	COc1ccc2[nH]cc(CCN)c2c1	CID:1833	phase I
BRD-K53815609	NC(=O)NN=Cc1ccc(o1)[N+](=O)[O-]	CID:1839	phase I
BRD-K11163873	O=c1[nH]c2ccccc2c3ccccc13	CID:1853	phase I
BRD-A42187224	NCC(O)c1cc(O)c(O)cc1F	CID:1862	phase I
BRD-K00184207	O=Cc1c2[nH]c3ccccc3c2cc4[nH]c5ccccc5c14	CID:1863	phase I
BRD-K83064458	Cn1c2ncn(CCO)c2c(=O)n(C)c1=O	CID:1892	phase I
BRD-K04430056	[O-][N+](=O)c1cccc2cn[nH]c12	CID:1893	phase I
BRD-A52771319	Nc1ncnc2n(C3OC4COP(=O)(O)OC4C3O)c(Br)nc12	CID:1913	phase I
BRD-K81473089	Nc1c2CCCCc2nc2ccccc12	CID:1935	phase I
BRD-K32188552	CC(C)(C(N)=N)\N=N\C(C)(C)C(N)=N	CID:1969	phase I
BRD-A29260609	CCCC(=O)Nc1ccc(OCC(O)CNC(C)C)c(c1)C(C)=O	CID:1978	phase I
BRD-A80567352	CC(=O)OC1CN2CC[C@H]1CC2	CID:1979	phase I
BRD-K67563174	COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)OCC(O)=O)c2c1	CID:1981	phase I
BRD-K41524689	CC(=O)Nc1ccc(O)cc1	CID:1983	phase I
BRD-K43457670	CC(=O)Nc1nnc(s1)S(N)(=O)=O	CID:1986	phase I
BRD-K52960356	CC(=O)c1ccc(cc1)S(=O)(=O)NC(=O)NC1CCCCC1	CID:1989	phase I
BRD-K33483813	CC(=O)Nc1ccc(CC(O)=O)cc1	CID:2018	phase I
BRD-A42383464	CC(C)C1NC(=O)C(NC(=O)c2ccc(C)c3oc4c(C)c(=O)c(N)c(C(=O)NC5C(C)OC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C6CCCN6C(=O)C(NC5=O)C(C)C)c4nc23)C(C)OC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C7CCCN7C1=O	CID:2019	phase I
BRD-K60907894	CCN(CC)CCOC(=O)C(c1ccccc1)c1ccccc1	CID:2031	phase I
BRD-K67506692	Oc1cc(C=C(C#N)C#N)ccc1[N+](=O)[O-]	CID:2046	phase I
BRD-K57926513	Cc1cc2ncc(nc2cc1C)c3ccccc3	CID:2048	phase I
BRD-K76064317	COc1cc2ncc(nc2cc1OC)-c1ccccc1	CID:2049	phase I
BRD-K68336408	COc1cc2ncnc(Nc3cccc(Cl)c3)c2cc1OC	CID:2051	phase I
BRD-K49657628	Oc1ccc(C=C(C#N)C#N)cc1O	CID:2052	phase I
BRD-K81209512	Oc1ccc(C=C(C#N)C(=O)Nc2ccccc2)cc1O	CID:2055	phase I
BRD-K72783841	Oc1ccc(C=C(C#N)C(=O)NCCCc2ccccc2)cc1O	CID:2058	phase I
BRD-K14441456	Oc1ccc(C=C(C#N)C(=O)NCCCCc2ccccc2)cc1O	CID:2059	phase I
BRD-K03670461	Oc1cc(C=C(C#N)C#N)cc(O)c1O	CID:2061	phase I
BRD-K08132273	COc1cc(C=C(C#N)C(=O)N)cc(CSc2nc3ccccc3s2)c1O	CID:2062	phase I
BRD-K41996876	COc1ccc(C=C(C#N)C#N)cc1	CID:2063	phase I
BRD-K36737713	COC(=O)c1ccc(NCc2cc(O)ccc2O)cc1	CID:2064	phase I
BRD-K51223576	NC(=O)C(=Cc1ccc(O)c(O)c1)C#N	CID:2065	phase I
BRD-A14966924	CC(N)C(=O)OC(C)(C)Cc1ccc(Cl)cc1	CID:2081	phase I
BRD-K79131256	CCCSc1ccc2[nH]c(NC(=O)OC)nc2c1	CID:2082	phase I
BRD-A88254928	CC(C)(C)NCC(O)c1ccc(O)c(CO)c1	CID:2083	phase I
BRD-K75527158	NCCCC(O)(P(O)(O)=O)P(O)(O)=O	CID:2088	phase I
BRD-A42335949	CCCCC(CC)CNC(=N)NC(=N)NCCCCCCNC(=N)NC(=N)NCC(CC)CCCC	CID:2090	phase I
BRD-A09056319	COc1cc2nc(nc(N)c2cc1OC)N(C)CCCNC(=O)C1CCCO1	CID:2092	phase I
BRD-K46742498	Cc1[nH]cnc1CN1CCc2c(C1=O)c1ccccc1n2C	CID:2099	phase I
BRD-A17745711	CC(N)Cc1c[nH]c2ccc(O)cc12	CID:2107	phase I
BRD-A82892199	CC(C)CCCC(C)CCCC(C)CCCC1(C)CCc2c(C)c(O)c(C)c(C)c2O1	CID:2116	phase I
BRD-K32398298	Cc1nnc2CN=C(c3ccccc3)c3cc(Cl)ccc3-n12	CID:2118	phase I
BRD-A00993607	CC(C)NCC(O)COc1ccccc1CC=C	CID:2119	phase I
BRD-K35498378	OC(=O)CN1C(=O)c2cccc3cccc(C1=O)c23	CID:2120	phase I
BRD-A56675431	NS(=O)(=O)c1cc2c(NC(CSCC=C)NS2(=O)=O)cc1Cl	CID:2122	phase I
BRD-K67043667	CN(C)c1nc(nc(n1)N(C)C)N(C)C	CID:2123	phase I
BRD-K92000912	Cc1c(nn(c1-c1ccc(I)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1	CID:2125	phase I
BRD-K06854232	CC1(C)CCC(C)(C)c2cc(ccc12)C(=O)Nc1ccc(cc1)C(O)=O	CID:2126	phase I
BRD-K21667562	CCCCCC=CCC=CCC=CCC=CCCCC(=O)Nc1ccc(O)cc1	CID:2127	phase I
BRD-A11813248	CN(CCc1ccc(Cl)c(Cl)c1)CC(O)COc1ccc(NS(C)(=O)=O)cc1	CID:2129	phase I
BRD-K70330367	NC12CC3CC(CC(C3)C1)C2	CID:2130	phase I
BRD-A16478930	CC(=O)OCC(=O)C12OC3(CCCC3)OC1CC1C3CCC4=CC(=O)C=CC4(C)C3(F)C(O)CC21C	CID:2133	phase I
BRD-K73947551	NCCCNCCSP(O)(O)=O	CID:2141	phase I
BRD-A28095882	CN1C2CCC1CC(C2)OC(c3ccccc3)c4ccccc4N	CID:2143	phase I
BRD-A25234499	CCC1(CCC(=O)NC1=O)c1ccc(N)cc1	CID:2145	phase I
BRD-K65544384	Nc1ccc(cc1)C(=O)NCC(O)=O	CID:2148	phase I
BRD-K20484910	Cc1c(N)c(=O)n(-c2ccccc2)n1C	CID:2151	phase I
BRD-K97799481	Cn1c2nc[nH]c2c(=O)n(C)c1=O	CID:2153	phase I
BRD-K17561142	CCCCc1oc2ccccc2c1C(=O)c1cc(I)c(OCCN(CC)CC)c(I)c1	CID:2157	phase I
BRD-A60197193	CCN1CCCC1CNC(=O)c1cc(c(N)cc1OC)S(=O)(=O)CC	CID:2159	phase I
BRD-K53737926	CN(C)CCC=C1c2ccccc2CCc2ccccc12	CID:2160	phase I
BRD-K29530284	CC(C)c1ccc2oc3nc(N)c(cc3c(=O)c2c1)C(O)=O	CID:2161	phase I
BRD-A22032524	CCOC(=O)C1=C(NC(=C(C1C2=CC=CC=C2Cl)C(=O)OC)C)COCCN	CID:2162	phase I
BRD-K91290917	CCN(CC)Cc1cc(Nc2ccnc3cc(Cl)ccc23)ccc1O	CID:2165	phase I
BRD-K02265150	Clc1ccc2Oc3ccccc3N=C(N3CCNCC3)c2c1	CID:2170	phase I
BRD-A16754160	CC1(C)SC2C(NC(=O)C(N)c3ccccc3)C(=O)N2C1C(=O)O	CID:2174	phase I
BRD-A39172021	CCOC(=O)OC(C)OC1=C(N(C)S(=O)(=O)c2ccccc12)C(=O)Nc1ccccn1	CID:2176	phase I
BRD-K52172416	CC(C)(C#N)c1cc(Cn2cncn2)cc(c1)C(C)(C)C#N	CID:2187	phase I
BRD-K92490248	COc1ccc(cc1)-c1cc(=S)ss1	CID:2194	phase I
BRD-K88611939	COc1ccc(cc1)C(=O)N1CCCC1=O	CID:2196	phase I
BRD-K99300445	C(N(Cc1ccccc1)c1ccccc1)C1=NCCN1	CID:2200	phase I
BRD-K46937689	Cc1cc(=O)n(-c2ccccc2)n1C	CID:2206	phase I
BRD-K23922020	CN1CCC=C(C1)C(=O)OCC#C	CID:2229	phase I
BRD-K17110974	COc1cccc2c1cc([N+](=O)[O-])c3c(cc4OCOc4c23)C(=O)O	CID:2236	phase I
BRD-K11433652	CC(=O)Oc1ccccc1C(O)=O	CID:2244	phase I
BRD-K37249724	COc1ccc(CCN2CCC(CC2)Nc2nc3ccccc3n2Cc2ccc(F)cc2)cc1	CID:2247	phase I
BRD-A20239487	CC(C)NCC(O)COc1ccc(CC(N)=O)cc1	CID:2249	phase I
BRD-A82307304	CC(C)c1c(C(=O)Nc2ccccc2)c(c(-c2ccc(F)cc2)n1CCC(O)CC(O)CC(O)=O)-c1ccccc1	CID:2250	phase I
BRD-A44133049	CN1C(=O)COc2c1cc(Cl)cc2C(=O)NC1CN2CCC1CC2	CID:2264	phase I
BRD-K32821942	Cn1cnc(c1Sc1[nH]cnc2ncnc12)[N+]([O-])=O	CID:2265	phase I
BRD-A68888262	CN1CCCC(CC1)n1nc(Cc2ccc(Cl)cc2)c2ccccc2c1=O	CID:2267	phase I
BRD-A84174873	NCC(CC(O)=O)c1ccc(Cl)cc1	CID:2284	phase I
BRD-A16694057	CC(C)(c1ccc(OCC2CO2)cc1)c3ccc(OCC4CO4)cc3	CID:2286	phase I
BRD-K40919711	CC(=O)OCOC(=O)CN(CC(=O)OCOC(=O)C)c1ccccc1OCCOc2ccccc2N(CC(=O)OCOC(=O)C)CC(=O)OCOC(=O)C	CID:2293	phase I
BRD-A05457250	COC(=O)C1=C(C)NC(C)=C(C1c1ccccc1C(F)(F)F)[N+]([O-])=O	CID:2303	phase I
BRD-K14993104	CCC1(C)CC(=O)NC(=O)C1	CID:2310	phase I
BRD-A15131297	CCOC(=O)C(CCc1ccccc1)NC2CCc3ccccc3N(CC(=O)O)C2=O	CID:2311	phase I
BRD-A80017228	NS(=O)(=O)c1cc2c(NC(Cc3ccccc3)NS2(=O)=O)cc1C(F)(F)F	CID:2315	phase I
BRD-A22305049	CC(Cc1cccc(c1)C(F)(F)F)NCCOC(=O)c1ccccc1	CID:2318	phase I
BRD-K02571615	CC(N(Cc1cnc(C)nc1N)C=O)=C(CCOP(O)(O)=O)SC(=O)c1ccccc1	CID:2320	phase I
BRD-A42423104	CC(COc1ccccc1Cc2ccccc2)N3CCCCC3	CID:2326	phase I
BRD-A61194565	NC(CO)C(=O)NNCc1ccc(O)c(O)c1O	CID:2327	phase I
BRD-K11717138	CCc1oc2ccccc2c1C(=O)c1cc(Br)c(O)c(Br)c1	CID:2333	phase I
BRD-K72723676	CC(C)(C)CC(C)(C)c1ccc(OCCOCC[N+](C)(C)Cc2ccccc2)cc1	CID:2335	phase I
BRD-K09668667	c1ccc2c(c1)cc3ccc4cccc5ccc2c3c45	CID:2336	phase I
BRD-K75466013	CCOC(=O)c1ccc(N)cc1	CID:2337	phase I
BRD-K21450440	NS(=O)(=O)c1cc2c(cc1Cl)N=C(CSCc1ccccc1)NS2(=O)=O	CID:2343	phase I
BRD-A25067867	CN1C2CCC1CC(C2)OC(c3ccccc3)c4ccccc4	CID:2344	phase I
BRD-A91008255	CC(C)COCC(CN(Cc1ccccc1)c1ccccc1)N1CCCC1	CID:2351	phase I
BRD-A15034104	COc1c(O)cc2C(=O)OC3C(O)C(O)C(CO)OC3c2c1O	CID:2356	phase I
BRD-K91315211	CNCCc1ccccn1	CID:2366	phase I
BRD-A02759312	CC(C)NCC(O)COc1ccc(CCOCC2CC2)cc1	CID:2369	phase I
BRD-A99833829	CC(C[N+](C)(C)C)OC(N)=O	CID:2370	phase I
BRD-A29485665	CC(O)(CS(=O)(=O)c1ccc(F)cc1)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F	CID:2375	phase I
BRD-K18779551	CNCCCCOc1ccccc1Cc1ccccc1	CID:2377	phase I
BRD-A94543220	c1cn(cn1)C(c1ccccc1)c1ccc(cc1)-c1ccccc1	CID:2378	phase I
BRD-A00546892	OC(CCN1CCCCC1)(C1CC2CC1C=C2)c1ccccc1	CID:2381	phase I
BRD-K12357156	Oc1ccc(C=C(C#N)C(=O)NCc2ccccc2)cc1O	CID:2390	phase I
BRD-K39987650	CC(=O)Oc1ccc(cc1)C(c1ccc(OC(C)=O)cc1)c1ccccn1	CID:2391	phase I
BRD-K31342827	CN(C)CCCn1cc(C2=C(C(=O)NC2=O)c3c[nH]c4ccccc34)c5ccccc15	CID:2396	phase I
BRD-K49448285	O=C1NC(=O)C(=C1c2c[nH]c3ccccc23)c4c[nH]c5ccccc45	CID:2399	phase I
BRD-A89175223	CC(C)NCC(O)COc1ccc(COCCOC(C)C)cc1	CID:2405	phase I
BRD-K39120595	Oc1c(Cl)cc(Cl)cc1Sc1cc(Cl)cc(Cl)c1O	CID:2406	phase I
BRD-K94379058	COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)N3CCOCC3)c2c1	CID:2415	phase I
BRD-K31054881	COc1ccccc1N1CCN(CCN2C(=O)CC3(CCCC3)CC2=O)CC1	CID:2419	phase I
BRD-A17065207	CC1CCCC=CC2CC(O)CC2C(O)C=CC(=O)O1	CID:2430	phase I
BRD-K49669424	CC[N+](C)(C)Cc1ccccc1Br	CID:2431	phase I
BRD-K68264559	Brc1c(NC2=NCCN2)ccc2nccnc12	CID:2435	phase I
BRD-K17868609	CN1CCC(CC1)c1c[nH]c2ccc(O)cc12	CID:2438	phase I
BRD-K47631482	CN(Cc1cc(Br)cc(Br)c1N)C1CCCCC1	CID:2442	phase I
BRD-A69960130	CC(C)CC1N2C(=O)C(NC(=O)C3CN(C)C4Cc5c(Br)[nH]c6cccc(C4=C3)c56)(OC2(O)C7CCCN7C1=O)C(C)C	CID:2443	phase I
BRD-K78643075	OC1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)c1ccc(Br)cc1	CID:2448	phase I
BRD-K55344148	C1CN=C(N1)c1ccc2ccccc2n1	CID:2457	phase I
BRD-A04706586	CCCC(=O)Nc1ncnc2n(cnc12)C3OC4COP(=O)(O)OC4C3OC(=O)CCC	CID:2460	phase I
BRD-A82238138	CCCC1OC2CC3C4CCC5=CC(=O)C=CC5(C)C4C(O)CC3(C)C2(O1)C(=O)CO	CID:2462	phase I
BRD-K36660044	CCCCOc1ccc(CC(=O)NO)cc1	CID:2466	phase I
BRD-K19462402	COc1cc(OC)c(C(=O)CCCN2CCCC2)c(OC)c1	CID:2467	phase I
BRD-K38197229	CCCCNc1cc(cc(c1Oc1ccccc1)S(N)(=O)=O)C(O)=O	CID:2471	phase I
BRD-A01636364	CCCCN1CCCCC1C(=O)Nc1c(C)cccc1C	CID:2474	phase I
BRD-K93461745	O=C1CC2(CCCC2)CC(=O)N1CCCCN1CCN(CC1)c1ncccn1	CID:2477	phase I
BRD-K23204545	CS(=O)(=O)OCCCCOS(C)(=O)=O	CID:2478	phase I
BRD-K99622919	CCCCN(CCCC)CCCOC(=O)c1ccc(N)cc1	CID:2480	phase I
BRD-K71350836	CC(C)CC1(CC=C)C(=O)NC(=O)NC1=O	CID:2481	phase I
BRD-K27217864	CCCCOC(=O)c1ccc(N)cc1	CID:2482	phase I
BRD-K90630139	CN(Cc1ccc(cc1)C(C)(C)C)Cc1cccc2ccccc12	CID:2484	phase I
BRD-A68891053	CC(C=Cc1cccc(Oc2ccc(F)cc2)c1)N(O)C(=O)N	CID:2491	phase I
BRD-A53416814	CCCCCCCCCCCCCC=CC(O)C(CO)NC(=O)C	CID:2505	phase I
BRD-A63043573	CCNC(=O)N(CCCN(C)C)C(=O)C1CC2C(Cc3c[nH]c4cccc2c34)N(CC=C)C1	CID:2512	phase I
BRD-K02404261	Cn1cnc2n(C)c(=O)n(C)c(=O)c12	CID:2519	phase I
BRD-A09533288	COc1ccc(CCN(C)CCCC(C#N)(C(C)C)c2ccc(OC)c(OC)c2)cc1OC	CID:2520	phase I
BRD-A98283014	Clc1ccc(cc1)C(c2ccc(Cl)cc2)[n+]3ccn(CC(OCc4ccc(Cl)cc4Cl)c5ccc(Cl)cc5Cl)c3	CID:2531	phase I
BRD-A84045418	CCCCC(NC(=O)C(CC(C)C)NC(=O)OCc1ccccc1)C=O	CID:2532	phase I
BRD-A30437061	CCC1(O)C(=O)OCc2c1cc3-c4nc5ccccc5cc4Cn3c2=O	CID:2538	phase I
BRD-A65671304	CCOc1nc2cccc(C(=O)OC(C)OC(=O)OC3CCCCC3)c2n1Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1	CID:2540	phase I
BRD-K84091759	CCOc1nc2cccc(C(O)=O)c2n1Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1	CID:2541	phase I
BRD-K75037734	C[N+](C)(C)CCOC(N)=O	CID:2551	phase I
BRD-K71799949	NC(=O)N1c2ccccc2C=Cc2ccccc12	CID:2554	phase I
BRD-K06181161	CCN(CC)CCOCCOC(=O)C1(CCCC1)c1ccccc1	CID:2562	phase I
BRD-A69512159	CC(Cc1ccc(O)c(O)c1)(NN)C(=O)O	CID:2563	phase I
BRD-A29426959	CN(C)CCOC(c1ccc(Cl)cc1)c1ccccn1	CID:2564	phase I
BRD-K53570330	CNC(=O)Oc1cccc2CC(C)(C)Oc21	CID:2566	phase I
BRD-A99939097	CCCC(C)(COC(N)=O)COC(=O)NC(C)C	CID:2576	phase I
BRD-K11630072	CCCCCCNC(=O)n1cc(F)c(=O)[nH]c1=O	CID:2577	phase I
BRD-A17411484	CC(C(O)=O)c1ccc2c(c1)[nH]c1ccc(Cl)cc21	CID:2581	phase I
BRD-A42167015	CC(C)(C)NCC(O)COc1cccc2NC(=O)CCc12	CID:2583	phase I
BRD-A10977446	COc1ccccc1OCCNCC(O)COc1cccc2[nH]c3ccccc3c12	CID:2585	phase I
BRD-K15616905	Clc1cccc(NN=C(C#N)C#N)c1	CID:2603	phase I
BRD-K71860425	Nc1cc(Nc2ccc(cc2)S(=O)(=O)N)ncn1	CID:2608	phase I
BRD-A65282128	Cc1nnc(SCC2=C(N3C(SC2)C(NC(=O)Cn4cnnn4)C3=O)C(=O)O)s1	CID:2618	phase I
BRD-K02637541	Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(F)(F)F	CID:2662	phase I
BRD-A95602221	CCN(CC)C(=O)Nc1ccc(OCC(O)CNC(C)(C)C)c(c1)C(C)=O	CID:2663	phase I
BRD-A42571354	OC(=O)COCCN1CCN(CC1)C(c1ccccc1)c1ccc(Cl)cc1	CID:2678	phase I
BRD-A31575449	Cn1cc(nc1c2ccc(OCC(O)CNCCOc3ccc(O)c(c3)C(=O)N)cc2)C(F)(F)F	CID:2685	phase I
BRD-A34706053	CC(C)(C)NCC(O)COc1cccc2[nH]c(=O)[nH]c12	CID:2687	phase I
BRD-A35623999	Clc1ccc2NC(=O)CSC(c3ccccc3Cl)c2c1	CID:2688	phase I
BRD-K18909381	CN1CCN(CC1)c2nc3cc(ccc3n4cccc24)C(F)(F)F	CID:2689	phase I
BRD-K49049886	Nc1nc2ccc(Cl)cc2c2nc(nn12)-c1ccco1	CID:2690	phase I
BRD-A81866333	CCNC(=O)C1OC(C(O)C1O)n2cnc3c(N)nc(NCCc4ccc(CCC(=O)O)cc4)nc23	CID:2691	phase I
BRD-K29458283	OC(=O)CCCc1ccc(cc1)N(CCCl)CCCl	CID:2708	phase I
BRD-A57133233	CN1CCN(CC1)C(c1ccccc1)c1ccc(Cl)cc1	CID:2710	phase I
BRD-K52256627	Clc1ccc(NC(=N)NC(=N)NCCCCCCNC(=N)NC(=N)Nc2ccc(Cl)cc2)cc1	CID:2713	phase I
BRD-A20348246	CN1C(c2ccc(Cl)cc2)S(=O)(=O)CCC1=O	CID:2717	phase I
BRD-A91699651	CCN(CC)CCCC(C)Nc1ccnc2cc(Cl)ccc12	CID:2719	phase I
BRD-K88682005	NS(=O)(=O)c1cc2c(cc1Cl)N=CNS2(=O)=O	CID:2720	phase I
BRD-K17075857	Oc1c(Cl)cc(Cl)c2cccnc12	CID:2722	phase I
BRD-A39230911	NC(=O)OCC(O)COc1ccc(Cl)cc1	CID:2724	phase I
BRD-A04553218	CN(C)CCC(c1ccc(Cl)cc1)c1ccccn1	CID:2725	phase I
BRD-K89997465	CN(C)CCCN1c2ccccc2Sc2ccc(Cl)cc12	CID:2726	phase I
BRD-K81091703	CN(C)CCC=C1c2ccccc2Sc2ccc(Cl)cc12	CID:2729	phase I
BRD-A26384407	NS(=O)(=O)c1cc(ccc1Cl)C1(O)NC(=O)c2ccccc12	CID:2732	phase I
BRD-K98174813	Clc1ccc2oc(=O)[nH]c2c1	CID:2733	phase I
BRD-K52313696	CC(=O)Nc1ccc(cc1)C(=O)Nc1ccccc1N	CID:2746	phase I
BRD-K13044802	Cc1cc(C2CCCCC2)n(O)c(=O)c1	CID:2749	phase I
BRD-A93000692	CC1(COc2ccc(CC3SC(=O)NC3=O)cc2)CCCCC1	CID:2750	phase I
BRD-A07875874	COCCOC(=O)C1=C(C)NC(=C(C1c2cccc(c2)[N+](=O)[O-])C(=O)OCC=Cc3ccccc3)C	CID:2752	phase I
BRD-K28578425	CN(C1CCCCC1)C(=O)CCCOc1ccc2[nH]c(=O)ccc2c1	CID:2753	phase I
BRD-K67017579	O=C1CCc2cc(OCCCCc3nnnn3C3CCCCC3)ccc2N1	CID:2754	phase I
BRD-A65440446	CC(C)NCC(O)c1ccc(N)c(c1)C#N	CID:2755	phase I
BRD-K18618618	CNC(=NC#N)NCCSCc1nc[nH]c1C	CID:2756	phase I
BRD-K74927006	C(C=Cc1ccccc1)N1CCN(CC1)C(c1ccccc1)c1ccccc1	CID:2761	phase I
BRD-A49358627	CC(C)(Oc1ccc(cc1)C1CC1(Cl)Cl)C(O)=O	CID:2763	phase I
BRD-K04804440	OC(=O)c1cn(C2CC2)c2cc(N3CCNCC3)c(F)cc2c1=O	CID:2764	phase I
BRD-K54142781	C(Oc1ccccc1C1CC1)C1=NCCN1	CID:2765	phase I
BRD-K24630133	Cl[Pt++]Cl	CID:2768	phase I
BRD-K01228321	Cl[Pt]Cl	CID:2770	phase I
BRD-A47598013	CN(C)CCCC1(OCc2cc(ccc12)C#N)c1ccc(F)cc1	CID:2771	phase I
BRD-K00675675	O=C(NCCCCN1CCOCC1)c2cc3ccccc3o2	CID:2777	phase I
BRD-K17294426	COc1cc(N)c(Cl)cc1C(=O)NC1CCN(Cc2ccccc2)CC1	CID:2780	phase I
BRD-K04704168	Clc1ccc(Cn2c(CN3CCCC3)nc3ccccc23)cc1	CID:2782	phase I
BRD-A75726477	CC(C)(C)NCC(O)c1cc(Cl)c(N)c(Cl)c1	CID:2783	phase I
BRD-K09255212	Oc1c(I)cc(Cl)c2cccnc12	CID:2788	phase I
BRD-K71430621	Clc1ccc(CNC(=N)SCCCc2c[nH]cn2)cc1	CID:2790	phase I
BRD-K56614220	CC(C)\N=c1/cc2n(-c3ccc(Cl)cc3)c3ccccc3nc2cc1Nc1ccc(Cl)cc1	CID:2794	phase I
BRD-K45252063	CCOC(=O)C(C)(C)Oc1ccc(Cl)cc1	CID:2796	phase I
BRD-K19111024	CC(C)(Oc1ccc(Cl)cc1)C(O)=O	CID:2797	phase I
BRD-K02680176	CCCCCCC[N+](CC)(CC)CCCCc1ccc(Cl)cc1	CID:2798	phase I
BRD-K91328526	CCN(CC)CCOc1ccc(cc1)C(=C(Cl)c1ccccc1)c1ccccc1	CID:2800	phase I
BRD-K52989797	CN(C)CCCN1c2ccccc2CCc2ccc(Cl)cc12	CID:2801	phase I
BRD-K98530306	Clc1cccc(Cl)c1N=C1NCCN1	CID:2803	phase I
BRD-A80908310	Clc1ccc(cc1)C(OCCN1CCCCC1)c1ccccc1	CID:2805	phase I
BRD-A93269281	COC(=O)C(N1CCc2sccc2C1)c3ccccc3Cl	CID:2806	phase I
BRD-K15916496	Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1ccnc1	CID:2812	phase I
BRD-A51410489	COC(=O)C1C(O)CCC2CN3CCc4c([nH]c5ccccc45)C3CC12	CID:2866	phase I
BRD-A24951056	NC(C1CC1)(C(O)=O)c1ccc(cc1)P(O)(O)=O	CID:2878	phase I
BRD-K20920669	OC(COc1cccc2oc(cc(=O)c12)C(O)=O)COc1cccc2oc(cc(=O)c12)C(O)=O	CID:2882	phase I
BRD-K13240564	CCN(C(=O)C=CC)c1ccccc1C	CID:2883	phase I
BRD-A37837077	COc1cc2nc(nc(N)c2cc1OC)N1CCN(C2CCCCC12)C(=O)c1ccco1	CID:2894	phase I
BRD-K42348709	CN(C)CCC=C1c2ccccc2C=Cc2ccccc12	CID:2895	phase I
BRD-A62184259	CC1CC(C)C(=O)C(C1)C(O)CC2CC(=O)NC(=O)C2	CID:2900	phase I
BRD-A41250306	NS(=O)(=O)c1cc2c(NC(CC3CCCC3)NS2(=O)=O)cc1Cl	CID:2904	phase I
BRD-A77291778	CN(C)CCOC(=O)C(c1ccccc1)C1(O)CCCC1	CID:2905	phase I
BRD-A09722536	ClCCN(CCCl)P1(=O)NCCCO1	CID:2907	phase I
BRD-A64290322	CCC1NC(=O)C(C(O)C(C)CC=CC)N(C)C(=O)C(C(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)C(C)NC(=O)C(C)NC(=O)C(CC(C)C)N(C)C(=O)C(NC(=O)C(CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C	CID:2909	phase I
BRD-K28143534	CN1CCC(CC1)=C1c2ccccc2C=Cc2ccccc12	CID:2913	phase I
BRD-A77118605	SC(=S)OC1CC2CC1C1CCCC21	CID:2941	phase I
BRD-K35520305	CN(C)\N=N\c1[nH]cnc1C(N)=O	CID:2942	phase I
BRD-K93325701	COc1c(C=O)c(O)cc2C(=O)c3ccccc3C(=O)c12	CID:2948	phase I
BRD-A20243730	CC12CCC3C(CCC4=Cc5oncc5CC34C)C2CCC1(O)C#C	CID:2949	phase I
BRD-K10065684	Oc1cccc2C(=O)c3cccc(O)c3C(=O)c12	CID:2950	phase I
BRD-K31333309	[O-][N+](=O)c1ccc(cc1)c2ccc(C=NN3CC(=O)NC3=O)o2	CID:2952	phase I
BRD-K62363391	Nc1ccc(cc1)S(=O)(=O)c1ccc(N)cc1	CID:2955	phase I
BRD-A68929948	CC(NC(=O)Cc1cc(F)cc(F)c1)C(=O)NC(C(=O)OC(C)(C)C)c2ccccc2	CID:2956	phase I
BRD-A37630846	COc1cccc2C(=O)c3c(O)c4CC(O)(CC(OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(=O)C	CID:2958	phase I
BRD-K06878038	Cc1c(O)c(=O)ccn1C	CID:2972	phase I
BRD-K37792168	CCCCn1c(=O)n(CCCC)c2ncn(CC(=O)C)c2c1=O	CID:2984	phase I
BRD-K60274257	CN([N+][O-])c1cc(O)ccc1O	CID:2990	phase I
BRD-K77685957	Cc1cc(N)c2ccccc2[n+]1CCCCCCCCCC[n+]1c(C)cc(N)c2ccccc12	CID:2993	phase I
BRD-K60762818	CNCCCN1c2ccccc2CCc2ccccc12	CID:2995	phase I
BRD-A35108200	CC1CC2C3CCC4=CC(=O)C=CC4(C)C3(F)C(O)CC2(C)C1(O)C(=O)CO	CID:3003	phase I
BRD-K54665485	Cc1nc2sccn2c(=O)c1CCN1CCC(CC1)=C(c1ccccc1)c1ccc(F)cc1	CID:3012	phase I
BRD-K16508793	CN1c2ccc(Cl)cc2C(=NCC1=O)c1ccccc1	CID:3016	phase I
BRD-K73109821	CC1=Nc2ccc(Cl)cc2S(=O)(=O)N1	CID:3019	phase I
BRD-K99121711	CCCCOc1cc(C(=O)NCCN(CC)CC)c2ccccc2n1	CID:3025	phase I
BRD-K08252256	OC(=O)Cc1ccccc1Nc1c(Cl)cccc1Cl	CID:3033	phase I
BRD-K71499074	NS(=O)(=O)c1cc(Cl)c(Cl)c(c1)S(N)(=O)=O	CID:3038	phase I
BRD-K68507560	CCN(CC)CCOC(=O)C1(CCCCC1)C1CCCCC1	CID:3042	phase I
BRD-A20131130	CC1OC(CC1O)n1cnc2c(N)ncnc12	CID:3044	phase I
BRD-A85777636	ClC1=C(Cl)C2(Cl)C3C4CC(C5OC54)C3C1(Cl)C2(Cl)Cl	CID:3048	phase I
BRD-K55106630	CC=C(C(=CC)c1ccc(O)cc1)c1ccc(O)cc1	CID:3049	phase I
BRD-K45542189	CCN(CC)C(=O)N1CCN(C)CC1	CID:3052	phase I
BRD-K40621224	OC(=O)CN(CCN(CC(O)=O)CC(O)=O)CCN(CC(O)=O)CC(O)=O	CID:3053	phase I
BRD-K17084514	CCC(=C(CC)c1ccc(O)cc1)c1ccc(O)cc1	CID:3054	phase I
BRD-K01663662	OC(CCCN1CCCCC1)(c1ccccc1)c1ccccc1	CID:3055	phase I
BRD-K22031190	OC(=O)c1cc(ccc1O)-c1ccc(F)cc1F	CID:3059	phase I
BRD-A44701612	CC(C)C1(NC(=O)C2CC3C(Cc4c[nH]c5cccc3c45)N(C)C2)OC6(O)C7CCCN7C(=O)C(Cc8ccccc8)N6C1=O	CID:3065	phase I
BRD-A54845972	CN1CC(CC2C1Cc3c[nH]c4cccc2c34)C(=O)NC5(C)OC6(O)C7CCCN7C(=O)C(Cc8ccccc8)N6C5=O	CID:3066	phase I
BRD-K37846922	C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12	CID:3071	phase I
BRD-K48722258	COc1cc(cc(OC)c1OC)C(=O)OCCCN1CCCN(CCCOC(=O)c2cc(OC)c(OC)c(OC)c2)CC1	CID:3074	phase I
BRD-A69636825	COc1ccc(cc1)C1Sc2ccccc2N(CCN(C)C)C(=O)C1OC(C)=O	CID:3076	phase I
BRD-K23541596	CN(C)CCCSC(N)=N	CID:3077	phase I
BRD-K43687498	CC1(C)OC(=O)NC1=O	CID:3081	phase I
BRD-K47278471	CN(C)CCOC(c1ccccc1)c1ccccc1	CID:3100	phase I
BRD-K65814004	[I+]1c2ccccc2-c2ccccc12	CID:3101	phase I
BRD-K22936972	CN1CCC(CC1)OC(c1ccccc1)c1ccccc1	CID:3103	phase I
BRD-A47494775	CNCC(O)c1ccc(OC(=O)C(C)(C)C)c(OC(=O)C(C)(C)C)c1	CID:3105	phase I
BRD-K82577285	CCCN(CCC)CCc1ccc(O)c(O)c1	CID:3106	phase I
BRD-K86301799	OCCN(CCO)c1nc(N2CCCCC2)c2nc(nc(N3CCCCC3)c2n1)N(CCO)CCO	CID:3108	phase I
BRD-K76812510	CN(CS(O)(=O)=O)c1c(C)n(C)n(-c2ccccc2)c1=O	CID:3111	phase I
BRD-A29734509	CC(C)N(CCC(C(N)=O)(c1ccccc1)c1ccccn1)C(C)C	CID:3114	phase I
BRD-K32744045	CCN(CC)C(=S)SSC(=S)N(CC)CC	CID:3117	phase I
BRD-K41260949	CCCC(CCC)C(O)=O	CID:3121	phase I
BRD-A56012032	OC(=O)CNC(=O)C(CS)Cc1ccccc1	CID:3132	phase I
BRD-K60487568	CN(C)c1ccc(C=C2C(=O)Nc3ccccc23)cc1	CID:3135	phase I
BRD-K38305202	Clc1ccc2n(C3CCN(CCCn4c5ccccc5[nH]c4=O)CC3)c(=O)[nH]c2c1	CID:3151	phase I
BRD-A49160188	COc1cc2CC(CC3CCN(Cc4ccccc4)CC3)C(=O)c2cc1OC	CID:3152	phase I
BRD-A46179541	CCN1CC(CCN2CCOCC2)C(C1=O)(c1ccccc1)c1ccccc1	CID:3156	phase I
BRD-A13188892	COc1cc2nc(nc(N)c2cc1OC)N1CCN(CC1)C(=O)C1COc2ccccc2O1	CID:3157	phase I
BRD-K36616567	CN(C)CCC=C1c2ccccc2COc3ccccc13	CID:3158	phase I
BRD-A44008656	CN(C)CCOC(C)(c1ccccc1)c1ccccn1	CID:3162	phase I
BRD-K97158071	Fc1ccc(cc1)C(=O)CCCN1CCC(=CC1)n1c2ccccc2[nH]c1=O	CID:3168	phase I
BRD-A29349577	OCC(O)CN1CCN(CC1)c1ccccc1	CID:3169	phase I
BRD-K06221026	CS(=O)(=O)c1ccc(cc1)-c1cc(Br)sc1-c1ccc(F)cc1	CID:3177	phase I
BRD-K72259270	CCCCOc1ccc(cc1)C(=O)CCN1CCCCC1	CID:3180	phase I
BRD-A00827783	Cn1c2ncn(CC(O)CO)c2c(=O)n(C)c1=O	CID:3182	phase I
BRD-K41713976	Cc1cccc(CCN2CCC(CC2)C(=O)c2ccc(NS(C)(=O)=O)cc2)n1	CID:3185	phase I
BRD-K29359156	O=c1n([se]c2ccccc12)-c1ccccc1	CID:3194	phase I
BRD-A51820102	Clc1ccc(COC(Cn2ccnc2)c2ccc(Cl)cc2Cl)cc1	CID:3198	phase I
BRD-K81128206	CC[N+](C)(C)c1cccc(O)c1	CID:3202	phase I
BRD-K85985071	Cc1c2[nH]c3ccccc3c2c(C)c4cnccc14	CID:3213	phase I
BRD-K15010214	CCOCCn1c(nc2ccccc12)N1CCCN(C)CC1	CID:3219	phase I
BRD-K58685305	Cc1cc(O)c2C(=O)c3c(O)cc(O)cc3C(=O)c2c1	CID:3220	phase I
BRD-K78113049	CCn1cc(C(O)=O)c(=O)c2cc(F)c(nc12)N1CCNCC1	CID:3229	phase I
BRD-K39339537	COc1cc(C)nn1-c1nc(C)cc(OC)n1	CID:3242	phase I
BRD-A88080608	CC12CCC3C(=CCc4cc(O)ccc34)C1CCC2=O	CID:3247	phase I
BRD-K88741031	COC(=O)C=Cc1cc(O)ccc1O	CID:3248	phase I
BRD-A73581086	CC(CO)NC(=O)C1CN(C)C2Cc3c[nH]c4cccc(C2=C1)c34	CID:3250	phase I
BRD-A44827100	CCOC(=O)CCC(=O)OC1C(CC(C)OC1OC2C(C)C(OC3CC(C)(OC)C(O)C(C)O3)C(C)C(=O)OC(CC)C(C)(O)C(O)C(C)C(=O)C(C)CC2(C)O)N(C)C	CID:3256	phase I
BRD-A36066264	CC12CCC3C(CCc4cc(OC(=O)c5ccccc5)ccc34)C2CCC1O	CID:3262	phase I
BRD-A88939772	CC12CCC3C(CCc4cc(O)ccc34)C2CC(O)C1O	CID:3269	phase I
BRD-K96042922	OCCNC(=O)Cn1ccnc1[N+]([O-])=O	CID:3276	phase I
BRD-K64755930	CCOC(=O)c1cnc2n(CC)ncc2c1NN=C(C)C	CID:3277	phase I
BRD-K63630713	CCC(=C)C(=O)c1ccc(OCC(O)=O)c(Cl)c1Cl	CID:3278	phase I
BRD-A74500471	CCC(CO)NCCNC(CC)CO	CID:3279	phase I
BRD-K36756879	CCOc1ccc(Cc2nccc3cc(OCC)c(OCC)cc23)cc1OCC	CID:3280	phase I
BRD-A43286952	CC12CCC3C(CCc4cc(O)ccc34)C1CCC2(O)C#C	CID:3285	phase I
BRD-K08556791	CCCSP(=O)(OCC)SCCC	CID:3289	phase I
BRD-A16311756	CCN(CC)C(C)CN1c2ccccc2Sc2ccccc12	CID:3290	phase I
BRD-A99633051	CCC1(C)CC(=O)NC1=O	CID:3291	phase I
BRD-A30205217	CCN1C(=O)NC(C1=O)c1ccccc1	CID:3292	phase I
BRD-K56792340	CCOc1ccc2NC(C)(C)C=C(C)c2c1	CID:3293	phase I
BRD-K37949327	CC(O)(P(O)(O)=O)P(O)(O)=O	CID:3305	phase I
BRD-A09925278	CCNCC(O)c1cccc(O)c1	CID:3306	phase I
BRD-A74667430	CCc1cccc2c3CCOC(CC)(CC(O)=O)c3[nH]c12	CID:3308	phase I
BRD-K36248164	CCOC(=O)C=C(C)C=CC=C(C)C=Cc1c(C)cc(OC)c(C)c1C	CID:3312	phase I
BRD-K32977963	COc1cc(CC=C)ccc1O	CID:3314	phase I
BRD-K45033733	CC(=O)OCC(CCn1cnc2cnc(N)nc12)COC(C)=O	CID:3324	phase I
BRD-K00673382	NC(N)=Nc1nc(CSCC\C(N)=N/S(N)(=O)=O)cs1	CID:3325	phase I
BRD-A08255417	CC(Cc1ccccc1)N(C)Cc1c(C(C)C)c(=O)n(-c2ccccc2)n1C	CID:3326	phase I
BRD-K14821540	FC(F)(F)Oc1ccc(NN=C(C#N)C#N)cc1	CID:3330	phase I
BRD-K99107520	NC(=O)OCC(COC(N)=O)c1ccccc1	CID:3331	phase I
BRD-K91740057	OC(=O)Cc1ccc(cc1)-c1ccccc1	CID:3332	phase I
BRD-A30815329	CCOC(=O)C1=C(C)NC(C)=C(C1c1cccc(Cl)c1Cl)C(=O)OC	CID:3333	phase I
BRD-K51318897	COC(=O)Nc1nc2ccc(Sc3ccccc3)cc2[nH]1	CID:3334	phase I
BRD-K12513978	OC(=O)CCC(=O)c1ccc(cc1)-c1ccccc1	CID:3335	phase I
BRD-A71033472	CC(NCCC(c1ccccc1)c1ccccc1)c1ccccc1	CID:3336	phase I
BRD-A66284731	CCCCC(O)c1ccccc1	CID:3338	phase I
BRD-K50388907	CC(C)OC(=O)C(C)(C)Oc1ccc(cc1)C(=O)c1ccc(Cl)cc1	CID:3339	phase I
BRD-A50684349	Oc1ccc(cc1)C1CNCCc2c(Cl)c(O)c(O)cc12	CID:3341	phase I
BRD-A97104540	CC(Cc1ccc(O)cc1)NCC(O)c1cc(O)cc(O)c1	CID:3343	phase I
BRD-K26739552	O=C1NCC2(CCN(CCc3ccccc3)CC2)O1	CID:3344	phase I
BRD-A73368467	CC(C)(C(O)=O)c1ccc(cc1)C(O)CCCN1CCC(CC1)C(O)(c1ccccc1)c1ccccc1	CID:3348	phase I
BRD-K37688416	Clc1ccc(OCC(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)cc1	CID:3351	phase I
BRD-A50675702	Nc1c(c(nn1-c1c(Cl)cc(cc1Cl)C(F)(F)F)C#N)S(=O)C(F)(F)F	CID:3352	phase I
BRD-K47639036	Cc1c(oc2c(cccc2c1=O)C(=O)OCCN1CCCCC1)-c1ccccc1	CID:3354	phase I
BRD-A09472452	FC(F)(F)COc1ccc(OCC(F)(F)F)c(c1)C(=O)NCC1CCCCN1	CID:3356	phase I
BRD-A80638690	OCC1OC(CC1O)n1cc(F)c(=O)[nH]c1=O	CID:3363	phase I
BRD-K05977355	OC(Cn1cncn1)(Cn1cncn1)c1ccc(F)cc1F	CID:3365	phase I
BRD-K82143716	Nc1nc(=O)[nH]cc1F	CID:3366	phase I
BRD-K44067360	OC(=O)c1ccccc1Nc1cccc(c1)C(F)(F)F	CID:3371	phase I
BRD-K55127134	OCCN1CCN(CCCN2c3ccccc3Sc3ccc(cc23)C(F)(F)F)CC1	CID:3372	phase I
BRD-K98769987	CCOC(=O)c1ncn-2c1CN(C)C(=O)c1cc(F)ccc-21	CID:3373	phase I
BRD-A69777949	CC1CCc2cc(F)cc3c2n1cc(C(O)=O)c3=O	CID:3374	phase I
BRD-K12184470	Fc1ccc(cc1)C(N2CCN(CC=Cc3ccccc3)CC2)c4ccc(F)cc4	CID:3378	phase I
BRD-K24844714	Fc1c[nH]c(=O)[nH]c1=O	CID:3385	phase I
BRD-A31159102	CNCCC(Oc1ccc(cc1)C(F)(F)F)c1ccccc1	CID:3386	phase I
BRD-A21490874	CC1(O)CCC2C3CCC4=CC(=O)CCC4(C)C3(F)C(O)CC12C	CID:3387	phase I
BRD-A86044036	CC(C(O)=O)c1ccc(c(F)c1)-c1ccccc1	CID:3394	phase I
BRD-K77947974	Fc1ccc(cc1)C(CCCN1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(F)cc1	CID:3396	phase I
BRD-K28307902	CC(C)C(=O)Nc1ccc(c(c1)C(F)(F)F)[N+]([O-])=O	CID:3397	phase I
BRD-K72676686	COCCCCC(=NOCCN)c1ccc(cc1)C(F)(F)F	CID:3404	phase I
BRD-K56810756	Cc1cn[nH]c1	CID:3406	phase I
BRD-A70449690	CC(=O)OC1C(O)C2C(C)(C)CCC(O)C2(C)C2(O)C(=O)CC(C)(OC12C)C=C	CID:3413	phase I
BRD-K28687144	OC(=O)c1ccccc1OP(O)(O)=O	CID:3418	phase I
BRD-K78959463	COC(=O)c1c(C)[nH]c(C)c1C(=O)c1ccccc1Cc1ccccc1	CID:3423	phase I
BRD-A35713041	[O-][N+](=O)c1ccc(C=NN2CC(CN3CCOCC3)OC2=O)o1	CID:3434	phase I
BRD-K78010432	NS(=O)(=O)c1cc(C(O)=O)c(NCc2ccco2)cc1Cl	CID:3440	phase I
BRD-K87049188	CCCCc1ccc(nc1)C(=O)O	CID:3442	phase I
BRD-K62737565	NCC1(CC(O)=O)CCCCC1	CID:3446	phase I
BRD-K59256312	CCOC(=O)c1ccc(OC(=O)CCCCCNC(N)=N)cc1	CID:3447	phase I
BRD-K89104321	Oc1noc2CNCCc12	CID:3448	phase I
BRD-A49148672	COc1ccc2CN(C)CCC34C=CC(O)CC4Oc1c23	CID:3449	phase I
BRD-K43106192	CC[N+](CC)(CC)CCOc1cccc(OCC[N+](CC)(CC)CC)c1OCC[N+](CC)(CC)CC	CID:3450	phase I
BRD-K32501161	Fc1ccc(cc1)C(OCCN1CCN(CCCc2ccccc2)CC1)c1ccc(F)cc1	CID:3455	phase I
BRD-K50135270	C(CN1CCN(CCOC(c2ccccc2)c2ccccc2)CC1)Cc1ccccc1	CID:3456	phase I
BRD-K11129031	Cc1ccc(C)c(OCCCC(C)(C)C(O)=O)c1	CID:3463	phase I
BRD-A38076815	OCC(O)COC(=O)c1ccccc1Nc1ccnc2cc(Cl)ccc12	CID:3474	phase I
BRD-A61154809	Cc1ccc(cc1)S(=O)(=O)NC(=O)NN1CC2CCCC2C1	CID:3475	phase I
BRD-K12219985	Cc1cnc(cn1)C(=O)NCCc1ccc(cc1)S(=O)(=O)NC(=O)NC1CCCCC1	CID:3478	phase I
BRD-K36927236	COc1ccc(Cl)cc1C(=O)NCCc2ccc(cc2)S(=O)(=O)NC(=O)NC3CCCCC3	CID:3488	phase I
BRD-A73859745	CC(CCC(=O)NCC(=O)O)C1CCC2C3CCC4CC(O)CCC4(C)C3CC(O)C12C	CID:3493	phase I
BRD-A81233518	C[N+]1(C)CCC(C1)OC(=O)C(O)(C1CCCC1)c1ccccc1	CID:3494	phase I
BRD-K19295594	CC(C)c1c(O)c(O)c(C=O)c2c(O)c(c(C)cc12)-c1c(C)cc2c(C(C)C)c(O)c(O)c(C=O)c2c1O	CID:3503	phase I
BRD-A93659613	COC(=O)N1CCN(C(CN2CCCC2)C1)C(=O)Cc3ccc(Cl)c(Cl)c3	CID:3505	phase I
BRD-A90515964	COc1ccccc1OCC(O)CO	CID:3516	phase I
BRD-K67847053	NC(=N)NN=Cc1c(Cl)cccc1Cl	CID:3517	phase I
BRD-K32830106	NC(=N)NC(=O)Cc1c(Cl)cccc1Cl	CID:3519	phase I
BRD-K24240364	CC1=NN=C(c2ccc(N)cc2)c2cc3OCOc3cc2C1	CID:3538	phase I
BRD-K18742343	CNCCNS(=O)(=O)c1cccc2cnccc12	CID:3540	phase I
BRD-A55756846	CC1CNCCN1S(=O)(=O)c2cccc3cnccc23	CID:3542	phase I
BRD-K70577657	NCCNS(=O)(=O)c1cccc2cnccc12	CID:3544	phase I
BRD-K72462751	O=S(=O)(N1CCNCC1)c1cccc2cnccc12	CID:3545	phase I
BRD-K05434375	NC(=N)NCCNS(=O)(=O)c1cccc2cnccc12	CID:3546	phase I
BRD-K76617868	O=S(=O)(N1CCCNCC1)c1cccc2cnccc12	CID:3547	phase I
BRD-A13807286	CCOC(=O)C(C#N)C1c2cc(Br)ccc2OC(N)=C1C(=O)OCC	CID:3549	phase I
BRD-K67783091	OC1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)c1ccc(Cl)cc1	CID:3559	phase I
BRD-K13238168	Clc1cc(Cl)c(OCC#CI)cc1Cl	CID:3561	phase I
BRD-K56064827	COCc1cc(O)c(O)c(O)c1c2c(O)c(O)c(O)cc2COC	CID:3568	phase I
BRD-A39646320	CC1NC(=O)C2CCCN2C(=O)C(CCCCCC(=O)C2CO2)NC(=O)C(C)NC1=O	CID:3571	phase I
BRD-A21329147	C[N+]1(C)CCOC(O)(C1)c2ccc(cc2)c3ccc(cc3)C4(O)C[N+](C)(C)CCO4	CID:3585	phase I
BRD-A32988684	CC(N)CCCC(C)(C)O	CID:3590	phase I
BRD-K99792991	Oc1c(Cl)cc(Cl)c(Cl)c1Cc1c(O)c(Cl)cc(Cl)c1Cl	CID:3598	phase I
BRD-K10598093	C[N+](C)(C)CCCCCC[N+](C)(C)C	CID:3604	phase I
BRD-A01078468	CCC(C(CC)c1ccc(O)cc1)c1ccc(O)cc1	CID:3606	phase I
BRD-A18605525	CCCCC(CC)CN1CN(CC(CC)CCCC)CC(C)(N)C1	CID:3607	phase I
BRD-K99946902	CCCCCCc1ccc(O)cc1O	CID:3610	phase I
BRD-K37691127	CC(C)c1cccc(=O)c(O)c1	CID:3611	phase I
BRD-K04710043	CC(=O)NCCCCCCNC(=O)C	CID:3616	phase I
BRD-A22769835	CN1CCCN(CC1)C(c1ccccc1)c1ccc(Cl)cc1	CID:3627	phase I
BRD-K50406511	CCN(CC)CCNc1ccc(CO)c2sc3ccccc3c(=O)c12	CID:3634	phase I
BRD-K13078532	NS(=O)(=O)c1cc2c(NCNS2(=O)=O)cc1Cl	CID:3639	phase I
BRD-A73635141	CC12CC(O)C3C(CCC4=CC(=O)CCC34C)C2CCC1(O)C(=O)CO	CID:3640	phase I
BRD-K37447567	COc1c2OCOc2cc3CCN(C)Cc13	CID:3646	phase I
BRD-K36862742	NS(=O)(=O)c1cc2c(NCNS2(=O)=O)cc1C(F)(F)F	CID:3647	phase I
BRD-A99117172	CCN(CCO)CCCC(C)Nc1ccnc2cc(Cl)ccc12	CID:3652	phase I
BRD-A98299281	Nc1c2C(O)CCCc2nc2ccccc12	CID:3655	phase I
BRD-A62428732	OCCOCCN1CCN(CC1)C(c1ccccc1)c1ccc(Cl)cc1	CID:3658	phase I
BRD-A20527803	CNC(=O)C1OC(C(O)C1O)n2cnc3c(NCc4cccc(I)c4)ncnc23	CID:3668	phase I
BRD-K16444452	CC(C)C(=O)c1c(nn2ccccc12)C(C)C	CID:3671	phase I
BRD-A17655518	CC(C)Cc1ccc(cc1)C(C)C(O)=O	CID:3672	phase I
BRD-K87024524	NNCCc1ccccc1	CID:3675	phase I
BRD-K52662033	CCN(CC)CC(=O)Nc1c(C)cccc1C	CID:3676	phase I
BRD-K18194590	CNC(C)(C)Cc1ccccc1	CID:3677	phase I
BRD-K89055274	CCN(CCCc1ccccc1)CCCc1ccccc1	CID:3678	phase I
BRD-A78942461	CC(C)NC(C)C(O)COc1ccc(C)c2CCCc21	CID:3682	phase I
BRD-A37776212	CN(C(CN1CCCC1)c2cccc(OCC(=O)O)c2)C(=O)Cc3ccc(Cl)c(Cl)c3	CID:3683	phase I
BRD-K37516142	COC1=C(OC)C(=O)C(CCCCCCCCCCO)=C(C)C1=O	CID:3686	phase I
BRD-A24191444	CC(C(O)c1ccc(O)cc1)N1CCC(Cc2ccccc2)CC1	CID:3689	phase I
BRD-A67097164	ClCCNP1(=O)OCCCN1CCCl	CID:3690	phase I
BRD-K38436528	CN(C)CCCN1c2ccccc2CCc2ccccc12	CID:3696	phase I
BRD-A95869247	CC1Cc2ccccc2N1NC(=O)c1ccc(Cl)c(c1)S(N)(=O)=O	CID:3702	phase I
BRD-K01815685	OCc1c[nH]c2ccccc12	CID:3712	phase I
BRD-K57222227	COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)O)c2c1	CID:3715	phase I
BRD-A44090213	CC(C(O)=O)c1ccc(cc1)N1Cc2ccccc2C1=O	CID:3718	phase I
BRD-A08660406	CC(=O)N(CC(O)CN(C(C)=O)c1c(I)c(C(=O)NCC(O)CO)c(I)c(C(=O)NCC(O)CO)c1I)c1c(I)c(C(=O)NCC(O)CO)c(I)c(C(=O)NCC(O)CO)c1I	CID:3724	phase I
BRD-A60217728	CC(=O)N(CC(O)CO)c1c(I)c(C(=O)NCC(O)CO)c(I)c(C(=O)NCC(O)CO)c1I	CID:3730	phase I
BRD-A42628519	CCC(Cc1c(I)cc(I)c(N)c1I)C(=O)O	CID:3735	phase I
BRD-A72075775	COCC(=O)Nc1c(I)c(C(=O)NCC(O)CO)c(I)c(C(=O)N(C)CC(O)CO)c1I	CID:3736	phase I
BRD-K67261995	OC(=O)c1c(I)cc(I)c(NC(=O)CCCCC(=O)Nc2c(I)cc(I)c(C(=O)O)c2I)c1I	CID:3739	phase I
BRD-A65818372	OCCN(C(=O)CO)c1c(I)c(C(=O)NCC(O)CO)c(I)c(C(=O)NCC(O)CO)c1I	CID:3741	phase I
BRD-K79124250	CNC(=O)c1c(I)c(N(C)C(C)=O)c(I)c(C(=O)NCC(=O)Nc2c(I)c(C(O)=O)c(I)c(C(=O)NCCO)c2I)c1I	CID:3742	phase I
BRD-A05352148	CC(C)[N+]1(C)C2CCC1CC(C2)OC(=O)C(CO)c1ccccc1	CID:3746	phase I
BRD-K93618743	CC(C)Oc1ccc2c(c1)occ(-c1ccccc1)c2=O	CID:3747	phase I
BRD-K88568253	CC(C)NNC(=O)c1ccncc1	CID:3748	phase I
BRD-K60038276	CCCCC1=NC2(CCCC2)C(=O)N1Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1	CID:3749	phase I
BRD-K74195153	Nc1nc(N)nc(n1)-c1cc(Cl)ccc1Cl	CID:3752	phase I
BRD-K93332168	Cc1cc(no1)C(=O)NNCc1ccccc1	CID:3759	phase I
BRD-K87202646	NNC(=O)c1ccncc1	CID:3767	phase I
BRD-A74269027	CC(COc1ccccc1)NC(C)C(O)c2ccc(O)cc2	CID:3783	phase I
BRD-A90799790	COC(=O)C1=C(C)NC(C)=C(C1c1cccc2nonc12)C(=O)OC(C)C	CID:3784	phase I
BRD-K76097666	ONC(=O)CCCN1C(=O)c2cccc3cccc(C1=O)c23	CID:3785	phase I
BRD-K96740444	COc1ccc(cc1OC)C(=O)NCc1ccc(OCCN(C)C)cc1	CID:3792	phase I
BRD-A34817987	CCC(C)n1ncn(c2ccc(cc2)N3CCN(CC3)c4ccc(OCC5COC(Cn6cncn6)(O5)c7ccc(Cl)cc7Cl)cc4)c1=O	CID:3793	phase I
BRD-K52850071	COc1cc2ncnc(Nc3ccc(O)c(Br)c3)c2cc1OC	CID:3795	phase I
BRD-K68407802	COc1cc2ncnc(Nc3cc(Br)c(O)c(Br)c3)c2cc1OC	CID:3796	phase I
BRD-K40624912	CC(C)N(CCC(=O)c1ccc2ccccc2c1)Cc1ccccc1	CID:3797	phase I
BRD-K95676198	C=CC(=O)c1ccc2ccccc2c1	CID:3799	phase I
BRD-K22010301	COc1oc(=O)c2cc(N)ccc2c1Cl	CID:3803	phase I
BRD-K37312348	Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1	CID:3820	phase I
BRD-K49671696	Fc1ccc(cc1)C(=O)C1CCN(CCn2c(=O)[nH]c3ccccc3c2=O)CC1	CID:3822	phase I
BRD-A76019558	CC(=O)N1CCN(CC1)c2ccc(OCC3COC(Cn4ccnc4)(O3)c5ccc(Cl)cc5Cl)cc2	CID:3823	phase I
BRD-A97739905	CC(C(O)=O)c1cccc(c1)C(=O)c1ccccc1	CID:3825	phase I
BRD-A40639672	OC(=O)C1CCn2c1ccc2C(=O)c1ccccc1	CID:3826	phase I
BRD-K28936863	CN1CCC(CC1)=C1c2ccsc2C(=O)Cc2ccccc12	CID:3827	phase I
BRD-K80353807	COc1c2ccoc2c(OC)c2oc(C)cc(=O)c12	CID:3828	phase I
BRD-K65667145	C(Nc1ncnc2[nH]cnc12)c1ccco1	CID:3830	phase I
BRD-A81177136	CN(C(Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N4CCN(CC4)c5ccccc5)S(=O)(=O)c6cccc7cnccc67	CID:3838	phase I
BRD-A07440155	CC(CCc1ccccc1)NCC(O)c1ccc(O)c(c1)C(N)=O	CID:3869	phase I
BRD-K93460210	Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl	CID:3878	phase I
BRD-A49172652	Cc1c(OCC(F)(F)F)ccnc1CS(=O)c1nc2ccccc2[nH]1	CID:3883	phase I
BRD-K23583188	OC(=O)c1cc(ccc1O)N(Cc2ccccc2O)Cc3cc(O)ccc3O	CID:3894	phase I
BRD-K80725632	OC(=O)c1cc(NCc2cc(O)ccc2O)ccc1O	CID:3896	phase I
BRD-K78692225	Cc1oncc1C(=O)Nc1ccc(cc1)C(F)(F)F	CID:3899	phase I
BRD-K88789588	N#Cc1ccc(cc1)C(c1ccc(cc1)C#N)n1cncn1	CID:3902	phase I
BRD-A32836748	CC(C)CC(NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)C(N)Cc2ccc(O)cc2)C(=O)O	CID:3903	phase I
BRD-A46393198	C1CN2CC(N=C2S1)c1ccccc1	CID:3913	phase I
BRD-K56596464	CC[N+](CC)(CC)CC(=O)Nc1c(C)cccc1C	CID:3925	phase I
BRD-K62996583	Cc1cccc(C)c1NC(=O)CN1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1	CID:3926	phase I
BRD-K59332007	O=C1N(c2ccccc2C1(Cc1ccncc1)Cc1ccncc1)c1ccccc1	CID:3932	phase I
BRD-K82147103	CN(CCCN1c2ccccc2CCc2ccccc12)CC(=O)c1ccc(Cl)cc1	CID:3947	phase I
BRD-A75850590	CCn1cc(C(O)=O)c(=O)c2cc(F)c(N3CCNC(C)C3)c(F)c12	CID:3948	phase I
BRD-K62858456	COc1ccc(CN2CCN(CC2)C(c2ccc(F)cc2)c2ccc(F)cc2)c(OC)c1OC	CID:3949	phase I
BRD-A15501135	CC(=CCc1c(O)c(CC=C(C)C)c2OC(CC(=O)c2c1O)c3ccc(O)cc3)C	CID:3951	phase I
BRD-K96670504	OC(=O)c1nn(Cc2ccc(Cl)c(Cl)c2)c3ccccc13	CID:3953	phase I
BRD-K61250553	CN(C)C(=O)C(CCN1CCC(O)(CC1)c1ccc(Cl)cc1)(c1ccccc1)c1ccccc1	CID:3955	phase I
BRD-K82795137	CCOC(=O)N1CCC(CC1)=C1c2ccc(Cl)cc2CCc2cccnc12	CID:3957	phase I
BRD-A11990600	OC1N=C(c2ccccc2Cl)c2cc(Cl)ccc2NC1=O	CID:3958	phase I
BRD-A29854054	CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1	CID:3960	phase I
BRD-K76205745	CCCCc1nc(Cl)c(CO)n1Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1	CID:3961	phase I
BRD-K39915878	CN1CCN(CC1)C1=Nc2ccccc2Oc2ccc(Cl)cc12	CID:3964	phase I
BRD-A43082555	CC(C(O)=O)c1ccc(CC2CCCC2=O)cc1	CID:3965	phase I
BRD-K74765201	CCCc1c(OCCCCc2nnn[nH]2)ccc(C(C)=O)c1O	CID:3969	phase I
BRD-A12016240	CN1C2CCC1CC(C2)NC(=O)c3nn(C)c4ccccc34	CID:3970	phase I
BRD-K22385716	O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCNCC1	CID:3971	phase I
BRD-K27305650	O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCOCC1	CID:3973	phase I
BRD-K62792802	O=C1C=C(Nc2ccccc2)C(=O)c3cccnc13	CID:3976	phase I
BRD-K45528773	CN(C)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO	CID:3994	phase I
BRD-K30649484	NCc1ccc(cc1)S(N)(=O)=O	CID:3998	phase I
BRD-K35458079	CC1=NN(C(=O)C1)c1ccccc1	CID:4021	phase I
BRD-K77987382	COC(=O)Nc1nc2ccc(cc2[nH]1)C(=O)c1ccccc1	CID:4030	phase I
BRD-A09467419	CCN(CCCCOC(=O)c1ccc(OC)c(OC)c1)C(C)Cc1ccc(OC)cc1	CID:4031	phase I
BRD-A20119038	CNC1(C)C2CCC(C2)C1(C)C	CID:4032	phase I
BRD-A50311610	Cc1cccc(CN2CCN(CC2)C(c2ccccc2)c2ccc(Cl)cc2)c1	CID:4034	phase I
BRD-K50398167	Cc1ccc(Cl)c(Nc2ccccc2C(O)=O)c1Cl	CID:4037	phase I
BRD-K10314788	CN(C)CCOC(=O)COc1ccc(Cl)cc1	CID:4039	phase I
BRD-K92778217	Cc1cccc(Nc2ccccc2C(O)=O)c1C	CID:4044	phase I
BRD-K20655524	CCN(CC)CCNC(=O)COc1ccc(OC)cc1	CID:4045	phase I
BRD-A89585551	OC(C1CCCCN1)c1cc(nc2c(cccc12)C(F)(F)F)C(F)(F)F	CID:4046	phase I
BRD-A08200164	NC(Cc1ccc(cc1)N(CCCl)CCCl)C(O)=O	CID:4053	phase I
BRD-A79803969	CC12CC3CC(C)(C1)CC(N)(C3)C2	CID:4054	phase I
BRD-K78126613	CC1=CC(=O)c2ccccc2C1=O	CID:4055	phase I
BRD-A62421304	C[N+]1(C)CCCC(C1)OC(=O)C(O)(c1ccccc1)c1ccccc1	CID:4057	phase I
BRD-A55469827	Cc1ccccc1OCC(O)CO	CID:4059	phase I
BRD-A83937277	CCC1(NC(=O)N(C)C1=O)c1ccccc1	CID:4060	phase I
BRD-A03216249	CN1CCCCC1C(=O)Nc1c(C)cccc1C	CID:4062	phase I
BRD-K65417056	CCCNC(C)(C)COC(=O)c1ccccc1	CID:4065	phase I
BRD-K28849549	Nc1ccc(O)c(c1)C(O)=O	CID:4075	phase I
BRD-A14395271	CN1CCCCC1CCN1c2ccccc2Sc2ccc(cc12)S(C)=O	CID:4078	phase I
BRD-A07780951	CC(C)NCC(O)c1cc(O)cc(O)c1	CID:4086	phase I
BRD-A30435184	CN1CC(CNC(=O)OCc2ccccc2)CC3C1Cc4cn(C)c5cccc3c45	CID:4090	phase I
BRD-K79602928	CN(C)C(=N)NC(N)=N	CID:4091	phase I
BRD-K09859624	CC[N+](C)(CC)CCOC(=O)C1c2ccccc2Oc2ccccc12	CID:4097	phase I
BRD-K47323024	CN(C)CCN(Cc1cccs1)c1ccccn1	CID:4098	phase I
BRD-K13356952	CC(=O)N=c1sc(nn1C)S(N)(=O)=O	CID:4100	phase I
BRD-K30114692	C1N2CN3CN1CN(C2)C3	CID:4101	phase I
BRD-A02189320	CSCCC(N)C(=O)NC(CC(C)C)C(=O)NC(Cc1ccccc1)C(=O)O	CID:4105	phase I
BRD-A07932845	CSc1ccc2Sc3ccccc3CC(N3CCN(C)CC3)c2c1	CID:4106	phase I
BRD-A31521121	COc1ccccc1OCC(O)COC(N)=O	CID:4107	phase I
BRD-A55424491	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(cc1)C(=O)NC(CCC(O)=O)C(O)=O	CID:4112	phase I
BRD-K63430059	COc1c2occc2cc2ccc(=O)oc12	CID:4114	phase I
BRD-K66195174	COc1ccc(cc1)C(c2ccc(OC)cc2)C(Cl)(Cl)Cl	CID:4115	phase I
BRD-K12539581	COC(=O)Nc1nc2cc(ccc2[nH]1)C(=O)c1cccs1	CID:4122	phase I
BRD-K46531780	Cc1cc(ccc1OCCOCC[N+](C)(C)Cc1ccccc1)C(C)(C)CC(C)(C)C	CID:4135	phase I
BRD-K16406336	CN(C)c1ccc2nc3ccc(cc3[s+]c2c1)N(C)C	CID:4139	phase I
BRD-A63667919	CCC(CO)NC(=O)C1CN(C)C2Cc3c[nH]c4cccc(C2=C1)c34	CID:4140	phase I
BRD-K45437867	Cc1ccc(C[N+](C)(C)C)o1	CID:4141	phase I
BRD-A08062015	CC1(O)CCC2C3CCC4=CC(=O)CCC4(C)C3CCC12C	CID:4160	phase I
BRD-A98725278	CCC(CO)NC(=O)C1CN(C)C2Cc3cn(C)c4cccc(C2=C1)c34	CID:4163	phase I
BRD-K58265391	Cc1cc2CCCS(=O)(=O)c2cc1S(N)(=O)=O	CID:4165	phase I
BRD-A33711280	CN1CCCC(CC2c3ccccc3Sc3ccccc23)C1	CID:4167	phase I
BRD-K75641298	CCN(CC)CCNC(=O)c1cc(Cl)c(N)cc1OC	CID:4168	phase I
BRD-A61793559	CC1Nc2cc(Cl)c(cc2C(=O)N1c1ccccc1C)S(N)(=O)=O	CID:4170	phase I
BRD-A03623303	COCCc1ccc(OCC(O)CNC(C)C)cc1	CID:4171	phase I
BRD-K52020312	Cc1ncc(n1CCO)[N+]([O-])=O	CID:4173	phase I
BRD-K46862739	CC(C)(C(=O)c1cccnc1)c1cccnc1	CID:4174	phase I
BRD-A64092382	CC(N)COc1c(C)cccc1C	CID:4178	phase I
BRD-A19661776	CN1CCN2C(C1)c1ccccc1Cc1ccccc21	CID:4184	phase I
BRD-A82396632	Clc1ccc(COC(Cn2ccnc2)c2ccc(Cl)cc2Cl)c(Cl)c1	CID:4189	phase I
BRD-K00532621	Cc1ncc2CN=C(c3ccccc3F)c4cc(Cl)ccc4-n12	CID:4192	phase I
BRD-A79981887	COc1ccc(OC)c(c1)C(O)CNC(=O)CN	CID:4195	phase I
BRD-A44780397	CC#CC1(O)CCC2C3CCC4=CC(=O)CCC4=C3C(CC21C)c5ccc(cc5)N(C)C	CID:4196	phase I
BRD-K67080878	Cc1[nH]c(=O)c(cc1-c1ccncc1)C#N	CID:4197	phase I
BRD-K02867583	Cc1cc(nnc1NCCN1CCOCC1)-c1ccccc1	CID:4199	phase I
BRD-A64977602	CN1CCN2C(C1)c1ccccc1Cc1cccnc21	CID:4205	phase I
BRD-A31204924	ClC(Cl)C(c1ccc(Cl)cc1)c1ccccc1Cl	CID:4211	phase I
BRD-K21680192	OCCNCCNc1ccc(NCCNCCO)c2C(=O)c3c(O)ccc(O)c3C(=O)c12	CID:4212	phase I
BRD-K93201660	Ic1cccc2c(cccc12)S(=O)(=O)N3CCCNCC3	CID:4216	phase I
BRD-K68402494	Clc1cccc2c(cccc12)S(=O)(=O)N1CCCNCC1	CID:4217	phase I
BRD-K07237224	Clc1ccc(cc1)C(=O)NCCN1CCOCC1	CID:4235	phase I
BRD-A16332958	NC(=O)CS(=O)C(c1ccccc1)c1ccccc1	CID:4236	phase I
BRD-K49372556	COc1ccc(cc1)c2noc(CC(=O)O)c2c3ccc(OC)cc3	CID:4237	phase I
BRD-K35531059	CCOC(=O)/N=c\1/c[n+]([n-]o1)N2CCOCC2	CID:4238	phase I
BRD-A43392971	CC1C(=O)OC2CCN3CC=C(COC(=O)C(C)(O)C1(C)O)C23	CID:4246	phase I
BRD-K74820615	CN1CCCN=C1C=Cc1sccc1C	CID:4250	phase I
BRD-K81144366	CC(C)c1cc(OC(C)=O)c(C)cc1OCCN(C)C	CID:4260	phase I
BRD-K77908580	Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1	CID:4261	phase I
BRD-A99449986	CCCCCCCCN1C(=O)C(=C(C)C1(C)O)C(=O)C	CID:4262	phase I
BRD-K31542390	COc1c(C)c2COC(=O)c2c(O)c1CC=C(C)CCC(=O)O	CID:4272	phase I
BRD-K81521265	O=C(NC1CCCCC1)NC2CCCCC2	CID:4277	phase I
BRD-K94080537	CCN(CC)C(=O)c1cccc(C)c1	CID:4284	phase I
BRD-K44899736	NCCNC(=O)c1ccc(Cl)cc1	CID:4289	phase I
BRD-K94887716	FC(F)(F)c1cccc(c1)N2CCNCC2	CID:4296	phase I
BRD-K78084463	NCCCCNS(=O)(=O)c1ccc2ccccc2c1	CID:4298	phase I
BRD-K45068323	NCCCCNS(=O)(=O)c1ccc2c(Cl)cccc2c1	CID:4299	phase I
BRD-K68341547	NCCCCCCNS(=O)(=O)c1ccc2c(Cl)cccc2c1	CID:4306	phase I
BRD-A47633927	CC(C)CC(NC(=O)OCC1c2ccccc2-c3ccccc13)C(=O)O	CID:4308	phase I
BRD-K41868777	NCCCCCCNS(=O)(=O)c1cccc2ccccc12	CID:4314	phase I
BRD-K98297262	CCN1C(=O)C=CC1=O	CID:4362	phase I
BRD-A61470182	CSCCC(NC=O)C(=O)NC(C)C(=O)O	CID:4363	phase I
BRD-K61951118	CNC(=O)c1cc2c(cn1)[nH]c1ccccc21	CID:4375	phase I
BRD-K73251053	CN(CCCOc1ccc(Cl)cc1Cl)CC#C	CID:4380	phase I
BRD-K31987754	CCCCCCCCC=CCCCCCCCC(=O)NCCO	CID:4383	phase I
BRD-A85234536	OCC1OC(C(O)C1O)n2cnc3c(NC4CCCC4)ncnc23	CID:4402	phase I
BRD-K65146499	COc1ccc2cc(CCC(C)=O)ccc2c1	CID:4409	phase I
BRD-A24397426	CC1CCc2c(N3CCC(O)CC3)c(F)cc3c2n1cc(C(O)=O)c3=O	CID:4410	phase I
BRD-A97454584	CC(C)(C)NCC(O)COc1cccc2CC(O)C(O)Cc12	CID:4411	phase I
BRD-A67862938	CCN(CC)CCOC(=O)C(CC1CCCO1)Cc1cccc2ccccc12	CID:4417	phase I
BRD-A01787639	COc1ccccc1N1CCN(CC(O)COc2cccc3ccccc23)CC1	CID:4418	phase I
BRD-K47886988	CCn1cc(C(O)=O)c(=O)c2ccc(C)nc12	CID:4421	phase I
BRD-A37541666	Oc1ccc2CC3N(CC=C)CCC4(C5Oc1c24)C3(O)CCC5=O	CID:4425	phase I
BRD-A41833852	Oc1ccc2CC3N(CC=C)CCC4(C5Oc1c24)C3(O)CCC5=NNC(=O)c6ccccc6	CID:4426	phase I
BRD-A83855350	Oc1ccc2CC3N(CC4CC4)CCC5(C6Oc1c25)C3(O)CCC6=O	CID:4428	phase I
BRD-A21723284	Oc1ccc2CC3N(CC4CC4)CCC5(C6Oc1c25)C3(O)Cc7c6oc8ccccc78	CID:4429	phase I
BRD-A82656074	Oc1ccc2CC3N(CC4CC4)CCC5(C6Oc1c25)C3(O)Cc7c6[nH]c8ccccc78	CID:4430	phase I
BRD-K69195780	COc1ccccc1N1CCN(CCCCN2C(=O)c3ccccc3C2=O)CC1	CID:4431	phase I
BRD-K77641333	C(C1=NCCN1)c1cccc2ccccc12	CID:4436	phase I
BRD-K90789829	CCc1nn(CCCN2CCN(CC2)c2cccc(Cl)c2)c(=O)n1CCOc1ccccc1	CID:4449	phase I
BRD-A78877355	CN1CCOC(c2ccccc2)c2ccccc2C1	CID:4450	phase I
BRD-A66927094	CNc1cc(OC)c(cc1Cl)C(=O)NC2CCN(Cc3ccccc3)C2C	CID:4452	phase I
BRD-K18922609	CN(C)C(=O)Oc1cccc(c1)[N+](C)(C)C	CID:4456	phase I
BRD-K15502390	Cc1ccnc2c1NC(=O)c1cccnc1N2C1CC1	CID:4463	phase I
BRD-K12102668	O=C(CCNNC(=O)c1ccncc1)NCc1ccccc1	CID:4472	phase I
BRD-A26711594	COC(=O)C1=C(C)NC(C)=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)OCCN(C)Cc1ccccc1	CID:4474	phase I
BRD-K35960502	Oc1ccc(Cl)cc1C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O	CID:4477	phase I
BRD-K96354014	COC(=O)C1=C(C)NC(C)=C(C1c1ccccc1[N+]([O-])=O)C(=O)OC	CID:4485	phase I
BRD-K32311154	Cn1c(NCCN(CCO)CCCc2ccc(cc2)[N+]([O-])=O)cc(=O)n(C)c1=O	CID:4486	phase I
BRD-K47407372	Cc1c(NC(=O)c2cccnc2)c(=O)n(-c2ccccc2)n1C	CID:4487	phase I
BRD-K98763141	OC(=O)c1cccnc1Nc1cccc(c1)C(F)(F)F	CID:4488	phase I
BRD-K23566484	CC1(C)NC(=O)N(C1=O)c1ccc(c(c1)C(F)(F)F)[N+]([O-])=O	CID:4493	phase I
BRD-K76775527	CS(=O)(=O)Nc1ccc(cc1Oc1ccccc1)[N+]([O-])=O	CID:4495	phase I
BRD-K70883034	CN1c2ccc(cc2C(=NCC1=O)c1ccccc1)[N+]([O-])=O	CID:4496	phase I
BRD-A58048407	COCCOC(=O)C1=C(C)NC(C)=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)OC(C)C	CID:4497	phase I
BRD-A84465106	COC(=O)C1=C(C)NC(C)=C(C1c1ccccc1[N+]([O-])=O)C(=O)OCC(C)C	CID:4499	phase I
BRD-A95696066	CNCCC(Oc1ccccc1OC)c1ccccc1	CID:4500	phase I
BRD-K57930253	[O-][N+](=O)c1ccc2NC(=O)CN=C(c3ccccc3)c2c1	CID:4506	phase I
BRD-A02006392	CCOC(=O)C1=C(C)NC(C)=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)OC	CID:4507	phase I
BRD-K92193792	CNC(NCCSCc1csc(CN(C)C)n1)=C[N+]([O-])=O	CID:4513	phase I
BRD-K42221274	OC(=O)C1=CCCN(CCON=C(c2ccccc2)c2ccccc2)C1	CID:4515	phase I
BRD-A29644307	CN1CC(c2ccccc2)c2cccc(N)c2C1	CID:4528	phase I
BRD-A11135865	Oc1ccc2CC3N(CC4CC4)CCC5(C6Oc1c25)C3(O)Cc7c8CC9(O)C%10Cc%11ccc(O)c%12OC(c8[nH]c67)C9(CCN%10CC%13CC%13)c%12%11	CID:4533	phase I
BRD-K11196887	CCn1cc(C(O)=O)c(=O)c2cc(F)c(cc12)N1CCNCC1	CID:4539	phase I
BRD-K91263825	CNCCC=C1c2ccccc2CCc2ccccc12	CID:4543	phase I
BRD-K54210043	Oc1ccc(cc1n2c(=O)[nH]c3cc(ccc23)C(F)(F)F)C(F)(F)F	CID:4552	phase I
BRD-A36267905	CC(CCc1ccccc1)NC(C)C(O)c1ccc(O)cc1	CID:4567	phase I
BRD-K48029790	CCCCCCCCCCCCCCCCCCc1ccc(cc1)C(=O)C=CC(=O)O	CID:4579	phase I
BRD-A14240607	NCC(O)c1ccc(O)cc1	CID:4581	phase I
BRD-A24228527	CC1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(O)=O)c3=O	CID:4583	phase I
BRD-K82731415	Cn1cnc2c(NCc3ccccc3)nc(NCCO)nc12	CID:4592	phase I
BRD-A55962179	COc1ccc2nc([nH]c2c1)S(=O)Cc1ncc(C)c(OC)c1C	CID:4594	phase I
BRD-A19736161	Cc1nccn1CC1CCc2c(C1=O)c1ccccc1n2C	CID:4595	phase I
BRD-A53576514	CN(C)CCOC(c1ccccc1)c1ccccc1C	CID:4601	phase I
BRD-A46747628	CC1OC(OC2CC(O)C3(CO)C4C(O)CC5(C)C(CCC5(O)C4CCC3(O)C2)C6=CC(=O)OC6)C(O)C(O)C1O	CID:4605	phase I
BRD-A03044413	Cc1onc(c1C(=O)NC1C2SC(C)(C)C(N2C1=O)C(O)=O)-c1ccccc1	CID:4608	phase I
BRD-K25394294	OC(=O)CCc1nc(c(o1)-c1ccccc1)-c1ccccc1	CID:4614	phase I
BRD-K56940463	CN(C(=O)CN(CCO)CC(=O)N(C)C(C)(C)Cc1ccccc1)C(C)(C)Cc1ccccc1	CID:4621	phase I
BRD-K52075715	CCCOc1ccc2nc(NC(=O)OC)[nH]c2c1	CID:4622	phase I
BRD-K88538023	Clc1ccc(CON=C(Cn2ccnc2)c3ccc(Cl)cc3Cl)c(Cl)c1	CID:4623	phase I
BRD-K41809988	NCCc1cc(O)c(O)cc1O	CID:4624	phase I
BRD-K73394555	CCn1cc(C(O)=O)c(=O)c2cc3OCOc3cc12	CID:4628	phase I
BRD-K21936341	O=C1CCCN1CC#CCN1CCCC1	CID:4630	phase I
BRD-A43671941	CC(C)NCC(O)COc1ccccc1OCC=C	CID:4631	phase I
BRD-K59037100	COc1ccc(C(=O)c2ccccc2)c(O)c1	CID:4632	phase I
BRD-K04185004	CCCCOc1cc(ccc1N)C(=O)OCCN(CC)CC	CID:4633	phase I
BRD-A65013509	CCN(CC)CC#CCOC(=O)C(O)(C1CCCCC1)c1ccccc1	CID:4634	phase I
BRD-K16195444	Cc1cc(c(O)c(C)c1CC1=NCCN1)C(C)(C)C	CID:4636	phase I
BRD-A33749298	CCCCC1C(=O)N(N(C1=O)c1ccc(O)cc1)c1ccccc1	CID:4641	phase I
BRD-K19525698	OC(=O)C=Cc1ccc(Cn2ccnc2)cc1	CID:4646	phase I
BRD-K80267133	Nc1ccc(C(O)=O)c(O)c1	CID:4649	phase I
BRD-A23723433	CC(=O)OC1C2=C(C)C(CC(O)(C(OC(=O)c3ccccc3)C4C5(COC5CC(O)C4(C)C1=O)OC(=O)C)C2(C)C)OC(=O)C(O)C(NC(=O)c6ccccc6)c7ccccc7	CID:4666	phase I
BRD-K68095457	CCCCCCCCCCCCCCCC(=O)NCCO	CID:4671	phase I
BRD-A22380646	COc1ccnc(CS(=O)c2nc3cc(OC(F)F)ccc3[nH]2)c1OC	CID:4679	phase I
BRD-K15567136	COc1ccc(Cc2nccc3cc(OC)c(OC)cc23)cc1OC	CID:4680	phase I
BRD-K40992116	Oc1ccc(Cl)cc1	CID:4684	phase I
BRD-K83597974	CN(CC#C)Cc1ccccc1	CID:4688	phase I
BRD-A62326914	Fc1ccc(cc1)C2CCNCC2COc3ccc4OCOc4c3	CID:4691	phase I
BRD-A29289453	COC(=O)C1=C(C)NC(C)=C(C1C)C(=O)OCCSc1ccccc1	CID:4698	phase I
BRD-A63836183	CN(C)c1ccc(Cn2cnc3CN(C(Cc32)C(=O)O)C(=O)C(c4ccccc4)c5ccccc5)cc1C	CID:4701	phase I
BRD-K48735772	CNc1cc2c(Nc3cccc(Br)c3)ncnc2cn1	CID:4707	phase I
BRD-K77133231	[O-][N+](=O)c1ccc(cc1)c2nc(c([nH]2)c3ccncc3)c4ccc(F)cc4	CID:4712	phase I
BRD-K62810658	COc1cccc(-c2cc(=O)c3ccccc3o2)c1N	CID:4713	phase I
BRD-A80793822	NC1=NC(=O)C(O1)c1ccccc1	CID:4723	phase I
BRD-A43150328	COC1=CC(=O)OC1(O)C(=C)C	CID:4728	phase I
BRD-A84702196	CC1(C)SC2C(NC(=O)COc3ccccc3)C(=O)N2C1C(=O)O	CID:4731	phase I
BRD-K13183738	NC(=N)c1ccc(OCCCCCOc2ccc(cc2)C(N)=N)cc1	CID:4735	phase I
BRD-A44448661	CCCC(C)C1(CC)C(=O)NC(=O)NC1=O	CID:4737	phase I
BRD-K57569181	CC(=O)CCCCn1c(=O)n(C)c2ncn(C)c2c1=O	CID:4740	phase I
BRD-A19633847	C(C(C1CCCCC1)C1CCCCC1)C1CCCCN1	CID:4746	phase I
BRD-K10995081	OCCN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc23)CC1	CID:4748	phase I
BRD-K38323065	CCOc1ccc(NC(C)=O)cc1	CID:4754	phase I
BRD-K76304753	Nc1ccc(\N=N\c2ccccc2)c(N)n1	CID:4756	phase I
BRD-K70592963	O=C1C(C(=O)c2ccccc12)c1ccccc1	CID:4760	phase I
BRD-A23072235	CN(C)CCC(c1ccccc1)c1ccccn1	CID:4761	phase I
BRD-K19227686	Oc1ccc(cc1)C1(OC(=O)c2ccccc12)c1ccc(O)cc1	CID:4764	phase I
BRD-A67799922	CC(COc1ccccc1)N(CCCl)Cc1ccccc1	CID:4768	phase I
BRD-K22009844	NC(=O)OCCCc1ccccc1	CID:4770	phase I
BRD-K96319534	CC(C)(N)Cc1ccccc1	CID:4771	phase I
BRD-K67102207	OC(=O)CCCc1ccccc1	CID:4775	phase I
BRD-K31491153	NC(=N)NC(=N)Nc1ccccc1	CID:4780	phase I
BRD-K10843433	CCCCC1C(=O)N(N(C1=O)c1ccccc1)c1ccccc1	CID:4781	phase I
BRD-K33422401	FS(=O)(=O)Cc1ccccc1	CID:4784	phase I
BRD-K15563106	Oc1ccc(CCC(=O)c2c(O)cc(O)cc2O)cc1	CID:4788	phase I
BRD-A15079084	CCCCCCCCCCCCCC(=O)OC1C(C)C2(O)C3C=C(C)C(=O)C3(O)CC(=CC2C4C(C)(C)C41OC(=O)C)CO	CID:4792	phase I
BRD-K64659768	OC(=O)c1ccccc1C(=O)Nc1ccc(cc1)S(=O)(=O)Nc1nccs1	CID:4806	phase I
BRD-K77771411	COc1nc(C)nc(Cl)c1NC1=NCCN1	CID:4810	phase I
BRD-K26241953	Oc1cc(O)cc(C=Cc2ccc(O)c(O)c2)c1	CID:4813	phase I
BRD-K67277431	COc1ccc(cc1C(=O)NCc1cccnc1)C(=O)NCc1cccnc1	CID:4814	phase I
BRD-K66874953	Cc1ccc(cc1)C(=O)Cn1c2CCCCc2sc1=N	CID:4817	phase I
BRD-K88090157	CN1CCC(CC1)=C1c2ccccc2Sc2ccccc12	CID:4822	phase I
BRD-A22897758	CC(C(C)(C)C)\N=C(/NC#N)Nc1ccncc1	CID:4826	phase I
BRD-A97701745	CC(C)NCC(O)COc1cccc2[nH]ccc12	CID:4828	phase I
BRD-A48430263	CCc1ccc(CCOc2ccc(CC3SC(=O)NC3=O)cc2)nc1	CID:4829	phase I
BRD-K26801045	NC(=O)C1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)N1CCCCC1	CID:4830	phase I
BRD-K08999871	CCn1cc(C(O)=O)c(=O)c2cnc(nc12)N1CCNCC1	CID:4831	phase I
BRD-A97479839	CCN1CCCC(C1)OC(=O)C(c1ccccc1)c1ccccc1	CID:4839	phase I
BRD-K19456237	NC(=O)CN1CCCC1=O	CID:4843	phase I
BRD-K25224017	Cc1nc2ccccn2c(=O)c1CCN1CCC(CC1)C(=O)c1ccc(F)cc1	CID:4847	phase I
BRD-K89375097	CN1CCN(CC(=O)N2c3ccccc3C(=O)Nc3cccnc23)CC1	CID:4848	phase I
BRD-K87990216	NS(=O)(=O)c1cc(cc(N2CCCC2)c1Oc1ccccc1)C(O)=O	CID:4849	phase I
BRD-K47936004	C(N1CCN(CC1)c1ncccn1)c1ccc2OCOc2c1	CID:4850	phase I
BRD-K37682401	CCn1cc(C(O)=O)c(=O)c2cnc(nc12)N1CCCC1	CID:4855	phase I
BRD-K11853856	CN(C)CC(=O)Nc1ccc2[nH]c(=O)c3ccccc3c2c1	CID:4858	phase I
BRD-A16746338	COc1cc(cc(OC)c1OC)C1C2C(COC2=O)C(O)c2cc3OCOc3cc12	CID:4865	phase I
BRD-K95785537	CC(C)(C)n1nc(-c2ccc(Cl)cc2)c2c(N)ncnc12	CID:4878	phase I
BRD-K16977723	Nc1ncnc2n(ncc12)c3ccccc3	CID:4879	phase I
BRD-A41304429	CC(C)NCC(O)COc1ccc(NC(C)=O)cc1	CID:4883	phase I
BRD-K61327230	C[n+]1ccccc1C=NO	CID:4884	phase I
BRD-K46523383	CCCCOc1ccc(OCCCN2CCOCC2)cc1	CID:4886	phase I
BRD-K97045029	O=C(Nc1cccc2c1oc(cc2=O)-c1nnn[nH]1)c1ccc(OCCCCc2ccccc2)cc1	CID:4887	phase I
BRD-A64610707	CC(C(O)=O)c1ccc2Oc3ncccc3Cc2c1	CID:4888	phase I
BRD-A11170096	CCC(C)C(=O)OC1CC(O)C=C2C=CC(C)C(CCC(O)CC(O)CC(O)=O)C12	CID:4889	phase I
BRD-A21858158	O=C(C1CCCCC1)N1CC2N(CCc3ccccc23)C(=O)C1	CID:4891	phase I
BRD-K49111258	COc1cc2nc(nc(N)c2cc1OC)N3CCN(CC3)C(=O)c4ccco4	CID:4893	phase I
BRD-A53952395	CCCNC(C)C(=O)Nc1ccccc1C	CID:4906	phase I
BRD-A55913614	COc1cc(NC(C)CCCN)c2ncccc2c1	CID:4908	phase I
BRD-K32247306	CCC1(C(=O)NCNC1=O)c1ccccc1	CID:4909	phase I
BRD-K46317332	CCCC(C(=O)OCCN(CC)CC)(c1ccccc1)c1ccccc1	CID:4910	phase I
BRD-K95237249	CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(O)=O	CID:4911	phase I
BRD-K72029282	CC(C)(Sc1cc(c(O)c(c1)C(C)(C)C)C(C)(C)C)Sc1cc(c(O)c(c1)C(C)(C)C)C(C)(C)C	CID:4912	phase I
BRD-K75089421	CCN(CC)CCNC(=O)c1ccc(N)cc1	CID:4913	phase I
BRD-K24616672	CCN(CC)CCOC(=O)c1ccc(N)cc1	CID:4914	phase I
BRD-K13032584	CNNCc1ccc(cc1)C(=O)NC(C)C	CID:4915	phase I
BRD-A22684332	CCC(NC(C)C)C(O)c1ccc(O)c2[nH]c(=O)ccc12	CID:4916	phase I
BRD-K19352500	CN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc23)CC1	CID:4917	phase I
BRD-A31800922	OC(CCN1CCCC1)(C1CCCCC1)c1ccccc1	CID:4919	phase I
BRD-A44863528	CCCN(CCC)C(=O)C(CCC(O)=O)NC(=O)c1ccccc1	CID:4922	phase I
BRD-K28183345	CC(C)NC(=N)NC(=N)Nc1ccc(Cl)cc1	CID:4923	phase I
BRD-K06980535	CN(C)CCCN1c2ccccc2Sc2ccccc12	CID:4926	phase I
BRD-A46335897	CC(CN1c2ccccc2Sc2ccccc12)N(C)C	CID:4927	phase I
BRD-K99029477	COc1nc(NC(C)C)nc(NC(C)C)n1	CID:4928	phase I
BRD-A87715314	CC(C)NCC(O)c1ccc2ccccc2c1	CID:4930	phase I
BRD-A26334849	CCCNCC(O)COc1ccccc1C(=O)CCc1ccccc1	CID:4932	phase I
BRD-K90885812	CC(C)[N+](C)(CCOC(=O)C1c2ccccc2Oc2ccccc12)C(C)C	CID:4934	phase I
BRD-K79116891	CCCOc1ccc(cc1N)C(=O)OCCN(CC)CC	CID:4935	phase I
BRD-K59273480	CCCn1cnc2n(C)c(=O)n(CCCCC(C)=O)c(=O)c12	CID:4938	phase I
BRD-K14821965	CC[N+](C)(CC)CCC[n+]1c(-c2ccccc2)c2cc(N)ccc2c2ccc(N)cc12	CID:4939	phase I
BRD-K82255054	CC(C)c1cccc(C(C)C)c1O	CID:4943	phase I
BRD-A10070317	CC(C)NCC(O)COc1cccc2ccccc12	CID:4946	phase I
BRD-K83302049	CN1CCc2cc3OCOc3cc2C(=O)Cc4ccc5OCOc5c4C1	CID:4970	phase I
BRD-K42098891	CNCCCC1c2ccccc2C=Cc2ccccc12	CID:4976	phase I
BRD-K63072637	CN1CCCN=C1C=Cc1cccs1	CID:4989	phase I
BRD-K69688083	CN(C)C(=O)Oc1ccc[n+](C)c1	CID:4991	phase I
BRD-K97564742	COc1ccc(cc1)CN(CCN(C)C)c1ccccn1	CID:4992	phase I
BRD-K88429204	CCc1nc(N)nc(N)c1-c1ccc(Cl)cc1	CID:4993	phase I
BRD-K36116267	CCC1(CC)C(=O)NC=CC1=O	CID:4994	phase I
BRD-K11663430	ONC(=O)CCCCCCC(=O)Nc1cccnc1	CID:4996	phase I
BRD-K68867920	OCCOCCN1CCN(CC1)C1=Nc2ccccc2Sc2ccccc12	CID:5002	phase I
BRD-K77925998	C1CN(CCN1)c1ccc2ccccc2n1	CID:5011	phase I
BRD-K62056274	CN1CCN(CC1)c1ccc2ccccc2n1	CID:5013	phase I
BRD-K40782193	Cc1cccc(C)c1NC(=O)C[N+](C)(C)C	CID:5014	phase I
BRD-A39390670	COCCCOc1ccnc(CS(=O)c2nc3ccccc3[nH]2)c1C	CID:5029	phase I
BRD-A54236247	CNC(C)C(O)c1ccccc1	CID:5032	phase I
BRD-K39520573	Oc1c(Br)cc(C=C2C(=O)Nc3ccc(I)cc23)cc1Br	CID:5034	phase I
BRD-K63828191	Oc1ccc(cc1)-c1sc2cc(O)ccc2c1C(=O)c1ccc(OCCN2CCCCC2)cc1	CID:5035	phase I
BRD-K85333151	CC(C)Nc1c(C)n(C)n(-c2ccccc2)c1=O	CID:5037	phase I
BRD-K30816563	CNC(=C[N+](=O)[O-])NCCSCc1ccc(CN(C)C)o1	CID:5039	phase I
BRD-A15909516	OC(=O)C(Cc1cc(=O)[nH]c2ccccc12)NC(=O)c1ccc(Cl)cc1	CID:5042	phase I
BRD-A71765365	COC1C(CC2CN3CCc4c([nH]c5cc(OC)ccc45)C3CC2C1C(=O)OC)OC(=O)c6cc(OC)c(OC)c(OC)c6	CID:5052	phase I
BRD-A83431637	CC(=CC1C(C(=O)OCc2coc(Cc3ccccc3)c2)C1(C)C)C	CID:5053	phase I
BRD-K85603128	CC(=O)Oc1cccc(O)c1	CID:5055	phase I
BRD-K25591257	Oc1ccc(C=Cc2cc(O)cc(O)c2)cc1	CID:5056	phase I
BRD-A68281735	CCCCCC(O)c1cccc(OCc2ccc3ccccc3n2)c1	CID:5059	phase I
BRD-K56047318	O=C(NCCCCCCNC(=O)ON=C1CCCCC1)ON=C1CCCCC1	CID:5063	phase I
BRD-A96255180	NC(=O)c1ncn(n1)C1OC(CO)C(O)C1O	CID:5064	phase I
BRD-K21283037	Nc1nc2ccc(OC(F)(F)F)cc2s1	CID:5070	phase I
BRD-A63346720	CC1CN(CCCn2c3ccccc3c4ccccc24)CC(C)N1	CID:5072	phase I
BRD-K53857191	Cc1nc2CCCCn2c(=O)c1CCN1CCC(CC1)c1noc2cc(F)ccc12	CID:5073	phase I
BRD-K40887525	Cc1nc2sccn2c(=O)c1CCN1CCC(CC1)=C(c1ccc(F)cc1)c1ccc(F)cc1	CID:5074	phase I
BRD-A03323675	CC(C)C(NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)NC(CC(O)C(Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1	CID:5076	phase I
BRD-K75699339	CN(C)CCc1c[nH]c2ccc(Cn3cncn3)cc12	CID:5078	phase I
BRD-K82823076	CCOC(=O)c1ncn-2c1CN(C)C(=O)c1cc(ccc-21)N=[N+]=[N-]	CID:5081	phase I
BRD-K06543683	Cn1cc(C2=C(C(=O)NC2=O)c2cn(CCCSC(N)=N)c3ccccc23)c2ccccc12	CID:5083	phase I
BRD-K21733600	CS(=O)(=O)c1ccc(cc1)C1=C(C(=O)OC1)c1ccccc1	CID:5090	phase I
BRD-A34255068	COc1ccc(cc1OC1CCCC1)C1CNC(=O)C1	CID:5092	phase I
BRD-K94266545	Cn1c(COC(N)=O)ncc1[N+]([O-])=O	CID:5094	phase I
BRD-K15933101	CCCN(CCC)CCc1cccc2NC(=O)Cc12	CID:5095	phase I
BRD-K39256324	CC(=O)c1c(O)c(C)c(O)c(Cc2c(O)c(C(=O)C=Cc3ccccc3)c4OC(C)(C)C=Cc4c2O)c1O	CID:5103	phase I
BRD-K22685337	Oc1ccc(cc1[N+]([O-])=O)[As](O)(O)=O	CID:5104	phase I
BRD-K81855038	CC(=O)OCC(=O)NCCCOc1cccc(CN2CCCCC2)c1	CID:5105	phase I
BRD-A01320529	OCc1cc(ccc1O)C(O)CNCCCCCCOCCCCc1ccccc1	CID:5152	phase I
BRD-K36395411	Cn1ccc2cc3N(CCc3cc12)C(=O)Nc1cccnc1	CID:5163	phase I
BRD-K54330070	Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1	CID:5169	phase I
BRD-K54729176	ONC(=O)CCCCCCC(=O)NO	CID:5173	phase I
BRD-K85871428	Cc1nc(c(o1)c2ccncc2)c3ccccc3	CID:5174	phase I
BRD-K05361803	CCCCCCCNS(=O)(=O)c1cccc2c(Cl)cccc12	CID:5175	phase I
BRD-A14566392	CN1C2CC(CC1C3OC32)OC(=O)C(CO)c4ccccc4	CID:5184	phase I
BRD-K22503835	ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23	CID:5186	phase I
BRD-K15868788	CCN(CC)CCOC(=O)c1cc(Cl)c(N)cc1OC	CID:5191	phase I
BRD-A23359898	CC(C)CC(N(C)C)C1(CCC1)c1ccc(Cl)cc1	CID:5210	phase I
BRD-A83815268	COc1cc(ccc1O)C2Oc3cc(ccc3OC2CO)C4Oc5cc(O)cc(O)c5C(=O)C4O	CID:5213	phase I
BRD-K32273377	Nc1ccc(cc1)S(=O)(=O)Nc1ncccn1	CID:5215	phase I
BRD-K96809896	Fc1ccc(cc1)-c1nc2SCCn2c1-c1ccncc1	CID:5228	phase I
BRD-K88868628	OC(=O)CI	CID:5240	phase I
BRD-A33168282	CC(C)NCC(O)c1ccc(NS(C)(=O)=O)cc1	CID:5253	phase I
BRD-K55468218	Fc1ccc(cc1)C(=O)CCCN1CCC2(CC1)N(CNC2=O)c1ccccc1	CID:5265	phase I
BRD-A72483914	O=C1NCN(c2ccccc2)C11CCN(CC2COc3ccccc3O2)CC1	CID:5268	phase I
BRD-K27710560	O=C1CCc2c(O1)ccc1ccccc21	CID:5269	phase I
BRD-A56987319	Nc1ncnc2n(cnc12)C1CCCO1	CID:5270	phase I
BRD-K93280214	COc1ccc(cc1)c2ccc(N)[n+](CCCC(=O)O)n2	CID:5275	phase I
BRD-K68332390	OC(=O)Cc1nn(Cc2ccc(Br)cc2F)c(=O)c3ccccc13	CID:5278	phase I
BRD-A71203467	COc1cc2CCN3Cc4c(OC)c(O)ccc4CC3c2cc1O	CID:5290	phase I
BRD-K92723993	CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1	CID:5291	phase I
BRD-A84066268	CC12CCC3C(CCC4(O)CC(O)CCC34C=O)C2(O)CCC1C5=CC(=O)OC5	CID:5303	phase I
BRD-K81418486	ONC(=O)CCCCCCC(=O)Nc1ccccc1	CID:5311	phase I
BRD-K01950558	OC(=O)CCC(=O)Nc1ccc(cc1)S(=O)(=O)Nc1nccs1	CID:5315	phase I
BRD-A70649075	Clc1ccc(CSC(Cn2ccnc2)c2ccc(Cl)cc2Cl)cc1	CID:5318	phase I
BRD-K59983611	Nc1ccc(cc1)S(=O)(=O)NC(=O)c1ccccc1	CID:5319	phase I
BRD-K21520694	CC(=O)NS(=O)(=O)c1ccc(N)cc1	CID:5320	phase I
BRD-K71125014	COc1cc(NS(=O)(=O)c2ccc(N)cc2)nc(OC)n1	CID:5323	phase I
BRD-K45086103	NC(=N)NS(=O)(=O)c1ccc(N)cc1	CID:5324	phase I
BRD-K93524252	Cc1ccnc(NS(=O)(=O)c2ccc(N)cc2)n1	CID:5325	phase I
BRD-K11640013	Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1	CID:5327	phase I
BRD-K31682896	Cc1nnc(NS(=O)(=O)c2ccc(N)cc2)s1	CID:5328	phase I
BRD-K28494619	Cc1cc(NS(=O)(=O)c2ccc(N)cc2)no1	CID:5329	phase I
BRD-K00938507	COc1ccc(NS(=O)(=O)c2ccc(N)cc2)nn1	CID:5330	phase I
BRD-K14116214	COc1cc(NS(=O)(=O)c2ccc(N)cc2)ncn1	CID:5332	phase I
BRD-K10671814	Nc1ccc(cc1)S(=O)(=O)Nc1ccnn1-c1ccccc1	CID:5335	phase I
BRD-K41406082	Nc1ccc(cc1)S(=O)(=O)Nc1ccccn1	CID:5336	phase I
BRD-K71133585	Nc1ccc(cc1)S(=O)(=O)Nc1cnc2ccccc2n1	CID:5338	phase I
BRD-K10670311	OC(=O)c1cc(ccc1O)\N=N\c1ccc(cc1)S(=O)(=O)Nc1ccccn1	CID:5339	phase I
BRD-K14705039	Nc1ccc(cc1)S(=O)(=O)Nc1nccs1	CID:5340	phase I
BRD-A36217750	O=C1C(CCS(=O)c2ccccc2)C(=O)N(N1c1ccccc1)c1ccccc1	CID:5342	phase I
BRD-K50859149	Cc1noc(NS(=O)(=O)c2ccc(N)cc2)c1C	CID:5344	phase I
BRD-A58955223	CS(=O)CCCCN=C=S	CID:5350	phase I
BRD-A03427350	CC1=C(CC(=O)O)c2cc(F)ccc2C1=Cc3ccc(cc3)S(=O)C	CID:5352	phase I
BRD-A34205397	CCCCCCCCNC(C)C(O)c1ccc(SC(C)C)cc1	CID:5354	phase I
BRD-A55272860	CCN1CCCC1CNC(=O)c1cc(ccc1OC)S(N)(=O)=O	CID:5355	phase I
BRD-K50938287	CNS(=O)(=O)Cc1ccc2[nH]cc(CCN(C)C)c2c1	CID:5358	phase I
BRD-A34006693	CC(C(O)=O)c1ccc(cc1)C(=O)c1cccs1	CID:5359	phase I
BRD-K70327167	Cc1ccc(cc1NC(=O)c1cccc(NC(=O)Nc2cccc(c2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(c3cc(cc(c23)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O)c1)C(=O)Nc1ccc(c2cc(cc(c12)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O	CID:5361	phase I
BRD-K78815826	CCCCC1(COC(=O)CCC(O)=O)C(=O)N(N(C1=O)c1ccccc1)c1ccccc1	CID:5362	phase I
BRD-K63516691	COC(=O)c1c(-c2cc(OC)c(OC)c(OC)c2)c2ccnc(OCc3ncccn3)c2c(=O)n1Cc1ccnc(C)c1	CID:5368	phase I
BRD-K75615183	Nc1nc2CCN(CC=C)CCc2s1	CID:5374	phase I
BRD-K43744935	CCC(=C(c1ccccc1)c2ccc(OCCN(C)C)cc2)c3ccccc3	CID:5376	phase I
BRD-A74980173	COc1c(N2CCNC(C)C2)c(F)cc2c1n(cc(C(O)=O)c2=O)C1CC1	CID:5379	phase I
BRD-K30743633	Clc1cnc(Oc2ccc(Oc3ncc(Cl)cc3Cl)cc2)c(Cl)c1	CID:5382	phase I
BRD-K34820100	CNC(=O)N(C)c1nnc(s1)C(C)(C)C	CID:5383	phase I
BRD-A79903587	Fc1cn(C2CCCO2)c(=O)[nH]c1=O	CID:5386	phase I
BRD-K06147391	CN1CCN(CC(=O)N2c3c(C)scc3C(=O)Nc3ccccc23)CC1	CID:5387	phase I
BRD-K51805276	COP(=S)(OC)Oc1ccc(Sc2ccc(OP(=S)(OC)OC)cc2)cc1	CID:5392	phase I
BRD-K32107296	Cn1nnc2c(ncn2c1=O)C(N)=O	CID:5394	phase I
BRD-A33833419	CN(C)CC1Cc2ccccc2C1=O	CID:5400	phase I
BRD-A22256192	COc1cc2nc(nc(N)c2cc1OC)N1CCN(CC1)C(=O)C1CCCO1	CID:5401	phase I
BRD-A50157456	CC(C)(C)NCC(O)c1cc(O)cc(O)c1	CID:5403	phase I
BRD-A06352418	CC(C)(C)c1ccc(cc1)C(O)CCCN1CCC(CC1)C(O)(c1ccccc1)c1ccccc1	CID:5405	phase I
BRD-A79479878	CC12CCC3C(CCC4=CC(=O)CCC34C)C2CCC1O	CID:5408	phase I
BRD-K45071273	CCCCNc1ccc(cc1)C(=O)OCCN(C)C	CID:5411	phase I
BRD-A43940795	COc1ccc2CC3N(CCc4cc(OC)c(OC)cc34)Cc2c1OC	CID:5417	phase I
BRD-A28856712	C1CN=C(N1)C1CCCc2ccccc12	CID:5419	phase I
BRD-A93255169	O=C1N(C2CCC(=O)NC2=O)C(=O)c2ccccc12	CID:5426	phase I
BRD-K34888156	Cn1cnc2n(C)c(=O)[nH]c(=O)c12	CID:5429	phase I
BRD-K77695569	c1nc(cs1)-c1nc2ccccc2[nH]1	CID:5430	phase I
BRD-K69600043	CCSc1ccc2Sc3ccccc3N(CCCN3CCN(C)CC3)c2c1	CID:5440	phase I
BRD-A84481105	CSc1ccc2Sc3ccccc3N(CCC3CCCCN3C)c2c1	CID:5452	phase I
BRD-K09631521	S=P(N1CC1)(N1CC1)N1CC1	CID:5453	phase I
BRD-K13387373	CCCCCCCCCCCCCCCC[N+](C)(C)CCN(Cc1ccc(OC)cc1)c1ncccn1	CID:5456	phase I
BRD-K57432881	CCN(CC)CCNC(=O)c1cc(ccc1OC)S(C)(=O)=O	CID:5467	phase I
BRD-A72988804	CC(C(O)=O)c1ccc(s1)C(=O)c1ccccc1	CID:5468	phase I
BRD-K00603606	Clc1ccccc1CN1CCc2sccc2C1	CID:5472	phase I
BRD-K89125793	CCS(=O)(=O)CCn1c(C)ncc1[N+]([O-])=O	CID:5479	phase I
BRD-A33084557	Clc1sccc1COC(Cn1ccnc1)c1ccc(Cl)cc1Cl	CID:5482	phase I
BRD-K06335600	Clc1ccc2nsnc2c1NC1=NCCN1	CID:5487	phase I
BRD-K45988865	COc1ccc(C=Cc2cc(OC)cc(OC)c2)c(OC)c1	CID:5491	phase I
BRD-K68553471	CCOC(=O)NNc1nncc2ccccc12	CID:5501	phase I
BRD-K32164935	Cc1ccc(cc1)S(=O)(=O)NC(=O)NN1CCCCCC1	CID:5503	phase I
BRD-K46211610	C(C1=NCCN1)c1ccccc1	CID:5504	phase I
BRD-K85119730	CCCCNC(=O)NS(=O)(=O)c1ccc(C)cc1	CID:5505	phase I
BRD-K82562631	Cc1ccc(cc1)C(=O)c1ccc(CC(O)=O)n1C	CID:5509	phase I
BRD-K44273375	CN(C(=S)Oc1ccc2ccccc2c1)c1cccc(C)c1	CID:5510	phase I
BRD-A59985574	CCC1(O)C(=O)OCc2c1cc1-c3nc4ccc(O)c(CN(C)C)c4cc3Cn1c2=O	CID:5515	phase I
BRD-K63460351	CN(C)CCOc1ccc(cc1)C(=C(CCCl)c1ccccc1)c1ccccc1	CID:5516	phase I
BRD-A41450521	NC1CCN(C1)c1nc2n(cc(C(O)=O)c(=O)c2cc1F)-c1ccc(F)cc1F	CID:5517	phase I
BRD-K34154330	CCCCNc1c(C(=O)OCC)c(C)nc2n(CC)ncc12	CID:5522	phase I
BRD-K19533706	COc1ccc(C=CC(=O)Nc2ccccc2C(=O)O)cc1OC	CID:5527	phase I
BRD-K95763993	CCN(CC)c1cc(C)nc2ncnn12	CID:5531	phase I
BRD-K70778732	Clc1cccc(c1)N1CCN(CCCn2nc3ccccn3c2=O)CC1	CID:5533	phase I
BRD-K08619838	C(C#CCN1CCCC1)N1CCCC1	CID:5534	phase I
BRD-K84663978	COc1cc2CCn3c(c\c(=N/c4c(C)cc(C)cc4C)n(C)c3=O)-c2cc1OC	CID:5537	phase I
BRD-K06926592	CC(=CC=CC(=CC(=O)O)C)C=CC1=C(C)CCCC1(C)C	CID:5538	phase I
BRD-K92049597	Nc1nc(N)c2nc(-c3ccccc3)c(N)nc2n1	CID:5546	phase I
BRD-A28940325	NS(=O)(=O)c1cc2c(NC(NS2(=O)=O)C(Cl)Cl)cc1Cl	CID:5560	phase I
BRD-K41731458	Oc1cc(Cl)ccc1Oc1ccc(Cl)cc1Cl	CID:5564	phase I
BRD-K89732114	CN1CCN(CCCN2c3ccccc3Sc3ccc(cc23)C(F)(F)F)CC1	CID:5566	phase I
BRD-K63675182	CN(C)CCCN1c2ccccc2Sc2ccc(cc12)C(F)(F)F	CID:5568	phase I
BRD-A48180038	OC(CCN1CCCCC1)(C1CCCCC1)c1ccccc1	CID:5572	phase I
BRD-A92630576	CCC(COC(=O)c1cc(OC)c(OC)c(OC)c1)(N(C)C)c1ccccc1	CID:5573	phase I
BRD-A49225603	CC(CN(C)C)CN1c2ccccc2Sc2ccccc12	CID:5574	phase I
BRD-K16606819	CN1C(=O)OC(C)(C)C1=O	CID:5576	phase I
BRD-K34415467	COc1cc(cc(OC)c1OC)C(=O)NCc1ccc(OCCN(C)C)cc1	CID:5577	phase I
BRD-K07208025	COc1cc(Cc2cnc(N)nc2N)cc(OC)c1OC	CID:5578	phase I
BRD-A19195498	CC(CN(C)C)CN1c2ccccc2CCc2ccccc12	CID:5584	phase I
BRD-K54790157	Cc1cc2cc3c(C)cc(=O)oc3c(C)c2o1	CID:5585	phase I
BRD-K57033106	CN(C)CCN(Cc1ccccc1)c1ccccn1	CID:5587	phase I
BRD-K56231354	Cc1ccc(cc1)C(=CCN2CCCC2)c3ccccn3	CID:5588	phase I
BRD-A13084692	Cc1c(C)c2OC(C)(COc3ccc(CC4SC(=O)NC4=O)cc3)CCc2c(C)c1O	CID:5591	phase I
BRD-A79672927	CCN(Cc1ccncc1)C(=O)C(CO)c1ccccc1	CID:5593	phase I
BRD-A83859836	CN1C2CCC1CC(C2)OC(=O)c3c[nH]c4ccccc34	CID:5595	phase I
BRD-A68589262	COc1cc(cc(OC)c1OC)C(=O)NC1CCCNC1	CID:5597	phase I
BRD-K00959089	FC(F)(F)C(=O)CC(=O)c1cccs1	CID:5601	phase I
BRD-K68246049	CC(=Cc1ccc(cc1)C(=O)O)c2ccc3c(c2)C(C)(C)CCC3(C)C	CID:5602	phase I
BRD-K40255344	CC(C)(C)c1cc(C=C(C#N)C#N)cc(c1O)C(C)(C)C	CID:5614	phase I
BRD-K70281171	CCCN(CCC)C1Cc2cc(OC)c(OC)cc2C1	CID:5626	phase I
BRD-K46419649	NC(=C(C#N)C(=C(N)Sc1ccccc1N)C#N)Sc2ccccc2N	CID:5637	phase I
BRD-K73196317	COc1ccccc1N1CCN(CCCNc2cc(=O)n(C)c(=O)n2C)CC1	CID:5639	phase I
BRD-K24297741	CCOC(N)=O	CID:5641	phase I
BRD-A14792000	CCCCC(=O)N(Cc1ccc(cc1)-c1ccccc1-c1nn[nH]n1)C(C(C)C)C(O)=O	CID:5650	phase I
BRD-A51714012	COc1ccc(cc1)C(CN(C)C)C1(O)CCCCC1	CID:5656	phase I
BRD-A07893380	NC(CCC(O)=O)C=C	CID:5665	phase I
BRD-A59198242	CCOc1ccccc1OCC1CNCCO1	CID:5666	phase I
BRD-A22783572	CCC1(O)CC2CN(C1)CCc3c([nH]c4ccccc34)C(C2)(C(=O)OC)c5cc6c(cc5OC)N(C)C7C86CCN9CC=CC(CC)(C98)C(C(=O)OC)C7(O)C(=O)OC	CID:5667	phase I
BRD-A19374631	CCOC(=O)C1=CC2(CC)CCCN3CCc4c(C32)n1c5ccccc45	CID:5673	phase I
BRD-K90259198	NCCCCCCNS(=O)(=O)c1cccc2c(Cl)cccc12	CID:5681	phase I
BRD-K69812556	COc1ccccc1N1CCN(CCN(C(=O)C2CCCCC2)c2ccccn2)CC1	CID:5684	phase I
BRD-A75409952	COCC1OC(=O)c2coc3c2C1(C)C1=C(C2CCC(=O)C2(C)CC1OC(C)=O)C3=O	CID:5691	phase I
BRD-K01902415	Cc1cccc(Nc2cc(Cl)nc(SCC(O)=O)n2)c1C	CID:5694	phase I
BRD-K21565985	Cc1cccc(C)c1NC1=NCCCS1	CID:5707	phase I
BRD-K08356259	Cc1cc(cc(C)c1CC1=NCCN1)C(C)(C)C	CID:5709	phase I
BRD-A58280226	CC(N)C1CCC(CC1)C(=O)Nc2ccncc2	CID:5711	phase I
BRD-K60476892	OCc1ccc(o1)c2nn(Cc3ccccc3)c4ccccc24	CID:5712	phase I
BRD-A04026261	CCCCCCCCNC(=O)C(Cc1ccc(OCc2ccncc2)cc1)NC(=O)C3CCC(CN)CC3	CID:5713	phase I
BRD-K06208435	COc1ccc(CCN(C)CCc2ccc(OC)c(OC)c2)cc1OC	CID:5714	phase I
BRD-K71289571	COc1cc(ccc1Cc1cn(C)c2ccc(NC(=O)OC3CCCC3)cc12)C(=O)NS(=O)(=O)c1ccccc1C	CID:5717	phase I
BRD-K92657060	CCN(C(C)=O)c1cccc(c1)-c1ccnc2c(cnn12)C#N	CID:5719	phase I
BRD-K37561857	COc1cc(ccc1OC(F)F)-c1ccc(=O)[nH]n1	CID:5723	phase I
BRD-K73789395	CN(C)c1cccc(c1)C(=O)Nc1ccc(C)c(NC(=O)c2ccc(O)cc2)c1	CID:5730	phase I
BRD-K44876623	CN(C)C(=O)Cc1c(nc2ccc(C)cn12)-c1ccc(C)cc1	CID:5732	phase I
BRD-K48300629	NS(=O)(=O)Cc1noc2ccccc12	CID:5734	phase I
BRD-A34309505	CN1CCN(CC1)C(=O)OC2N(C(=O)c3nccnc23)c4ccc(Cl)cn4	CID:5735	phase I
BRD-K38775274	C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:5743	phase I
BRD-K86161929	CC(=O)OCC(=O)[C@@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3C(=O)C[C@]12C	CID:5745	phase I
BRD-A14208071	CC[N+](C)(CC)CCOC(=O)C(O)(C1CCCCC1)c1ccccc1	CID:5749	phase I
BRD-K73589401	C[C@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)CO	CID:5753	phase I
BRD-K93568044	C[C@@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CC[C@]1(O)C(=O)CO	CID:5754	phase I
BRD-K17016787	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@@H]1C[C@@H](O)[C@@H]2O	CID:5756	phase I
BRD-K18910433	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@@H]1CC[C@@H]2O	CID:5757	phase I
BRD-K95921201	CO[C@H]1[C@@H](C[C@@H]2CN3CCc4c([nH]c5cc(OC)ccc45)[C@H]3C[C@@H]2[C@@H]1C(=O)OC)OC(=O)c1cc(OC)c(OC)c(OC)c1	CID:5770	phase I
BRD-K90333595	Cc1ccc(cc1)N(CC1=NCCN1)c1cccc(O)c1	CID:5775	phase I
BRD-K47832606	OC[C@H]1O[C@H](C[C@@H]1O)n2cc(F)c(=O)[nH]c2=O	CID:5790	phase I
BRD-K61236135	OC(=O)Cc1cc(I)c(Oc2ccc(O)c(I)c2)c(I)c1	CID:5803	phase I
BRD-K37264083	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	CID:5808	phase I
BRD-K39981244	NC[C@@H](O)c1ccc(O)c(O)c1	CID:5814	phase I
BRD-K30685142	N[C@@H](Cc1cc(I)c(Oc2cc(I)c(O)c(I)c2)c(I)c1)C(O)=O	CID:5819	phase I
BRD-K96037667	CC(=O)O[C@]1(CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@@H]4[C@H]3CC[C@]12C)C#C	CID:5832	phase I
BRD-K90027355	CC(=O)S[C@@H]1CC2=CC(=O)CC[C@]2(C)[C@H]2CC[C@@]3(C)[C@@H](CC[C@@]33CCC(=O)O3)[C@H]12	CID:5833	phase I
BRD-K44942604	C[N+]1(CCCCC[N+]2(C)CCCC2)CCCC1	CID:5850	phase I
BRD-A22101059	COP(=O)(OC)C(O)C(Cl)(Cl)Cl	CID:5853	phase I
BRD-K81839095	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@@H]1CCC2=O	CID:5870	phase I
BRD-K94070024	C[C@H]1C[C@H]2[C@@H]3CC[C@](O)(C(=O)COC(=O)C)[C@@]3(C)C[C@H](O)[C@@H]2[C@@]4(C)C=CC(=O)C=C14	CID:5877	phase I
BRD-A11132253	NC(=O)c1ccc[n+](c1)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OC[C@H]2O[C@H]([C@H](O)[C@@H]2O)n2cnc3c(N)ncnc23)[C@@H](O)[C@H]1O	CID:5893	phase I
BRD-K63993117	CC(=O)Nc1ccc-2c(Cc3ccccc-23)c1	CID:5897	phase I
BRD-K56745457	OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n2ncc(=O)[nH]c2=O	CID:5901	phase I
BRD-K55191674	CC1(C)S[C@@H]2[C@H](NC(=O)Cc3ccccc3)C(=O)N2[C@H]1C(O)=O	CID:5904	phase I
BRD-K76634210	OC[C@H]1O[C@H](C[C@@H]1O)n1cc(I)c(=O)[nH]c1=O	CID:5905	phase I
BRD-K96253961	C[C@H](N)[C@H](O)c1cccc(O)c1	CID:5906	phase I
BRD-K85090592	CC[C@H]1[C@@H](Cc2cncn2C)COC1=O	CID:5910	phase I
BRD-K15522385	CN(C)CCCSc1ccccc1NC(=O)C=Cc2ccccc2	CID:5913	phase I
BRD-K57718010	C1CCc2nnnn2CC1	CID:5917	phase I
BRD-K89152108	N[C@@H](Cc1cc(I)c(Oc2ccc(O)c(I)c2)c(I)c1)C(O)=O	CID:5920	phase I
BRD-K24610782	CCN(CC)[N+][O-]	CID:5921	phase I
BRD-K24169676	ClC(Cl)(Cl)Cl	CID:5943	phase I
BRD-K80684056	C[C@]12[C@@H]3CC[C@@H](O3)[C@@]1(C)C(=O)OC2=O	CID:5944	phase I
BRD-K08111712	OC[C@@H](NC(=O)C(Cl)Cl)[C@H](O)c1ccc(cc1)[N+]([O-])=O	CID:5959	phase I
BRD-K83896451	N[C@@H](CCC(N)=O)C(O)=O	CID:5961	phase I
BRD-K51471001	CN(CCCCCCCCCCN(C)C(=O)Oc1cccc(c1)[N+](C)(C)C)C(=O)Oc1cccc(c1)[N+](C)(C)C	CID:5966	phase I
BRD-K25650355	CNC(=O)Oc1ccc2N(C)[C@H]3N(C)CC[C@@]3(C)c2c1	CID:5983	phase I
BRD-K48195008	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@@H]1CC[C@@]2(O)C#C	CID:5991	phase I
BRD-K64994968	CC(=O)[C@H]1CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:5994	phase I
BRD-K90553655	CCC(=O)O[C@H]1CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:5995	phase I
BRD-K99621550	COc1cc2CCN(C)[C@H]3Cc4ccc(Oc5c(O)c(OC)cc6CC[N+](C)(C)[C@H](Cc7ccc(O)c(Oc1cc23)c7)c56)cc4	CID:6000	phase I
BRD-K66090100	Cc1c2ccccc2c(C)c3c1ccc4ccccc43	CID:6001	phase I
BRD-K84036904	C[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:6010	phase I
BRD-A47564106	COc1cc2CCN3CC(CC(C)C)C(=O)CC3c2cc1OC	CID:6018	phase I
BRD-K08327065	NC[C@H]1O[C@H](O[C@@H]2[C@@H](N)C[C@@H](N)[C@H](O[C@H]3O[C@H](CO)[C@@H](O)[C@H](N)[C@H]3O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1O	CID:6032	phase I
BRD-K18673820	Nc1nc(=O)c2nc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(O)=O)C(O)=O)cnc2[nH]1	CID:6037	phase I
BRD-K34730807	N[C@@H](Cc1ccc(O)c(O)c1)C(O)=O	CID:6047	phase I
BRD-K37814297	CN(C)CCCN1c2ccccc2Sc2ccc(cc12)C(C)=O	CID:6077	phase I
BRD-A39189014	COc1ccc(OC)c(c1)C(O)C(C)N	CID:6082	phase I
BRD-K85767870	Nc1ncnc2n(cnc12)[C@@H]3O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]3O	CID:6083	phase I
BRD-K53123955	[O-][N+](=O)c1cnc(s1)N1CCNC1=O	CID:6093	phase I
BRD-K66353228	Nc1nc2cc(Cl)ccc2o1	CID:6103	phase I
BRD-K91960538	CN(C)[N+][O-]	CID:6124	phase I
BRD-K93441486	C[N+]1(C)CCC(CC1)=C(c1ccccc1)c1ccccc1	CID:6127	phase I
BRD-K32610195	C[C@@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CCC1=O	CID:6128	phase I
BRD-K54208592	CNC(=O)Oc1cccc2ccccc12	CID:6129	phase I
BRD-K98521173	C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)CO	CID:6166	phase I
BRD-K00259736	COc1cc2CC[C@H](NC(C)=O)c3cc(=O)c(OC)ccc3-c2c(OC)c1OC	CID:6167	phase I
BRD-K84595254	C[C@@]12CC[C@H]3[C@@H](CC[C@]4(O)C[C@@H](O)CC[C@]34C=O)[C@@]2(O)CC[C@@H]1C5=CC(=O)OC5	CID:6185	phase I
BRD-K96786677	Cc1onc(c1C(=O)N[C@H]1[C@H]2SC(C)(C)[C@@H](N2C1=O)C(O)=O)-c1ccccc1	CID:6196	phase I
BRD-K36055864	C[C@H]1C[C@H](C)C(=O)[C@@H](C1)[C@H](O)CC1CC(=O)NC(=O)C1	CID:6197	phase I
BRD-K88785477	ClC(Cl)Cl	CID:6212	phase I
BRD-K94353609	CC1(C)O[C@@H]2C[C@H]3[C@@H]4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:6215	phase I
BRD-K92073408	C[C@@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@H]34)[C@@H]2CC[C@@]1(O)C#C	CID:6230	phase I
BRD-K80334323	C[C@@]12CC[C@H]3[C@@H](CCC4=C3CCC(=O)C4)[C@@H]2CC[C@@]1(O)C#C	CID:6231	phase I
BRD-K87226815	N[C@@H]1CONC1=O	CID:6234	phase I
BRD-K68432770	CC1(C)S[C@@H]2[C@H](NC(=O)[C@H](N)c3ccccc3)C(=O)N2[C@H]1C(O)=O	CID:6249	phase I
BRD-K33106058	Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)n1	CID:6253	phase I
BRD-K03243820	OC[C@H]1O[C@H](C[C@@H]1O)n1cc(c(=O)[nH]c1=O)C(F)(F)F	CID:6256	phase I
BRD-K82216340	C[C@H]1C[C@H]2[C@@H]3CC[C@](OC(=O)C)(C(=O)C)[C@@]3(C)CC[C@@H]2[C@@]4(C)CCC(=O)C=C14	CID:6279	phase I
BRD-K60923938	COc1ccc(cc1OC)C(=O)O[C@H]2CC[C@@]3(C)[C@@H]4CC[C@@H]5[C@@]3(C[C@@]6(O)[C@@H]7CN8C[C@@H](C)CC[C@H]8[C@@](C)(O)[C@@]7(O)[C@@H](O)C[C@@]56O)O[C@@]42O	CID:6280	phase I
BRD-K31920458	COc1ccc2[C@H]3CC[C@@]4(C)[C@@H](CC[C@@]4(O)C#C)[C@@H]3CCc2c1	CID:6291	phase I
BRD-A59303141	CCC1NC(=O)c2cc(c(Cl)cc2N1)S(N)(=O)=O	CID:6307	phase I
BRD-K53790871	CC1(C)O[C@@H]2C[C@H]3[C@@H]4CCC5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:6436	phase I
BRD-K92758126	C[C@@]12[C@H]3[C@H](C(O)=O)[C@@]45CC(=C)[C@@](O)(C4)CC[C@H]5[C@]3(OC1=O)C=C[C@@H]2O	CID:6466	phase I
BRD-K46435528	ClC=C(Cl)Cl	CID:6575	phase I
BRD-K13664374	OC(=O)C(Cl)Cl	CID:6597	phase I
BRD-K71075093	CN1C(C)(C)CCCC1(C)C	CID:6603	phase I
BRD-K41494493	CC(C)(c1ccc(O)cc1)c2ccc(O)cc2	CID:6623	phase I
BRD-K32021043	Nc1ccc(cc1)S(=O)(=O)Nc1ccc(Cl)nn1	CID:6634	phase I
BRD-K90976994	C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@H]3[C@H](CC(=O)[C@]12C)[C@@]4(C)CCC(=O)C[C@H]4CC3=O	CID:6674	phase I
BRD-K81062487	C[C@H](CCC(=O)NCCS(=O)(=O)O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:6675	phase I
BRD-K76872913	O=C1c2ccccc2-c3cccc4cccc1c34	CID:6697	phase I
BRD-K79501723	CN1CCN(CC1)C(c1ccccc1)c1ccccc1	CID:6726	phase I
BRD-K73824630	Cc1c[nH]c2ccccc12	CID:6736	phase I
BRD-K35240538	C[C@H]1C[C@H]2[C@@H]3CC[C@](O)(C(=O)CO)[C@@]3(C)C[C@H](O)[C@@H]2[C@@]4(C)C=CC(=O)C=C14	CID:6741	phase I
BRD-A08027849	CC(CCC(O)=O)[C@H]1CC[C@H]2[C@@H]3CC[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:6742	phase I
BRD-K08316444	COc1cc2OC[C@H]3Oc4c5C[C@@H](Oc5ccc4C(=O)[C@H]3c2cc1OC)C(=C)C	CID:6758	phase I
BRD-K25741894	COc1ccc2c(OC)c3ccoc3nc2c1OC	CID:6760	phase I
BRD-K14200658	CCOC(=O)Oc1c(OC)cc(cc1OC)C(=O)O[C@@H]2C[C@@H]3CN4CCc5c([nH]c6cc(OC)ccc56)[C@H]4C[C@@H]3[C@@H]([C@H]2OC)C(=O)OC	CID:6769	phase I
BRD-A68723818	CN(C)CCC(c1ccc(Br)cc1)c1ccccn1	CID:6834	phase I
BRD-A18043272	CN1C(=O)CC(C1=O)c1ccccc1	CID:6839	phase I
BRD-K18250272	CCCOc1cc(N)ccc1C(=O)OCCN(CC)CC	CID:6843	phase I
BRD-K70327191	O=C(Oc1cccc2cccnc12)c1ccccc1	CID:6855	phase I
BRD-K73391359	CCCCc1cc2ccccc2c(OCCN(C)C)n1	CID:6857	phase I
BRD-K84175871	CN[C@@H](C)[C@@H](O)c1ccccc1	CID:7028	phase I
BRD-A37288617	CCN(CC)C(C)C(=O)c1ccccc1	CID:7029	phase I
BRD-K18436203	C1Cc2ccccc2CN1	CID:7046	phase I
BRD-K53032901	FC(F)(F)c1ccc2Sc3ccccc3Nc2c1	CID:7082	phase I
BRD-K59597909	N1c2ccccc2Sc2ccccc12	CID:7108	phase I
BRD-A04327189	CNCC(O)c1ccc(O)cc1	CID:7172	phase I
BRD-K08287586	CCCCOC(=O)c1ccc(O)cc1	CID:7184	phase I
BRD-K33459542	Cc1ccccc1NC(=N)Nc1ccccc1C	CID:7333	phase I
BRD-K54028654	OC[C@H]1O[C@H](O[C@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1O	CID:7427	phase I
BRD-K76133116	NCc1ccccc1	CID:7504	phase I
BRD-K76600340	OCc1cccnc1	CID:7510	phase I
BRD-A37942872	CC1CC(CC(C)(C)N1C)OC(=O)C(O)c1ccccc1	CID:7534	phase I
BRD-K54262262	Oc1ccc(OCc2ccccc2)cc1	CID:7638	phase I
BRD-K91699951	CCCCNc1ccc(cc1)C(=O)OCCOCCOCCOCCOCCOCCOCCOCCOCCOC	CID:7699	phase I
BRD-K20075662	NCCc1cc[nH]n1	CID:7741	phase I
BRD-K65278478	c1ccoc1	CID:8029	phase I
BRD-K33235400	C=CCCCCCCCCC=O	CID:8187	phase I
BRD-K41298358	NCCNCCNCCNCCN	CID:8197	phase I
BRD-K34685430	CC[C@@H](CO)NC(=O)[C@H]1CN(C)[C@@H]2Cc3c[nH]c4cccc(C2=C1)c34	CID:8226	phase I
BRD-K11399644	NC(=N)NC(=N)NCCc1ccccc1	CID:8249	phase I
BRD-K15842202	COc1cc(cc(OC)c1OC)C(=O)O	CID:8357	phase I
BRD-A34751532	CC1CC(CC(C)(C)C1)OC(=O)c1ccccc1O	CID:8362	phase I
BRD-K40619305	Cc1occc(=O)c1O	CID:8369	phase I
BRD-K71013094	NC[C@@H]1O[C@H](O[C@H]2[C@@H](O)[C@H](O[C@@H]3[C@@H](O)[C@H](N)C[C@H](N)[C@H]3O[C@H]4O[C@H](CN)[C@@H](O)[C@H](O)[C@H]4N)O[C@@H]2CO)[C@H](N)[C@@H](O)[C@@H]1O	CID:8378	phase I
BRD-K59570838	COc1ccc(CCN)cc1OC	CID:8421	phase I
BRD-K01555864	O=C(CC(=O)c1ccccc1)c2ccccc2	CID:8433	phase I
BRD-K94848716	NC(=O)Nc1ccc(cc1)[As](O)(O)=O	CID:8480	phase I
BRD-K01567962	O=C1c2ccccc2-c2n[nH]c3cccc1c23	CID:8515	phase I
BRD-K28595280	CNC[C@H](O)[C@@H](O)[C@H](O)[C@H](O)CO	CID:8567	phase I
BRD-K22193694	COc1ccc(C(=O)c2ccccc2O)c(O)c1	CID:8569	phase I
BRD-K72034655	COc1c(oc2cc3oc(=O)ccc3cc12)C(C)C	CID:8616	phase I
BRD-K43880410	CC(=O)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:8955	phase I
BRD-K35586044	COC(=O)[C@H]1[C@@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12	CID:8969	phase I
BRD-K79511609	Nc1nc(Cl)nc2n(cnc12)[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O	CID:8974	phase I
BRD-K72238567	Nc1nc(F)nc2n(cnc12)[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O	CID:8975	phase I
BRD-K18574842	CCOc1ccc2ccccc2c1C(=O)N[C@H]1[C@H]2SC(C)(C)[C@@H](N2C1=O)C(O)=O	CID:8982	phase I
BRD-K68620903	CC(=O)[C@H]1CC[C@H]2[C@@H]3C=CC4=CC(=O)CC[C@@]4(C)[C@@H]3CC[C@]12C	CID:9051	phase I
BRD-K97808269	OC[C@H]1O[C@H](O)C[C@@H](O)[C@@H]1O	CID:9062	phase I
BRD-K09784055	c1ccc2c(c1)c3cccc4ccc5cccc2c5c43	CID:9128	phase I
BRD-K04368295	c1cc2ccccc2o1	CID:9223	phase I
BRD-K59946561	N[C@@H](Cc1cc(I)c(O)c(I)c1)C(=O)O	CID:9305	phase I
BRD-K85030058	CCN(CC)CCOC(=O)C(O)(c1ccccc1)c2ccccc2	CID:9330	phase I
BRD-K38055836	CCN(CC)C(=O)c1ccc(O)c(OC)c1	CID:9363	phase I
BRD-K43786866	OCCN1CCN(CCCN2c3ccccc3C=Cc3ccccc23)CC1	CID:9417	phase I
BRD-K79145749	CN(C)CCN1C(=O)c2ccccc2N(C)c3ccccc13	CID:9419	phase I
BRD-K08619574	CN(C)S(=O)(=O)c1ccc2Sc3ccccc3N(CCCN3CCN(C)CC3)c2c1	CID:9429	phase I
BRD-K03406345	Nc1ncn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1	CID:9444	phase I
BRD-K71696703	CC(=O)Oc1cc(ccc1C(O)=O)C(F)(F)F	CID:9458	phase I
BRD-K57886322	CC(=O)OCC(=O)[C@]12OC(C)(C)O[C@@H]2C[C@H]3[C@@H]4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@@]31C	CID:9642	phase I
BRD-A41995253	COc1cc2N3C4[C@@H]5C(CC3=O)OCC=C3CN6CC[C@]4([C@@H]6C[C@H]53)c2cc1OC	CID:9649	phase I
BRD-K49481516	COc1ccc2CN(C)CC[C@@]34C=C[C@H](O)C[C@@H]3Oc1c24	CID:9651	phase I
BRD-K35941380	CC[C@@H](CO)NC(=O)[C@H]1CN(C)[C@@H]2Cc3cn(C)c4cccc(C2=C1)c34	CID:9681	phase I
BRD-A94624445	CCCC(=O)Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP(O)(=O)O[C@H]2[C@H]1OC(=O)CCC	CID:9687	phase I
BRD-K03642198	Clc1ccccc1CNCC2CCC(CNCc3ccccc3Cl)CC2	CID:9705	phase I
BRD-K79134921	CNCCc1ccc(O)cc1	CID:9727	phase I
BRD-K39188321	C[C@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:9782	phase I
BRD-A10662413	CC(Cc1ccccc1)NCCC(c1ccccc1)c1ccccc1	CID:9801	phase I
BRD-K20986251	C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@@H]3CC[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:9903	phase I
BRD-K52080565	C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@H]34)[C@@H]1CC[C@@H]2O	CID:9904	phase I
BRD-A01826957	CN(CCO)CC(O)Cn1cnc2n(C)c(=O)n(C)c(=O)c12	CID:9913	phase I
BRD-K63165456	CNCCC=C1c2ccccc2C=Cc2ccccc12	CID:9918	phase I
BRD-K35128472	Nc1ncc2nc[nH]c2n1	CID:9955	phase I
BRD-K18135438	C[C@H](CCC(O)=O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:10133	phase I
BRD-K54771420	C[C@H](CCC(=O)NCC(=O)O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:10140	phase I
BRD-K03440695	COc1cc-2c(C[C@@H]3N(C)CCc4cc(O)c(OC)c2c34)cc1O	CID:10154	phase I
BRD-K25836724	C[C@@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CC[C@H]1O	CID:10204	phase I
BRD-K36137799	CC1=CC(=O)c2c(O)cccc2C1=O	CID:10205	phase I
BRD-K07117950	CC(=CCOc1c2occc2cc3ccc(=O)oc13)C	CID:10212	phase I
BRD-K03067624	CC[C@H]1CN2CCc3cc(OC)c(OC)cc3[C@@H]2C[C@@H]1C[C@H]1NCCc2cc(OC)c(OC)cc12	CID:10219	phase I
BRD-K78294846	COc1ccc2ccc(=O)oc2c1CC=C(C)C	CID:10228	phase I
BRD-A07824748	O=C1CC(Oc2ccccc12)c3ccccc3	CID:10251	phase I
BRD-A75140635	COc1cc2CCNC(C)c2cc1OC	CID:10302	phase I
BRD-K59773493	ONC(=O)c1ccccc1	CID:10313	phase I
BRD-K36162096	OC(=O)c1ccnc(c1)C(=O)O	CID:10365	phase I
BRD-K72166146	CN1C[C@@H](C[C@H]2[C@H]1Cc1c[nH]c3cccc2c13)C(=O)N[C@]1(C)O[C@@]2(O)[C@@H]3CCCN3C(=O)[C@H](Cc3ccccc3)N2C1=O	CID:10531	phase I
BRD-K47869605	COc1cc(cc(OC)c1OC)[C@H]1[C@@H]2[C@H](COC2=O)[C@@H](O)c2cc3OCOc3cc12	CID:10607	phase I
BRD-K38903228	COc1ccc(cc1O)[C@@H]2CC(=O)c3c(O)cc(O[C@@H]4O[C@H](CO[C@@H]5O[C@@H](C)[C@H](O)[C@@H](O)[C@H]5O)[C@@H](O)[C@H](O)[C@H]4O)cc3O2	CID:10621	phase I
BRD-K99615199	C[C@H]1C[C@H]2[C@@H]3CC[C@](O)(C(C)=O)[C@@]3(C)CC[C@@H]2[C@@]2(C)CCC(=O)C=C12	CID:10631	phase I
BRD-K18523449	C[C@]1(O)CC[C@H]2[C@@H]3CC[C@H]4CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:10633	phase I
BRD-K82561139	COc1ccn(C)c(=O)c1C#N	CID:10666	phase I
BRD-K51980294	COc1cc(cc(OC)c1O)C(=O)O	CID:10742	phase I
BRD-K46585355	CC(=O)Oc1ccccc1C(=O)Oc1ccccc1C(O)=O	CID:10745	phase I
BRD-K81209159	COc1ccc2ccc(=O)oc2c1	CID:10748	phase I
BRD-A09062839	CCC(C)(CN(C)C)OC(=O)c1ccccc1	CID:10767	phase I
BRD-A97730597	CC(CNC1CCCCC1)OC(=O)c1ccccc1	CID:10770	phase I
BRD-K50422030	Cc1ncsc1CCCl	CID:10783	phase I
BRD-A30693873	O=C(Nc1ccccc1)OCC(CN1CCCCC1)OC(=O)Nc1ccccc1	CID:10831	phase I
BRD-A29082194	C[C@@]12CCC3C(CC[C@@H]4C[C@@H](O)CC[C@@]43C)[C@@]2(O)C[C@H](O)[C@@H]1C5=CC(=O)OC5	CID:11012	phase I
BRD-K95788524	CC(C)c1ccc(C)c(C(=O)O)c1O	CID:11052	phase I
BRD-A35033682	Oc1cc(O)c2C(=O)CC(Oc2c1)c3ccc(O)c(O)c3	CID:11095	phase I
BRD-A19053259	CN1C2CCCC1CC(=O)C2	CID:11096	phase I
BRD-K27062708	COc1ccc(cc1)C(Cl)=C(c1ccc(OC)cc1)c1ccc(OC)cc1	CID:11289	phase I
BRD-K19507340	CC(=O)O[C@@]1(CC[C@H]2[C@@H]3C=C(C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C)C(C)=O	CID:11683	phase I
BRD-K88965984	[O-][N+](=O)c1ccc-2c(Cc3ccccc-23)c1	CID:11831	phase I
BRD-K59058747	CC(=O)N[C@@H](CS)C(O)=O	CID:12035	phase I
BRD-A68930007	C[C@@H]1O[C@@H](O[C@H]2C[C@@H](O)[C@]3(CO)C4[C@H](O)C[C@]5(C)[C@H](CC[C@]5(O)C4CC[C@]3(O)C2)C2=CC(=O)OC2)[C@H](O)[C@H](O)[C@H]1O	CID:12420	phase I
BRD-K00198051	OCCN1CCN(CCC=C2c3ccccc3Sc3ccc(Cl)cc23)CC1	CID:12454	phase I
BRD-K53220666	COc1cc(cc(OC)c1OC)C(=O)N1CCOCC1	CID:12478	phase I
BRD-K15567837	C[C@H]1CCC[C@@H](C)N1NC(=O)c2ccc(Cl)c(c2)S(=O)(=O)N	CID:12492	phase I
BRD-K78683072	Cl[Sn](c1ccccc1)(c1ccccc1)c1ccccc1	CID:12540	phase I
BRD-K28542495	CN(C)CCCOc1nn(Cc2ccccc2)c2ccccc12	CID:12555	phase I
BRD-K63550407	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O	CID:12560	phase I
BRD-K35189033	CC[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@H]34)[C@@H]1CC[C@@]2(O)C#C	CID:13109	phase I
BRD-K01188359	CC[C@]1(O)C[C@@H]2CN(C1)CCc3c([nH]c4ccccc34)[C@@](C2)(C(=O)OC)c5cc6c(cc5OC)N(C)[C@@H]7[C@@]86CCN9CC=C[C@](CC)([C@H]98)[C@@H](OC(=O)C)[C@]7(O)C(=O)OC	CID:13342	phase I
BRD-K41903098	CCOC(=O)C1(CCN(CCC(C#N)(c2ccccc2)c3ccccc3)CC1)c4ccccc4	CID:13505	phase I
BRD-K42596464	CCN(CC)CCc1nc(no1)-c1ccccc1	CID:13738	phase I
BRD-K26104851	Oc1ccc(cc1)C(=O)NN=Cc2ccc(o2)[N+](=O)[O-]	CID:13764	phase I
BRD-K39391626	CC[C@]1(O)CC[C@H]2[C@@H]3CCC4=CCCC[C@@H]4[C@H]3CC[C@]12C	CID:13765	phase I
BRD-K66766661	CCCCC(=O)O[C@H]1CC[C@H]2[C@@H]3CCc4cc(O)ccc4[C@H]3CC[C@]12C	CID:13791	phase I
BRD-K14221570	Cc1cc(ccc1N=Nc2cc(c3ccccc3c2N)S(=O)(=O)O)c4ccc(N=Nc5cc(c6ccccc6c5N)S(=O)(=O)O)c(C)c4	CID:13817	phase I
BRD-K37984227	[O-][N+](=O)c1ccc(C=NNC(=O)CN2CCOCC2)o1	CID:14165	phase I
BRD-A61273891	COc1cc2OC3OC=CC3c2c2oc(=O)c3C(=O)CCc3c12	CID:14403	phase I
BRD-A57957888	CC(=O)NC1CCSC1=O	CID:14520	phase I
BRD-K96527333	CC(=O)O[C@H]1CC[C@]2(C)[C@H]3CC[C@@]4(C)[C@@H](CCC4=O)[C@@H]3CC=C2C1	CID:14709	phase I
BRD-A80928489	CCCCCCCCCCCCCCCC(=O)OCC(O)CO	CID:14900	phase I
BRD-K22081896	OC(=O)CC(CC(O)=O)C(O)=O	CID:14925	phase I
BRD-K27871032	CN1C[C@H](CO)C=C2[C@H]1Cc3c[nH]c4cccc2c34	CID:14987	phase I
BRD-K39356024	CC(=O)[C@H]1[C@@H](C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C)C#N	CID:15032	phase I
BRD-K37606513	NC(=O)c1ccncc1	CID:15074	phase I
BRD-K88145757	CCCC[Sn](Cl)(CCCC)CCCC	CID:15096	phase I
BRD-K00824317	CC1(C)O[C@@H]2C[C@H]3[C@@H]4C[C@H](F)C5=CC(=O)CC[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:15209	phase I
BRD-A54635441	CCC(=O)OC(Cc1ccccc1)(C(C)CN(C)C)c1ccccc1	CID:15330	phase I
BRD-K40902647	CC[C@]1(CCCN2CCc3c4[C@@H]21)C[C@](O)(C(=O)OC)n4c5ccccc35	CID:15376	phase I
BRD-K92984783	CC1CCN(CCCC(=O)c2ccc(F)cc2)CC1	CID:15387	phase I
BRD-K45861246	Fc1ccc(cc1)C(=O)CCCN1CCN(CC1)c1ccccn1	CID:15443	phase I
BRD-A94709349	Cc1cc(C)cc(OCC2CNC(=O)O2)c1	CID:15459	phase I
BRD-K18619710	C[C@@]12[C@H](CC[C@]1(O)[C@@H]1CC[C@@H]3C[C@@H](O)CC[C@]3(C)[C@H]1C[C@H]2O)C1=CC(=O)OC1	CID:15478	phase I
BRD-K11905747	CN[C@@H]1[C@H](O)[C@H](NC)[C@H]2O[C@]3(O)[C@@H](O[C@H](C)CC3=O)O[C@@H]2[C@H]1O	CID:15541	phase I
BRD-A24817035	COc1ccc(CC2N(C)CCc3cc(OC)c(OC)cc23)cc1OC	CID:15548	phase I
BRD-K02603382	Cc1nccc2ccccc12	CID:15592	phase I
BRD-K90697689	Clc1cc2Oc3cc(Cl)c(Cl)cc3Oc2cc1Cl	CID:15625	phase I
BRD-K97061094	OC(C1CCNCC1)(c1ccccc1)c1ccccc1	CID:15723	phase I
BRD-K93859331	Cc1ccc2[nH]cc(CCN)c2c1	CID:15760	phase I
BRD-A51916548	CC(N)Cc1cccc(c1)C(F)(F)F	CID:15897	phase I
BRD-K36452089	CC(C)(C)c1cc(O)ccc1O	CID:16043	phase I
BRD-K97181089	NC(=N)NC(=O)c1nc(Cl)c(N)nc1N	CID:16231	phase I
BRD-K01292756	Fc1ccc(cc1)C(CCCN1CCC(CC1)n1c2ccccc2[nH]c1=O)c1ccc(F)cc1	CID:16362	phase I
BRD-K79425933	Fc1ccc(cc1)C(=O)CCCN1CCC(CC1)n1c2ccccc2[nH]c1=O	CID:16363	phase I
BRD-K07223205	CN(C)CCCN1c2ccc(O)cc2Sc2ccc(Cl)cc12	CID:16414	phase I
BRD-K61496577	C[C@@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:16490	phase I
BRD-K73978287	C[C@@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CC[C@]1(O)C(=O)COC(=O)CCC(=O)O	CID:16623	phase I
BRD-K56700933	S=C=NCCc1ccccc1	CID:16741	phase I
BRD-K43807558	COc1cc(CCCO)ccc1O	CID:16822	phase I
BRD-K22947005	CN(C)CC[C@@H](c1ccc(Br)cc1)c2ccccn2	CID:16960	phase I
BRD-K74534237	CC(C)c1cc(c(C)cc1OC(=O)N1CCCCC1)[N+](C)(C)C	CID:17104	phase I
BRD-K55250441	COc1ncnc(NS(=O)(=O)c2ccc(N)cc2)c1OC	CID:17134	phase I
BRD-K82259334	CCOC(=O)[C@@](C)(N)Cc1ccc(O)c(O)c1	CID:17277	phase I
BRD-K56483981	COc1cc(ccc1\N=N\c1ccc2c(cc(c(N)c2c1O)S(O)(=O)=O)S(O)(=O)=O)-c1ccc(\N=N\c2ccc3c(cc(c(N)c3c2O)S(O)(=O)=O)S(O)(=O)=O)c(OC)c1	CID:17461	phase I
BRD-K71055333	Oc1ccc(O)c(c1)S(O)(=O)=O	CID:17507	phase I
BRD-K00656370	Nc1cc2c3ccccc3ccc2c4ccccc14	CID:17534	phase I
BRD-K66792149	NC1=C(Cl)C(=O)c2ccccc2C1=O	CID:17748	phase I
BRD-K93880783	Cc1cn([C@@H]2O[C@H](CO)C=C2)c(=O)[nH]c1=O	CID:18283	phase I
BRD-K05673000	Cc1onc(c1C(=O)N[C@H]1[C@H]2SC(C)(C)[C@@H](N2C1=O)C(O)=O)-c1c(Cl)cccc1Cl	CID:18381	phase I
BRD-K12057390	CC(=O)Oc1ccc(cc1)c2cc(=O)c3c(OC(=O)C)cc(OC(=O)C)cc3o2	CID:18721	phase I
BRD-A30142024	OC(CS)C(O)CS	CID:19001	phase I
BRD-K89046952	CC1(C)S[C@@H]2[C@H](NC(=O)C3(N)CCCCC3)C(=O)N2[C@H]1C(=O)O	CID:19003	phase I
BRD-K13169950	Oc1ccc([N+][O-])c2cccnc12	CID:19103	phase I
BRD-K47029922	N[C@@H]1C[C@H]1c1ccccc1	CID:19493	phase I
BRD-K10974103	CN(C(=O)C(Cl)Cl)c1ccc(OC(=O)c2ccco2)cc1	CID:19529	phase I
BRD-K47878171	C[N+](C)(CCOc1ccccc1)Cc1ccccc1	CID:19667	phase I
BRD-K16277217	CC(=O)c1ccc2Sc3ccccc3N(CCCN3CCC(CCO)CC3)c2c1	CID:19675	phase I
BRD-K93034159	Nc1nc(Cl)nc2n(cnc12)[C@H]1C[C@H](O)[C@@H](CO)O1	CID:20279	phase I
BRD-A22152765	CC[N+](CC)(CC)CCC(O)(C1CCCCC1)c1ccccc1	CID:20299	phase I
BRD-K94325918	OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n2cnc3c(NCc4ccco4)ncnc23	CID:20345	phase I
BRD-A18246003	CCCCC(CC)COC(=O)c1ccccc1C(O)=O	CID:20393	phase I
BRD-K18905250	CCc1cccc(CC)c1N=C1NCCN1	CID:20864	phase I
BRD-A42346008	CNCC(O)c1ccc(O)c(OC)c1	CID:21100	phase I
BRD-K88366685	COc1ccc(CN2CCNCC2)c(OC)c1OC	CID:21109	phase I
BRD-K92830582	CC(C)NC[C@@H](O)COc1cccc2ccccc12	CID:21138	phase I
BRD-A04020513	CCCCS(=N)(=O)CCC(N)C(=O)O	CID:21157	phase I
BRD-K97810537	CCC(=O)OCC(=O)[C@@]1(OC(=O)CC)[C@@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]12C	CID:21700	phase I
BRD-K72093121	Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O	CID:21704	phase I
BRD-A69917777	CC(CC(C(N)=O)(c1ccccc1)c1ccccc1)N(C)C	CID:22565	phase I
BRD-K15834839	CCOC(=O)Nc1nc2ccccc2[nH]1	CID:22752	phase I
BRD-A04308630	COC(=O)C1=COC(O)C2C1CC=C2CO	CID:23340	phase I
BRD-K25310650	COc1cc(C)c(Cc2cnc(N)nc2N)cc1OC	CID:23418	phase I
BRD-K74773935	Cn1cc(CCN)c2ccccc12	CID:23492	phase I
BRD-K04170657	COc1cc(C(=O)O)c2Oc3c(C=O)c(O)cc(C)c3C(=O)Oc2c1C	CID:23725	phase I
BRD-A65280694	CCc1c(C)[nH]c2CCC(CN3CCOCC3)C(=O)c12	CID:23897	phase I
BRD-K85925969	Nc1ccn([C@H]2CC[C@@H](CO)O2)c(=O)n1	CID:24066	phase I
BRD-K90864987	Cl[Co]Cl	CID:24288	phase I
BRD-K37890730	CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccccc4cc3Cn1c2=O	CID:24360	phase I
BRD-K26756156	Cl[Cd]Cl	CID:24633	phase I
BRD-A02367930	C[C@]12CCC3C(CCc4cc(O)ccc34)C1CC[C@@]2(O)C#C	CID:24707	phase I
BRD-K51751936	CC(=O)OCC(=O)[C@H]1CC[C@H]2[C@@H]3CC[C@H]4C[C@H](O)CC[C@]4(C)[C@H]3C(=O)C[C@]12C	CID:24733	phase I
BRD-K04156788	Brc1ccccc1C(=O)Nc2ccccc2	CID:25126	phase I
BRD-K83257731	CN(C)CCN(Cc1ccc(Cl)cc1)c1ccccn1	CID:25295	phase I
BRD-K72542090	OP(O)(=O)C(Cl)(Cl)P(O)(O)=O	CID:25419	phase I
BRD-K88575585	NCCc1csc2ccc(O)cc12	CID:25600	phase I
BRD-K88809146	N[C@H]1C[C@@H]1c1ccccc1	CID:26070	phase I
BRD-A70182876	CCCC1C(=O)N2N(C1=O)c1cc(C)ccc1N=C2N(C)C	CID:26098	phase I
BRD-K69122748	CC(=O)Oc1cccc2C(=O)c3cc(cc(OC(C)=O)c3C(=O)c12)C(O)=O	CID:26248	phase I
BRD-A30582499	CCNC1(CCCCC1=O)c1cccs1	CID:26533	phase I
BRD-K02407574	CCCCc1ccc2[nH]c(NC(=O)OC)nc2c1	CID:26596	phase I
BRD-K86434416	C[C@H](Cc1ccccc1)N(C)CC#C	CID:26757	phase I
BRD-K27853494	C[C@@H](N)[C@@H](O)c1ccccc1	CID:26934	phase I
BRD-A43809092	CC(CN(C)C)C(C)(O)Cc1ccc(Cl)cc1	CID:26937	phase I
BRD-K30240666	CN1CCC[C@@H]1CCO[C@](C)(c1ccccc1)c1ccc(Cl)cc1	CID:26987	phase I
BRD-K79711234	CS(=O)(=O)c1ccc(cc1)[C@@H](O)[C@@H](CO)NC(=O)C(Cl)Cl	CID:27200	phase I
BRD-K75958195	CN1CCC(CC1)=C1c2ccsc2CCc2ccccc12	CID:27400	phase I
BRD-K90733503	CC1=C(N2[C@H](SC1)[C@H](NC(=O)[C@H](N)c1ccccc1)C2=O)C(O)=O	CID:27447	phase I
BRD-K16551401	Cn1c2CCNCCc2c2ccccc12	CID:27559	phase I
BRD-A37492983	CC(CN(C(C)=O)c1c(I)cc(I)c(N)c1I)C(O)=O	CID:27648	phase I
BRD-K82225283	O[C@H]1CO[C@@H]2[C@@H](CO[C@H]12)O[N+]([O-])=O	CID:27661	phase I
BRD-K14920963	OC(=O)c1ccccc1-c1c2cc(I)c(O)c(I)c2oc2c(I)c(=O)c(I)cc12	CID:27873	phase I
BRD-K68552125	CCCCCCCCCCCCCC(=O)O[C@@H]1[C@@H](C)[C@]2(O)[C@@H]3C=C(C)C(=O)[C@@]3(O)CC(CO)=C[C@H]2[C@@H]2C(C)(C)[C@]12OC(C)=O	CID:27924	phase I
BRD-A42759514	Cc1ncc(n1CC(O)CCl)[N+]([O-])=O	CID:28061	phase I
BRD-K48970916	C[C@@]12CC[C@H]3[C@@H](CCC4=Cc5oncc5C[C@]34C)[C@@H]2CC[C@@]1(O)C#C	CID:28417	phase I
BRD-K56699285	CN1C[C@H](CNC(=O)OCc2ccccc2)C[C@H]2[C@H]1Cc1cn(C)c3cccc2c13	CID:28693	phase I
BRD-K84102257	COc1cc(cc(OC)c1OC)C(=O)N2CCN(CC2)c3ccccn3	CID:28761	phase I
BRD-K16077845	OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)-c1ccccc1	CID:28871	phase I
BRD-A06779035	COc1cc(cc(OC)c1OC)C(O)CN	CID:28894	phase I
BRD-K34411947	CN([N+][O-])C(=O)N[C@H]1[C@@H](O)O[C@H](CO)[C@@H](O)[C@@H]1O	CID:29327	phase I
BRD-A75144621	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)O[C@H]1[C@@H](O)C[C@H](O[C@H]2[C@@H](O)C[C@H](O[C@H]3CC[C@@]4(C)[C@H](CC[C@@H]5[C@@H]4C[C@@H](O)[C@]4(C)C(CC[C@]54O)C4=CC(=O)OC4)C3)O[C@@H]2C)O[C@@H]1C	CID:30322	phase I
BRD-K43389675	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O	CID:30323	phase I
BRD-A02990301	CC(Oc1c(Cl)cccc1Cl)C1=NCCN1	CID:30668	phase I
BRD-K87156652	CCOC(=O)n1ccn(C)c1=S	CID:31072	phase I
BRD-K42978307	C1COCCO1	CID:31275	phase I
BRD-K77554836	C[C@]12C[C@H](O)[C@@]3(F)[C@@H](CCC4=CC(=O)C=C[C@]34C)[C@@H]1C[C@@H](O)[C@]2(O)C(=O)CO	CID:31307	phase I
BRD-K68386748	ClC(Cl)=C(Cl)Cl	CID:31373	phase I
BRD-K91301684	COc1ccc2[C@@H](OC(=O)c2c1OC)[C@@H]1N(C)CCc2cc3OCOc3c(OC)c12	CID:31411	phase I
BRD-K82261406	COc1ccc(C[C@@H]2NC[C@@H](O)[C@@H]2OC(=O)C)cc1	CID:31549	phase I
BRD-K92093830	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(=O)CO	CID:31703	phase I
BRD-A59174698	CC(NCCc1ccc(O)cc1)C(O)c1ccc(O)cc1	CID:31729	phase I
BRD-A00100033	CC1CS(=O)(=O)CCN1N=Cc1ccc(o1)[N+]([O-])=O	CID:31772	phase I
BRD-A70514680	CCCNC(C)C(=O)Nc1c(C)csc1C(=O)OC	CID:32170	phase I
BRD-A17555397	NC(Cc1csc2ccc(O)cc12)C(O)=O	CID:32334	phase I
BRD-K10799896	CCC(=O)O[C@@]1([C@@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C)C(=O)CCl	CID:32798	phase I
BRD-A56518012	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(=O)CO	CID:32875	phase I
BRD-K39462424	CN(C)CC[C@@H](c1ccc(Cl)cc1)c1ccccn1	CID:33036	phase I
BRD-K51465424	C[C@H](NCCc1ccc(O)cc1)[C@H](O)c2ccc(O)cc2	CID:33572	phase I
BRD-K55044200	CC1(C)S[C@@H]2[C@H](NC(=O)[C@H](N)c3ccc(O)cc3)C(=O)N2[C@H]1C(O)=O	CID:33613	phase I
BRD-K08806317	CC(C)(C)NC[C@H](O)COc1nsnc1N1CCOCC1	CID:33624	phase I
BRD-K15409150	OC1(CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1)c1ccc(Cl)c(c1)C(F)(F)F	CID:33630	phase I
BRD-K04412738	COc1cccc(c1)[C@@]2(O)CCCC[C@@H]2CN(C)C	CID:33741	phase I
BRD-K76810206	CO[C@]12C[C@@H](COC(=O)c3cncc(Br)c3)CN(C)[C@@H]1Cc1cn(C)c3cccc2c13	CID:34040	phase I
BRD-K04196797	NC(=O)N1c2ccccc2CC(=O)c2ccccc12	CID:34312	phase I
BRD-K78712176	C[C@@](Cc1ccc(O)c(O)c1)(NN)C(O)=O	CID:34359	phase I
BRD-K21548250	CCOC(=O)Nc1ccc2Sc3ccccc3N(C(=O)CCN3CCOCC3)c2c1	CID:34633	phase I
BRD-A04831598	NC1CCc2ccccc2C1	CID:34677	phase I
BRD-A24429032	Oc1ccc(CCNCC2CCc3ccccc3C2=O)cc1	CID:34772	phase I
BRD-K72903603	Cc1cn([C@H]2C[C@H](N=[N+]=[N-])[C@@H](CO)O2)c(=O)[nH]c1=O	CID:35370	phase I
BRD-K73541271	OCCOCCOC(=O)c1ccccc1Nc1cccc(c1)C(F)(F)F	CID:35375	phase I
BRD-K86003836	COC(=O)Nc1nc2cc(ccc2[nH]1)C(=O)c1ccc(F)cc1	CID:35802	phase I
BRD-K41051431	CC1(C)S[C@@H]2[C@H](\N=C\N3CCCCCC3)C(=O)N2[C@H]1C(O)=O	CID:36273	phase I
BRD-A54880345	CCOC(=O)c1cncn1C(C)c1ccccc1	CID:36339	phase I
BRD-K37798499	COc1cc(cc(OC)c1O)[C@H]1[C@@H]2[C@H](COC2=O)[C@H](O[C@@H]2O[C@@H]3CO[C@@H](C)O[C@H]3[C@H](O)[C@H]2O)c2cc3OCOc3cc12	CID:36462	phase I
BRD-A78322124	CC(CCc1ccc(O)cc1)NCCc1ccc(O)c(O)c1	CID:36811	phase I
BRD-A61866602	COc1ccc2[nH]cc(CC(C)N)c2c1	CID:36906	phase I
BRD-A77864279	CN(C)C1CCc2c(C1)ccc(O)c2O	CID:37033	phase I
BRD-A11776908	Clc1ccc(C(Cn2ccnc2)OCC=C)c(Cl)c1	CID:37175	phase I
BRD-A51964809	CCCCN(CCCC)CCC(O)c1cc2c(Cl)cc(Cl)cc2c2cc(ccc12)C(F)(F)F	CID:37393	phase I
BRD-K70821460	Cc1nc[nH]c1CCN	CID:37463	phase I
BRD-K60369935	NC(=O)c1ncn(n1)[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	CID:37542	phase I
BRD-K88043978	NCC[C@H](O)C(=O)N[C@@H]1C[C@H](N)[C@@H](O[C@H]2O[C@H](CN)[C@@H](O)[C@H](O)[C@H]2O)[C@H](O)[C@H]1O[C@H]1O[C@H](CO)[C@@H](O)[C@H](N)[C@H]1O	CID:37768	phase I
BRD-K99984802	Cc1c(Nc2ncccc2C(O)=O)cccc1C(F)(F)F	CID:38081	phase I
BRD-A65444648	OCN1C(NC(=O)NCNC(=O)NC2N(CO)C(=O)NC2=O)C(=O)NC1=O	CID:38258	phase I
BRD-K34098590	OC(=O)COc1ccc(C(=O)c2cccs2)c(Cl)c1Cl	CID:38409	phase I
BRD-K48578705	C[C@](N)(Cc1ccc(O)c(O)c1)C(O)=O	CID:38853	phase I
BRD-A92670106	CC(N)C(=O)Nc1c(C)cccc1C	CID:38945	phase I
BRD-K46018455	CC(C)(Oc1ccc(CCNC(=O)c2ccc(Cl)cc2)cc1)C(O)=O	CID:39042	phase I
BRD-A87606379	CC(C)(C)NCC(O)COc1cccc2C[C@@H](O)[C@@H](O)Cc12	CID:39147	phase I
BRD-K24023109	COc1ccc(cc1)[C@@H]1Sc2ccccc2N(CCN(C)C)C(=O)[C@@H]1OC(C)=O	CID:39186	phase I
BRD-K78513633	OC(=O)c1nn(Cc2ccc(Cl)cc2Cl)c2ccccc12	CID:39562	phase I
BRD-K20168442	CC(=O)O[C@H]1[C@H](C[C@H]2[C@@H]3CC[C@H]4C[C@H](OC(=O)C)[C@H](C[C@]4(C)[C@H]3CC[C@]12C)N5CCCCC5)[N+]6(C)CCCCC6	CID:39765	phase I
BRD-K14965640	CC(C)Cc1ccc(cc1)[C@H](C)C(O)=O	CID:39912	phase I
BRD-K00766422	OC(=O)C[C@H](NC(=O)CP(O)(O)=O)C(O)=O	CID:39981	phase I
BRD-K65716359	Oc1ccc(C(=O)c2cc(O)c(O)c(O)c2)c(O)c1O	CID:40399	phase I
BRD-A19134330	CNc1ccc2oc(C[C@@H]3OC4(CC[C@@H]3C)O[C@H](C(C)C(=O)c5ccc[nH]5)[C@H](C)C[C@H]4C)nc2c1C(=O)O	CID:40486	phase I
BRD-K96862998	Cc1ccc(=O)n(c1)-c1ccccc1	CID:40632	phase I
BRD-A17846016	Cc1c(C)c2OC(C)(CCc2c(C)c1O)C(O)=O	CID:40634	phase I
BRD-K40645748	O[C@H]([C@H]1CCCCN1)c2cc(nc3c(cccc23)C(F)(F)F)C(F)(F)F	CID:40692	phase I
BRD-K59753975	CC[C@]1(O)C[C@H]2CN(C1)CCc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C)[C@@H]1[C@]22CCN3CC=C[C@](CC)([C@@H]23)[C@@H](O)[C@]1(O)C(N)=O	CID:40839	phase I
BRD-A33447119	COC(=O)Nc1nc2ccc(cc2[nH]1)S(=O)c1ccccc1	CID:40854	phase I
BRD-A02710418	CCC1(CCCCN(C)C1)c1cccc(O)c1	CID:41049	phase I
BRD-K90699611	COc1cc(C)c(C=CC(C)=CC=CC(C)=CC(O)=O)c(C)c1C	CID:41317	phase I
BRD-K96471533	CC(=O)Oc1ccccc1C(=O)Nc1ncc(s1)[N+]([O-])=O	CID:41684	phase I
BRD-A16444946	C[C@H]1O[C@H](O[C@@H]2[C@@H](CO)O[C@H](O[C@@H]3[C@@H](CO)OC(O)[C@H](O)[C@H]3O)[C@H](O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1N[C@H]1C=C(CO)[C@@H](O)[C@H](O)[C@H]1O	CID:41774	phase I
BRD-K30480208	CC(C)NC(=O)NS(=O)(=O)c1cnccc1Nc1cccc(C)c1	CID:41781	phase I
BRD-K04548931	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(=O)CO	CID:41867	phase I
BRD-K94173644	CN(C)CC=C(c1ccc(Br)cc1)c2cccnc2	CID:41987	phase I
BRD-K48470486	CO[C@]1(NC(=O)CSCC#N)[C@H]2SCC(=C(N2C1=O)C(=O)O)CSc3nnnn3C	CID:42008	phase I
BRD-A19952358	Cc1cc(C(C#N)c2ccc(Cl)cc2)c(Cl)cc1NC(=O)c1cc(I)cc(I)c1O	CID:42574	phase I
BRD-A71390734	CC1OC(CC(N)C1O)O[C@H]1C[C@@](O)(Cc2c(O)c3C(=O)c4ccccc4C(=O)c3c(O)c12)C(C)=O	CID:42594	phase I
BRD-K29627430	OCC=C1O[C@@H]2CC(=O)N2[C@H]1C(O)=O	CID:42617	phase I
BRD-K86958018	CCCCCCCCC=CCCCCCCCC(=O)NCc1ccc(O)c(OC)c1	CID:42760	phase I
BRD-K69650333	C[C@@H]1O[C@H](C[C@H](N)[C@@H]1O)O[C@H]1C[C@@](O)(Cc2c(O)c3C(=O)c4ccccc4C(=O)c3c(O)c12)C(C)=O	CID:42890	phase I
BRD-A50310035	CCCCC(C)(O)CC=C[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)OC	CID:42955	phase I
BRD-A03061970	COc1cc2[nH]nnc2cc1C(=O)NCC1CCCN1CC=C	CID:43008	phase I
BRD-K97521363	Nc1cc(C(Cl)=C(Cl)Cl)c(cc1S(N)(=O)=O)S(N)(=O)=O	CID:43231	phase I
BRD-K00206590	CCC(C)(C)N=C(NC#N)Nc1cccnc1	CID:43345	phase I
BRD-K37848908	NCc1ccccc1CC(=O)N[C@H]2[C@H]3SCC(=C(N3C2=O)C(=O)O)CSc4nnnn4CC(=O)O	CID:43507	phase I
BRD-K86873305	CCN1CCN(C(=O)N[C@@H](C(=O)N[C@H]2[C@H]3SC(C)(C)[C@@H](N3C2=O)C(O)=O)c2ccccc2)C(=O)C1=O	CID:43672	phase I
BRD-K02275692	CN(C)CCn1nnnc1SCC1=C(N2[C@H](SC1)[C@H](NC(=O)Cc1csc(N)n1)C2=O)C(O)=O	CID:43708	phase I
BRD-K37991163	Fc1ccc(cc1)[C@@H]1CCNC[C@H]1COc1ccc2OCOc2c1	CID:43815	phase I
BRD-K54529596	C[C@H](CS)C(=O)N1CCC[C@H]1C(O)=O	CID:44093	phase I
BRD-K17953061	CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n3c4ccccc4c5c6CNC(=O)c6c7c8ccccc8n2c7c35	CID:44259	phase I
BRD-A48323445	COc1cc2C(C)NCCc2cc1O	CID:46695	phase I
BRD-A20862232	COc1cc2CCNC(C)c2cc1O	CID:46697	phase I
BRD-A63546914	COc1cc2CCN(C)C(CCc3ccc(Cl)cc3)c2cc1O	CID:46740	phase I
BRD-A75935363	COc1ccc(CC2c3cc(OC)c(OC)cc3CC[N+]2(C)CCC(=O)OCCCCCOC(=O)CC[N+]2(C)CCc3cc(OC)c(OC)cc3C2Cc2ccc(OC)c(OC)c2)cc1OC	CID:47319	phase I
BRD-A16665823	Clc1ccc(CCC(Cn2ccnc2)Sc2c(Cl)cccc2Cl)cc1	CID:47472	phase I
BRD-K97752965	[O-][N+](=O)OCCNC(=O)c1cccnc1	CID:47528	phase I
BRD-K74141488	CN(C\C=C\c1ccccc1)Cc1cccc2ccccc12	CID:47641	phase I
BRD-K60770992	CCCN1C[C@H](CSC)C[C@H]2[C@H]1Cc1c[nH]c3cccc2c13	CID:47811	phase I
BRD-K09602097	CC(=O)O[C@H]1[C@@H](O)[C@H]2C(C)(C)CC[C@H](O)[C@]2(C)[C@@]2(O)C(=O)C[C@@](C)(O[C@]12C)C=C	CID:47936	phase I
BRD-K63242551	CC1=C(N2[C@H](SC1)[C@H](NC(=O)[C@H](N)c3ccc(O)cc3)C2=O)C(=O)O	CID:47965	phase I
BRD-A98378129	FC(F)(F)c1cccc(Nc2ncccc2C(=O)OC2OC(=O)c3ccccc23)c1	CID:48229	phase I
BRD-K15715913	CN1CCN(CC1)C2=Nc3cc(F)ccc3Cc4ccccc24	CID:49381	phase I
BRD-K81916719	CSc1nc2cc(Cl)c(Oc3cccc(Cl)c3Cl)cc2[nH]1	CID:50248	phase I
BRD-K11107424	CNC(=NC#N)NCCSCc1csc(N=C(N)N)n1	CID:50287	phase I
BRD-K56334280	CN(C)CCN1C(=O)c2cccc3cc(N)cc(C1=O)c23	CID:50515	phase I
BRD-K70507123	Cn1c2ncn(CC3OCCO3)c2c(=O)n(C)c1=O	CID:50942	phase I
BRD-K20338176	N[C@@H](C(=O)N[C@H]1[C@H]2SCC(Cl)=C(N2C1=O)C(O)=O)c1ccccc1	CID:51039	phase I
BRD-K55034111	CCn1cc(C(O)=O)c(=O)c2cc(F)c(cc12)N1CCN(C)CC1	CID:51081	phase I
BRD-K67445247	NP(N)(=O)NC(=O)c1ccc(F)cc1	CID:51173	phase I
BRD-K04188046	Oc1ccc(cc1O)C(=O)Cn2ccnc2	CID:52780	phase I
BRD-K91289464	CO[C@]1(NC(=O)C2SC(=C(C(=O)N)C(=O)O)S2)[C@H]3SCC(=C(N3C1=O)C(=O)O)CSc4nnnn4C	CID:53025	phase I
BRD-K09416995	CC[C@H](C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@@H]12	CID:53232	phase I
BRD-K50720187	CCOC(=O)Nc1ccc(NCc2ccc(F)cc2)nc1N	CID:53276	phase I
BRD-K70490179	C[C@H]1CN(CCCn2c3ccccc3c3ccccc23)C[C@@H](C)N1	CID:53389	phase I
BRD-K12437696	C[C@H]1[C@H](NC(=O)C(=NOC(C)(C)C(=O)O)c2csc(N)n2)C(=O)N1S(=O)(=O)O	CID:54117	phase I
BRD-K59935627	CC(C)(ON=C(C(=O)N[C@H]1[C@H]2SCC(C[n+]3ccccc3)=C(N2C1=O)C(O)=O)c1csc(N)n1)C(O)=O	CID:54197	phase I
BRD-K22134346	CCC(C)(C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@@H]12	CID:54454	phase I
BRD-A26112980	CC1NCCc2cc(O)c(O)cc12	CID:54456	phase I
BRD-A18696154	C1CN=C(N1)C1COc2ccccc2O1	CID:54459	phase I
BRD-K54094468	CCN1CCC[C@H]1CNC(=O)c1c(OC)ccc(Br)c1OC	CID:54477	phase I
BRD-K26548821	CCCN1CCC[C@@H]2Cc3n[nH]cc3C[C@@H]12	CID:54562	phase I
BRD-K41410256	OC(=O)CCNC(=O)c1ccc(cc1)N=Nc1ccc(O)c(c1)C(O)=O	CID:54585	phase I
BRD-K60511616	CC[C@H](C)C(=O)O[C@H]1C[C@H](O)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(O)=O)[C@@H]12	CID:54687	phase I
BRD-K86882815	CCNC(=O)N(CCCN(C)C)C(=O)[C@@H]1C[C@H]2[C@@H](Cc3c[nH]c4cccc2c34)N(CC=C)C1	CID:54746	phase I
BRD-A17462676	CN(C)C(=O)Oc1cc(OC(=O)N(C)C)cc(c1)C(O)CNC(C)(C)C	CID:54766	phase I
BRD-K20141153	CNCC[C@@H](Oc1ccccc1C)c1ccccc1	CID:54841	phase I
BRD-K72222507	CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1Cc2ccccc2C[C@H]1C(O)=O	CID:54892	phase I
BRD-A52647795	CC(C#CCN1CCCC1)N(C)C(C)=O	CID:55005	phase I
BRD-K37270826	CC#C[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CCC4=C3[C@H](C[C@]12C)c1ccc(cc1)N(C)C	CID:55245	phase I
BRD-A76934284	CCCN1CCCC(C1)c1cccc(O)c1	CID:55445	phase I
BRD-A41722204	COc1cc(ccc1c2nc3ccncc3[nH]2)S(=O)C	CID:55690	phase I
BRD-K08525451	OC(=O)c1cn(-c2ccc(F)cc2)c2cc(N3CCNCC3)c(F)cc2c1=O	CID:56208	phase I
BRD-K39716612	CC(C)n1c(C=C[C@H](O)C[C@H](O)CC(O)=O)c(-c2ccc(F)cc2)c2ccccc12	CID:56719	phase I
BRD-A97674275	COc1ccccc1OCC(O)CN1CCN(CC(=O)Nc2c(C)cccc2C)CC1	CID:56959	phase I
BRD-K90574421	O=C1N(CCCCN2CCN(CC2)c2ncccn2)S(=O)(=O)c2ccccc12	CID:56971	phase I
BRD-K13261168	CCCN1CCC[C@@H]2Cc3nc(N)ncc3C[C@@H]12	CID:57242	phase I
BRD-K50417881	CCN1CCC[C@H]1CNC(=O)c1c(O)c(CC)cc(Cl)c1OC	CID:57267	phase I
BRD-K01095011	CC(C)(C)NC(=O)[C@H]1CC[C@H]2[C@@H]3CC[C@H]4NC(=O)C=C[C@]4(C)[C@H]3CC[C@]12C	CID:57363	phase I
BRD-K82484965	OC(=O)c1ccc2[nH]cc(CCCCN3CCC(=CC3)c3ccccc3)c2c1	CID:57364	phase I
BRD-K26657438	CC(C)Cn1cnc2c(N)nc3ccccc3c12	CID:57469	phase I
BRD-A87479750	NC(=O)N1C(=O)C(C(=O)c2cccs2)c2cc(Cl)ccc12	CID:57946	phase I
BRD-K79353516	CN1Cc2ccccc2[C@H]3[C@H]1Cc4c[nH]c5cccc3c45	CID:58144	phase I
BRD-K62374253	CN1CCN(CC1)c1c(F)cc2c3c1SCCn3cc(C(O)=O)c2=O	CID:58258	phase I
BRD-A25619068	N#Cc1ccc(cc1)C1CCCc2cncn12	CID:59693	phase I
BRD-A07395371	COC(=O)CCc1ccc(OCC(O)CNC(C)C)cc1	CID:59768	phase I
BRD-A93964801	NC1CCN(C1)c1c(F)cc2c(c1Cl)n(cc(C(O)=O)c2=O)C1CC1	CID:60063	phase I
BRD-K69116396	Fc1ccc(cc1)-n1cc(C2CCN(CCN3CCNC3=O)CC2)c2cc(Cl)ccc12	CID:60149	phase I
BRD-K33127281	COc1ccc(cc1C12CC3CC(CC(C3)C1)C2)-c1ccc2cc(ccc2c1)C(O)=O	CID:60164	phase I
BRD-K33425534	C[C@@]12CC[C@H]3[C@@H](CC(=C)C4=CC(=O)C=C[C@]34C)[C@@H]2CCC1=O	CID:60198	phase I
BRD-K07612980	C[C@H]1CN(C[C@@H](C)N1)c1c(F)c(N)c2c(c1F)n(cc(C(O)=O)c2=O)C1CC1	CID:60464	phase I
BRD-A56359832	CC(N(O)C(N)=O)c1cc2ccccc2s1	CID:60490	phase I
BRD-A36074203	CC(Cc1ccccc1)(NC(=O)CN)c1ccccc1	CID:60511	phase I
BRD-K27721098	COC(=O)[C@@H](N1CCc2sccc2C1)c1ccccc1Cl	CID:60606	phase I
BRD-K60160658	Cc1ccsc1C(=CCCN1CCC[C@H](C1)C(O)=O)c1sccc1C	CID:60648	phase I
BRD-K71926323	CN1CCN(CC1)c1c(F)cc2c3c1OCN(C)n3cc(C(O)=O)c2=O	CID:60651	phase I
BRD-K09549677	COCC(=O)O[C@]1(CCN(C)CCCc2nc3ccccc3[nH]2)CCc2cc(F)ccc2[C@@H]1C(C)C	CID:60663	phase I
BRD-K55696337	CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccc(O)c(CN(C)C)c4cc3Cn1c2=O	CID:60700	phase I
BRD-A61392169	OC(CN1CCC(Cc2ccc(F)cc2)CC1)c1ccc(Cl)cc1	CID:60703	phase I
BRD-K47679368	Nc1c(CC(O)=O)cccc1C(=O)c1ccc(Br)cc1	CID:60726	phase I
BRD-K15108141	Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)C2(F)F)c(=O)n1	CID:60750	phase I
BRD-A99164655	Oc1cc2CCC3NCc4ccccc4C3c2cc1O	CID:60759	phase I
BRD-A50764878	O=C1CC2(CCCC2)CC(=O)N1CCNCC1COc2ccccc2O1	CID:60769	phase I
BRD-K08998509	Fc1ccc(cc1)N1CCN(CCCN2c3cccc4cccc(c34)S2(=O)=O)CC1	CID:60785	phase I
BRD-K70358946	Clc1cccc(N2CCN(CCCCOc3ccc4CCC(=O)Nc4c3)CC2)c1Cl	CID:60795	phase I
BRD-K69726342	CC(C)c1c(C(=O)Nc2ccccc2)c(c(-c2ccc(F)cc2)n1CC[C@@H](O)C[C@@H](O)CC(O)=O)-c1ccccc1	CID:60823	phase I
BRD-K02992638	Nc1ccn([C@@H]2CS[C@H](CO)O2)c(=O)n1	CID:60825	phase I
BRD-K71103788	CNCC[C@H](Oc1cccc2ccccc12)c1cccs1	CID:60835	phase I
BRD-K08547377	CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCC(CC3)N3CCCCC3)cc12	CID:60838	phase I
BRD-K45158365	CCCCC(=O)N(Cc1ccc(cc1)-c1ccccc1-c1nn[nH]n1)[C@@H](C(C)C)C(O)=O	CID:60846	phase I
BRD-K08681769	CCCCCN(C)CCC(O)(P(O)(O)=O)P(O)(O)=O	CID:60852	phase I
BRD-K29582115	Clc1cc2NC(=O)Cc2cc1CCN1CCN(CC1)c1nsc2ccccc12	CID:60854	phase I
BRD-K54314721	CN(C)CCc1c[nH]c2ccc(C[C@H]3COC(=O)N3)cc12	CID:60857	phase I
BRD-K43860855	NC(=N)NCc1cccc(I)c1	CID:60860	phase I
BRD-K37130586	CN(C)CCC=C1c2ccccc2COc2ccc(CC(O)=O)cc12	CID:60865	phase I
BRD-A72066420	COP(=O)(OC)OC(c1ccc(Cl)cc1)P(=O)(OC)OC	CID:60910	phase I
BRD-K39503511	CC(C)(C)Sc1c(CC(C)(C)C(O)=O)n(Cc2ccc(Cl)cc2)c2ccc(OCc3ccc4ccccc4n3)cc12	CID:60923	phase I
BRD-K96720755	COc1ccc(cc1OC)S(=O)(=O)N1[C@@H](C(=O)N2CCC[C@H]2C(N)=O)[C@](O)(c2cc(Cl)ccc12)c1ccccc1Cl	CID:60943	phase I
BRD-K99673372	CC(C)(O)c1ccccc1CC[C@@H](SCC1(CC(O)=O)CC1)c1cccc(C=Cc2ccc3ccc(Cl)cc3n2)c1	CID:60951	phase I
BRD-K61192372	CCCCCOC(=O)Nc1nc(=O)n(cc1F)[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O	CID:60953	phase I
BRD-K62289640	CC(C)c1ccc2c(CC[C@H]3[C@](C)(CN)CCC[C@]23C)c1	CID:62034	phase I
BRD-K62929068	N(Cc1ccccc1)c1ncnc2nc[nH]c12	CID:62389	phase I
BRD-K52219182	CCCn1c2nc(N)nn2cc(C)c1=O	CID:62824	phase I
BRD-K83836748	CN(C)CCN1c2ccccc2Sc2ccc(Cl)cc12	CID:62861	phase I
BRD-K02410399	Clc1ccc2Sc3ccccc3N(CCCN3CCN(CC3)C3C4CC5CC(C4)CC3C5)c2c1	CID:62872	phase I
BRD-K58901278	CNCCCN1c2ccccc2Sc2ccc(Cl)cc12	CID:62875	phase I
BRD-K40758068	FC(F)(F)[C@]1(OC(=O)Nc2ccc(Cl)cc12)C#CC1CC1	CID:64139	phase I
BRD-K74117820	Cc1c(O)cccc1C(=O)N[C@@H](CSc1ccccc1)[C@H](O)CN1C[C@H]2CCCC[C@H]2C[C@H]1C(=O)NC(C)(C)C	CID:64143	phase I
BRD-A41630653	COc1ccc2CC3C4CCCC[C@@]4(CCN3C)c2c1	CID:64650	phase I
BRD-K94441233	CC[C@H](C)C(=O)O[C@H]1CCC=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@@H]12	CID:64715	phase I
BRD-K68185022	C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]2[C@H]1C)C(=O)O	CID:64945	phase I
BRD-K45401373	CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)C(O)=O	CID:64971	phase I
BRD-K53523901	COc1cc(C[C@@H]2[C@@H](Cc3ccc(OC)c(OC)c3)COC2=O)ccc1O	CID:64981	phase I
BRD-K19059335	Clc1ccc2NC(=O)CN=C(c3ccc[nH]3)c2c1	CID:64983	phase I
BRD-K33240821	C(N1CCCNCCNCCCNCC1)c1ccc(CN2CCCNCCNCCCNCC2)cc1	CID:65015	phase I
BRD-K51730347	O=c1c(c1-c1ccccc1)-c1ccccc1	CID:65057	phase I
BRD-K55591206	Oc1cc(O)c2C[C@@H](OC(=O)c3cc(O)c(O)c(O)c3)[C@H](Oc2c1)c1cc(O)c(O)c(O)c1	CID:65064	phase I
BRD-K80970344	SC(=S)N1CCCC1	CID:65351	phase I
BRD-K91733562	COc1cc(C[C@@H](CO)[C@H](CO)Cc2ccc(O)c(OC)c2)ccc1O	CID:65373	phase I
BRD-K80431395	Cn1nc(N)c2cn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c3ncnc1c23	CID:65399	phase I
BRD-K75868704	C[C@H](O)C(=O)Nc1c(I)c(C(=O)NC(CO)CO)c(I)c(C(=O)NC(CO)CO)c1I	CID:65492	phase I
BRD-K66818636	CC(=O)CCCCn1cnc2n(C)c(=O)n(C)c(=O)c12	CID:65599	phase I
BRD-K92446736	COc1ccc(CCN(C)CCCN2CCc3cc(OC)c(OC)cc3CC2=O)cc1OC	CID:65637	phase I
BRD-K79759031	C[C@@H]1CC[C@H]2[C@@H](C)[C@@H](OC(=O)CCC(=O)O)O[C@@H]3O[C@@]4(C)CC[C@@H]1[C@@]23OO4	CID:65664	phase I
BRD-K32755366	CO[C@H]1[C@H](O)C[C@@H]2CN3CCc4c([nH]c5cc(OC)ccc45)[C@H]3C[C@@H]2[C@@H]1C(=O)O	CID:65747	phase I
BRD-K02227374	CCN(CC)C(=O)[C@@]1(C[C@@H]1CN)c1ccccc1	CID:65833	phase I
BRD-K55424922	Clc1cccc(SC2CCNCC2)n1	CID:65854	phase I
BRD-K32814891	CCOc1ccccc1O[C@H]([C@@H]1CNCCO1)c1ccccc1	CID:65856	phase I
BRD-A95939040	Clc1ccc(C(Cn2ccnc2)OCc2csc3c(Cl)cccc23)c(Cl)c1	CID:65863	phase I
BRD-K28115081	Cc1nnc2CN=C(c3cc(CCC(=O)N4CCOCC4)sc3-n12)c1ccccc1Cl	CID:65889	phase I
BRD-K21884483	CN(C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1)c1nccc(=O)[nH]1	CID:65906	phase I
BRD-A26032986	CC1(CN2CCC(CC2)n2c3ccccc3[nH]c2=O)OCc2ccccc2-n2cccc12	CID:65909	phase I
BRD-K44442813	OC(=O)[C@@H]1CSCN1C(=O)[C@@H]1CCC(=O)N1	CID:65944	phase I
BRD-K66412701	C[C@H]1COc2c(c(F)cc3c2n1cc(C(O)=O)c3=O)C1(N)CC1	CID:65957	phase I
BRD-K82846253	CCOc1cc(CC(=O)N[C@@H](CC(C)C)c2ccccc2N2CCCCC2)ccc1C(O)=O	CID:65981	phase I
BRD-K73999723	CCCc1nc2c(C)cc(cc2n1Cc1ccc(cc1)-c1ccccc1C(O)=O)-c1nc2ccccc2n1C	CID:65999	phase I
BRD-K21317336	Cc1ccc(cc1)N(CC1=NCCN1)c1ccc(O)cc1	CID:66148	phase I
BRD-K58626373	CCN[C@@H](C)Cc1cccc(c1)C(F)(F)F	CID:66265	phase I
BRD-K59406868	OC(=O)c1ccccc1Nc1cccc2C(=O)c3c(Nc4ccccc4C(O)=O)cccc3C(=O)c12	CID:66490	phase I
BRD-K12260308	COc1cc(O)c(C(=O)C)c(OC)c1	CID:66654	phase I
BRD-K53595844	N1c2ccccc2Oc2ccccc12	CID:67278	phase I
BRD-K61443650	CC[Hg]Sc1ccccc1C(O)=O	CID:67361	phase I
BRD-K01779529	OC(=O)C(=O)CF	CID:67946	phase I
BRD-K94689771	Oc1cc(O)c2C(=O)C[C@H](Oc2c1)c1ccccc1	CID:68071	phase I
BRD-K25186396	COc1ccc(cc1)-c1cc(=O)c2c(OC)c(OC)c(OC)c(OC)c2o1	CID:68077	phase I
BRD-K29178788	COc1c2ccoc2nc3ccccc13	CID:68085	phase I
BRD-K94512704	Fc1ccc(OCCCN2CCC3(CC2)N(CNC3=O)c4ccccc4)cc1	CID:68186	phase I
BRD-K91781484	S=c1ccss1	CID:68296	phase I
BRD-K64514229	Cc1cc(ccc1Oc1ccc(SC(F)(F)F)cc1)-n1c(=O)[nH]c(=O)n(C)c1=O	CID:68591	phase I
BRD-A66563878	CC(c1cnc[nH]1)c2cccc(C)c2C	CID:68602	phase I
BRD-K82036761	CN[C@H]1CC[C@@H](c2ccc(Cl)c(Cl)c2)c2ccccc12	CID:68617	phase I
BRD-K01638814	C1CC1C(NC1=NCCO1)C1CC1	CID:68712	phase I
BRD-K05851096	CCOC(=O)C1=C(C)NC(C)=C(C1c1ccccc1C=CC(=O)OC(C)(C)C)C(=O)OCC	CID:68733	phase I
BRD-A54490543	Cc1ccc2n3CCNC4CCCc(c34)c2c1	CID:68802	phase I
BRD-K74913225	CCN[C@H]1CN(CCCOC)S(=O)(=O)c2sc(cc12)S(N)(=O)=O	CID:68844	phase I
BRD-K91336023	CN(C)S(=O)(=O)N[C@H]1C[C@H]2[C@@H](Cc3cn(C)c4cccc2c34)N(C)C1	CID:68848	phase I
BRD-A53077924	CN1c2ccccc2C(NCCCCCCC(O)=O)c2ccc(Cl)cc2S1(=O)=O	CID:68870	phase I
BRD-K39621635	CO[C@H]1O[C@@H]2O[C@@]3(C)CC[C@H]4[C@H](C)CC[C@@H]([C@H]1C)[C@@]24OO3	CID:68911	phase I
BRD-A68318914	CC1NC(=O)NC1=O	CID:69216	phase I
BRD-K44004064	Cn1c2ncn(CC(O)=O)c2c(=O)n(C)c1=O	CID:69550	phase I
BRD-K94158209	COc1cc(CC(O)=O)cc(OC)c1OC	CID:70372	phase I
BRD-A94494639	CN(C)CCCN1c2ccccc2S(=O)c2ccc(Cl)cc12	CID:70413	phase I
BRD-K73700643	CC(=O)NCCc1c[nH]c2ccccc12	CID:70547	phase I
BRD-K92980438	OC(=O)C(=O)CBr	CID:70684	phase I
BRD-K01160827	O=S1c2ccccc2Nc3ccccc13	CID:71014	phase I
BRD-K16828188	CN1c2ccccc2Sc2ccccc12	CID:71015	phase I
BRD-K76534306	CCN1CCN(CC1)c1cc2n(cc(C(O)=O)c(=O)c2cc1F)C1CC1	CID:71188	phase I
BRD-K40227168	CC[C@@]12CCCN3CCc4c([C@H]13)n(C(=O)C2)c1ccccc41	CID:71203	phase I
BRD-K39746403	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2OC(=O)CC)N(C)C)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O	CID:71277	phase I
BRD-K86887724	CN(CCOc1ccc(NS(C)(=O)=O)cc1)CCc1ccc(NS(C)(=O)=O)cc1	CID:71329	phase I
BRD-K28137194	ClC(=Cn1cncn1)c2ccc(Cl)cc2Cl	CID:71333	phase I
BRD-K72816382	CCC(CC)(CC(=O)Nc1cccc(C=Cc2nc(cs2)C3CCC3)c1)C(=O)O	CID:71350	phase I
BRD-K48722833	COc1cc(ccc1OCCCN1CCC(CC1)c1noc2cc(F)ccc12)C(C)=O	CID:71360	phase I
BRD-K07265709	C[C@@H](CN1CC(=O)NC(=O)C1)N1CC(=O)NC(=O)C1	CID:71384	phase I
BRD-K17674993	C[C@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(OC(=O)C)C(=O)COC(=O)C	CID:71414	phase I
BRD-A10303790	CC1(C)S[C@@H]2[C@H](NC(=O)[C@H](N)c3ccccc3)C(=O)N2[C@H]1C(=O)OC4OC(=O)c5ccccc45	CID:71447	phase I
BRD-K84566043	C[N+]1(CCC(C(=O)N)(c2ccccc2)c3ccccc3)CCCCC1	CID:71490	phase I
BRD-K06557128	C[C@@H](c1ncncc1F)[C@](O)(Cn1cncn1)c1ccc(F)cc1F	CID:71616	phase I
BRD-K57291914	NC(=N)NC(=N)N1CCOCC1	CID:71655	phase I
BRD-K68538666	OC(=O)COC(=O)Cc1ccccc1Nc1c(Cl)cccc1Cl	CID:71771	phase I
BRD-A62057054	OC(C1CCN(CCc2ccccc2)CC1)c1ccccc1	CID:71781	phase I
BRD-A70083328	CC(O)Cn1c(C)ncc1[N+]([O-])=O	CID:71815	phase I
BRD-A11605036	COc1c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)cc3CCC(NC(=O)C)c4cc(=O)c(SC)ccc4-c3c1OC	CID:72067	phase I
BRD-A91992993	CNC(=Nc1ccc(cc1)C2=NNC(=O)CC2C)NC#N	CID:72124	phase I
BRD-K59574735	CC(C)C[C@H](NC(=O)[C@@H](O)[C@H](N)Cc1ccccc1)C(O)=O	CID:72172	phase I
BRD-K35559145	COc1ccc2Sc3ccccc3N(C[C@H](C)CN(C)C)c2c1	CID:72287	phase I
BRD-K98493452	Oc1ccc(cc1CC=C)-c1cc(CC=C)ccc1O	CID:72303	phase I
BRD-K06753942	COc1ccc(cc1OC)-c1cc(=O)c2c(OC)c(OC)c(OC)c(OC)c2o1	CID:72344	phase I
BRD-K06792661	O[C@H]1C=C2[C@@H](NC(=O)c3c(O)c4OCOc4cc23)[C@H](O)[C@@H]1O	CID:72376	phase I
BRD-K88625236	CCCCCCCCCc1ccc(OCCOCCOCCOCCOCCOCCOCCOCCOCCO)cc1	CID:72385	phase I
BRD-K92413528	OC(=O)[C@@H]1CSC(=O)N1	CID:72390	phase I
BRD-K43245338	CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc2ccccc2)C=O	CID:72430	phase I
BRD-K32681104	Nc1ccccc1S(N)(=O)=O	CID:72894	phase I
BRD-K55478147	ONC(=O)c1ccncc1	CID:72967	phase I
BRD-K88849294	CCCCCc1c(C(=O)O)c(O)cc2OC(=O)c3c(cc(OC)cc3Oc12)C(=O)CCCC	CID:73157	phase I
BRD-K11801786	ONC(=N)c1cc(O)c(O)c(O)c1	CID:73313	phase I
BRD-K52397688	CCNC(=O)N1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1	CID:73333	phase I
BRD-K43813806	CN(CC=Cc1ccccc1)Cc1cccc2ccccc12	CID:73342	phase I
BRD-K26134695	CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C=O	CID:73364	phase I
BRD-K19360254	CC(C)[C@@H]1N2C(=O)[C@](NC(=O)[C@H]3CN(C)[C@@H]4Cc5c[nH]c6cccc(C4=C3)c56)(O[C@@]2(O)[C@@H]7CCCN7C1=O)C(C)C	CID:73453	phase I
BRD-K70980943	COc1ccc2Sc3ccccc3Nc2c1	CID:74490	phase I
BRD-K06817181	BrC1C(Br)C(Br)C(Br)C(Br)C1Br	CID:74603	phase I
BRD-K13195996	COc1cc(cc(O)c1OC)C(O)=O	CID:74709	phase I
BRD-K88329126	COc1cc(c(O)cc1C(C)(C)C)C(C)(C)C	CID:74812	phase I
BRD-K10283649	NCCc1ccccc1O	CID:74865	phase I
BRD-K78075916	NCCCN1c2ccccc2Sc2ccc(Cl)cc12	CID:74981	phase I
BRD-A65771317	NCCCN1c2ccccc2S(=O)c2ccc(Cl)cc12	CID:75220	phase I
BRD-K17874705	NCCc1ccccn1	CID:75919	phase I
BRD-K20985754	COc1ccc(OC)c(CCN)c1	CID:76632	phase I
BRD-K32795028	C(c1ccccc1)n2ccnc2	CID:77918	phase I
BRD-K10706131	CCN(C)C(=O)Oc1cccc(c1)[C@H](C)N(C)C	CID:77991	phase I
BRD-A97437073	CN(CCOc1ccc(CC2SC(=O)NC2=O)cc1)c1ccccn1	CID:77999	phase I
BRD-K45542213	C1CNC2=NCCCN2C1	CID:79873	phase I
BRD-K26947839	CC(=O)c1ccc2Sc3ccccc3Nc2c1	CID:81131	phase I
BRD-K51066026	Nc1ccc2c[nH]nc2c1	CID:81423	phase I
BRD-K49577446	CC1(C)O[C@@H]2C[C@H]3[C@@H]4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:82153	phase I
BRD-K04809113	OCCc1ccc(O)c(O)c1	CID:82755	phase I
BRD-K17896185	CCC(=O)N(C1CCN(CCc2ccc(cc2)N=C=S)CC1)c1ccccc1	CID:84008	phase I
BRD-K49668410	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC	CID:84029	phase I
BRD-K99502674	CCN1CCC[C@H]1CNC(=O)c1cc(I)cc(OC)c1OC	CID:86101	phase I
BRD-K23986500	COc1cc2Sc3ccc(Cl)cc3N(CCCN(C)C)c2cc1OC	CID:87327	phase I
BRD-K43913647	COc1ccc2[nH]c3C(=O)NCCc3c2c1	CID:87372	phase I
BRD-K96146874	CCCC(CCC)C(=O)NO	CID:88129	phase I
BRD-K05395900	CN1CCC[C@H]1c1cccnc1	CID:89594	phase I
BRD-K34441861	CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1Cc2cc(OC)c(OC)cc2C[C@H]1C(O)=O	CID:91270	phase I
BRD-K13994703	CC(C)NC[C@H](O)COc1cccc2ccccc12	CID:91536	phase I
BRD-K99595596	C[C@@H]1NCCc2cc(O)c(O)cc12	CID:91588	phase I
BRD-K80396088	COc1ccc2c(c1)C(=O)N(CCc1ccc(cc1)S(=O)(=O)NC(=O)NC1CCCCC1)C(=O)C2(C)C	CID:91610	phase I
BRD-K96043519	Cc1nc(CCN)c[nH]1	CID:91613	phase I
BRD-K27351809	CC(=O)O[C@@]1(CC[C@H]2[C@@H]3C=C(C)C4=CC(=O)CC[C@@H]4[C@H]3CC[C@]12C)C(C)=O	CID:91668	phase I
BRD-K08996725	C(CNc1nc2ccccc2s1)COc1cccc(CN2CCCCC2)c1	CID:91769	phase I
BRD-A17081056	CC1NCCc2ccccc12	CID:92214	phase I
BRD-A49046702	OC(=O)C1CCCN(CCC=C(c2ccccc2)c2ccccc2)C1	CID:92409	phase I
BRD-A48261811	C[C@@H]1CCN([C@H](C1)C(O)=O)C(=O)[C@H](CCCN=C(N)N)NS(=O)(=O)c1cccc2CC(C)CNc12	CID:92722	phase I
BRD-K99451608	CC(C)[C@H](N1CCCNC1=O)C(=O)N[C@H](C[C@H](O)[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C)Cc1ccccc1	CID:92727	phase I
BRD-K06467078	COC(=O)[C@@H]1[C@@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12	CID:92766	phase I
BRD-K65411918	N[C@@H](Cc1cc(I)c(Oc2ccc(O)cc2)c(I)c1)C(O)=O	CID:92859	phase I
BRD-K24526313	CC1(C)Oc2ccc(cc2[C@H]([C@@H]1O)N1CCCC1=O)C#N	CID:93504	phase I
BRD-K84571636	CCCCCCCC(=O)CCc1ccc(O)c(OC)c1	CID:94378	phase I
BRD-K69032158	CC[C@H](C)[C@H](N)C(=O)N1CCC[C@H]1C(=O)N[C@@H]([C@@H](C)CC)C(=O)O	CID:94701	phase I
BRD-K31030218	CCCCc1oc2ccccc2c1C(=O)c3ccc(O)cc3	CID:96670	phase I
BRD-A59215453	CN1C(CC(O)c2ccccc2)CCCC1CC(O)c3ccccc3	CID:96946	phase I
BRD-K63784565	CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccc(O)cc4cc3Cn1c2=O	CID:97226	phase I
BRD-A37867643	OCC(O)Cc1ccc2OCOc2c1	CID:97807	phase I
BRD-K49759007	Cc1c(O)c(=O)n(-c2ccccc2)n1C	CID:98889	phase I
BRD-K87714311	OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cccnc1=O	CID:100016	phase I
BRD-A65550283	CC(=CCCC(C)(OC1OC(COC2OC(CO)C(O)C2O)C(O)C(O)C1O)C3CCC4(C)C3C(O)CC5C6(C)CCC(OC7OC(CO)C(O)C(O)C7OC8OC(CO)C(O)C(O)C8O)C(C)(C)C6CCC54C)C	CID:100018	phase I
BRD-K67484673	OC(=O)c1nn(Cc2ccc(Cl)cc2)c2ccccc12	CID:100493	phase I
BRD-K95847244	CC(=O)NCCc1ccc(O)c(O)c1	CID:100526	phase I
BRD-K34437622	Oc1ncc(F)cn1	CID:101498	phase I
BRD-K66206289	CN1[C@H](C[C@H](O)c2ccccc2)CCC[C@@H]1CC(=O)c1ccccc1	CID:101616	phase I
BRD-K24994810	C[C@]12CC[C@H]3[C@@H](CC[C@H]4C[C@H](O)CC[C@]34C)[C@@H]1CC=C2	CID:101989	phase I
BRD-K81807412	CNc1ncnc2n(cnc12)[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	CID:102175	phase I
BRD-A27143604	Oc1ccc(CC(C#N)c2ccc(O)cc2)cc1	CID:102614	phase I
BRD-K41445866	CC(=O)[C@H]1CC[C@H]2[C@@H]3CC[C@H]4C[C@H](O)CC[C@]4(C)[C@H]3C(=O)C[C@]12C	CID:104845	phase I
BRD-K13296708	Cc1c(nn(c1-c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1	CID:104850	phase I
BRD-K74763371	COc1ccccc1Oc1c(NS(=O)(=O)c2ccc(cc2)C(C)(C)C)nc(nc1OCCO)-c1ncccn1	CID:104865	phase I
BRD-A90311807	CC1(C)CC1C(=O)NC(=CCCCCSCC(N)C(=O)O)C(=O)O	CID:104867	phase I
BRD-A72703248	COc1ccc(CCCOC(Cn2ccnc2)c2ccc(OC)cc2)cc1	CID:104956	phase I
BRD-K14844937	CCc1c(ncc2[nH]c3cc(OC)c(OC)cc3c12)C(=O)OC	CID:104999	phase I
BRD-A96456596	CCCc1c(OCC(O)COc2ccc3c(oc(cc3=O)C(O)=O)c2CCC)ccc(C(C)=O)c1O	CID:105007	phase I
BRD-K38251852	CC(C)(O)[C@H]1O[C@H]2CC[C@]3(C)[C@]4(C)[C@H](Cc5c4[nH]c6ccccc56)CC[C@@]3(O)C2=CC1=O	CID:105008	phase I
BRD-K49061529	CCOC(=O)c1cc2c(cn1)[nH]c3ccccc32	CID:105078	phase I
BRD-K71339761	CNCCCN1c2ccc(O)cc2Sc2ccc(Cl)cc12	CID:107410	phase I
BRD-K28680267	COC(=O)c1cc2c(cn1)[nH]c3ccccc32	CID:107704	phase I
BRD-K97440753	CC(C)[C@@]1(NC(=O)[C@@H]2C[C@H]3[C@@H](Cc4c[nH]c5cccc3c45)N(C)C2)O[C@@]2(O)[C@@H]3CCCN3C(=O)[C@H](Cc3ccccc3)N2C1=O	CID:107715	phase I
BRD-A08187463	CC(=O)SCC(Cc1ccccc1)C(=O)NCC(=O)OCc1ccccc1	CID:107751	phase I
BRD-K11911061	COc1ccc(NC(=O)c2ccc(cc2)-c2ccc(cc2C)-c2noc(C)n2)cc1N1CCN(C)CC1	CID:107780	phase I
BRD-K92731339	CCC[C@H](N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@H]1C(O)=O)C(=O)OCC	CID:107807	phase I
BRD-K32696739	C1Cc2c(CN1)[nH]c3ccccc23	CID:107838	phase I
BRD-A00520476	CCN(CC)CC1CCCCN1CC(=O)N1c2ccccc2C(=O)Nc2cccnc12	CID:107867	phase I
BRD-K79905821	COc1ccc(cc1)-c1ccc(=N)n(CCCC(O)=O)n1	CID:107896	phase I
BRD-K50660797	Oc1cc(O)c2C[C@@H](OC(=O)c3cc(O)c(O)c(O)c3)[C@H](Oc2c1)c1ccc(O)c(O)c1	CID:107905	phase I
BRD-K94270326	CN1CCc2cc(Cl)c(O)cc2[C@@H]3[C@@H]1CCc4ccccc34	CID:107930	phase I
BRD-K61401890	COc1cc2OC[C@H]3Oc4c5C=CC(C)(C)Oc5ccc4C(=O)[C@H]3c2cc1OC	CID:107935	phase I
BRD-K00662280	Cc1nnc2ccc(nn12)-c1cccc(c1)C(F)(F)F	CID:107950	phase I
BRD-K83508485	CN(Cc1ccccc1)C(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)c1cn(C)c2ccccc12	CID:107967	phase I
BRD-K45882009	COc1cc(CNC(=O)CCCCCCC(C)C)ccc1O	CID:107982	phase I
BRD-K39484304	CC(C)[C@@]12O[C@H]2[C@@H]3O[C@]34[C@]5(O[C@H]5C[C@H]6C7=C(CC[C@@]64C)C(=O)OC7)[C@@H]1O	CID:107985	phase I
BRD-K19554809	Clc1cncc(n1)N2CCNCC2	CID:107992	phase I
BRD-A20589515	NC(C(O)=O)c1cc(O)cc(O)c1	CID:108001	phase I
BRD-K00234327	COc1ccc2[nH]cc(C3=CCNCC3)c2c1	CID:108029	phase I
BRD-K84709232	Oc1ccc(C=CC(=O)OCCc2ccccc2)cc1O	CID:108042	phase I
BRD-A15435692	OC(CCCN1CCN(CC1)c1ncc(F)cn1)c1ccc(F)cc1	CID:108046	phase I
BRD-K19653414	CN(C)CCCN1c2ccccc2CCc2cc(O)ccc12	CID:108051	phase I
BRD-K80315159	CCN(CC)CCOc1ccc(Cc2ccccc2)cc1	CID:108092	phase I
BRD-A65597028	COC1(COc2ccccc2O1)C1=NCCN1	CID:108094	phase I
BRD-K87158025	NC(NCc1ccccc1)=NC(=O)c1nc(Cl)c(N)nc1N	CID:108107	phase I
BRD-K55748775	Cc1nc2c(OCc3ccccc3)cccn2c1CC#N	CID:108137	phase I
BRD-K36627727	CC1(C)CCC(C)(C)c2cc(NC(=O)c3ccc(cc3)C(O)=O)ccc12	CID:108143	phase I
BRD-A65615053	COc1cc(N)c(Cl)cc1C(=O)NC1CN2CCC1CC2	CID:108182	phase I
BRD-K93645900	CN1CC(=O)N2[C@H](Cc3c([nH]c4ccccc34)[C@H]2c2ccc3OCOc3c2)C1=O	CID:110635	phase I
BRD-K41049123	Nc1nc(N)c(nc1Cl)C(=O)NC(=N)NCc1ccc(Cl)c(Cl)c1	CID:114771	phase I
BRD-K11298197	CS(=O)(=O)c1ccc(cc1)[C@@H](O)[C@@H](CF)NC(=O)C(Cl)Cl	CID:114811	phase I
BRD-K47539947	CCCCCCCCCCCCCCSCC(O)=O	CID:114924	phase I
BRD-K67100011	CC(C)(C)C(=O)OCOC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](\N=C\N1CCCCCC1)C2=O	CID:115163	phase I
BRD-K68392338	CCOC(=O)c1ncc2[nH]c3cccc(OC(C)C)c3c2c1C	CID:115210	phase I
BRD-K85503079	O=C1[C@H]2CCCC[C@H]2C(=O)N1CCCCN1CCN(CC1)c1nsc2ccccc12	CID:115368	phase I
BRD-K08807999	CC(=O)Oc1ccccc1C(=O)Oc1cccc(CO[N+]([O-])=O)c1	CID:119032	phase I
BRD-K25075681	COc1cccc(OC)c1-c1cc(nn1-c1ccnc2cc(Cl)ccc12)C(=O)NC1(C2CC3CC(C2)CC1C3)C(O)=O	CID:119192	phase I
BRD-K13629382	CN1CC[C@]2(C)[C@H]1N(C)c1ccc(O)cc21	CID:119198	phase I
BRD-A12426960	OC1(CF)CCOC(=O)C1	CID:119214	phase I
BRD-K49945136	Cn1cc(C(=O)OCC2CCN(CCNS(C)(=O)=O)CC2)c2ccccc12	CID:119376	phase I
BRD-A47706533	CCCCS(=N)(=O)CC[C@H](N)C(O)=O	CID:119565	phase I
BRD-K06388322	CCCN[C@H]1CCc2nc(N)sc2C1	CID:119570	phase I
BRD-A39052811	CCOc1cc(N)c(Cl)cc1C(=O)NCC1CN(Cc2ccc(F)cc2)CCO1	CID:119584	phase I
BRD-K12994359	Cc1onc(c1-c1ccc(cc1)S(N)(=O)=O)-c1ccccc1	CID:119607	phase I
BRD-K13800121	CCC(=O)NS(=O)(=O)c1ccc(cc1)-c1c(C)onc1-c1ccccc1	CID:119828	phase I
BRD-K41670583	OC(=O)c1cc([nH]n1)c2ccccc2	CID:121025	phase I
BRD-K65981456	CC(=O)NCCc1ccc(O)cc1	CID:121051	phase I
BRD-K96834847	CNCCCN1c2ccccc2CCc2cc(O)ccc12	CID:121249	phase I
BRD-K45117373	CC(=O)N(O)[C@H]1[C@H](O)C(C)(C)Oc2ccc(cc12)C#N	CID:121878	phase I
BRD-K33882852	CCOC(=O)c1ncc2[nH]c3ccc(OCc4ccccc4)cc3c2c1COC	CID:121926	phase I
BRD-K14282469	Nc1ccc(CCN2CCN(CC2)c3cccc(c3)C(F)(F)F)cc1	CID:121930	phase I
BRD-K92492521	CCc1cc(C(C)=O)c(O)cc1OCCCCCC(C)(C)c1nnn[nH]1	CID:122023	phase I
BRD-K89402695	Cc1c(CC(C)(C)C(O)=O)n(Cc2ccc(Cl)cc2)c2ccc(F)cc12	CID:122070	phase I
BRD-K35629949	OC(=O)Cn1c(cc2ccccc12)C(=O)Nc1nc(cs1)-c1ccccc1Cl	CID:122077	phase I
BRD-K58442346	NCCc1ccc(O)c(OS(O)(=O)=O)c1	CID:122136	phase I
BRD-A24122750	NCC(CS(O)(=O)=O)c1ccc(Cl)cc1	CID:122150	phase I
BRD-K67013324	CC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12	CID:122162	phase I
BRD-K56509348	CN(C)c1cccc2c(cccc12)S(=O)(=O)Nc1onc(C)c1C	CID:122272	phase I
BRD-K62103095	CN1CCc2c(Cl)ccc(OCC=C(C)C)c2CC1	CID:122295	phase I
BRD-K88544581	CCCCCCCCCCC(C)(C)C(=O)Nc1c(OC)cc(OC)cc1OC	CID:122327	phase I
BRD-K60174629	O=C[C@@H]1CCCN1C(=O)[C@@H]2CCCN2C(=O)OCc3ccccc3	CID:122623	phase I
BRD-A99182808	CC(=O)C1C(=O)C=C2Oc3c(c(O)c(C)c(O)c3C(C)=O)[C@]2(C)C1=O	CID:122718	phase I
BRD-K34469523	CC(C)(C)NC[C@H](O)c1ccc(O)c(CO)c1	CID:123600	phase I
BRD-K54770957	Cc1ccc(cn1)-c1ncc(Cl)cc1-c1ccc(cc1)S(C)(=O)=O	CID:123619	phase I
BRD-K14312455	C[C@]1(Cn2ccnn2)[C@@H](N2[C@@H](CC2=O)S1(=O)=O)C(O)=O	CID:123630	phase I
BRD-K64052750	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCOCC1	CID:123631	phase I
BRD-K85242180	CCCOC(=O)c1cc2c(cn1)[nH]c3ccccc32	CID:123662	phase I
BRD-A03359064	OC(CNCCNC(=O)Nc1ccccc1)COc1ccccc1C#N	CID:123686	phase I
BRD-K15519488	C1CCN(CC1)C1(CCCCC1)c1cc2ccccc2s1	CID:123692	phase I
BRD-A10355991	NC1(CCCCC1=O)c2ccccc2Cl	CID:123767	phase I
BRD-A67552655	CCOC(=O)C1(CCCCCCOc2ccc(Cl)cc2)CO1	CID:123823	phase I
BRD-K33811357	NCCc1ccc(OS(O)(=O)=O)c(O)c1	CID:123932	phase I
BRD-K34034388	C(CN1CCN(CC=Cc2ccccc2)CC1)OC(c3ccccc3)c4ccccc4	CID:123956	phase I
BRD-K81876028	O=c1ccc2[nH]cc(C3=CCNCC3)c2[nH]1	CID:124007	phase I
BRD-K82357231	Clc1ccc2c(CCc3cccnc3C2=C2CCNCC2)c1	CID:124087	phase I
BRD-K25875056	Clc1cccc2c(cccc12)S(=O)(=O)NCCCCCCc1ccccc1	CID:124172	phase I
BRD-K43978949	[O-][N+]1=C(C(=O)c2ccccc12)c1ccccn1	CID:124334	phase I
BRD-K76274772	CCCCCCCCCCCCCC(=O)N[C@H](C)[C@@H](O)c1ccccc1	CID:124735	phase I
BRD-A66435872	CC(CCCCC(=O)Nc1ccc(cc1)C(F)(F)F)NCCc1c[nH]cn1	CID:124846	phase I
BRD-K91862102	Nc1ccc(CCN2CN(c3ccccc3)C3(CCN(CCCC(=O)c4ccc(F)cc4)CC3)C2=O)cc1	CID:125085	phase I
BRD-K27803479	NCCCN1c2cc(Cl)ccc2Sc2cc(O)c(O)cc12	CID:125358	phase I
BRD-K04976539	Nc1ccc(cc1)c2cc(=O)c3cc(O)ccc3o2	CID:125519	phase I
BRD-K01649396	CN[C@@H]1C[C@H](c2ccccc12)c1ccc(Cl)c(Cl)c1	CID:126280	phase I
BRD-K17008822	CN(CCN1CCCC1)CCc1ccc(Cl)c(Cl)c1	CID:126388	phase I
BRD-K57304726	O=C(OCCN1CCOCC1)C1(CCCCC1)c1ccccc1	CID:126402	phase I
BRD-K23192422	C[C@]12O[C@H](C[C@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13	CID:126565	phase I
BRD-K39670393	Cc1nc(N)sc1CCN	CID:126688	phase I
BRD-K77677632	Cn1ccc2cc(NC(=O)Nc3cccnc3)ccc12	CID:126769	phase I
BRD-K59456551	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(cc1)C(=O)N[C@@H](CCC(O)=O)C(O)=O	CID:126941	phase I
BRD-K80778372	CN1Cc2c(ncn2-c2ccsc2C1=O)C(=O)OC(C)(C)C	CID:127382	phase I
BRD-A26845397	CC(C)NCC(O)COc1ccccc1-n1cccc1	CID:127404	phase I
BRD-K84895041	OC(=O)COc1cccc(c1)-c1ocnc1-c1nc(c(o1)-c1ccccc1)-c1ccccc1	CID:127861	phase I
BRD-K78844995	Ic1ccc(cc1)C(=O)NCCN1CCCCC1	CID:127898	phase I
BRD-K26160755	Clc1cccc2CN(Cc12)C1=NCCN1	CID:127951	phase I
BRD-K46441700	CN(C)CCCc1cc(ccc1O)C(=O)Nc2ccc(cc2)c3ccncc3	CID:128018	phase I
BRD-K19284129	COC(=O)[C@@H]1C[C@H](OC(C)=O)C(=O)[C@H]2[C@@]1(C)CC[C@H]1C(=O)O[C@@H](C[C@]21C)c1ccoc1	CID:128563	phase I
BRD-K86940927	[N-]=[N+]=Nc1ccc(CCN2CCN(CC2)c2cccc(C(F)(F)F)c2)cc1	CID:128737	phase I
BRD-K88358234	FC(F)(F)c1cccc(c1)C1=CCN(CCc2ccc3ccccc3c2)CC1	CID:128919	phase I
BRD-K52721684	CC1(C)Oc2ccc(cc2[C@@H](OC2=CC(=O)CC2)[C@@H]1O)C#N	CID:129348	phase I
BRD-A85472596	CS(=O)(=O)c1ccc(Cn2c3C(CC(O)=O)CCCc3c3cc(F)cc(F)c23)cc1	CID:129360	phase I
BRD-K81729199	CCN(CC)CCCCC1CCN(CC(=O)N2c3ccccc3C(=O)Nc3cccnc23)CC1	CID:129989	phase I
BRD-K44133266	CC1(C)[C@@H](N2[C@@H](CC2=O)S1(=O)=O)C(O)=O	CID:130313	phase I
BRD-K51290057	CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)C=Cc2ccc(cc2)C(=O)O	CID:130325	phase I
BRD-K27237442	CN1CCc2cc(Cl)c(O)cc2[C@H](C1)c1cccc2ccoc12	CID:130424	phase I
BRD-K78485176	CCCc1nc(C(C)(C)O)c(C(=O)OCc2oc(=O)oc2C)n1Cc1ccc(cc1)-c1ccccc1-c1nn[nH]n1	CID:130881	phase I
BRD-A67433117	OC1C(=CC(=O)O)CCCc2ccccc12	CID:131414	phase I
BRD-K09397065	NC1CCN(CC1)c1cccc(Cl)n1	CID:131747	phase I
BRD-K46766488	COc1ccc2cccc(N3CCN(CCNC(=O)c4ccc(F)cc4)CC3)c2c1	CID:131906	phase I
BRD-K18816859	CS(=O)(=O)Nc1ccc(Cc2noc(n2)-c2ccc3[nH]cc(CCN)c3c2)cc1	CID:132059	phase I
BRD-A04668240	CCOC(OCC)P(=O)(O)CCCNCc1ccc(Cl)c(Cl)c1	CID:132252	phase I
BRD-K28470988	CC(Oc1ccc(O)cc1)(P(O)(O)=O)P(O)(O)=O	CID:132449	phase I
BRD-K11634954	Fc1ccc(cc1)C(OCCN2CCN(CC=Cc3ccccc3)CC2)c4ccc(F)cc4	CID:132475	phase I
BRD-K09778810	CCCCCCN(CCCCCC)C(=O)Cc1c([nH]c2ccccc12)-c1ccc(F)cc1	CID:132496	phase I
BRD-K51662849	CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(C)C)CC(=O)NO	CID:132519	phase I
BRD-K15791587	FC(F)(F)c1cc(CO[C@H]2CCCN[C@H]2c2ccccc2)cc(c1)C(F)(F)F	CID:132846	phase I
BRD-K22227508	C/N=C(\N)/NCCC[C@H](N)C(=O)O	CID:132862	phase I
BRD-K04877770	CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC[C@@H](NC[C@@H](N)CS)C(C)C)C(=O)O	CID:132887	phase I
BRD-A70268693	CC(C(=O)OC1CC2CCC(C1)N2C)c1ccc(Br)cc1	CID:133002	phase I
BRD-K13211965	Cc1c(noc1-c1ccc(Cl)cc1)C1CCN(CCc2ccccc2)CC1	CID:133008	phase I
BRD-K50018155	COc1cc(N)c(Cl)cc1C(=O)CCC1CCN(CCNS(C)(=O)=O)CC1	CID:133076	phase I
BRD-A40807648	CN1CCCC1c1cncc(c1)C#C	CID:133106	phase I
BRD-K15467014	CN(C)CCCN1c2ccc(cc2CCc3cc(ccc13)[N+](=O)[O-])[N+](=O)[O-]	CID:133407	phase I
BRD-A04260165	CN1CCc2c(Cl)c(O)c(O)cc2C(C1)c3cccc(C)c3	CID:133538	phase I
BRD-A10903566	CCn1ccnc1CC1COc2ccccc2O1	CID:133621	phase I
BRD-K05181463	OC1(CCN(Cc2c[nH]c3ccccc23)CC1)c4ccc(Cl)cc4	CID:133633	phase I
BRD-K37542305	C[N+](C)(C)Cc1cccc(c1)\N=N\c1cccc(C[N+](C)(C)C)c1	CID:133795	phase I
BRD-K86570333	CCCCN1C(=O)C(=O)N(CCCC)C1=S	CID:134014	phase I
BRD-K48367671	CC(C)COc1ccc(cc1C#N)-c1nc(C)c(s1)C(O)=O	CID:134018	phase I
BRD-K04389336	C[C@H](CCc1ccccc1)NC[C@H](O)c1ccc(O)c(c1)C(N)=O	CID:134044	phase I
BRD-K45479396	C(COc1ccc2OCOc2c1)CN1CCN(CC1)c1ccccc1	CID:134117	phase I
BRD-K53987533	FC(F)(F)c1ccc2Sc3ccccc3N(CCCN4CCN(CCCl)CC4)c2c1	CID:134141	phase I
BRD-K17693482	CC(=O)OCCNC(=O)c1cccnc1	CID:134230	phase I
BRD-K74212935	CC(C)C[C@@H]1N2C(=O)[C@](NC(=O)[C@H]3CN(C)[C@@H]4Cc5c[nH]c6cccc(C4=C3)c56)(O[C@@]2(O)[C@@H]7CCCN7C1=O)C(C)C	CID:134551	phase I
BRD-K66782112	NC(=O)CCCCn1ccc(N=C(N)NCC(F)(F)F)n1	CID:134778	phase I
BRD-K89271983	COc1cc(SC)ccc1c2nc3ccncc3[nH]2	CID:135179	phase I
BRD-K28907958	OC(=O)c1ccc2cc(ccc2c1)-c1ccc(O)c(c1)C12CC3CC(CC(C3)C1)C2	CID:135411	phase I
BRD-K84996949	COc1ccc(cc1OC)-c1cc(=O)c2c(OC)c(OC)c(OC)cc2o1	CID:145659	phase I
BRD-K70301876	CN(C)CCC[C@]1(OCc2cc(ccc12)C#N)c1ccc(F)cc1	CID:146570	phase I
BRD-K47335880	Clc1ccc(OCCCCCC\N=C(\NC#N)Nc2ccncc2)cc1	CID:148198	phase I
BRD-K09471561	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(O)=O)c3=O	CID:149096	phase I
BRD-K48099440	CCCCC[C@H](O)C=C[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(O)=O	CID:149351	phase I
BRD-K27450477	CCCCCC[C@@H]([C@@H](C)O)n1cnc2c(N)ncnc12	CID:149784	phase I
BRD-K42260897	O[C@@H](CC[C@@H]1[C@H](N(C1=O)c1ccc(F)cc1)c1ccc(O)cc1)c1ccc(F)cc1	CID:150311	phase I
BRD-K49612115	NCCc1ccc(O)cc1O	CID:150962	phase I
BRD-K70163715	Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1	CID:151194	phase I
BRD-A68631409	CN1C2N(CCc3c2[nH]c2ccccc32)C(=O)c2ccccc12	CID:151289	phase I
BRD-K85853281	C[C@@H]1O[C@H](C[C@H](N)[C@@H]1O)O[C@@H]1C[C@](O)(Cc2c(O)c3C(=O)c4ccccc4C(=O)c3c(O)c12)C(C)=O	CID:151582	phase I
BRD-K04701986	OC(=O)CCc1cc(I)c(O)c(I)c1	CID:151819	phase I
BRD-K24304282	N[C@@H](Cc1ccc(O)cc1O)C(O)=O	CID:152670	phase I
BRD-K66615216	COc1c(N2C[C@@H]3CCCN[C@@H]3C2)c(F)cc2c1n(cc(C(O)=O)c2=O)C1CC1	CID:152946	phase I
BRD-K49808142	NCCc1ccc(OS(O)(=O)=O)cc1	CID:153005	phase I
BRD-A47884604	CC(C)(C)NCC(O)COc1cccc2[nH]c(cc12)C#N	CID:155346	phase I
BRD-K53878242	COCc1nc2c(=O)n(C)c(=O)n(CC(C)C)c2[nH]1	CID:155806	phase I
BRD-K32645441	CCCN(CCC)CCc1c[nH]c2ccc(cc12)C(=O)N	CID:156314	phase I
BRD-K47289124	CNc1cc(OC)c(cc1Cl)C(=O)N[C@@H]2CCN(Cc3ccccc3)[C@@H]2C	CID:156333	phase I
BRD-K59197931	COc1ccc2cc(ccc2c1)[C@H](C)C(O)=O	CID:156391	phase I
BRD-K50168500	Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl	CID:156414	phase I
BRD-K73838513	C[C@@H](NCCCc1cccc(c1)C(F)(F)F)c1cccc2ccccc12	CID:156419	phase I
BRD-K74065929	Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C	CID:156422	phase I
BRD-K83144676	CCCc1nc(c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1-c1nn[nH]n1)C(C)(C)O	CID:158781	phase I
BRD-K64157027	O[C@@H](CNCCOc1ccc(CC(O)=O)cc1)c1ccccc1	CID:158794	phase I
BRD-K62965247	Cn1cncc1[C@@](N)(c1ccc(Cl)cc1)c1ccc2n(C)c(=O)cc(-c3cccc(Cl)c3)c2c1	CID:159324	phase I
BRD-K92159000	NCCCN1c2ccccc2CCc2ccccc12	CID:159642	phase I
BRD-K37365015	CN(C)CCCN1c2cc(Cl)ccc2Sc2cc(O)c(O)cc12	CID:159916	phase I
BRD-A52660433	C1CCC(CC1)c1ccc2n3CCNC4CCCc(c34)c2c1	CID:160020	phase I
BRD-K07691486	CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1	CID:160355	phase I
BRD-A09073503	CN(C)CCC[N+]1([O-])c2ccccc2Sc2ccc(Cl)cc12	CID:160588	phase I
BRD-A10396145	COc1cc(CC(O)CO)ccc1O	CID:161566	phase I
BRD-A85860691	CN1C(=O)C23CC4(C(Nc5ccccc54)N3C(=O)C1(CO)SS2)C67CC8(SSC9(CO)N(C)C8=O)N(C7Nc%10ccccc%106)C9=O	CID:161591	phase I
BRD-K48869804	Oc1ccccc1N1CC=C(NC1=O)c1cccc(c1)[N+]([O-])=O	CID:161930	phase I
BRD-K90711641	NCCC(=O)NCCc1ccc(O)c(O)c1	CID:162755	phase I
BRD-A39747742	CCCCC(=O)O[C@H]1CCC2C3CCc4cc(O)ccc4C3CC[C@]12C	CID:163332	phase I
BRD-K43468059	CCC[C@H]1CC2=C(C[C@@H](CC)CC3=C1C(=O)OC3=O)C(=O)OC2=O	CID:164723	phase I
BRD-K40367460	CN(C)CCCN1c2ccccc2S(=O)(=O)c2ccc(Cl)cc12	CID:165214	phase I
BRD-K66989831	CCCCCCCCCCCCCCCc1cccc(O)c1C(O)=O	CID:167551	phase I
BRD-K96119599	C[C@H]1[C@@H]2CCC(=C3[C@@H]([C@H]2OC1=O)C(=CC3=O)C)C	CID:167683	phase I
BRD-K13544237	CCCN1CCc2cccc-3c2[C@H]1Cc4ccc(O)c(O)c43	CID:167715	phase I
BRD-K46272620	CC(C)[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O	CID:168182	phase I
BRD-K60060639	CC[N+](C)(CC)CC(=O)Nc1c(C)cccc1C	CID:168868	phase I
BRD-K33299843	COc1ccc2cc(ccc2c1)[C@@H](C)C(=O)O	CID:169118	phase I
BRD-K14643723	NCCc1ccc(cc1)S(=O)(=O)N	CID:169682	phase I
BRD-K63979671	CCc1cccc(CC)c1NC(=O)CN(CC(O)=O)CC(O)=O	CID:170344	phase I
BRD-A52530852	COc1ccc(cc1O)C(O)CO	CID:170451	phase I
BRD-K03222093	CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)CC=CC)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C	CID:171409	phase I
BRD-K89210380	OC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12	CID:171548	phase I
BRD-K16701932	NCC(=O)NCC(=O)N[C@@H](CCCNC(=O)CP(O)(O)=O)C(O)=O	CID:172813	phase I
BRD-K12120659	NC(=N)c1ccc(cc1)N1CCN(CC1)C1CCN(CC(O)=O)CC1	CID:173614	phase I
BRD-K68190965	COc1ccc(CNC(=O)C=Cc2ccc3[nH]cc(CCN(C)C)c3c2)cc1	CID:173615	phase I
BRD-K44993696	CC(C)NC[C@H](O)COc1ccc(CC(N)=O)cc1	CID:175540	phase I
BRD-K50938786	CCCN1CCCC[C@H]1C(=O)Nc1c(C)cccc1C	CID:175805	phase I
BRD-A37704979	CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1	CID:176155	phase I
BRD-K61177364	CCCN(CC1CC1)c1nc(C)nc(Nc2c(Cl)cc(Cl)cc2Cl)c1Cl	CID:176157	phase I
BRD-K59184148	Cn1cc(C2=C(C(=O)NC2=O)c2ccc(Cl)cc2Cl)c2ccccc12	CID:176158	phase I
BRD-K79404599	Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12	CID:176167	phase I
BRD-K19605405	Nc1nc(NCCc2ccc(O)cc2)nc2nc(nn12)-c1ccco1	CID:176407	phase I
BRD-K81225797	Nc1nc2n(CCc3ccccc3)ncc2c2nc(nn12)-c1ccco1	CID:176408	phase I
BRD-K70401845	COCCOc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCOC	CID:176870	phase I
BRD-K05906022	CC1(C)O[C@H]2CC(=O)OC[C@@]23[C@H]1CC(=O)[C@]4(C)[C@@H]3CC[C@@]5(C)[C@@H](OC(=O)[C@H]6O[C@]654)c7ccoc7	CID:179651	phase I
BRD-K58930050	C[C@]12N[C@H](Cc3ccccc13)c1ccccc21	CID:180081	phase I
BRD-K68075732	CC(C)NC[C@@H](O)COc1ccc(CC(N)=O)cc1	CID:180559	phase I
BRD-K18812295	O=C1C=CC(=O)c2c1ccc3c2ccc4ccccc43	CID:180933	phase I
BRD-K46836114	Oc1ccc(cc1)c2cc(=O)c3cc(O)ccc3o2	CID:182362	phase I
BRD-A17453586	O=C1CC2(CCCC2)CC(=O)N1CCCCNCC1COc2ccccc2O1	CID:182585	phase I
BRD-K01868942	COc1cc(N)c(Cl)cc1C(=O)OCCCN1CCCCC1	CID:182593	phase I
BRD-K20995441	CN([C@@H]1CCCC[C@@H]1N1CCCC1)C(=O)c1ccc(Cl)c(Cl)c1	CID:183470	phase I
BRD-K46142322	CCCCN1CCC(CCC(=O)c2cc(Cl)c(N)cc2OC)CC1	CID:183782	phase I
BRD-K09767179	NC(=O)c1nc(=O)[nH]c(=O)[nH]1	CID:188244	phase I
BRD-K36864847	CN(C)CCN(C)CCc1ccc(Cl)c(Cl)c1	CID:188914	phase I
BRD-K95767742	COc1cc2[nH]cc(CCNC(C)=O)c2cc1OC	CID:189748	phase I
BRD-K72015216	Cc1ccc2c(CCN)c[nH]c2c1	CID:190006	phase I
BRD-K56621596	NCCc1ccc(O)c(O)c1O	CID:193386	phase I
BRD-K36651625	C=CC(=O)N1CCN(CC1)C(=O)C=C	CID:193422	phase I
BRD-A04332542	CC(=O)NCC(O)c1ccc(O)cc1	CID:193691	phase I
BRD-A15530910	CC(C)OC(=O)c1cc2c(OCC(O)CNC(C)(C)C)cccc2[nH]1	CID:193949	phase I
BRD-A42264566	CCOc1cc(ccc1O)C(O)CO	CID:194138	phase I
BRD-K19309090	C(CN1CCOCC1)Nc1cc2CCCc3ccccc3-c2nn1	CID:195165	phase I
BRD-A29322418	C[C@]12CCC3C(C=CC4=CC(=O)CC[C@]34C)C1CC[C@@]2(O)CCC(O)=O	CID:195915	phase I
BRD-A60294240	CCOC1O[C@H]([C@@H](COCc2ccccc2)OCc2ccccc2)[C@H](OCc2ccccc2)[C@H]1O	CID:196122	phase I
BRD-K30990140	COc1ccc(cc1)-c1nc(sc1-c1ccc(OC)cc1)C(=O)N1CCN(C)CC1	CID:196841	phase I
BRD-K55703048	CN1CCc2c(C1)c1cc(C)ccc1n2CCc1ccc(C)nc1	CID:197033	phase I
BRD-A22707317	CC#CCOC(=O)c1c(C)nc2sc3CC(O)CCc3c2c1N	CID:197690	phase I
BRD-A34578416	COC(C(Oc1nc(C)cc(C)n1)C(=O)O)(c2ccccc2)c3ccccc3	CID:197712	phase I
BRD-K32828673	CN1Cc2c3OCOc3ccc2[C@H]4[C@@H](O)Cc5cc6OCOc6cc5[C@H]41	CID:197810	phase I
BRD-K02715688	COc1ccc2[C@H](OC(=O)c2c1OC)[C@@H]1N(C)CCc2cc3OCOc3cc12	CID:197835	phase I
BRD-K81029756	COc1ccc(cc1)[C@H]2Sc3ccccc3N(CCN(C)C)C(=O)[C@H]2OC(=O)C	CID:198107	phase I
BRD-K67680372	OC(=O)C1=CCCN(CCOC(c2ccc(cc2)C(F)(F)F)c2ccc(cc2)C(F)(F)F)C1	CID:198693	phase I
BRD-K19216856	Oc1cc(O)c2C[C@@H](OC(=O)c3cc(O)c(O)c(O)c3)[C@@H](Oc2c1)c4cc(O)c(O)c(O)c4	CID:199472	phase I
BRD-K88365400	NCCC[C@H](N)CC(=O)N[C@H]1CNC(=O)[C@@H](NC(=O)C(NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC1=O)=CNC(N)=O)[C@H]1C[C@H](O)N=C(N)N1	CID:200244	phase I
BRD-K74176882	OC(=O)c1ccccc1Nc2ccc(cc2)[N+](=O)[O-]	CID:201986	phase I
BRD-K38310698	CO[C@H]1C[C@H](O[C@H]2[C@H](C)[C@@H](O[C@@H]3O[C@H](C)C[C@@H]([C@H]3OC(=O)C)N(C)C)[C@@H](C)C[C@@]4(CO4)C(=O)[C@H](C)[C@@H](OC(=O)C)[C@@H](C)[C@@H](C)OC(=O)[C@@H]2C)O[C@@H](C)[C@@H]1OC(=O)C	CID:202225	phase I
BRD-A65797496	CN1[C@H]2CC[C@@H]1CC(C2)OC1c2ccccc2CCc2ccccc12	CID:203911	phase I
BRD-K19687926	CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1	CID:208908	phase I
BRD-K77286328	C1CCC(CC1)Nc2nc(Nc3ccc(cc3)N4CCOCC4)nc5[nH]cnc25	CID:210332	phase I
BRD-K09887211	C1CCC(CC1)(N1CCOCC1)c1cccs1	CID:210739	phase I
BRD-K23984367	CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)ccn1	CID:216239	phase I
BRD-A24381660	CC1CCC[C@H](O)CCCCCc2cc(O)cc(O)c2C(=O)O1	CID:216284	phase I
BRD-A17883755	Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O	CID:216326	phase I
BRD-A12230535	COc1ccc(C2=NC(C(N2C(=O)N2CCNC(=O)C2)c2ccc(Cl)cc2)c2ccc(Cl)cc2)c(OC(C)C)c1	CID:216345	phase I
BRD-A56592690	CCC(C)SSc1ncc[nH]1	CID:219104	phase I
BRD-A96485169	CCOC(=O)C1CN(Cc2ccccc2)C(=O)C1=O	CID:219271	phase I
BRD-K74112339	ONC(=O)Cc1ccccc1	CID:220184	phase I
BRD-K43164539	C[C@H](CCC(O)=O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:221493	phase I
BRD-A83326220	Oc1ccc2C3c4cc(O)c(O)cc4CC3(O)COc2c1	CID:222515	phase I
BRD-K41170226	C[C@H](CCC(O)=O)[C@H]1CC[C@H]2[C@@H]3CC[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:222528	phase I
BRD-K43736954	C[C@@]12CC(=O)[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CC[C@]1(O)C(=O)CO	CID:222786	phase I
BRD-K04046242	C[C@@]12CC[C@H]3C(=CCc4cc(O)ccc34)[C@@H]2CCC1=O	CID:223368	phase I
BRD-K29173907	CC(=O)OCC(=O)[C@@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]12C	CID:224246	phase I
BRD-A93477898	OC(Cc1ccncc1)C(Cl)(Cl)Cl	CID:224859	phase I
BRD-A56245458	CC12CCC3C(CCC4=CC(=O)CCC34C)C2CCC1(O)C(=O)CO	CID:227112	phase I
BRD-K88679075	C[C@]1(O)CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@@]21C	CID:229021	phase I
BRD-K33308633	O=C1C=CC(=O)C2=C1C1c3ccccc3C2c2ccccc12	CID:230748	phase I
BRD-K67439147	Cc1cccc(C=Cc2ccccc2)n1	CID:235382	phase I
BRD-K47635719	C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)COC(=O)C	CID:236702	phase I
BRD-K99411983	COC1=C[C@H]2[C@H](C3=C2c4c(OC)c(OC)c(OC)cc4CC[C@@H]3NC(=O)C)C1=O	CID:244898	phase I
BRD-K56515112	C[C@H]1C[C@H]2[C@@H]3CC[C@H](C(=O)C)[C@@]3(C)C[C@H](O)[C@@H]2[C@@]4(C)CCC(=O)C=C14	CID:247839	phase I
BRD-A31180007	NC(Cc1ccc(O)cc1O)C(O)=O	CID:251462	phase I
BRD-K40853697	Cc1ccc(cc1)S(=O)(=O)OCC(=O)Nc1ccc(C(O)=O)c(O)c1	CID:252682	phase I
BRD-K64451768	c1cc(ccn1)-c1sc(c(c1-c1ccncc1)-c1ccncc1)-c1ccncc1	CID:253078	phase I
BRD-K91370081	COc1ccc(C[C@H]2NC[C@H](O)[C@H]2OC(C)=O)cc1	CID:253602	phase I
BRD-K38324426	Cc1ccc(cc1)S(=O)(=O)NC2CCCCCCC2	CID:260972	phase I
BRD-K68143200	OCCSC1=C(SCCO)C(=O)c2ccccc2C1=O	CID:262093	phase I
BRD-K66043364	COc1ccc2[C@@H](OC(=O)c2c1OC)[C@H]1N(C)CCc2cc3OCOc3c(OC)c12	CID:262535	phase I
BRD-K88378636	C[C@@H]([C@H]1CC[C@H]2[C@@H]3C[C@H]4O[C@]45[C@@H](O)C=CC(=O)[C@]5(C)[C@H]3CC[C@]12C)[C@H]6CC(=C(CO)C(=O)O6)C	CID:265237	phase I
BRD-A81585303	NC(=O)c1ncn(C2OC(CO)C(O)C2O)c1N	CID:266934	phase I
BRD-K28100108	CCOC(=O)c1c2C(=O)c3ccccc3C(=O)c2n4ccccc14	CID:273769	phase I
BRD-K89237706	COc1ccc2[C@H](OC(=O)c2c1OC)[C@@H]3N(C)CCc4cc5OCOc5c(OC)c34	CID:275196	phase I
BRD-K59637651	OC(=O)c1c(Br)c(Br)c(Br)c(Br)c1c2c3ccc(O)cc3oc4cc(=O)ccc24	CID:275510	phase I
BRD-A08877921	COC1=CC23CCCN3CCc4cc5OCOc5cc4C2C1O	CID:278679	phase I
BRD-K76674262	COC(=O)C[C@](O)(CCCC(C)(C)O)C(=O)O[C@H]1[C@H]2c3cc4OCOc4cc3CCN3CCC[C@]23C=C1OC	CID:285033	phase I
BRD-K11981252	OC(=O)CCC(=O)Nc1ccccc1C(=O)O	CID:287263	phase I
BRD-A42649439	Cn1nc(N)c2cn(C3OC(CO)C(O)C3O)c4ncnc1c24	CID:290486	phase I
BRD-K31841256	Cc1ccc(NC(=O)COc2ccc(Cl)cc2Cl)c(c1)[N+](=O)[O-]	CID:295425	phase I
BRD-K82135108	CN(NC(=O)CC(=O)NN(C)C(=S)c1ccccc1)C(=S)c1ccccc1	CID:300471	phase I
BRD-K37727696	COC(=O)CSc1nc2ccccc2[nH]1	CID:302929	phase I
BRD-K78633253	COC(=O)c1ccccc1NC(=O)c1ccc(F)cc1	CID:310557	phase I
BRD-K71731651	COc1cc(OC)c(NC(=O)Nc2cc(C)on2)cc1Cl	CID:311434	phase I
BRD-K87343924	COC[C@H]1OC(=O)c2coc3c2[C@@]1(C)C1=C([C@@H]2CCC(=O)[C@@]2(C)C[C@H]1OC(C)=O)C3=O	CID:312145	phase I
BRD-K15318909	OCC1(CO)N2CCC(CC2)C1=O	CID:322968	phase I
BRD-K20510412	Cc1ccc(cc1)C(=O)/N=c\2/cccc[nH]2	CID:327120	phase I
BRD-K96799727	NS(=O)(=O)C#Cc1ccccc1	CID:327653	phase I
BRD-A77050075	CC(C)(O)C(O)COc1c2occc2cc3ccc(=O)oc13	CID:328236	phase I
BRD-K36377456	CC(C)(O)[C@@H]1Cc2cc3ccc(=O)oc3cc2O1	CID:334704	phase I
BRD-K89225759	COc1ccc2c(=O)c(coc2c1)c3cc4OCOc4cc3OC	CID:343083	phase I
BRD-K81925089	CCCN(CCC)c1nc(N)c2ccccc2n1	CID:345945	phase I
BRD-K45845523	COc1ccc(CC(O)=O)c(OC)c1	CID:350555	phase I
BRD-K63178889	COc1ccc2Nc3cc(Cl)ccc3Sc2c1	CID:350929	phase I
BRD-K92683369	Cn1c(cc(=O)c2ccccc12)c3ccc4OCOc4c3	CID:353825	phase I
BRD-A82371568	Nc1nc(Cl)nc2n(cnc12)C3OC(CO)C(O)C3F	CID:354624	phase I
BRD-K94841585	OC(=O)c1cc(O)c2C(=O)c3c(O)cc(O)cc3C(=O)c2c1	CID:361510	phase I
BRD-K63587518	COc1ccc(cc1)S(=O)(=O)N(C)CC(=O)O	CID:362743	phase I
BRD-A95445494	Oc1ccc2C3Oc4cc5OCOc5cc4C3COc2c1	CID:363863	phase I
BRD-K63151507	Cn1cnnc1Sc1c(ncn1C)[N+]([O-])=O	CID:364622	phase I
BRD-K37392901	Cc1ccc(C=C2CNCC(=Cc3ccc(C)cc3)C2=O)cc1	CID:365287	phase I
BRD-K53597484	CO[C@@H]1[C@@H](CC[C@]2(CO2)[C@H]1[C@@]1(C)O[C@@H]1CC=C(C)C)OC(=O)NC(=O)CCl	CID:369976	phase I
BRD-K83691318	c1ccc2[nH]c(nc2c1)c3nc4ccccc4s3	CID:373878	phase I
BRD-K00317371	OCc1ccc(s1)-c1ccc(o1)-c1ccc(CO)s1	CID:374536	phase I
BRD-A30590053	O=C(NCCCN1CCCCCC1)C(C1CCCCC1)c1ccccc1	CID:378811	phase I
BRD-K03109492	ClC1=C(NCCN2CCOCC2)C(=O)c2ncccc2C1=O	CID:379077	phase I
BRD-A74907996	Oc1ccc(cc1)C2COc3cc(O)ccc3C2	CID:382975	phase I
BRD-K95885906	COc1ccc(cc1OC)-c1oc2cc(OC)c(OC)c(OC)c2c(=O)c1OC	CID:386331	phase I
BRD-K88510285	CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnccn1)B(O)O	CID:387447	phase I
BRD-K51485625	CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@H](C[C@H](O)[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1	CID:392622	phase I
BRD-K37618799	Clc1ccc2nc(NC(=O)Cc3ccccc3)n3nc(nc3c2c1)-c1ccco1	CID:393595	phase I
BRD-K75532464	CSCC[C@H](NC(=O)c1ccc(NC[C@@H](N)CS)cc1-c1ccccc1)C(O)=O	CID:395754	phase I
BRD-K35553576	BrCC(=O)NCCc1c[nH]c2ccccc12	CID:399698	phase I
BRD-A80213327	CCN(CC)CCCC(C)Nc1nc(C)cc(Nc2ccc3nc(C)cc(N)c3c2)n1	CID:409805	phase I
BRD-K25701726	C[N+](C)(C)CC(=O)c1ccc(O)c(O)c1	CID:412800	phase I
BRD-A13982089	C[N+](C)(C)CC(O)c1ccc(O)c(O)c1	CID:414684	phase I
BRD-A81795050	CCN(CC)CCOC1CCC2(C)C3CCC4(C)C(CCC4=O)C3CC=C2C1	CID:415541	phase I
BRD-K54906270	COc1ccc2[nH]c3C(=NCCc3c2c1)C	CID:417052	phase I
BRD-K09485525	CN(C)c1ccccc1CN1CCCN(Cc2ccccc2N(C)C)C1c1ccncc1	CID:421610	phase I
BRD-K08713111	NCCc1ccc(OCc2ccccc2)c(OCc3ccccc3)c1	CID:423869	phase I
BRD-K31268420	Nc1nnc2[nH]c3ccccc3nc12	CID:438981	phase I
BRD-K35708212	C[C@@H]1O[C@@H](O[C@H]2C[C@@H](O)[C@]3(CO)[C@H]4[C@H](O)C[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)C6=CC(=O)OC6)[C@H](O)[C@H](O)[C@H]1O	CID:439501	phase I
BRD-K64614248	OC[C@H]1O[C@@H](Oc2ccccc2CO)[C@H](O)[C@@H](O)[C@@H]1O	CID:439503	phase I
BRD-K19107160	CC[C@H]1OC(=O)C[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)[C@@H](O[C@H]3C[C@@](C)(O)[C@@H](O)[C@H](C)O3)[C@@H]([C@H]2O)N(C)C)[C@@H](CC=O)C[C@@H](C)C(=O)C=CC(=C[C@@H]1CO[C@@H]4O[C@H](C)[C@@H](O)[C@@H](OC)[C@H]4OC)C	CID:439504	phase I
BRD-A79067928	COc1cc(cc(OC)c1O)[C@H]2[C@@H]3[C@H](COC3=O)[C@H](OC4OC5COC(C)OC5C(O)C4O)c6cc7OCOc7cc26	CID:439525	phase I
BRD-K36007650	COc1ccc(C[C@H](N)C(=O)N[C@H]2[C@@H](O)[C@@H](O[C@@H]2CO)n3cnc4c(ncnc34)N(C)C)cc1	CID:439530	phase I
BRD-K94649603	O[C@@H]1[C@H](Oc2cc(O)cc(O)c2C1=O)c1ccc(O)c(O)c1	CID:439533	phase I
BRD-A80574334	OC(C(C(O)=O)C(=O)C(O)=O)C(O)=O	CID:439620	phase I
BRD-K62609077	COc1ccc2C[C@@H]3N(CCc4cc(OC)c(O)cc34)Cc2c1O	CID:439654	phase I
BRD-K01976263	N[C@@H](CCl)C(=O)O	CID:439772	phase I
BRD-K08037784	OC[C@H]1O[C@@H](Oc2ccc(O)cc2)[C@H](O)[C@@H](O)[C@@H]1O	CID:440936	phase I
BRD-K59632282	COc1ccc2nccc([C@H](O)[C@H]3C[C@@H]4CC[N@]3C[C@@H]4C=C)c2c1	CID:441074	phase I
BRD-K01612348	C[C@@H](O)[C@@H]1[C@H]2[C@@H](C)C(=C(N2C1=O)C(=O)O)S[C@@H]3CN[C@@H](C3)C(=O)N(C)C	CID:441130	phase I
BRD-K08273968	COc1cc(OC)c(Cl)c2O[C@]3([C@H](C)CC(=O)C=C3OC)C(=O)c12	CID:441140	phase I
BRD-K55375480	CC[C@]1(CC[C@@H](O1)[C@]2(C)CC[C@]3(C[C@H](O)[C@@H](C)[C@H](O3)[C@@H](C)[C@@H](OC)[C@H](C)C(=O)O)O2)[C@@H]4O[C@H](C[C@@H]4C)[C@H]5O[C@@](O)(CO)[C@H](C)C[C@@H]5C	CID:441145	phase I
BRD-K70976396	CO[C@]1(NC(=O)Cc2cccs2)[C@H]2SCC(COC(N)=O)=C(N2C1=O)C(O)=O	CID:441199	phase I
BRD-K09963420	CC(C)(C)NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2CN1C[C@@H](O)[C@H](Cc3ccccc3)NC(=O)[C@H](CC(=O)N)NC(=O)c4ccc5ccccc5n4	CID:441243	phase I
BRD-A28746609	CC(=O)O[C@@H]1C2=C(C)[C@H](C[C@@](O)([C@@H](OC(=O)c3ccccc3)C3[C@@]4(CO[C@@H]4C[C@H](O)[C@@]3(C)C1=O)OC(C)=O)C2(C)C)OC(=O)[C@H](O)[C@@H](NC(=O)c1ccccc1)c1ccccc1	CID:441276	phase I
BRD-K44779798	OCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO	CID:441314	phase I
BRD-K65377893	CC(=O)OCC1=C(N2[C@H](SC1)[C@H](N)C2=O)C(O)=O	CID:441328	phase I
BRD-K60640630	C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]2(C)[C@@]1(OC(=O)c5ccco5)C(=O)CCl	CID:441336	phase I
BRD-K86204871	CC(C)N1CCN(CC1)c1ccc(OC[C@H]2CO[C@@](Cn3cncn3)(O2)c2ccc(Cl)cc2Cl)cc1	CID:441383	phase I
BRD-K66876909	CC(=O)NC[C@H]1CN(C(=O)O1)c1ccc(N2CCOCC2)c(F)c1	CID:441401	phase I
BRD-K71003802	CN1CCC2=C[C@H](O)[C@H]3OC(=O)c4cc5OCOc5cc4[C@H]3[C@H]12	CID:441594	phase I
BRD-A88282067	CCN1C[C@]2(COC)CC[C@H](OC)[C@]3([C@@H]4C[C@H]5[C@H](OC)[C@@H]4[C@@]6(C[C@@H]5OC)OCO[C@]76[C@@H](O)[C@@H]32)C17	CID:441724	phase I
BRD-A99177642	CCN1C[C@]2(C)CC[C@H](OC)[C@@]34[C@@H]2[C@H](OC(=O)C)[C@@]5(OCO[C@]65C[C@H](OC)[C@H]7C[C@]4(O)[C@@H]6[C@H]7OC)C13	CID:441728	phase I
BRD-A54445976	CCN1C[C@]2(C)CC[C@H](O)[C@]3([C@@H]2C[C@H]4C13)[C@@H]5C[C@H](O)[C@H]6C[C@]45[C@H](O)C6=C	CID:441749	phase I
BRD-K08486545	CO[C@H]1C[C@H](O[C@H]2CC[C@]3(C=O)[C@H]4CC[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)C6=CC(=O)OC6)O[C@H](C)[C@H]1O	CID:441853	phase I
BRD-K07476834	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)O[C@H]1CC[C@]2(C=O)[C@H]3CC[C@]4(C)[C@H](CC[C@]4(O)[C@@H]3CC[C@]2(O)C1)C1=CC(=O)OC1	CID:441860	phase I
BRD-K67265981	CC(C)c1cc2[C@@H]3C[C@H]4C(C)(C)CCC[C@]4(C(=O)O3)c2c(O)c1O	CID:442009	phase I
BRD-K68077509	COc1cc2N3[C@H]4[C@H]5[C@H]6C[C@@H]7N(CC[C@@]74c2cc1OC)CC6=CCO[C@H]5CC3=O	CID:442021	phase I
BRD-K63945320	CC(C)CC(=O)O[C@@H]1[C@H](OC(=O)C)c2c(OC1(C)C)ccc3ccc(=O)oc23	CID:442128	phase I
BRD-K80348542	CC[C@H]1CN2CCc3cc(OC)c(OC)cc3[C@@H]2C[C@@H]1C[C@H]4NCCc5cc(O)c(OC)cc45	CID:442195	phase I
BRD-K89853519	O[C@H]1Cc2ccc(O)cc2O[C@@H]1c3ccc(O)c(O)c3	CID:442397	phase I
BRD-K02953697	C[C@@H]1O[C@@H](O[C@@H]2[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]2Oc3cc(O)c4C(=O)C[C@H](Oc4c3)c5ccc(O)cc5)[C@H](O)[C@H](O)[C@H]1O	CID:442428	phase I
BRD-K39944607	C[C@@H]1Cc2c(Cl)cc(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)c(O)c2C(=O)O1	CID:442530	phase I
BRD-A61856038	OC[C@H]1O[C@@H](Oc2ccccc2COC(=O)C3(O)C=CCCC3=O)[C@H](OC(=O)c4ccccc4)[C@@H](O)[C@@H]1O	CID:442544	phase I
BRD-K26117720	CCCCC[C@H](O)CC(=O)CCc1ccc(O)c(OC)c1	CID:442793	phase I
BRD-K49071277	O=C1O[C@@]23C[C@@H](C=CC2=C1)N1CCCC[C@H]31	CID:442872	phase I
BRD-K13819402	C1CN2Cc3ccccc3N=C2C1	CID:442894	phase I
BRD-A99571536	COc1c2CC(Oc2nc3ccccc13)C(C)(O)CO	CID:442897	phase I
BRD-A06390036	CC[C@H]1CN2CCC1C[C@@H]2[C@@H](O)c1ccnc2ccc(OC)cc12	CID:442912	phase I
BRD-K58938839	C[C@@H]1[C@@H]2NC[C@@H](C)C[C@H]2O[C@@]31CC[C@H]4[C@@H]5CC=C6C[C@@H](O)CC[C@]6(C)[C@H]5CC4=C3C	CID:442972	phase I
BRD-K35923252	CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)C)C=O	CID:443118	phase I
BRD-K31792052	Cc1ccc(cc1)c2cn3c4CCCCc4sc3n2	CID:443278	phase I
BRD-K24473282	CC(C)NC[C@H](O)c1ccc(O)c(O)c1	CID:443372	phase I
BRD-K31238592	CN1C(=O)[C@@H](NC(=O)c2cc3ccccc3[nH]2)N=C(c4ccccc4)c5ccccc15	CID:443375	phase I
BRD-K14807180	CSc1cc2CCN(C(=O)Nc3cccnc3)c2cc1C(F)(F)F	CID:443389	phase I
BRD-A76093993	CC1(C)Oc2ccc(C#N)cc2C(C1O)N3CCCC3=O	CID:443423	phase I
BRD-K54316499	CC(C)N(CC[C@H](c1ccccc1)c1cc(C)ccc1O)C(C)C	CID:443879	phase I
BRD-K81709173	CC1(C)O[C@@H]2C[C@H]3[C@@H]4CCC5=CC(=O)CC[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CCl	CID:443943	phase I
BRD-A45543382	CN(C(C)=O)c1c(I)c(NC(C)=O)c(I)c(C(=O)N[C@H]2C(O)O[C@H](CO)[C@@H](O)[C@@H]2O)c1I	CID:443944	phase I
BRD-K51677086	CCOC(=O)CCC(=O)O[C@H]1[C@H](O[C@@H]2[C@@H](C)[C@H](O[C@H]3C[C@@](C)(OC)[C@@H](O)[C@H](C)O3)[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@]2(C)O)O[C@H](C)C[C@@H]1N(C)C	CID:443953	phase I
BRD-K53318339	CCOC(=O)C1=C[C@]2(CC)CCCN3CCc4c([C@H]23)n1c1ccccc41	CID:443955	phase I
BRD-K86284654	CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2C(CCC[C@]12C)=CC=C1C[C@@H](O)C[C@H](O)C1=C	CID:443990	phase I
BRD-K10467831	C[C@@H]1CC2=C(CCC(=O)C2)[C@H]3CC[C@@]4(C)[C@@H](CC[C@@]4(O)C#C)[C@H]13	CID:444008	phase I
BRD-K39983086	CCOC(=O)O[C@@]1(CC[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@]12C)C(=O)OCCl	CID:444025	phase I
BRD-K95773607	NC(=O)C([C@@H]1CCN(CCc2ccc3OCCc3c2)C1)(c1ccccc1)c1ccccc1	CID:444031	phase I
BRD-K62310379	CCC(=O)O[C@@]1([C@H](C)C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]12C)C(=O)SCF	CID:444036	phase I
BRD-K44276885	C[C@H]1O[C@H](O[C@@H]2[C@@H](CO)O[C@H](O[C@@H]3[C@@H](CO)O[C@@H](O)[C@H](O)[C@H]3O)[C@H](O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1N[C@H]1C=C(CO)[C@@H](O)[C@H](O)[C@H]1O	CID:444254	phase I
BRD-K68202742	C[C@H](\C=C(C)\C=C\C(=O)NO)C(=O)c1ccc(cc1)N(C)C	CID:444732	phase I
BRD-K71879491	CC(/C=C/C1=C(C)CCCC1(C)C)=C\C=C\C(C)=C\C(O)=O	CID:444795	phase I
BRD-K24656285	CC(=CCC/C(=C/CC/C(=C/CO)/C)/C)C	CID:445070	phase I
BRD-K80738081	Oc1ccc(cc1)\C=C\c1cc(O)cc(O)c1	CID:445154	phase I
BRD-K22429181	CC(\C=C\C=C(C)\C=C\C1=C(C)CCCC1(C)C)=C/CO	CID:445354	phase I
BRD-K39965020	CC\C=C/C\C=C/C\C=C/C\C=C/C\C=C/C\C=C/CCC(O)=O	CID:445580	phase I
BRD-K70131229	N[C@H]1[C@@H](O)O[C@H](CO)[C@@H](O)[C@@H]1O	CID:445621	phase I
BRD-K69608737	CO[C@@H]1C[C@@H](CC[C@H]1O)\C=C(/C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@]2(O)O[C@@H]([C@H](C[C@H]2C)OC)[C@H](C[C@@H](C)C\C(C)=C\[C@@H](CC=C)C(=O)C[C@H](O)[C@H]1C)OC	CID:445643	phase I
BRD-A57226833	CC(C)=CCC\C(C)=C\CC\C(C)=C\COP(O)(=O)OP(O)(O)=O	CID:445713	phase I
BRD-K66296774	CC(C)n1c(\C=C\[C@@H](O)C[C@@H](O)CC(O)=O)c(-c2ccc(F)cc2)c2ccccc12	CID:446155	phase I
BRD-K81169441	COCc1c(nc(C(C)C)c(/C=C/[C@@H](O)C[C@@H](O)CC(=O)O)c1c2ccc(F)cc2)C(C)C	CID:446156	phase I
BRD-K82941592	CC(C)c1nc(nc(-c2ccc(F)cc2)c1\C=C\[C@@H](O)C[C@@H](O)CC(O)=O)N(C)S(C)(=O)=O	CID:446157	phase I
BRD-K47192521	CC\C=C/C\C=C/C\C=C/C\C=C/C\C=C/CCCC(O)=O	CID:446284	phase I
BRD-K67097529	CCOP(=O)(OCC)C(=Cc1cc(c(O)c(c1)C(C)(C)C)C(C)(C)C)P(=O)(OCC)OCC	CID:446313	phase I
BRD-K69023402	CCCCCCCC(=O)O[C@@H]1[C@@H](OC(=O)/C(=C\C)/C)C(=C2[C@@H]3OC(=O)[C@@](C)(O)[C@@]3(O)[C@H](C[C@](C)(OC(=O)C)[C@@H]12)OC(=O)CCC)C	CID:446378	phase I
BRD-K63750851	COc1c(C)c2COC(=O)c2c(O)c1C\C=C(/C)CCC(O)=O	CID:446541	phase I
BRD-K15262564	C[C@H](O)[C@H](C)[C@@H]1O[C@H]1C[C@H]1CO[C@@H](C\C(C)=C\C(=O)OCCCCCCCCC(O)=O)[C@H](O)[C@@H]1O	CID:446596	phase I
BRD-A32065788	CCCCCCCCCCCCCCCCCCCC(=O)O[C@H](COC(=O)CCCCCCCCCCCCCC)COP(O)(=O)OCCN	CID:446872	phase I
BRD-K59753853	OC(=O)CCc1c([nH]c2cc(Cl)cc(Cl)c12)C(=O)O	CID:446916	phase I
BRD-K74501079	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O	CID:447043	phase I
BRD-A14999564	CC(C)=CCC\C(C)=C\CC\C(C)=C\CC\C(C)=C\COP(O)(=O)OP(O)(O)=O	CID:447277	phase I
BRD-K34170797	COC(=O)C=Cc1cccc(c1)N(Cc2ccc(cc2)c3ccc(cc3)N(C)C)C(=O)C4CCCCC4	CID:447713	phase I
BRD-K33818169	OC(=O)Cc1cccc(OCCCN(CC(c2ccccc2)c2ccccc2)Cc2cccc(c2Cl)C(F)(F)F)c1	CID:447905	phase I
BRD-K23383398	OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F	CID:447912	phase I
BRD-K06234293	c1[nH]nc(c1-c1ccnc2ccccc12)-c1ccccn1	CID:447966	phase I
BRD-K48935217	C[C@H]1CCC[C@@]2(C)O[C@H]2C[C@H](OC(=O)C[C@H](O)C(C)(C)C(=O)[C@H](C)[C@H]1O)C(\C)=C\c1csc(C)n1	CID:448013	phase I
BRD-K67860401	COc1ccc(CNC(=O)Nc2ncc(s2)[N+]([O-])=O)cc1	CID:448014	phase I
BRD-K75516118	COc1ccc(cc1OC1CCCC1)[C@@H]1CNC(=O)C1	CID:448055	phase I
BRD-K45330754	CC\C(c1ccc(O)cc1)=C(\CC)c1ccc(O)cc1	CID:448537	phase I
BRD-K71823332	C[C@H]1CCC[C@H]2O[C@H]2C[C@H](OC(=O)C[C@H](O)C(C)(C)C(=O)[C@H](C)[C@H]1O)C(\C)=C\c1csc(C)n1	CID:448799	phase I
BRD-K93658967	CCCCc1c([nH]c2nccnc12)c3ccc(O)cc3	CID:448912	phase I
BRD-K41564320	CC(C)[C@H](CO)Nc1nc(Nc2ccc(C(O)=O)c(Cl)c2)c2ncn(C(C)C)c2n1	CID:448991	phase I
BRD-K35483542	C/C(=C/C=C/C(=C/C(=O)O)/C)/C=C/C1=C(C)CCCC1(C)C	CID:449171	phase I
BRD-K45834949	C[C@@]12CCC[C@H]1[C@@H]1CC[C@H]3C[C@H](O)CC[C@]3(C)[C@H]1CC2	CID:449196	phase I
BRD-K53226837	N[C@H]1CONC1=O	CID:449215	phase I
BRD-K27737647	Brc1ccc(\C=C\CNCCNS(=O)(=O)c2cccc3cnccc23)cc1	CID:449241	phase I
BRD-K04210847	CC/C(=C(\c1ccc(O)cc1)/c2ccc(OCCN(C)C)cc2)/c3ccccc3	CID:449459	phase I
BRD-K79254416	Nc1ncn([C@H]2C[C@H](O)[C@@H](CO)O2)c(=O)n1	CID:451668	phase I
BRD-K57954781	Nc1ncnc2n(cnc12)[C@@H]3O[C@H](CO)C[C@@H]3O	CID:451875	phase I
BRD-K91145395	C[C@@H]1C[C@]2(OC(=O)C)[C@H]([C@@H]3C=C(CO)C[C@@]4(O)[C@@H](C=C(C)C4=O)[C@@]13O)C2(C)C	CID:454217	phase I
BRD-K70158168	CC(C)(C)NC(=O)[C@@H]1C[C@@H]2CCCC[C@H]2CN1C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)c1ccc2ccccc2n1	CID:454469	phase I
BRD-K29113274	CC(=O)N1CCN(CC1)c1ccc(OC[C@H]2CO[C@@](Cn3ccnc3)(O2)c2ccc(Cl)cc2Cl)cc1	CID:456201	phase I
BRD-K50836978	CC(C)[C@H](CO)Nc1nc(Nc2cccc(Cl)c2)c2ncn(C(C)C)c2n1	CID:456214	phase I
BRD-K76018977	CON=C(C(=O)N[C@H]1[C@H]2SCC(=C(N2C1=O)C(=O)O)COC(=O)C)c3csc(N)n3	CID:456256	phase I
BRD-K70578146	CC(C)[C@H]1NC(=O)[C@@H](NC(=O)c2ccc(C)c3oc4c(C)c(=O)c(N)c(C(=O)N[C@H]5[C@@H](C)OC(=O)[C@H](C(C)C)N(C)C(=O)CN(C)C(=O)[C@@H]6CCCN6C(=O)[C@H](NC5=O)C(C)C)c4nc23)[C@@H](C)OC(=O)[C@H](C(C)C)N(C)C(=O)CN(C)C(=O)[C@@H]2CCCN2C1=O	CID:457193	phase I
BRD-K16925374	CC(=O)Nc1ccc(NS(=O)(=O)C)cc1	CID:458876	phase I
BRD-K70751730	OC(=O)c1ccc(O)c2ncccc12	CID:459617	phase I
BRD-K80622725	Cc1nn(C)c2nc(=O)n(C)c(=O)c2n1	CID:460747	phase I
BRD-K60230970	CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C=O	CID:462382	phase I
BRD-K15891719	C[C@H](Cn1cnc2c(N)ncnc12)OCP(O)(O)=O	CID:464205	phase I
BRD-A63989068	CCC(C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]2CCCCN2C1=O	CID:467801	phase I
BRD-K54556307	CC[C@H](CO)NCCN[C@H](CC)CO	CID:470071	phase I
BRD-K06426971	Cc1nc2c(s1)C(=O)C=C(Nc1ccc(C)cc1)C2=O	CID:481747	phase I
BRD-A79314293	CC(=O)OCC1=C(N2C(SC1)[C@H](N)C2=O)C(O)=O	CID:483168	phase I
BRD-A04352665	CC(C)c1nnc(C)n1C1CC2CCC(C1)N2CC[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1	CID:483407	phase I
BRD-K92760278	Cc1cc2nc3c(nc(=O)[nH]c3=O)n(C[C@H](O)[C@H](O)[C@H](O)CO)c2cc1C	CID:493570	phase I
BRD-A32164164	CCN1CC2(COC(=O)c3ccccc3N4C(=O)CC(C)C4=O)CCC(OC)C5(C6CC7C(OC)C6C(O)(CC7OC)C8(O)C(OC)C52)C18	CID:494471	phase I
BRD-K86509404	Cn1cnc2nc(NCCO)nc(NCc3ccccc3)c12	CID:512292	phase I
BRD-K43014159	N[C@@H](Cc1ccc(OS(O)(=O)=O)cc1)C(O)=O	CID:514186	phase I
BRD-K22337096	N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)O	CID:515709	phase I
BRD-K62902879	COc1cc(ccc1OC(=O)C)C2=CCN(CC2)C(=O)C	CID:540740	phase I
BRD-A25170757	CNCC(O)c1cc(OCc2ccccc2)c(OCc3ccccc3)cc1F	CID:541830	phase I
BRD-A84524947	CNCC(O)c1cc(F)c(OCc2ccccc2)c(OCc3ccccc3)c1F	CID:541832	phase I
BRD-K60571253	CN(CC#CCN1CCCC1)C(=O)c2cccc(Cl)c2	CID:551033	phase I
BRD-A55609290	COc1ccc(C(O)CNC(C)C)c(F)c1OC	CID:551704	phase I
BRD-A72069525	COc1cc(cc(F)c1OC)C(O)CNC(C)C	CID:551940	phase I
BRD-K89486464	Oc1ccc(cc1O)C2=CCNCC2	CID:557589	phase I
BRD-K48576794	Cc1cc(NC(=O)CCl)no1	CID:566661	phase I
BRD-K48199208	CN(CC#CCN1CCC(O)CC1)C(=O)C	CID:567598	phase I
BRD-K11558771	Cc1cc(Cl)ccc1OCCCC(=O)NO	CID:568416	phase I
BRD-A98200599	OC1(NC(=O)c2ccccc2O1)c3ccccc3	CID:570188	phase I
BRD-K95118263	Nn1c(nc2ccccc2c1=O)C(=O)NCc3cccnc3	CID:572154	phase I
BRD-K81313552	OC(=O)CCC(=O)Nc1cccc(F)c1	CID:573894	phase I
BRD-K29668683	CN1CCN(CCc2ccc(Cl)c(Cl)c2)CC1	CID:574780	phase I
BRD-K71265179	Cc1ccc(cc1)C(=O)n2c3ccccc3c4ccccc24	CID:576989	phase I
BRD-K00878439	COc1ccc(CCNC(=O)C)cc1	CID:584258	phase I
BRD-A00150179	NC(Cc1c[nH]c2cccc(O)c12)C(O)=O	CID:589768	phase I
BRD-K74606027	OC(=O)CSc1c[nH]c2ccccc12	CID:590707	phase I
BRD-A76732176	COc1ccccc1CN2CC(CC2=O)C(=O)O	CID:590894	phase I
BRD-K49889622	COc1ccc(CCNC(C)=O)cc1O	CID:591256	phase I
BRD-K31477169	COC(=O)c1c(C)cc(OC)cc1O	CID:596344	phase I
BRD-A19918940	CC1(C)Oc2ccc3ccc(=O)oc3c2CC1O	CID:600670	phase I
BRD-K79857601	COc1cc(N=c2ssnc2Cl)c(OC)cc1Cl	CID:602897	phase I
BRD-K66896231	Nc1c2CCCc2nc2CCCCc12	CID:604519	phase I
BRD-A68890828	COc1ccc2N(C)C(=O)C(C)(CCN)c2c1	CID:605729	phase I
BRD-K93188295	COc1ccccc1N1CCN(CCN2C(=O)c3ccccc3C(C)(C)C2=O)CC1	CID:609483	phase I
BRD-K77508012	Cc1nn(C)c(C)c1Nc2nc(N)n[nH]2	CID:610065	phase I
BRD-K50133271	Cc1c(Cl)cccc1Nc1ccccc1C(O)=O	CID:610479	phase I
BRD-K93541117	CCCCCCN1CCN(CC1)c2cccc(Cl)c2	CID:610696	phase I
BRD-K70052774	NCCN1CCN(CC(=O)N2c3ccccc3C(=O)Nc4cccnc24)CC1	CID:611101	phase I
BRD-K57930080	COc1ccc(cc1OC)c2ccncc2	CID:612061	phase I
BRD-A91477472	CC1CCc2c(O)c3c(=O)cc(C)oc3cc2OC1	CID:612556	phase I
BRD-K89329876	CC(C)(C)c1ccc2cc(C#N)c(C#N)cc2c1	CID:613000	phase I
BRD-K03371390	COc1cc2c3CCNC(=O)c3[nH]c2cc1F	CID:616433	phase I
BRD-K43009525	N1c2ccccc2Nc3nc4ccccc4nc13	CID:616479	phase I
BRD-K43796186	C(Nc1ncnc2ccccc12)c3ccccc3	CID:616573	phase I
BRD-K97629076	Clc1ccc2Nc3cscc3C(=O)Nc2c1	CID:619526	phase I
BRD-K86456986	COc1c(F)cc2[nH]c3C(=O)NCCc3c2c1F	CID:619865	phase I
BRD-K52696183	CNCCCN1c2ccccc2CCc2ccc(Cl)cc12	CID:622606	phase I
BRD-A23226398	CC(=O)OC1CCC2C3CCc4cc(O)ccc4C3CCC12C	CID:628698	phase I
BRD-K32584078	OC(=O)c1ccc2nc(c3ccccc3)c(nc2c1)c4ccccc4	CID:629852	phase I
BRD-A98670841	CCC1(CCCN2CCC3(C4CC1)c5ccc(OC)c(O)c5N4C(=O)C)C23	CID:632854	phase I
BRD-K12765235	CC1(C)[C@H](CC[C@@]2(C)[C@H]1CC[C@]3(C)[C@@H]2C(=O)C=C4[C@@H]5C[C@](C)(CC[C@]5(C)CC[C@]43C)C(=O)O)OC(=O)CCC(=O)O	CID:636403	phase I
BRD-A42270467	COc1ccc2[nH]c(nc2n1)S(=O)Cc1ncc(C)c(OC)c1C	CID:636411	phase I
BRD-K10098805	COc1ccc(/C=C/c2cc(O)cc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c2)cc1O	CID:637213	phase I
BRD-K49060658	COc1ccc(cc1)\C=C\C	CID:637563	phase I
BRD-K03568070	CC(=CCC/C(=C/CO)/C)C	CID:637566	phase I
BRD-K24132293	COc1cc(/C=C/C(=O)N2CCC=CC2=O)cc(OC)c1OC	CID:637858	phase I
BRD-K59522102	O=C(\C=C\C=C\c1ccc2OCOc2c1)N1CCCCC1	CID:638024	phase I
BRD-K65331431	CC(=O)OC\C=C(C)\C=C\C=C(C)\C=C\C1=C(C)CCCC1(C)C	CID:638034	phase I
BRD-K33583600	Oc1ccc(cc1)\C=C\C(=O)c1ccc(O)cc1O	CID:638278	phase I
BRD-K77390737	COc1cc(O)c(CC=C(C)C)c(O)c1C(=O)/C=C/c2ccc(O)cc2	CID:639665	phase I
BRD-K36638830	C1CC[C@@H](NC1)c2cccnc2	CID:641266	phase I
BRD-K61559475	COc1cc(O)cc(O)c1C(=O)/C=C/c2ccccc2	CID:641785	phase I
BRD-K62353524	CCN(CC)c1ccc(C=NNC(=O)c2ccc(O)cc2)cc1	CID:644030	phase I
BRD-K93331255	NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSC[C@H](N)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N1)C(=O)NCC(N)=O	CID:644076	phase I
BRD-K93258693	[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc1ccccc1	CID:644213	phase I
BRD-K79090631	OCCCNc1cc(ccn1)c2ccnc(Nc3cccc(Cl)c3)n2	CID:644215	phase I
BRD-K81528515	Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F	CID:644241	phase I
BRD-K23875128	c1[nH]c2ccccc2c1c3ccncc3	CID:644354	phase I
BRD-A71657825	OC(=O)CCC(NS(=O)(=O)c1ccc(cc1)c2ccccc2)C(=O)O	CID:644601	phase I
BRD-K57019930	CCN(CC)S(=O)(=O)c1cccc2cc(C(=O)O)c(O)cc12	CID:645872	phase I
BRD-K34596778	CC=CCn1c(SCc2ccccc2)nc2n(C)c(=O)[nH]c(=O)c12	CID:646090	phase I
BRD-K56697208	CCCCCn1c(SCCc2ccccc2)nc3n(C)c(=O)[nH]c(=O)c13	CID:647508	phase I
BRD-A58482795	OC(CCN1CCOCC1)(C2CCCCC2)c3ccc(Cl)cc3	CID:650228	phase I
BRD-K44241590	COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:650361	phase I
BRD-A22514244	COc1ccc(cc1OC)c2nnn(CC(=O)N(C(C)C(=O)NC3CCCC3)C4CCCCC4)n2	CID:650573	phase I
BRD-K47448802	CCOC(=O)N1CCC(CC1)NCCNC(=O)c2ccccc2	CID:650899	phase I
BRD-K18587499	CCOC(=O)C1(CCN(Cc2cccc(c2)C(=O)O)CC1)c3ccccc3	CID:650919	phase I
BRD-K05326558	CCCn1c(SCC(=O)Nc2nc3CCCCc3s2)nc4n(C)c(=O)n(C)c(=O)c14	CID:653676	phase I
BRD-K81538844	Cc1cc2n(C)c3c(=O)n(Cc4ccccc4F)ncc3c2s1	CID:654376	phase I
BRD-K42841443	Oc1ccc(CNc2ccccc2F)c3cccnc13	CID:655278	phase I
BRD-K15640888	COc1ccc(cc1)S(=O)(=O)n2nc(OC(=O)c3ccccc3)cc2N	CID:655490	phase I
BRD-K46556543	C[C@]12CC[C@H]3[C@@H](C=CC4=CC(=O)CC[C@]34C)[C@@H]1CC[C@@]2(O)CCC(O)=O	CID:656615	phase I
BRD-K85383046	C[C@]1(Cc2cc(OCC(=O)O)c(Cl)c(Cl)c2C1=O)C3CCCC3	CID:656717	phase I
BRD-A83695761	CCS(=O)(=O)N(C)C1C(O)C(C)(C)Oc2ccc(C#N)cc12	CID:656731	phase I
BRD-K42748308	O=C1c2ccccc2C(Cc2ccncc2)(Cc2ccncc2)c2ccccc12	CID:656732	phase I
BRD-K32526544	CCn1c(=O)[nH]c2cc(Cl)c(Cl)cc12	CID:656765	phase I
BRD-K09295900	C[C@@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)C=C[C@]34C)[C@@H]2CC[C@]1(O)C(=O)COC(=O)CCC(=O)O	CID:656804	phase I
BRD-K66788707	Nc1nc(F)nc2n(cnc12)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O	CID:657237	phase I
BRD-K42635745	CCCCCCCCN[C@H](C)[C@@H](O)c1ccc(SC(C)C)cc1	CID:657255	phase I
BRD-K48168960	CCCc1cc(=O)[nH]c(=S)[nH]1	CID:657298	phase I
BRD-K14204120	CN\C(NCCSCc1ccc(CN(C)C)o1)=C\[N+]([O-])=O	CID:657345	phase I
BRD-A79226577	CN1[C@H]2CC[C@@H]1CC(C2)OC(=O)C1C=Nc2ccccc12	CID:657380	phase I
BRD-K14444135	CCc1c(C)[nH]c(=S)c(C#N)c1C	CID:658169	phase I
BRD-A77467113	Fc1ccc(cc1)C(=O)C(CN2CCOCC2)c3ccccc3	CID:659031	phase I
BRD-K92317137	O=S1(=O)Nc2c(ccc3cccnc23)-c4ccccc41	CID:659101	phase I
BRD-K14765469	O[C@@H]1CCCC[C@H]1N1CCC(CC1)c1ccccc1	CID:659840	phase I
BRD-K34968258	Cc1ccc(Cn2ncc3c(ncnc23)N4CCN(CC4)c5ccc(C)cc5)cc1	CID:661907	phase I
BRD-K15250199	Clc1ccc(CSc2nnc(o2)c3ccncc3)c(Cl)c1	CID:662619	phase I
BRD-K53833301	Clc1ccc(CSc2nnc(c3ccccn3)n2Cc4ccco4)c(Cl)c1	CID:662944	phase I
BRD-A76641868	CCN1CCN(CC1)c1nc2ccccc2nc1C(C#N)C(=O)OC1CCCCC1	CID:663281	phase I
BRD-K27484191	Brc1ccc(CSc2nnc(c3ccccn3)n2Cc4ccco4)cc1	CID:663290	phase I
BRD-K23935793	CN(C)c1oc(nc1C#N)c2ccc(OCc3ccc(Cl)cc3)cc2	CID:663459	phase I
BRD-K23217072	CC(Cl)=CCn1c(NCCc2ccccc2)nc2n(C)c(=O)n(C)c(=O)c12	CID:663872	phase I
BRD-K90826279	Cc1nc(SCc2nc3ccccc3[nH]2)c4oc5ccccc5c4n1	CID:664279	phase I
BRD-K85051645	O=C1CCCC2=C1C1(CCCC1)NC(Nc1nc3ccccc3o1)=N2	CID:664331	phase I
BRD-K05153001	CC(=O)C(C(=O)C)c1c(Cl)c(O)c(O)c2c(coc12)C(=O)c3ccccc3	CID:665013	phase I
BRD-K21640605	COc1ccccc1c2nnc(SCC(=O)c3ccc(O)c(O)c3)n2CC=C	CID:665093	phase I
BRD-K24598397	CC(C)(C)OC(=O)NCCc1nnc(o1)S(=O)(=O)Cc2ccc(Cl)cc2Cl	CID:665449	phase I
BRD-K87964538	Cc1cc(C)n(n1)c2nc(NCCCO)c3c4CCCCc4sc3n2	CID:665518	phase I
BRD-K73481389	CNC(=O)CCc1nc(no1)c2ccc(cc2)C(C)(C)C	CID:665654	phase I
BRD-K88668773	CCNC(=O)CCc1nc(no1)c2ccc(cc2)C(C)(C)C	CID:665747	phase I
BRD-K58679021	CCCCn1c(CN2CCN(CC2)c3cccc(Cl)c3)nc4n(C)c(=O)n(C)c(=O)c14	CID:666267	phase I
BRD-K55844427	Cc1nnc2sc(nn12)c3ccc(C)c(NC(=O)c4ccc(o4)c5cccc(Cl)c5)c3	CID:666410	phase I
BRD-K75360161	CCCc1cc(ccn1)C(S)=N	CID:666418	phase I
BRD-K24125544	COc1cc2CCN3C[C@@H](CC(C)C)C(=O)C[C@@H]3c2cc1OC	CID:667453	phase I
BRD-K59058766	CN(C)CC\C=C1/c2ccccc2Sc2ccc(Cl)cc12	CID:667466	phase I
BRD-K37694030	CN(C)CC\C=C1\c2ccccc2COc2ccccc12	CID:667468	phase I
BRD-K95309561	C\C=C(c1ccc(O)cc1)\C(c1ccc(O)cc1)=C\C	CID:667476	phase I
BRD-K54462405	CN(C)CC/C=C/1\c2ccccc2COc3ccccc13	CID:667477	phase I
BRD-K55055802	CCOC(=O)c1cncn1[C@H](C)c1ccccc1	CID:667484	phase I
BRD-K91601245	S=c1[nH]cnc2nc[nH]c12	CID:667490	phase I
BRD-K51033547	COc1cccc(c1)[C@]1(O)CCCC[C@H]1CN(C)C	CID:667511	phase I
BRD-K99260425	CCc1cccc2c3CCO[C@](CC)(CC(O)=O)c3[nH]c12	CID:667528	phase I
BRD-K43764301	C[C@H](C(=O)O)c1cccc(c1)C(=O)c2ccccc2	CID:667550	phase I
BRD-K96778649	NC(=S)/C(=C/c1ccc(O)c(O)c1)/C#N	CID:667601	phase I
BRD-K91509126	Oc1cc(O)cc(c1)\C=C\c1ccc(O)c(O)c1	CID:667639	phase I
BRD-K07212038	C/C=C(/C)\C(=O)O[C@@H]1Cc2c(OC1(C)C)ccc3ccc(=O)oc23	CID:668081	phase I
BRD-K63175663	COc1ccc(cc1)C(=O)Nc2cccc(NC(=O)C)c2	CID:669117	phase I
BRD-K61217870	CC(=O)Nc1cccc(NC(=O)c2cccc(Cl)c2)c1	CID:669190	phase I
BRD-K72192970	CC1=C(NC(=S)NC(=O)c2ccccc2)NCc3ccccc13	CID:670967	phase I
BRD-K41172353	O=C(Sc1cccc2ncccc12)c3ccccc3	CID:673329	phase I
BRD-K47693913	COc1c(OC[C@@H](O)C(C)(C)O)ccc2c(OC)c3ccoc3nc12	CID:673465	phase I
BRD-K87040771	CN(C)CCC(=O)c1coc2ccc(OC(=O)C)cc12	CID:674274	phase I
BRD-K56287385	COC(=O)CCc1[nH]c2ccccc2c1Sc3ccccc3	CID:674282	phase I
BRD-K41557448	COc1ccc2oc(cc(=O)c2c1)-c1ccccc1OC	CID:676288	phase I
BRD-K32480606	COc1ccc2oc(-c3ccccc3)c(OC)c(=O)c2c1	CID:676292	phase I
BRD-K01400178	Cc1c(OCC(=O)O)ccc2c(cc(=O)oc12)c3ccccc3	CID:679758	phase I
BRD-K43068349	CC(C)(C)c1ccc(C=CC(=O)Nc2ccc3OCCOc3c2)cc1	CID:680501	phase I
BRD-K30912208	CCN(CC)C(=O)c1sc(NC(=O)OC)c(C(N)=O)c1C	CID:681615	phase I
BRD-K66029294	[O-][N+](=O)c1ccc2c(c1)sn(-c1ccccc1)c2=O	CID:686211	phase I
BRD-K34952911	CNC(=O)CCc1cc2ccccc2[nH]1	CID:687114	phase I
BRD-K05197617	Cc1ccc2nc(Nc3ccccc3)cc(C)c2c1	CID:687170	phase I
BRD-K57179821	CCN(C(=O)\C=C\C)c1ccccc1C	CID:688020	phase I
BRD-K51671335	CCN1CCC[C@H]1CNC(=O)c1cc(ccc1OC)S(N)(=O)=O	CID:688272	phase I
BRD-K23644387	COc1ccc(cc1)-c1oc2ccccc2c(=O)c1OC	CID:688666	phase I
BRD-K58443469	Oc1ccc(cc1O)-c1cc(=O)c2ccc(O)c(O)c2o1	CID:688798	phase I
BRD-K80015639	Oc1ccc2oc(cc(=O)c2c1)-c1cccc(O)c1O	CID:688800	phase I
BRD-K09900591	OC(=O)\C=C\c1ccc(O)c(O)c1	CID:689043	phase I
BRD-K23673040	[O-][N+](=O)c1ccc(C=NNC(=O)CNc2cccc3ccccc23)o1	CID:690299	phase I
BRD-K99515112	CCN(CC)S(=O)(=O)c1cccc(c1)C(=O)Nc2nncs2	CID:691868	phase I
BRD-K67364256	O=C(NCc1cccnc1)c2cc3ccccc3oc2=O	CID:691928	phase I
BRD-K32836707	OC(=O)c1c[nH]c2c(Cl)c(Cl)ccc2c1=O	CID:693139	phase I
BRD-K94818765	S=c1[nH]nc(c2cccnc2)n1C3CCCCC3	CID:695345	phase I
BRD-K41227865	Sc1nnc2c3ccccc3n(Cc4ccccc4)c2n1	CID:695347	phase I
BRD-K77634909	NS(=O)(=O)c1nn2cc(nc2s1)-c1ccccc1	CID:698112	phase I
BRD-K38634661	Oc1ccc(CNc2cccc(F)c2)c2cccnc12	CID:698145	phase I
BRD-K03704870	CCc1ccc(OCC(=O)Nc2nnc[nH]2)cc1	CID:698942	phase I
BRD-K58900438	CCOC(=O)c1c(N)n(C2CCCCC2)c3nc4ccccc4nc13	CID:699552	phase I
BRD-K31754360	Cc1cc(ccc1F)S(=O)(=O)NCC(=O)O	CID:701150	phase I
BRD-K98025142	Cc1ccc(N2CCN(CC2)S(=O)(=O)N3CCCCC3)c(C)c1	CID:701237	phase I
BRD-K78867378	Cn1c(=O)c([N+](=O)[O-])c(Cl)c2ccccc12	CID:701939	phase I
BRD-K89391146	OC(=O)[C@H](Cc1c[nH]c2ccccc12)N1C(=O)c2ccccc2C1=O	CID:702558	phase I
BRD-K00203625	COc1cc(OC)cc(c1)C(=O)Nc2nc[nH]n2	CID:702927	phase I
BRD-K77432048	COc1ccc(Nc2nc(N)nc(CN3CCCCC3)n2)cc1	CID:704129	phase I
BRD-K21614065	Cc1cc(OCC(=O)Nc2nnc[nH]2)ccc1Cl	CID:704205	phase I
BRD-K85479953	Cc1cccc(Nc2nc(cs2)-c2ccncc2)c1	CID:704473	phase I
BRD-K71574320	C(Cn1c2nc(cn2c3ccccc13)c4ccccc4)N5CCOCC5	CID:706531	phase I
BRD-K76964878	NC(=O)[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21	CID:707029	phase I
BRD-K47128441	Nn1c(=O)c(Cc2ccco2)n[nH]c1=S	CID:708538	phase I
BRD-K39687892	Fc1cccc(Nc2nc(nc3ccccc23)c4ccncc4)c1	CID:710962	phase I
BRD-K95808480	O[C@H]1[C@H](Oc2cc(O)cc(O)c2C1=O)c3ccc(O)c(O)c3	CID:712318	phase I
BRD-K37393297	Cc1cc(C)nc(SCC(=O)c2ccc(O)c(O)c2)n1	CID:715454	phase I
BRD-K78388870	Clc1nssc1=Nc2ccc(C#N)cc2	CID:715698	phase I
BRD-K89595132	CN(C)CC[C@H](c1ccc(Cl)cc1)c2ccccn2	CID:716121	phase I
BRD-K19290969	CN1c2ccccc2Sc3cc(N)ccc13	CID:717880	phase I
BRD-K72462994	O=C(Nc1ccc(cc1)N2CCCCC2)c3ccncc3	CID:719365	phase I
BRD-K42834456	CN(C)c1ccc(/C=C/2\CSC(=S)NC2=O)cc1	CID:720272	phase I
BRD-K71322910	CCOC(=O)C1=C(CC2=C1CCCC2)NC(=S)Nc3ccccc3	CID:720932	phase I
BRD-K90735586	C1C=C(Nc2nnnn12)c3ccccc3	CID:727137	phase I
BRD-K96213252	CC(=O)Nc1ccc(NC(=O)c2ccccc2Br)cc1	CID:727425	phase I
BRD-K55498981	CCOC(=O)CCc1n[nH]c(=O)[nH]c1=O	CID:728578	phase I
BRD-K69003436	O=C(Cn1nnc2sc3CCCCc3c2c1=O)NCc4ccco4	CID:733669	phase I
BRD-K63116520	NCc1cccc(O)c1	CID:735894	phase I
BRD-K28362289	CC(=O)N1CCN(CC1)c2ccc(N)cc2	CID:736269	phase I
BRD-K23313025	OC(=O)c1cccnc1SCC(=O)c2cccc(c2)[N+](=O)[O-]	CID:741395	phase I
BRD-K37762845	COc1ccccc1NC(=O)CSc2nc3ccccc3o2	CID:742357	phase I
BRD-K93899689	OC(=O)CCNC(=O)c1cncc(Br)c1	CID:743143	phase I
BRD-K00390580	N#Cc1ccc(Oc2ccc(cc2)-c2ccccc2)cc1C#N	CID:746627	phase I
BRD-K35961280	Cc1cc2nc(SCCN3CCCC3)[nH]c2cc1C	CID:747185	phase I
BRD-K97701319	Nc1ccc(cc1)C(=O)Nc2ccc(O)c(c2)c3nc4ccccc4o3	CID:748328	phase I
BRD-K19875179	OC(=O)CCC(=O)Nc1ccc(Br)c2cccnc12	CID:752172	phase I
BRD-K20755323	Oc1ccc(Nc2nc(cs2)-c2ccc(Cl)cc2)cc1	CID:753704	phase I
BRD-K42308740	Cc1nnc(Sc2cc(C)nc3ccccc23)s1	CID:755405	phase I
BRD-K03568209	Oc1ccc2oc3C(=O)NCCCc3c2c1	CID:755673	phase I
BRD-K73125384	COc1ccccc1N(N=C2Sc3ccccc3C2=O)C(=O)C	CID:759940	phase I
BRD-K09635314	Cc1cc(C)c(c(C)c1)S(=O)(=O)Nc1cccc(c1)C(F)(F)F	CID:761523	phase I
BRD-K50659736	Cc1cccc(NC(=O)CCC(=O)O)c1	CID:763244	phase I
BRD-K33936059	CC(=O)Nc1ccc(/N=C/c2ccc(C)cc2)cc1	CID:767214	phase I
BRD-K67808578	COc1ccc2oc(=N)c(cc2c1)c3nc4ccccc4[nH]3	CID:768699	phase I
BRD-K46384212	Cc1cc(C)c(c(C)c1)S(=O)(=O)Nc1ccccc1C(F)(F)F	CID:770820	phase I
BRD-K17476933	Clc1ccc(C(=O)n2nnc3ccccc23)c(Cl)c1	CID:771910	phase I
BRD-K86350435	COc1ccc(CNc2cc(C)ccc2C)c(OC)c1	CID:775191	phase I
BRD-K03857568	Cc1ccc(Sc2c([N+](=O)[O-])c(=O)n(C)c3ccccc23)cc1	CID:776319	phase I
BRD-K05593511	Nc1ccccc1Nc2c(N)c(=O)oc3ccccc23	CID:777301	phase I
BRD-K01265221	CN(C)C1=C(Cl)C(=O)N(C1=O)c2ccc(Cl)c(Cl)c2	CID:779754	phase I
BRD-K33743361	COc1ccc(CNCc2cccc3ccccc23)cc1	CID:781301	phase I
BRD-K53932786	CCSc1nc(nc(n1)c2ccccc2)C(Cl)Cl	CID:781660	phase I
BRD-K88708949	Cc1ccc2nc(Nc3ccccc3)nc(c4ccccc4)c2c1	CID:782168	phase I
BRD-K61413806	COc1cc(CN2CCN(CC2)c3cc(C)ccc3C)ccc1O	CID:782696	phase I
BRD-K49861754	N#Cc1cc2ccc(cc2cc1C#N)N3CCOCC3	CID:784670	phase I
BRD-K11362964	Cc1cc(C)c(c(C)c1)S(=O)(=O)NCC(=O)O	CID:789791	phase I
BRD-K20112532	Nc1c(C#N)sc2nc(cc(c3ccc(Cl)cc3)c12)C4CC4	CID:790989	phase I
BRD-K98991361	CC(=O)Nc1cccc(NC(=O)c2ccccc2Cl)c1	CID:792012	phase I
BRD-K08463963	CCn1c(=O)c([N+](=O)[O-])c(Cl)c2ccccc12	CID:800048	phase I
BRD-K91349888	[O-][N+](=O)c1c(Cl)c2ccccc2n(Cc2ccccc2)c1=O	CID:800654	phase I
BRD-K68588778	Cc1c(C=O)c(C=O)c(C)n1Cc2ccccc2	CID:800760	phase I
BRD-K06191433	CN(C(C)=O)c1ccc(cc1)\N=C\c1c(O)ccc2ccccc12	CID:801047	phase I
BRD-K46285453	Fc1cccc(c1)C(=O)Nc2nc[nH]n2	CID:807820	phase I
BRD-K24632213	CC(C)Sc1nc2n(C)c(=O)[nH]c(=O)c2n1Cc3ccccc3	CID:814607	phase I
BRD-K25690923	Ic1cc(ncn1)-c1ccccc1	CID:817368	phase I
BRD-K58299615	Nc1ccc(cc1)-c1nc2ccc(cc2[nH]1)-c1nc2ccc(N)cc2[nH]1	CID:824226	phase I
BRD-K50776152	Cc1ccc(cc1)n2c(N)c(C#N)c(c(C#N)c2=O)c3ccccc3	CID:824820	phase I
BRD-K39829853	Oc1ccc(CNc2ccccc2Br)c2cccnc12	CID:830235	phase I
BRD-K06890060	Clc1cccc(Cl)c1C(=O)NCc2ccc3OCOc3c2	CID:831629	phase I
BRD-K05775306	COc1ccc2ccccc2c1CNCc3ccccn3	CID:834719	phase I
BRD-K07079548	Oc1ccc2C[C@H]3N(CC=C)CCc4cccc(c34)-c2c1O	CID:838674	phase I
BRD-K29699988	C1CCN(C1)c2nc(N3CCCC3)c4ccccc4n2	CID:839770	phase I
BRD-K69471245	Oc1ccccc1NC(=O)c1ccccn1	CID:842059	phase I
BRD-K84881516	O=C(Nc1nc2ccccc2s1)c1cccs1	CID:843289	phase I
BRD-K30536692	CCSc1cc(nc(n1)c2ccc(Cl)cc2)N3CCCC3	CID:852319	phase I
BRD-K94144010	CN1[C@@H](CCC1=O)c1cccnc1	CID:854019	phase I
BRD-K95349679	Cc1cccc(c1)c2nnc(SCC(=O)O)n2CC=C	CID:854343	phase I
BRD-K36111658	CCc1cc(=O)oc2cc(C)cc(OCC(=O)C(C)(C)C)c12	CID:855012	phase I
BRD-K00289828	CCc1cc2cc3OCOc3cc2nc1SCC(=O)OC(C)C	CID:855567	phase I
BRD-K68535470	Clc1ccc(cc1)C(=O)N1CCN(CC1)c1ccccn1	CID:870371	phase I
BRD-K37549600	CC(=O)Nc1nc(nc(n1)c2ccccc2OC(=O)C)c3ccccc3	CID:871154	phase I
BRD-K16309743	COc1ccccc1CN2CCN(Cc3cccnc3)CC2	CID:876559	phase I
BRD-K45114207	CN1C(=O)c2ccc(NC(=O)c3cccc4ccccc34)cc2C1=O	CID:877183	phase I
BRD-K38012662	CCC(=O)Nc1cccc(NC(=O)c2ccccc2Br)c1	CID:877874	phase I
BRD-K73707305	N#Cc1ccc(Oc2cccnc2)cc1C#N	CID:882273	phase I
BRD-K02641134	CC(C)(C)c1ccc(cc1)C(=O)Nc1cc(Cl)ccc1C(O)=O	CID:883362	phase I
BRD-K61993165	OC(=O)c1cccnc1SCCc2ccccc2	CID:888706	phase I
BRD-K83355732	CCOc1cc(CO)c(Br)cc1OCC(=O)O	CID:894165	phase I
BRD-K00859168	Cc1c(CC(=O)O)c(=O)oc2cc(OCC(=O)O)ccc12	CID:895450	phase I
BRD-K50289629	Clc1ccc(/C=C/C(=O)NC2=NCCS2)cc1Cl	CID:896331	phase I
BRD-K71554540	Cc1ccc(/C=C/C(=O)NC2=NCCS2)cc1	CID:897475	phase I
BRD-K03954795	COc1cc(nc(S)n1)c2ccccc2	CID:902452	phase I
BRD-K81142122	Cn1nc(nc2c(=O)n(C)c(=O)nc12)c3ccccn3	CID:906542	phase I
BRD-K45888792	C\C=C1\[C@@H]2Cc3nc(O)ccc3[C@@]1(N)CC(C)=C2	CID:907504	phase I
BRD-K24564544	Cc1cc(Cl)ccc1OCC(=O)NN=Cc1ccc[nH]1	CID:909513	phase I
BRD-K91913968	Clc1ccc(OCC(=O)NN=Cc2ccc[nH]2)c(Cl)c1	CID:910309	phase I
BRD-K86693415	CC(C)Oc1nc(nc2ccccc12)c3ccc(Cl)cc3	CID:914635	phase I
BRD-K83213280	Brc1ccc2N=C3CCCN3Cc2c1	CID:928277	phase I
BRD-K64885524	CCc1ccc2n(CC(=O)OC)c3nc4ccccc4nc3c2c1	CID:936254	phase I
BRD-K29582677	Fc1ccc(cc1)C(N1CCN(C\C=C\c2ccccc2)CC1)c1ccc(F)cc1	CID:941361	phase I
BRD-K97309399	CN(C)S(=O)(=O)c1ccc2Sc3ccccc3\C(=C/CCN3CCN(C)CC3)c2c1	CID:941650	phase I
BRD-K05542495	COc1ccc(cc1)c2nc(OC)c3ccccc3n2	CID:946273	phase I
BRD-K77014406	COc1cccc(c1)c2nc(OC(C)C)c3ccccc3n2	CID:946943	phase I
BRD-K78716413	CCc1nnc2sc(nn12)c3ccc(N)cc3	CID:952391	phase I
BRD-K79251086	Oc1ccc(CNc2ccccn2)c2cccnc12	CID:965010	phase I
BRD-K07572174	COc1cc(ccc1O)\C=C\C(=O)CC(=O)\C=C\c1ccc(O)c(OC)c1	CID:969516	phase I
BRD-K64985742	COc1ccc(Cl)cc1NC(=S)NCCn2cc(Cl)cn2	CID:971629	phase I
BRD-K74840245	CCOC(=O)Nc1cccc(NC(=O)c2cc(OC)cc(OC)c2)c1	CID:973303	phase I
BRD-K47084999	Cc1ccc(Nc2nc(=O)c3cccnc3s2)cc1	CID:973891	phase I
BRD-K36772364	O=C(CSc1cccc2cccnc12)N3CCCC3	CID:975656	phase I
BRD-K28112517	CCOc1ccc(cc1OCC)c2nc(no2)c3ccncc3	CID:976135	phase I
BRD-K63220166	Cc1ccc2n(CCN3CCOCC3)c4nc5ccccc5nc4c2c1	CID:976690	phase I
BRD-K08630646	COc1ccc(OC)c(NC(=O)c2ccc(CSc3ncnc4[nH]cnc34)cc2)c1	CID:980157	phase I
BRD-K17777116	CC1(C)C(C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(NC(=O)C4C(C)(C)C4(C)C)cc3)C1(C)C	CID:981129	phase I
BRD-K65503129	CCc1cc(-c2n[nH]c(C)c2-c2ccc3OCCOc3c2)c(O)cc1O	CID:984170	phase I
BRD-K56555032	CCn1c(COc2c(C)cccc2C)nnc1SCC(=O)N3CCN(CC3)c4ccccc4	CID:986349	phase I
BRD-K81609421	Cn1c(=O)n(C)c2nc(NCc3cccnc3)n(Cc4cccc(Br)c4)c2c1=O	CID:989617	phase I
BRD-K57016430	NC(=O)C1CCN(CC1)c2nc(cs2)c3ccc(Br)cc3	CID:990823	phase I
BRD-K92754162	Cc1ccc(NC(=O)c2ccc(o2)-c2cc(Cl)ccc2Cl)c(C)c1	CID:1007755	phase I
BRD-K05977823	CC(=O)Nc1ccc(NC(=S)NC(=O)c2ccc(cc2)C(C)(C)C)cc1	CID:1013376	phase I
BRD-K03122949	CC1CCN(CC1)S(=O)(=O)c2ccc(NC(=O)c3ccc(cc3)C(C)(C)C)cc2	CID:1013514	phase I
BRD-K91517665	Cc1ccc2oc(nc2c1)c3cccc(NC(=O)c4cc(ccc4Cl)n5cnnc5)c3	CID:1017704	phase I
BRD-K45031696	COc1nc(c2ccc3OCOc3c2)n(n1)c4ccc(NC(=O)CSc5ccccc5)cc4	CID:1029232	phase I
BRD-K12168891	Cc1ccc(cc1)n2c(N)c(C#N)c(c(C#N)c2=O)c3ccc(Cl)cc3	CID:1034641	phase I
BRD-K29715937	Cc1ccc(cc1)c2c(C#N)c(N)n(c3ccc(Cl)cc3)c(=O)c2C#N	CID:1034643	phase I
BRD-K48388979	CCOc1ccccc1C=NNC(=O)c2nnn(c2CN3CCCCCC3)c4nonc4N	CID:1036002	phase I
BRD-K25979535	CCOc1ccc(cc1)\N=c1/scc(-c2ccc(C)c(C)c2)n1CC	CID:1037728	phase I
BRD-K36638198	CC(C)(OC(=O)c1ccccc1)[C@@H]2Cc3cc4ccc(=O)oc4cc3O2	CID:1042895	phase I
BRD-K82395301	COc1cc(NC(=O)c2cc3ccccc3cc2OCC(=O)NC(C)(C)C)c(OC)cc1Cl	CID:1043828	phase I
BRD-K59036917	CCCC(=O)Nc1cccc(NC(=O)c2ccccc2Br)c1	CID:1048267	phase I
BRD-K81376179	COc1ccc(cc1OC)C(=O)Nc1sc2CCCCc2c1C(N)=O	CID:1048845	phase I
BRD-K47622659	Clc1cc(NC2CCCCC2)c3C(=O)c4ccccc4-c5onc1c53	CID:1049140	phase I
BRD-K86992982	Clc1ccc(NC(=O)Nc2nnc(s2)c3ccncc3)cc1Cl	CID:1075698	phase I
BRD-K22322324	CCc1nc2oc(C(=O)c3ccccc3)c(N)c2c4CC(C)(C)OCc14	CID:1075883	phase I
BRD-K15107389	O=C1c2ccccc2-c3c(NCCc4ccccc4)c(=O)[nH]c5cccc1c35	CID:1080352	phase I
BRD-K36817836	CCc1nc(SCC(=O)N2CCc3cc(OC)c(OC)cc3C2)c(C#N)cc1C	CID:1086218	phase I
BRD-K48924007	C(CN1CCOCC1)Sc2nc3ccccc3n2Cc4ccccc4	CID:1086976	phase I
BRD-K89306950	Cc1ccc(cc1)S(=O)(=O)n1c(N)nc2ccccc12	CID:1088438	phase I
BRD-K08799912	Nc1nc2ccccc2n1S(=O)(=O)c1ccc(Cl)cc1	CID:1088439	phase I
BRD-K18711687	Oc1ccc(CNc2ccccc2Cl)c2cccnc12	CID:1090316	phase I
BRD-K23149109	Oc1ccc(CNc2ccccc2C(F)(F)F)c2cccnc12	CID:1090321	phase I
BRD-K32644160	N(c1nnc(s1)c2ccncc2)c3cccc4ccccc34	CID:1090779	phase I
BRD-K13794505	CCn1nccc1C(=O)Nc2nc3ccccc3n2CCN4CCCCC4	CID:1091784	phase I
BRD-K90020768	CC(=O)Nc1cccc(c1)c2csc(Nc3cc(C)ccn3)n2	CID:1092458	phase I
BRD-K88735704	Nc1ccc2[nH]c(CCC(=O)O)nc2c1	CID:1093221	phase I
BRD-K74447990	CC(=O)c1cccc(NC(=O)c2cnn3c(C)cc(C)nc23)c1	CID:1097834	phase I
BRD-K06712146	COc1cc2CC(C)(C)n3c(cc4nc5ccccc5nc34)-c2cc1OC	CID:1103147	phase I
BRD-K40300908	Cc1ccc(cc1)n2nc3ccc(NC(=O)COc4ccccc4C)cc3n2	CID:1109840	phase I
BRD-K76211160	Fc1ccc(cc1)C(=O)Nc2cccnc2	CID:1118253	phase I
BRD-K05464208	COc1cc(SC)ccc1C(=O)N1CCC(Cc2ccccc2)CC1	CID:1126109	phase I
BRD-K82088145	Nc1ccccc1NC(=O)c1ccncc1	CID:1133081	phase I
BRD-K20880473	Nc1ccccc1NC(=O)c2cccnc2	CID:1133083	phase I
BRD-K32111336	Cc1cc2cc3OCCOc3cc2n2c(SCC(=O)Nc3nc(cs3)-c3ccccc3)nnc12	CID:1135867	phase I
BRD-K36267058	Cc1cccc(NC(=O)/C(=C/c2cn(CC(=O)NCc3ccco3)c4ccccc24)/C#N)c1	CID:1140587	phase I
BRD-K86631041	Cc1cc2cc3OCOc3cc2n2c(SCC(=O)Nc3nc(cs3)-c3ccccc3)nnc12	CID:1143390	phase I
BRD-K65200617	CC[C@@H]1CN2CCc3cc(OC)c(OC)cc3[C@H]2C[C@H]1C[C@@H]1NCCc2cc(OC)c(OC)cc12	CID:1151030	phase I
BRD-K05549170	Clc1ccc(cc1)S(=O)(=O)N[C@@H]1CCCC[C@H]1N1CCOCC1	CID:1167614	phase I
BRD-K66634822	Clc1ccc(cc1)S(=O)(=O)N[C@H]1CCCC[C@@H]1N1CCOCC1	CID:1167615	phase I
BRD-K57592392	Clc1ccc(cc1)S(=O)(=O)N[C@@H]1CCCC[C@@H]1N1CCOCC1	CID:1167616	phase I
BRD-K97330509	COc1ccc2c(cc(C)c3nnc(SCC(=O)Nc4cccc(c4)C(=O)C)n32)c1	CID:1172104	phase I
BRD-K96704748	COc1ccc(Oc2c(oc3cc(OCC(=O)Nc4ccccc4F)ccc3c2=O)C(F)(F)F)cc1	CID:1182101	phase I
BRD-K44494044	COC(=O)c1cc(Br)ccc1NC(=O)COc2ccc(cc2)C(C)(C)C	CID:1182617	phase I
BRD-K56658166	Brc1ccccc1OCC(=O)NCCc2nc3ccccc3[nH]2	CID:1183113	phase I
BRD-K50841342	Oc1c(CC=C)cccc1C=NNC(=O)CN2CCN(Cc3ccccc3)CC2	CID:1185541	phase I
BRD-K81441552	COc1ccc(cc1)C(=O)Nc2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F	CID:1188388	phase I
BRD-A98349433	CS(=O)(=O)c1ccc(S(=O)CC(=O)OCc2ccccc2)c(c1)[N+](=O)[O-]	CID:1189521	phase I
BRD-K75418381	COc1ccc(C)cc1NC(=O)c2ccc(OCC(=O)Nc3cc(Cl)ccc3Cl)cc2	CID:1189620	phase I
BRD-K77480336	COc1ccc(/N=c/2\cc(oc3ccc(O)cc23)c4ccc(OC)cc4)cc1	CID:1191868	phase I
BRD-K95673870	OCCn/1c(cs\c1=N/c2ccccc2)c3cccc(c3)N4C(=O)c5ccccc5C4=O	CID:1201964	phase I
BRD-K69569876	Nc1nc(CSc2nnnn2c3ccccc3)nc(Nc4ccccc4)n1	CID:1201976	phase I
BRD-K55420858	NC1=NC(=O)\C(S1)=C\c1ccc(O)cc1	CID:1206243	phase I
BRD-K89205986	Cc1c(/C=C/2\S/C(=N/c3ccccc3)/N(C4CCCC4)C2=O)c5ccccc5n1CC(=O)N	CID:1220374	phase I
BRD-K24677486	COC(=O)NN=Cc1ccc(o1)[N+](=O)[O-]	CID:1226495	phase I
BRD-K05831461	CC(C)C[C@@H](NC(C)=O)C(O)=O	CID:1241420	phase I
BRD-K42419294	OC(=O)c1ccc(NS(=O)(=O)c2cc3C(=O)NC(=O)c4cccc(c2)c43)cc1	CID:1242010	phase I
BRD-K88542532	COc1ccc(cc1)N(C(=O)c2cccnc2)S(=O)(=O)c3ccccc3	CID:1242547	phase I
BRD-K05649647	COc1ccc(cc1)N(C(=O)c2ccccc2)S(=O)(=O)c3cc(OC)ccc3OC	CID:1242560	phase I
BRD-K03176945	COc1ccc(cc1)N(C(=O)C2CCCCC2)S(=O)(=O)c3cc(OC)ccc3OC	CID:1242564	phase I
BRD-K84855138	Fc1ccccc1CNC(=O)c2cccs2	CID:1244199	phase I
BRD-K84389640	Cc1cccc(/N=C/2\SCC(=O)N2c3cccc(C)c3)c1	CID:1244300	phase I
BRD-K94035551	Brc1ccccc1CNC(=O)c1cccs1	CID:1246750	phase I
BRD-K61627029	CN(C)c1nc(N)nc(CSc2nnnn2c3ccccc3)n1	CID:1248117	phase I
BRD-K43739430	Oc1ccc(Br)cc1/C=N/c2ccc3nc(SCC(=O)Nc4ccccc4)sc3c2	CID:1248840	phase I
BRD-K92489476	CCOC(=O)c1cnc(SCC(=O)N2CCc3ccccc23)nc1N	CID:1249064	phase I
BRD-K19196783	Nc1nonc1n2nnc(C(=O)NN=Cc3ccccc3Br)c2CN4CCCC4	CID:1250001	phase I
BRD-K36111767	Clc1ccc(cc1)C(=O)N2CCN(CC2)c3ccnc4cc(Cl)ccc34	CID:1251584	phase I
BRD-K61359235	O=C(N1CCCc2ccccc12)c3cccc(c3)S(=O)(=O)NC4CCCCCC4	CID:1252831	phase I
BRD-K53011428	Fc1ccc(Nc2nnc(s2)c3ccncc3)cc1Cl	CID:1257201	phase I
BRD-K00551481	Cc1cc(nn1CC(=O)n2nc(C)c(Cl)c2C)[N+](=O)[O-]	CID:1257352	phase I
BRD-K31450967	CCN(CC)c1c(C#N)c(SCC(=O)c2cccs2)cc3CCCCc13	CID:1258678	phase I
BRD-K70917163	COc1ccc(CCn2c(N)cc(=O)[nH]c2=S)cc1OC	CID:1259573	phase I
BRD-K62578746	OC(C1CCN(CC1)C(S)=Nc1ccc(Cl)cc1)(c1ccccc1)c1ccccc1	CID:1261254	phase I
BRD-K66908362	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3cc(nc4c(C)cc(C)cc34)c5cccnc5)cc2)c1C	CID:1261290	phase I
BRD-K27539181	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3cc(nc4c(C)cc(C)cc34)c5ccccn5)cc2)c1C	CID:1261822	phase I
BRD-K31453413	Cc1cc(NS(=O)(=O)c2ccc(NC(=O)c3cc(nc4c(C)cc(C)cc34)c5ccccn5)cc2)no1	CID:1261872	phase I
BRD-K46961308	COc1cccc2cc(oc12)c3nnc(SCC(=O)Nc4cccc(Br)c4)n3C	CID:1262839	phase I
BRD-K82492171	CN(c1ccc(OCC(=O)O)cc1)S(=O)(=O)c2ccc(F)cc2	CID:1265060	phase I
BRD-K80184735	Brc1ccc(NC(=O)C2(CCCCC2)N(Cc2ccco2)C(=O)c2ccccn2)cc1	CID:1282817	phase I
BRD-K27881911	COc1ccc(Cn2c3ccc(Br)cc3c4nc5ccccc5nc24)cc1OC	CID:1287820	phase I
BRD-K48204702	Cc1ccc(cc1NC(=O)COc2ccccc2[N+](=O)[O-])c3nc4ccccc4[nH]3	CID:1288922	phase I
BRD-K02223034	Cc1nnc(SCC(=O)c2c(cc3ccccn23)c4ccc(C)cc4)s1	CID:1288929	phase I
BRD-K48823327	COc1cc(c(OC)cc1Cl)S(=O)(=O)n2nnc3ccccc23	CID:1289024	phase I
BRD-K06020002	FC(F)(F)c1ccc(Cl)c(Nc2nnc(s2)c3ccncc3)c1	CID:1294885	phase I
BRD-K14395638	CC(=O)c1cccc(NC(=O)Nc2nn(Cc3c(F)cccc3Cl)cc2Br)c1	CID:1297252	phase I
BRD-K14316227	Cc1ccc(cc1)S(=O)(=O)NC(=O)CSc2nc3ccccc3s2	CID:1299526	phase I
BRD-K10906552	Cn1c(SCC(=O)n2c3CCCCc3c4ccccc24)nnc1c5ccco5	CID:1300352	phase I
BRD-K27170250	Cc1cccnc1NC(=S)NC(=O)c2cncc(Br)c2	CID:1302558	phase I
BRD-K32949592	O=C(CS(=O)(=O)c1ccc2ccccc2c1)c3cc4ccccc4oc3=O	CID:1304413	phase I
BRD-K75458636	Clc1c(sc2ccccc12)C(=O)Nc3sc4CCCc4c3C(=O)NCc5ccco5	CID:1304563	phase I
BRD-K00954209	CC(=O)c1c(C)n(c2ccc(C)cc2)c3ccc(OC(=O)CN4C(=O)c5ccccc5C4=O)cc13	CID:1305613	phase I
BRD-K21672423	Cc1cc(C)c(C#N)c(SCCS(=O)(=O)c2nc3ccccc3s2)n1	CID:1317598	phase I
BRD-K91355947	[O-][N+](=O)c1ccc(OCC(=O)Nc2ccc3oc(nc3c2)c4ccc(F)cc4)cc1	CID:1326094	phase I
BRD-K47731572	CCOc1ccc(cc1)S(=O)(=O)Nc2nc3ccccc3nc2Nc4ccccc4	CID:1327854	phase I
BRD-K14609189	COc1ccc(c2nn(cc2/C=C\3/SC(=S)N(CCC(=O)O)C3=O)c4ccccc4)c(C)c1	CID:1328217	phase I
BRD-K32927008	COc1ccc(cc1)c2nnc(SCC(=O)Nc3cccc(c3)C(F)(F)F)n2c4ccccc4	CID:1329190	phase I
BRD-K53214709	CCc1ccc(O)c(NC(=S)NC(=O)COc2ccc(C)cc2C)c1	CID:1345154	phase I
BRD-K51696048	[O-][N+](=O)c1ccc(OCC(=O)Nc2ccc3oc(nc3c2)c4ccccc4Cl)cc1	CID:1349139	phase I
BRD-K54416256	Cn1cc[nH]c1=S	CID:1349907	phase I
BRD-K83637872	Cc1nn(c(C)c1C=NN2CCN(Cc3ccccc3)CC2)c4ccccc4	CID:1356208	phase I
BRD-K59980915	Oc1ccc(NC(=O)COc2ccc(Cl)cc2)cc1c3nc4ccccc4o3	CID:1363881	phase I
BRD-K41757249	Cc1ccc(cc1NC(=O)COc2ccccc2)c3nc4ccccc4o3	CID:1366986	phase I
BRD-K63712590	COc1ccc(cc1)-c1csc(NC(=O)CSc2nnc3c(C)cc4ccccc4n23)n1	CID:1374043	phase I
BRD-K73201151	COc1ccc(OC)c(c1)N2C(=O)C(=C(N3CCCCC3)C2=O)Cl	CID:1379247	phase I
BRD-K43131268	Cc1ccc(cc1)c2nnc(SCC(=O)c3ccc(O)c(O)c3)n2CC=C	CID:1394536	phase I
BRD-K48974000	Oc1ccc(cc1O)C(=O)CSc2nnc(c3cccc(Cl)c3)n2CC=C	CID:1398345	phase I
BRD-K57309821	COc1ccc2nc3n(CC(C)C)nc(NC(=O)CC(C)C)c3cc2c1	CID:1398674	phase I
BRD-K78056905	Cc1cccc(c1)c2nnc(SCC(=O)c3ccc(O)c(O)c3)n2CC=C	CID:1400246	phase I
BRD-K25522720	COc1ccc(cc1)c2nnc(SCC(=O)c3ccc(O)c(O)c3)n2CC=C	CID:1400698	phase I
BRD-K28075147	COc1ccc(cc1)c2coc3cc(OC(=O)C)cc(OC(=O)C)c3c2=O	CID:1403142	phase I
BRD-K40224283	COc1cccc(c1)c2nnc(SCC(=O)c3ccc(O)c(O)c3)n2CC=C	CID:1409759	phase I
BRD-K22832646	COc1cc(/C=C/2\SC(=NC2=O)N)ccc1O	CID:1417813	phase I
BRD-K26684619	OC(=O)c1cccnc1Nc2ccc(Cl)cc2	CID:1432578	phase I
BRD-K91134378	Cc1nc(N2CCN(CC2)C(=O)c3ccco3)c4c5CCCCc5sc4n1	CID:1434953	phase I
BRD-K75304533	Cc1nc(N2CCN(CC2)C(=O)c3cccs3)c4c5CCCCc5sc4n1	CID:1434956	phase I
BRD-K58982513	Cc1nc(N2CCN(CC2)C(=O)C2CCCCC2)c2c3CCCCc3sc2n1	CID:1434957	phase I
BRD-K02174945	Cc1nc(N2CCN(CC2)C(=O)COc2ccccc2C)c2c3CCCCc3sc2n1	CID:1434960	phase I
BRD-K70771662	Clc1ccc(cc1)C(=O)Nc2ccc(Sc3ccccc3)c(C#N)c2	CID:1471787	phase I
BRD-K50495309	COc1cc2ncnc(Nc3ccc(Oc4ccccc4)cc3)c2cc1OC	CID:1474853	phase I
BRD-K36287933	COc1ccc(cc1)C(=O)ON=C(C)c2nccs2	CID:1481893	phase I
BRD-K04363266	CC(=NOC(=O)c1ccc(Cl)cc1)c2nccs2	CID:1481894	phase I
BRD-K22215695	Cc1ccc(Cn2ncc3c(ncnc23)N4CCN(CC4)c5ccccc5C)cc1	CID:1502520	phase I
BRD-K19146323	Clc1ccc2c(ccnc2c1)N1CCN(CC1)C(=O)c1ccc(Cl)c(Cl)c1	CID:1505783	phase I
BRD-K63511615	Clc1cccc(c1)C(=O)N1CCN(CC1)c1ccnc2cc(Cl)ccc12	CID:1505784	phase I
BRD-K40151202	CCN(CC)C(=O)Cn1c2ccccc2c2nc3SCCn3c(=O)c12	CID:1507946	phase I
BRD-K49237419	Fc1ccc2c(c1)sn(-c1ccccc1)c2=O	CID:1510378	phase I
BRD-K45278408	Cc1ccccc1n2sc3cc(F)ccc3c2=O	CID:1510379	phase I
BRD-K67258146	Cc1ccc(C)c(c1)-n1sc2cc(F)ccc2c1=O	CID:1510389	phase I
BRD-K06432680	CCCN1CNc2c(C1)c(=O)[nH]c(=S)n2CCc3ccc(OC)c(OC)c3	CID:1512045	phase I
BRD-K51608872	CN(C)c1nc(N)nc(CSc2nnnn2c3cccc4ccccc34)n1	CID:1517919	phase I
BRD-K63513868	Cc1cccn2cc(COc3ccc(cc3)c4ccccc4)nc12	CID:1523656	phase I
BRD-K53566850	Cc1ccccc1N2CCN(CC2)c3ncnc4n(Cc5ccc(Cl)cc5)ncc34	CID:1542103	phase I
BRD-A13020530	COC(=O)CS(=O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F	CID:1543530	phase I
BRD-K17343332	Oc1c(Br)cc(Br)cc1C=NN2CCN(Cc3ccccc3)CC2	CID:1544274	phase I
BRD-K07220430	C(/C=C/c1ccccc1)N2CCN(CC2)C(c3ccccc3)c4ccccc4	CID:1547484	phase I
BRD-K66381707	Cn1c2ccc(/N=C/c3ccccc3O)cc2c4nc5ccccc5nc14	CID:1547739	phase I
BRD-K65389993	C1CCc2ncc(c3ccc(cc3)c4ccccc4)n2CC1	CID:1548076	phase I
BRD-K16336526	COc1cc(CNC(=O)CCCC/C=C\C(C)C)ccc1O	CID:1548942	phase I
BRD-K50590187	COc1cc(CNC(=O)CCCC\C=C\C(C)C)ccc1O	CID:1548943	phase I
BRD-K04218075	CCN(CC)CCOc1ccc(cc1)/C(=C(/Cl)\c2ccccc2)/c3ccccc3	CID:1548953	phase I
BRD-K29950728	CCN(CC)CCOc1ccc(cc1)C(=C(/Cl)c1ccccc1)\c1ccccc1	CID:1548955	phase I
BRD-K27184429	OC(=O)COCCN1CCN(CC1)[C@H](c1ccccc1)c1ccc(Cl)cc1	CID:1549000	phase I
BRD-K68132782	CN(C\C=C\C#CC(C)(C)C)Cc1cccc2ccccc12	CID:1549008	phase I
BRD-K85013741	CC(=CCC/C(=C/COc1ccc2ccc(=O)oc2c1)/C)C	CID:1550607	phase I
BRD-K79554012	CCCCOC(=O)CCN1C(=S)S\C(=C/c2ccccc2)C1=O	CID:1556232	phase I
BRD-K08478539	Brc1ccc2ncnc(NCC=C)c2c1	CID:1560402	phase I
BRD-K32862555	Clc1ccc(cc1)c2nc(C#N)c(NCC=C)o2	CID:1580719	phase I
BRD-K00555438	O=C(Nc1ccc(cc1)S(=O)(=O)Nc2nccs2)c3cc(nc4ccccc34)c5ccccc5	CID:1582687	phase I
BRD-K11758216	Clc1nc(NCc2ccccc2)c3ccccc3n1	CID:1604254	phase I
BRD-K94018295	Cn1c(SCC(=O)NN=Cc2ccc(s2)[N+](=O)[O-])nnc1c3ccc(Cl)cc3	CID:1607628	phase I
BRD-K58698715	CCCOc1ccc(cc1)c2nc(OC)c3ccccc3n2	CID:1612038	phase I
BRD-K96271548	COc1ccccc1/C=C\C(=O)O	CID:1622530	phase I
BRD-K42568865	CCCOc1ccc(cc1)c2nc(Oc3ccc(OC)cc3)c4ccccc4n2	CID:1634732	phase I
BRD-K74228917	CCOc1ccc2NC(C)(C)c3ss/c(=N\c4ccc(NC(=O)C)cc4)/c3-c2c1	CID:1635461	phase I
BRD-K19499941	CCCCCCCN(C(=O)CCl)c1cccc(C)c1	CID:1637653	phase I
BRD-K35716340	C(Cn1c2ccccc2c3ccccc13)c4nc5ccccc5[nH]4	CID:1641662	phase I
BRD-K82987299	CCOC(=O)c1cnc2c(C)c(C)ccc2c1NCCCN(C)C	CID:1645763	phase I
BRD-K93176058	CCCCCCCCc1ccc(cc1)-c1ccc(cc1)C(O)=O	CID:1714884	phase I
BRD-K45681478	ClC1=C(NCC=C)C(=O)c2ccccc2C1=O	CID:1716436	phase I
BRD-K12105018	Cc1c(NC(=O)COc2ccc(Br)cc2)cccc1c3nc4cc(Cl)ccc4o3	CID:1721551	phase I
BRD-K49814456	[O-][N+](=O)c1ccc(C=NNC(=O)CNc2cccc(c2)[N+](=O)[O-])o1	CID:1737777	phase I
BRD-K89814851	O=C(CSc1nc(ccc1C#N)c2cccs2)Nc3sc4CCCCc4c3C#N	CID:1772635	phase I
BRD-K57285282	COc1ccc(CN2C(=O)[C@@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)cc1	CID:1776583	phase I
BRD-K17830172	Cc1ccc(NC(=O)CCC(=O)NN=Cc2ccc(o2)[N+](=O)[O-])cc1C	CID:1789299	phase I
BRD-K63245238	CCOC(=O)c1c(NC(=S)NC(=O)c2ccc(OC)c(c2)[N+](=O)[O-])sc3CCCc13	CID:1797892	phase I
BRD-K89748981	CCCCc1ccc2nc(NC(=O)c3cccs3)sc2c1	CID:1814489	phase I
BRD-K35046132	CCCCc1ccc2nc(NC(=O)c3ccc(Br)o3)sc2c1	CID:1814490	phase I
BRD-K70960308	Cn1nnnc1SCCNC/C=C/c2ccccc2	CID:1817779	phase I
BRD-K93760529	CCOc1ccccc1CNCCN2CCOCC2	CID:1817873	phase I
BRD-K57836103	Cc1c(c2ccccc2)[n+]([O-])c(c(C)[n+]1[O-])c3ccc(Br)cc3	CID:1856447	phase I
BRD-K07530279	COc1ccc(Cl)cc1Nc2nnc(s2)c3ccncc3	CID:1864426	phase I
BRD-K00442147	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1ccccc1	CID:1871033	phase I
BRD-K99696746	CCCc1cc(ccn1)c2nc(cs2)c3ccc(C)cc3	CID:1889993	phase I
BRD-K95901403	Cc1ccc(cc1)S(=O)(=O)Nc1nc2ccccc2nc1Nc1ccc2nsnc2c1	CID:1893730	phase I
BRD-K23335153	C(CNC(c1ccccc1)c1ccccc1)NC(c1ccccc1)c1ccccc1	CID:1894361	phase I
BRD-K15164005	Clc1ccc(CN2C(=O)C(=O)c3ccccc23)cc1Cl	CID:1901244	phase I
BRD-K90090262	OC(=O)c1cc2cc(CSCCC#N)ccc2o1	CID:1916559	phase I
BRD-K34388789	OC(C1CCN(CC1)C(=Nc2ccc(F)cc2)S)(c3ccccc3)c4ccccc4	CID:1934050	phase I
BRD-K84114569	COCCNC(=S)Nc1nc(OC)cc(OC)n1	CID:1955478	phase I
BRD-K41790758	Cc1ccc(Nc2nc(=O)c3cccnc3s2)c(Br)c1	CID:1963150	phase I
BRD-K22384978	CN(C)CCCNc1oc(nc1C#N)c2ccccc2F	CID:1978813	phase I
BRD-K98381590	C[C@@H](Nc1nc(Cl)nc2ccccc12)c3ccccc3	CID:1993104	phase I
BRD-K72817452	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)c1ccccc1	CID:1998811	phase I
BRD-K61679744	Fc1ccc(cc1)C(=O)OCC#CCSc2nnc(o2)c3cccc4ccccc34	CID:1998940	phase I
BRD-K19433082	COc1ccc(cc1)C(=O)OCC#CCSc2nnc(o2)c3cccc4ccccc34	CID:1999882	phase I
BRD-K73143528	Brc1ccc(cc1)C(=O)OCC#CCSc2nnc(o2)c3cccc4ccccc34	CID:2013455	phase I
BRD-K11072542	COC(=O)c1cn(C(=O)c2cccc3ccccc23)c4ccccc14	CID:2016258	phase I
BRD-K68495126	O=C(OCC#CCSc1nnc(o1)c2cccc3ccccc23)c4cc5ccccc5o4	CID:2017368	phase I
BRD-K07061353	Clc1ccccc1c2nnc(SCC(=O)Nc3ccc(Br)cc3)n2c4ccccc4	CID:2046011	phase I
BRD-K74029109	OCCNc1nc(Nc2ccc(Cl)cc2)nc(n1)N3CCCC3	CID:2055451	phase I
BRD-K31851742	Cc1nn(CCCC(=O)O)c(C)c1[N+](=O)[O-]	CID:2057146	phase I
BRD-K95286134	CCCCc1ccc2nc(NC(=O)c3ccco3)sc2c1	CID:2066730	phase I
BRD-K66902379	CN(C)S(=O)(=O)c1cccc(c1)C(=O)N1CCN(CC1)c1cccc(C)c1C	CID:2090194	phase I
BRD-K13665914	C(C1CCN(CC1)c2ncnc3sccc23)c4ccccc4	CID:2100018	phase I
BRD-K05456756	Cc1cc(NC(=O)COC(=O)c2c(C)nn(Cc3ccccc3)c2Cl)no1	CID:2112466	phase I
BRD-K38985961	Cc1cc(C(=O)CN2C(=O)CCC2=O)c(C)n1Cc3ccccc3	CID:2113511	phase I
BRD-K24426149	CCCc1cc(NC(=O)CCl)n(n1)c2ccccc2	CID:2120347	phase I
BRD-K32536677	Clc1ccc(Cl)c(c1)c2ccc(/C=C(\C#N)/C(=O)Nc3cccc4ncccc34)o2	CID:2130404	phase I
BRD-K82924899	Cc1ccc2nc(NC(=O)CSc3nc4CCSc4c(=O)n3-c3ccccc3)sc2c1	CID:2155128	phase I
BRD-K60228169	Cc1cc(NC(=O)CS(=O)(=O)c2cn(Cc3cccc(F)c3)c4ccccc24)no1	CID:2157612	phase I
BRD-K14270862	Fc1cccc2sc(NC(=O)c3cccs3)nc12	CID:2159213	phase I
BRD-K18953385	OC(=O)c1ccccc1OCc2ccccc2Br	CID:2160985	phase I
BRD-K33720394	CC1(C)N[C@@H](Cc2c1[nH]c1ccccc21)C(O)=O	CID:2180476	phase I
BRD-K34966483	Brc1ccc(o1)C(=O)Nc2ccccc2c3ccccc3	CID:2183264	phase I
BRD-K75903201	CCCCC(=O)Nc1cccc(NC(=O)c2ccccc2Br)c1	CID:2186104	phase I
BRD-K11841836	Cc1nc2ccc(NC(=S)NCCCO)cc2nc1C	CID:2191501	phase I
BRD-K78701355	COc1ccc(OC)c(c1)S(=O)(=O)ON2C(=O)c3ccccc3C2=O	CID:2201555	phase I
BRD-K63954456	COc1cc(cc(Br)c1OCC(=O)O)c2nc3ccccc3s2	CID:2202512	phase I
BRD-A93893742	[O-][N+](=O)c1cc(ccc1S(=O)CC(=O)Oc2ccc(Cl)cc2)C(F)(F)F	CID:2203170	phase I
BRD-K32321439	COc1ccc(Cl)cc1NC(=O)CSc2nnc(c3cc4cc(Br)ccc4o3)n2C	CID:2207955	phase I
BRD-K94248251	CCn1cc(NC(=S)Nc2cc(Cl)ccc2OC)c(n1)C(=O)N	CID:2208391	phase I
BRD-K07877311	Clc1cc(NC(=O)CSc2nnc(c3ccccc3)n2c4ccccc4)ccc1Br	CID:2209276	phase I
BRD-K22988559	CCc1nnc(NC(=O)c2ccc(NS(=O)(=O)c3ccccc3)cc2)s1	CID:2210290	phase I
BRD-K69496360	COc1ccc(Cl)cc1NC(=S)NCCCN2CCCC2=O	CID:2211279	phase I
BRD-K70369221	Fc1ccc(cc1)C(=O)CSc2nnc(c3cccc(Br)c3)n2c4ccccc4	CID:2215989	phase I
BRD-K29767311	Clc1cccc(c1)c2nc(C#N)c(NCC=C)o2	CID:2218783	phase I
BRD-K16346331	CCOc1ccccc1C(=O)Oc2c(c(C)nn2c3ccccc3)S(=O)(=O)c4ccc(C)cc4	CID:2218860	phase I
BRD-K97631938	FC(F)(F)c1ccccc1NC(=O)Cn2cc(C(=O)c3ccco3)c4ccccc24	CID:2219490	phase I
BRD-K75329208	Cc1ccc(c(C)c1)S(=O)(=O)NC(=O)COc2cccc3ccccc23	CID:2222011	phase I
BRD-K95895342	Cc1cc(ccc1OCC(=O)O)S(=O)(=O)NC2CCCCC2	CID:2222056	phase I
BRD-K64738596	[O-][N+](=O)c1ccc2c(Cl)c(sc2c1)C(=O)NCCCN3CCOCC3	CID:2225472	phase I
BRD-K18814832	Cc1ccc(C)c(NS(=O)(=O)c2cc(ccc2Cl)C(=O)Nc3ccccc3c4ccccc4)c1	CID:2228302	phase I
BRD-K44931544	Cc1ccc(cc1S(=O)(=O)Nc2ccccc2)C(=O)Nc3ccccc3c4ccccc4	CID:2242162	phase I
BRD-K42541148	OC(=O)c1ccc(cc1)-c1ccc(\C=c2/sc3nc4ccccc4n3c2=O)o1	CID:2243732	phase I
BRD-K73238422	Clc1ccccc1\C=c1/sc2nc3cc(Br)cnc3n2c1=O	CID:2258411	phase I
BRD-K88013557	CCCC(=O)Nc1cccc(NC(=O)Cc2ccc(Cl)cc2)c1	CID:2274454	phase I
BRD-K61237522	Cc1ccc(NC(=O)CCC(=O)NN=Cc2ccco2)c(C)c1	CID:2275371	phase I
BRD-K70524666	Clc1cc(Cl)cc(c1)-c1ccc(\C=c2/sc3nc4cc(Br)cnc4n3c2=O)o1	CID:2300608	phase I
BRD-K32502880	O=C(NCCOc1ccccc1c2ccccc2)c3ccco3	CID:2300880	phase I
BRD-K02175743	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)c3cc(nc4ccccc34)c5ccccc5)cc2)n1	CID:2308203	phase I
BRD-K12707296	Cc1nn(c(N)c1Sc2ccc(F)cc2)c3nc(C)cc(C)n3	CID:2321431	phase I
BRD-K28296557	CC[n+]1c(/C=C/N(C)c2ccccc2)n(c3ccccc3)c4ccc(cc14)c5nc6ccccc6s5	CID:2326992	phase I
BRD-K70831943	Cc1ccc(cc1S(=O)(=O)N2CCCCC2)n3sc4ccccc4c3=O	CID:2327953	phase I
BRD-K96352593	Cc1cc(c(C)n1c2ccccc2)c3nnc4CCCCCn34	CID:2331284	phase I
BRD-K10806285	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3cc(nc4ccccc34)c5ccccc5Cl)cc2)c1C	CID:2332853	phase I
BRD-K65258912	CCc1nc2sc3CCCCc3c2c(=O)n1NC(=O)CCl	CID:2345373	phase I
BRD-K20401833	OC(c1ccc(NS(=O)(=O)c2cccs2)cc1)(C(F)(F)F)C(F)(F)F	CID:2360837	phase I
BRD-K23623876	Fc1cccc(C=NN=Cc2cccc(F)c2)c1	CID:2378095	phase I
BRD-K21918725	Cc1nn(c(N2CCCC2)c1C=NN=C(S)Nc3ccccc3F)c4ccccc4	CID:2379002	phase I
BRD-K42644990	O=S(=O)(Nc1nc2ccccc2nc1NCCC3=CCCCC3)c4ccccc4	CID:2387953	phase I
BRD-K62459624	ClCC(=O)N=c1sccn1Cc2ccccc2Cl	CID:2416356	phase I
BRD-K39345836	Cn1nnnc1Sc2ncnc3scc(c4ccccc4)c23	CID:2432214	phase I
BRD-K72504866	CN(C)S(=O)(=O)c1ccc(N2CCCC2)c(c1)C(=O)N3CCN(CC3)c4cccc(C)c4C	CID:2440433	phase I
BRD-K79390395	Cc1cc(C(=O)CCl)c(C)n1CCc2ccc(Cl)cc2	CID:2442307	phase I
BRD-K68313733	ClCC(=O)N(Cc1ccccc1OCC=C)c2ccc3OCOc3c2	CID:2449454	phase I
BRD-K26367064	CN(C)S(=O)(=O)c1ccc(N2CCCC2)c(c1)C(=O)N1CCN(CC1)c1ccccc1	CID:2466259	phase I
BRD-K42867405	Fc1ccccc1n2c(SCC(=O)Nc3ccc4CCCc4c3)nc5ccccc5c2=O	CID:2482839	phase I
BRD-K95495709	CCc1ccc2c(CN3CCc4cc(OC)c(OC)cc4C3)cc(=O)oc2c1	CID:2486932	phase I
BRD-K73099734	Fc1ccc(cc1Cl)-n1c(SCC(=O)Nc2ccc3CCCc3c2)nc2ccccc2c1=O	CID:2513861	phase I
BRD-K02986291	Clc1ccccc1NC(=O)COC(=O)CNC(=O)C2CCCCC2	CID:2547325	phase I
BRD-K51745483	O=C(CSc1nc2ccccc2c(=O)n1-c1ccccc1)Nc1ccc2CCCc2c1	CID:2557019	phase I
BRD-K03439359	Cc1cc(NC(=O)COC(=O)c2c(C)nn(Cc3ccccc3Cl)c2Cl)no1	CID:2571615	phase I
BRD-K57975631	O=S(=O)(N1CCN(CC1)S(=O)(=O)c1ccc2OCCOc2c1)c1cccc(c1)C#N	CID:2604410	phase I
BRD-K02421873	[O-][N+](=O)c1ccc(o1)C(=O)OCc2nnc(o2)c3ccccc3	CID:2630179	phase I
BRD-K88701661	OC(=O)[C@@H](S)[C@@H](S)C(O)=O	CID:2724354	phase I
BRD-K23478508	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)O[C@@H]2[C@@H](C)O[C@H](C[C@@H]2O)O[C@@H]3[C@@H](C)O[C@H](C[C@@H]3O)O[C@H]4CC[C@@]5(C)[C@H](CC[C@@H]6[C@@H]5C[C@@H](O)[C@]7(C)[C@H](CC[C@]67O)C8=CC(=O)OC8)C4	CID:2724385	phase I
BRD-K75649340	Nc1nc(S)c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1	CID:2724387	phase I
BRD-K19885561	Oc1ccccc1C(=O)Nc2ccc(NC(=O)c3ccc(Cl)cc3)cc2	CID:2725417	phase I
BRD-K33926001	CCOC(=O)c1cc(nc(O)c1C#N)c2ccc(Cl)cc2	CID:2726279	phase I
BRD-K34363599	OC(COc1ccc(F)cc1)(c2ccc(Cl)cc2)c3ccc(Cl)cc3	CID:2728620	phase I
BRD-A32241587	S=C1CC(Sc2ccccc2N1)c3ccccc3	CID:2728652	phase I
BRD-A18763547	OC(CN1CCNCC1)Cn1c2ccc(Br)cc2c2cc(Br)ccc12	CID:2729027	phase I
BRD-A56800788	CNS(=O)(=O)c1ccc(cc1S(=O)c2ccccc2C(=O)O)C(F)(F)F	CID:2729755	phase I
BRD-K44849676	Oc1cc2CCCN(Cc2cc1O)C(=S)NCCc1ccc(Cl)cc1	CID:2733484	phase I
BRD-K93754473	CC\C(c1ccccc1)=C(/c1ccccc1)c1ccc(OCCN(C)C)cc1	CID:2733526	phase I
BRD-A84189516	CC(=O)O[C@@H]1C2=C(C)[C@@H](O)C[C@@](O)([C@@H](OC(=O)c3ccccc3)C3[C@@]4(CO[C@@H]4C[C@H](O)[C@@]3(C)C1=O)OC(C)=O)C2(C)C	CID:2733529	phase I
BRD-K33572481	C[C@H](CCC(=O)NCCS(O)(=O)=O)[C@H]1CC[C@H]2[C@@H]3CC[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:2733768	phase I
BRD-A78295502	CC[C@H]1CN2CCC1C[C@H]2[C@H](O)c3ccnc4ccc(OC)cc34	CID:2734756	phase I
BRD-K50002132	CC[n+]1ccccc1Br	CID:2736301	phase I
BRD-K15196155	CC(C)n1nnc2cc(ccc12)C(O)=O	CID:2736690	phase I
BRD-K67867734	CCOC(=O)c1n[nH]c(=S)[nH]c1=O	CID:2739070	phase I
BRD-K82230692	CC(C)(C)NC(=O)N1CCN(CC1)c2ncccc2C(F)(F)F	CID:2741632	phase I
BRD-K58499478	Clc1ccc(cc1)C(=O)NNC(=O)c2csc(n2)c3cccs3	CID:2743956	phase I
BRD-K99532291	Cc1nc(cs1)C(=O)NNC(=O)c2ccc(Cl)cc2	CID:2744062	phase I
BRD-K53987746	CNC(=NN=Cc1c(cnn1c2ccc(F)cc2F)C(=O)OC)S	CID:2745684	phase I
BRD-K71382703	COC(=O)c1cnn(c1C=NN=C(S)Nc1ccc(Cl)cc1)-c1ccc(F)cc1F	CID:2745686	phase I
BRD-K06186994	COC(=O)c1cnn(c1C=NN=C(S)NC(C)(C)C)c2ccc(F)cc2F	CID:2745687	phase I
BRD-K88784410	COC(=O)c1cnn(c1C=NN=C(S)Nc1ccccc1)-c1ccc(F)cc1F	CID:2745688	phase I
BRD-K02313433	CNC(S)=NN=Cc1c(cnn1-c1ccc(Cl)cc1)C(=O)OC	CID:2745694	phase I
BRD-K32636001	COC(=O)c1cnn(c1C=NN=C(S)Nc1ccccc1)-c1ccc(Cl)cc1	CID:2745696	phase I
BRD-K73982490	Oc1nnc(Sc2ncc(s2)[N+]([O-])=O)n1-c1ccc2OCCOc2c1	CID:2747117	phase I
BRD-K51207550	CCc1cc(ccn1)C(S)=N	CID:2761171	phase I
BRD-K43069600	Cc1ccc(Sc2ccc(NC(=O)c3ccc(F)cc3)cc2C#N)cc1	CID:2769158	phase I
BRD-K40087974	COc1ccc(Sc2ccc(NC(=O)c3ccccc3Cl)cc2C#N)cc1	CID:2769229	phase I
BRD-K36087356	COc1ccc(Sc2ccc(NC(=O)c3cccc(Cl)c3)cc2C#N)cc1	CID:2769230	phase I
BRD-K00624509	C(OCc1nc2ccccc2[nH]1)c1nc2ccccc2[nH]1	CID:2772764	phase I
BRD-A18579359	CN(C)CC(O)Cn1c2ccc(Br)cc2c3cc(Br)ccc13	CID:2775510	phase I
BRD-K31843556	[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc1ccncc1	CID:2777391	phase I
BRD-K71835137	CCOC(=O)c1sc(SCc2ccccc2)c3C(=O)CC(C)(C)Cc13	CID:2778741	phase I
BRD-K79235952	CCOC(=O)c1sc(SC)c2C(=O)CCCc12	CID:2778748	phase I
BRD-K39580048	[O-][N+](=O)c1c(Cl)c2ccccc2[nH]c1=O	CID:2785467	phase I
BRD-A39121618	COc1ccc(NC(=O)c2ccc(OC(C)C(=O)O)cc2)cc1Cl	CID:2793096	phase I
BRD-K82685933	CN(C)/C=N/c1nnc(Sc2cc(C)nc3ccccc23)s1	CID:2799534	phase I
BRD-K50360938	CCOC(=O)CCSc1nnc(S)s1	CID:2802190	phase I
BRD-K24675965	Brc1ccc(NC(=O)N2NC(=O)[C@H]([C@@H]2c2ccccc2)c2ccccc2)cc1	CID:2802894	phase I
BRD-K92801790	C1c2sc(Nc3ccccc3)nc2-c4ccccc14	CID:2803032	phase I
BRD-K99311057	Fc1ccc(cc1)C(=O)CSc2nsc(SCC(=O)c3ccc(F)cc3)c2C#N	CID:2803059	phase I
BRD-A09984573	CSC1=C(C#N)C(=O)NC(S1)c2ccc(Cl)cc2	CID:2803185	phase I
BRD-A15113563	Clc1ccc(cc1Cl)C2Nc3ccccc3O2	CID:2806677	phase I
BRD-K26373640	NC(=O)c1sc(cc1N)-c1ccsc1	CID:2807869	phase I
BRD-K76565902	Clc1ccc2c(ccnc2c1)N1CCN(CC1)C(=O)c1cccs1	CID:2809486	phase I
BRD-K63488275	O=C(Nc1ccc2[nH]ccc2c1)c3cccs3	CID:2814135	phase I
BRD-A89067742	O=C(Nc1cccs1)N2CCN(CC2)C(=O)C3CCCO3	CID:2815576	phase I
BRD-K23841751	OC(=O)CSCC(=O)N1CCCN(CC1)c2ccc(cn2)C(F)(F)F	CID:2815616	phase I
BRD-K78549347	Clc1ccc(cc1)n2ncc(n2)C(=O)c3ccccc3	CID:2815801	phase I
BRD-K44136596	Cc1ccc(Cc2nn3c(nn(c4ccc(Cl)cc4)c3nc2=O)C(=O)c5cccs5)cc1	CID:2816236	phase I
BRD-K11147885	CNC(=O)NC(=O)CSc1nnc(c2ccncc2)n1Cc3ccccc3	CID:2816422	phase I
BRD-K26048285	Cc1cc(C)c2c3NC(=O)CN(C(=O)c3sc2n1)c4ccccc4C	CID:2817045	phase I
BRD-K93300946	Oc1ccc(CCNc2ccc(NCCc3ccc(O)cc3)c3C(=O)c4ccccc4C(=O)c23)cc1	CID:2817242	phase I
BRD-K14191038	FC(F)(F)C(NCc1ccccn1)(NC(=O)c2cccnc2)C(F)(F)F	CID:2817908	phase I
BRD-K55996963	CSc1nc(N)n(n1)c2cc(Cl)cc(Cl)c2	CID:2818504	phase I
BRD-K22931010	CC(C)(C)c1ccc(cc1)c2n[nH]c(NS(=O)(=O)c3ccccc3)c2Br	CID:2818982	phase I
BRD-K87375115	COc1cccc(c1)C(=O)C(=C(SC)SC)C#N	CID:2819095	phase I
BRD-K85493820	Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N	CID:2819152	phase I
BRD-K10817986	Cc1c(csc1C(=O)Nc2ccc(F)cc2F)S(=O)(=O)c3ccc(Cl)cc3	CID:2819320	phase I
BRD-K59761766	CSc1sc(C(=O)O)c2CC(C)(C)CC(=O)c12	CID:2819767	phase I
BRD-A84098870	CSc1sc(C(=O)NN)c2CCCC(O)c12	CID:2820091	phase I
BRD-K36264978	CSc1sc(c2ccn(n2)C(=O)Nc3ccccc3)c4CC(C)(C)CC(=O)c14	CID:2820118	phase I
BRD-K68344511	Nc1c(C#N)sc2sc(C#N)c(c3ccco3)c12	CID:2820134	phase I
BRD-K28120860	CC1(C)CC(=O)C=C(SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)S1	CID:2820381	phase I
BRD-A69336132	COc1cccc(NC(=S)N=S(=O)(C)c2ccccc2)c1	CID:2820633	phase I
BRD-A53746180	Clc1ccc(cc1)C2CC(=O)C=C(SCC(=O)c3ccccc3)S2	CID:2820696	phase I
BRD-K21788104	O=C(NNC(=O)c1ccccc1)c2csc(n2)c3cccnc3	CID:2824173	phase I
BRD-K65955264	CCCCCC[n+]1ccccc1\C=C\c1ccc(cc1)N(C)C	CID:2824731	phase I
BRD-A25416824	CC12CCC3C(CC=C4CC(O)CCC34CO)C2CCC1OC(=O)c5ccccc5	CID:2825553	phase I
BRD-A01960364	COc1ccc(cc1)C2C(C(=O)O)c3ccccc3C(=O)N2Cc4ccc(Cl)cc4	CID:2826386	phase I
BRD-A23747351	CC(NC(=O)c1ccccc1\N=C\c1c(O)ccc2ccccc12)c1ccccc1	CID:2827646	phase I
BRD-A36318220	CN1C(=S)NC(Cc2c[nH]c3ccccc23)C1=O	CID:2828334	phase I
BRD-A09164687	Cc1cc(C)c(OCC(O)CNC(C)(C)C)c(C)c1	CID:2830268	phase I
BRD-A77299732	ClC(Cl)(Cl)C(NC(=O)C=Cc1ccccc1)NC(=S)Nc2cccc3cccnc23	CID:2830510	phase I
BRD-A55565369	CCCC(NS(=O)(=O)c1ccc(C)cc1)C(=O)O	CID:2834096	phase I
BRD-A69439373	CN1CCN(CC(O)COCCC2(CC3CC4CC(C3)C2)C4)CC1	CID:2834356	phase I
BRD-A84389633	CN1C2CCC1CC(C2)OC(=O)c1cc(C)cc(C)c1	CID:2837530	phase I
BRD-A49734948	COc1cc(=O)n(C)c2c(OCC(O)C(C)(C)O)cccc12	CID:2837663	phase I
BRD-A98050686	CCN(CC)C(=O)C1CCCN(Cc2cccc(Cl)c2)C1	CID:2838441	phase I
BRD-K89692698	C1CN(CCO1)c2nnc(c3ccccc3)c(n2)c4ccccc4	CID:2842253	phase I
BRD-K10554164	OC(=O)CCN1C(=O)c2cccc3c(ccc(C1=O)c23)[N+](=O)[O-]	CID:2844045	phase I
BRD-K60070073	CC(C)(C)NC(=O)c1ccc2C(=O)c3ccccc3-c4onc1c42	CID:2847176	phase I
BRD-A65142661	COC1CCCCC1Nc2cc(C)ccc2C	CID:2850171	phase I
BRD-A43087975	COCC(C)NCc1ccc(OC)c(OC)c1OC	CID:2851120	phase I
BRD-A29721261	CC(C)c1ccc(NC(=O)C2CC3CCC2C3)cc1	CID:2852569	phase I
BRD-K90999434	O=C(CN1C2=NCCN2c2ccccc12)c1ccc(cc1)-c1ccccc1	CID:2853753	phase I
BRD-A00420644	CCN1C2C(C(=NC2Nc3ccccc13)OC)c4ccccc4	CID:2853908	phase I
BRD-K65050353	Cn1c2ccccc2c3nnc(SCCN4CCCCC4)nc13	CID:2857183	phase I
BRD-K59962020	Cc1cc2nc(NCCCO)n(CC(=O)c3cc(c(O)c(c3)C(C)(C)C)C(C)(C)C)c2cc1C	CID:2858523	phase I
BRD-K86682249	OC(=O)c1ccccc1c2ccc(C=c3sc4nc5cc(Br)cnc5n4c3=O)o2	CID:2861757	phase I
BRD-A57107094	COC(=O)C1=C(C)NC2=C(C1c3ccccc3)C(=O)CC(C2)c4ccc(Cl)cc4	CID:2864482	phase I
BRD-A36884011	COc1ccc(cc1)C(=O)Nc2ccccc2C(=O)NC(C(C)C)C(=O)O	CID:2868336	phase I
BRD-A35338386	CCNC(=O)C1OC(C(O)C1O)n2cnc3c(N)ncnc23	CID:2868392	phase I
BRD-K68548958	CC1=NN(C(=O)C\1=C\c1ccc(o1)-c1cc(C)c(C)cc1[N+]([O-])=O)c1ccc(cc1)C(O)=O	CID:2871948	phase I
BRD-A27640568	COc1ccc(C(NC(=O)c2ccccc2)c3ccc4cccnc4c3O)c(OC)c1	CID:2872362	phase I
BRD-A47816767	CC(C)C(=O)NC(c1ccco1)c2ccc3cccnc3c2O	CID:2876959	phase I
BRD-A62647958	CCOC(=O)C1=C(C)N=c2sc(=Cc3ccc(OCC(=O)O)cc3)c(=O)n2C1c4ccc(Cl)cc4	CID:2878586	phase I
BRD-A13195221	CCN(CC)c1ccc(cc1)C2Nc3ccccc3NC4=C2C(=O)CC(C4)c5ccccc5	CID:2878746	phase I
BRD-A45657137	CCOC(=O)C1=C(N=c2sc(=Cc3cc(OC)c(OC)c(OC)c3)c(=O)n2C1c4cccs4)c5ccccc5	CID:2885102	phase I
BRD-A67306036	OC(=O)C1C(C2CCC1O2)C(=O)NCCc3ccccc3	CID:2887234	phase I
BRD-K03644760	[O-][N+](=O)c1c(Nc2cc(Cl)cc(Cl)c2)c2ccccc2oc1=O	CID:2888950	phase I
BRD-A50388635	COc1ccc(cc1)C(=O)NC(c2ccc(OC)c(OC)c2)c3cc(Cl)c4cccnc4c3O	CID:2896739	phase I
BRD-K90041947	Cc1ccc(C=C2SC(=S)N(CCCC(=O)Nc3cccc(c3)C(O)=O)C2=O)cc1	CID:2905788	phase I
BRD-A48052484	Clc1ccc(cc1)S(=O)(=O)NC2CCCCC2N3CCOCC3	CID:2911646	phase I
BRD-K93095519	CCOc1cc(cc(Cl)c1OCC(=O)OC)\C=C1C(=O)N(N=C/1C)c1ccccc1	CID:2913564	phase I
BRD-K82034465	CC(=Cc1ccccc1)C=C1SC(=S)N(CCCC(=O)Nc2ccc(C(O)=O)c(O)c2)C1=O	CID:2914104	phase I
BRD-K54018158	CC(=Cc1ccccc1)C=C1SC(=S)N(CCCC(=O)Nc2ccc(cc2)C(O)=O)C1=O	CID:2914168	phase I
BRD-A54194844	CC(=O)NC(c1ccco1)c1cc(Cl)c2cccnc2c1O	CID:2921053	phase I
BRD-K84266862	CN(C)S(=O)(=O)c1cc(ccc1C)[N+]([O-])=O	CID:2921148	phase I
BRD-A36059655	COc1ccc2N3C(=NC(=O)C(Cc4ccccc4)C3=O)Sc2c1	CID:2928239	phase I
BRD-A67748489	CC(=O)NC1=NN(C(C)=O)C(C)(S1)c1ccccc1	CID:2930014	phase I
BRD-A16581344	CN(Cc1ccccc1)C(=O)C2CCCN(Cc3ccccc3C(F)(F)F)C2	CID:2930928	phase I
BRD-K36533576	[O-][N+](=O)c1ccc2c(Cl)c(sc2c1)C(=O)NCCCn1ccnc1	CID:2933863	phase I
BRD-K42629487	CCOc1ccc(NC(=S)N2CCC(CC2)C(O)(c3ccccc3)c4ccccc4)cc1	CID:2936384	phase I
BRD-K00640357	CCCN(CCC)c1ncnc2n(ncc12)c3ccc(OC)cc3	CID:2941340	phase I
BRD-A74699940	COC(Cc1nc2ccccc2s1)C(=O)O	CID:2941514	phase I
BRD-K96326565	CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccc([N+](=O)[O-])c(NCc4cccnc4)c3	CID:2941653	phase I
BRD-A89352139	O=C1C2CC=CCC2C(=O)N1c1nc(n[nH]1)-c1ccccc1	CID:2946732	phase I
BRD-K41924482	CS(=O)(=O)N(CC(=O)O)c1ccc(cc1)C2(CC3CC4CC(C3)C2)C4	CID:2946881	phase I
BRD-A02481876	CC(Nc1nc(nc2ccccc12)N3CCCC3)c4ccccc4	CID:2949965	phase I
BRD-A28422330	COc1ccc(cc1)C2CC(=NN2c3ccc(cc3)S(=O)(=O)N)c4ccccc4	CID:2950007	phase I
BRD-K95858622	COc1ccc(CNc2ccc(cc2)N2CCN(CC2)C(C)=O)cc1OC	CID:2950270	phase I
BRD-A61666925	NC(=O)C1CCN(CC1)C2CC(=O)N(C2=O)c3ccc(F)c(Cl)c3	CID:2951172	phase I
BRD-A88029023	CC(Oc1ccc(Cl)cc1C)C(=O)Nc2ccc(cc2)C(=O)Nc3ccccc3C(=O)O	CID:2951539	phase I
BRD-A72163687	CCC(=O)C1(CC(C)(C)OC1=O)Sc1nc2ccccc2[nH]1	CID:2951859	phase I
BRD-A56001686	CCOc1ccccc1NC(=O)C(C)Oc2ccc(OC)cc2	CID:2952127	phase I
BRD-K64310881	CCOc1ccccc1C(=O)Nc2cc(Cl)ccc2O	CID:2953683	phase I
BRD-A88504692	CCn1cc(C(C)NC(=S)Nc2cccc(c2)[N+](=O)[O-])c(C)n1	CID:2956635	phase I
BRD-A10330754	Clc1ccc(Cn2cc(NC(=S)NCC3CCCO3)cn2)cc1	CID:2956728	phase I
BRD-A36165599	COC(=O)c1c(C)c(C)sc1NC(=O)CC2Nc3cccc4cccc(NC2=O)c34	CID:2963476	phase I
BRD-A12643502	Oc1cccnc1NC(=O)CCC2COc3ccccc3O2	CID:2965120	phase I
BRD-A30455275	CCOc1ccc(NC(=O)C(C)Sc2ncnc3sc(cc23)c4ccccc4)cc1	CID:2976290	phase I
BRD-A07614565	CCOc1ccc(cc1)C(Nc2cccnc2)c3cc(Cl)c4cccnc4c3O	CID:2977478	phase I
BRD-A19928752	CC(Sc1ccc(C)cc1)C(=O)Nc2nc[nH]n2	CID:2977752	phase I
BRD-A72796238	CCOC(=O)C1=C(CN2CCc3ccccc23)NC(=O)NC1c4cccc(c4)[N+](=O)[O-]	CID:2978593	phase I
BRD-K27169919	CCOC(=O)CS(=O)(=O)c1nc(cc(n1)C(F)(F)F)c2ccc(F)cc2	CID:2980973	phase I
BRD-K51731619	NCCCN(Cc1ccco1)C2CCCC2	CID:2981024	phase I
BRD-K06800040	O=C1N(CCCSc2nnc[nH]2)C(=O)c3cccc4cccc1c34	CID:2981635	phase I
BRD-A96272097	COC(=O)CC1N(CCNC1=O)C(=O)OC(C)(C)C	CID:2986153	phase I
BRD-A78377521	CCOC(=O)C1=C(C)NC(=S)NC1c1cccc(O)c1	CID:2987927	phase I
BRD-K63350243	Fc1ccc2n(Cc3ccccc3)c4nc(SCCN5CCOCC5)nnc4c2c1	CID:2989846	phase I
BRD-K12623437	O=C(COC(=O)C1(CC2CC3CC(C2)C1)C3)NCc4ccco4	CID:2998659	phase I
BRD-A31429689	CC(OC(=O)c1cccc(NS(=O)(=O)C)c1)C(=O)Nc2ccc(cc2)N3CCOCC3	CID:2998821	phase I
BRD-K06666320	CCCn1c(NC(=O)c2cccc(c2)S(=O)(=O)N3CCCC3)nc4ccccc14	CID:3000022	phase I
BRD-K49384696	CCC[C@@H]1C[C@H](N(C)C1)C(=O)N[C@H]([C@@H](C)O)[C@H]1O[C@H](SC)[C@H](O)[C@@H](O)[C@H]1O	CID:3000540	phase I
BRD-K51095933	C[C@@]12CC[C@H]3[C@@H](CCc4cc(OS(=O)(=O)O)ccc34)[C@@H]2CCC1=O	CID:3001028	phase I
BRD-K70505054	CN\C(NCCSCc1ccc(CN(C)C)o1)=C/[N+]([O-])=O	CID:3001055	phase I
BRD-A71157293	C\C(N(Cc1cnc(C)nc1N)C=O)=C(\CCO)SSCC1CCCO1	CID:3002119	phase I
BRD-A11678676	COC[C@H]1OC(=O)c2coc3C(=O)C4=C([C@@H](C[C@@]5(C)C4CCC5=O)OC(=O)C)[C@]1(C)c23	CID:3003565	phase I
BRD-K51350053	CN(C)CCOc1ccc(cc1)C(\c1ccccc1)=C(\CCCl)c1ccccc1	CID:3005573	phase I
BRD-K18787491	N\C(Sc1ccccc1N)=C(C#N)/C(C#N)=C(\N)Sc1ccccc1N	CID:3006531	phase I
BRD-A43974499	CCOc1ccccc1OC(C2CNCCO2)c3ccccc3	CID:3022645	phase I
BRD-K59840856	Nc1nc2ccccc2n1S(=O)(=O)c1ccccc1	CID:3025920	phase I
BRD-K93331292	Nc1nc2ccccc2n1S(=O)(=O)c1ccc(cc1)[N+]([O-])=O	CID:3025945	phase I
BRD-K60690191	Cc1cccc(n1)C#Cc1ccccc1	CID:3025961	phase I
BRD-K43389698	CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCNCC3)s2)o1	CID:3025986	phase I
BRD-K34014345	COc1ccc2cc(ccc2c1)[C@H](C)CO	CID:3032818	phase I
BRD-K73589491	CN\C(NCCSCc1csc(CN(C)C)n1)=C/[N+]([O-])=O	CID:3033637	phase I
BRD-K00610438	Fc1ccc(cc1)C(=O)C1CCN(CCn2c(=S)[nH]c3ccccc3c2=O)CC1	CID:3033677	phase I
BRD-K04111260	CCN1CCC[C@H]1CNC(=O)c1c(O)c(Cl)cc(Cl)c1OC	CID:3033769	phase I
BRD-K63343048	CCCCCCCCCCC[C@@H](C[C@@H]1OC(=O)[C@H]1CCCCCC)OC(=O)[C@H](CC(C)C)NC=O	CID:3034010	phase I
BRD-K54006094	COc1ccc(C[C@H](C)NC[C@@H](O)c2ccc(O)c(NC=O)c2)cc1	CID:3034756	phase I
BRD-K68144790	C[C@H](CCC(=O)NCC(O)=O)[C@H]1CC[C@H]2[C@@H]3CC[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C	CID:3035026	phase I
BRD-K91623615	COc1ccc(cc1)S(=O)(=O)Nc1cccnc1Nc1ccc(O)cc1	CID:3035714	phase I
BRD-K51918615	Ic1ccc(CCNC(=N)SCCCc2c[nH]cn2)cc1	CID:3035746	phase I
BRD-K25906698	C(C1CCNCC1)c1c[nH]cn1	CID:3035842	phase I
BRD-K63874012	S=C(NC1CCCCC1)N1CCC(CC1)c1c[nH]cn1	CID:3035905	phase I
BRD-K55332332	CSc1ccc(cc1)[C@@H]1CN2CCC[C@@H]2c2ccccc12	CID:3036461	phase I
BRD-K57875380	CN1C[C@@H]2[C@@H](C1)c1cc(Cl)ccc1Oc1ccccc21	CID:3036780	phase I
BRD-K45435259	CN1CCc2cc(Cl)c(O)cc2[C@H](C1)c1ccccc1	CID:3036864	phase I
BRD-K17378184	COc1ccccc1N1CCN(CCCCNC(=O)c2ccc3ccccc3c2)CC1	CID:3038495	phase I
BRD-K89162000	COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1	CID:3038522	phase I
BRD-K91900765	Fc1ccc(Sc2ccc3c(-c4c(Cl)cccc4Cl)c(=O)ncn3n2)c(F)c1	CID:3038525	phase I
BRD-A68061604	Cc1ccc(cc1C)C(O)(C2CN3CCC2CC3)c4ccc(C)c(C)c4	CID:3044812	phase I
BRD-K42823101	CN(C)C[C@H](O)c1ccc(O)c(O)c1	CID:3054685	phase I
BRD-K68558722	COc1ccc(cc1F)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(F)F	CID:3058754	phase I
BRD-K49328571	Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CCO)CC1	CID:3062316	phase I
BRD-K77793136	Oc1nccc2c(cccc12)S(=O)(=O)N1CCCNCC1	CID:3064778	phase I
BRD-A26347577	OCC(O)c1ccc(O)cc1	CID:3081980	phase I
BRD-K58223721	NC(=O)C[C@H](NC(=O)Cc1ccc(O)cc1O)C(=O)O	CID:3082629	phase I
BRD-K73290745	CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc(Cl)c(Cl)c1	CID:3082718	phase I
BRD-K91844626	NCCc1c[nH]c2ccc(N)cc12	CID:3083677	phase I
BRD-K66944906	COc1cc2ccc(=O)oc2c(OC)c1OC	CID:3083928	phase I
BRD-A68009927	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(C)=O	CID:3085107	phase I
BRD-K83153774	CN1CCN2[C@@H](C1)c3ccccc3Cc4cccnc24	CID:3085219	phase I
BRD-K24652731	CC[C@H](C)[C@H]1O[C@]2(CC[C@@H]1C)C[C@@H]3C[C@@H](CC=C(C)[C@@H](O[C@H]4C[C@H](OC)[C@@H](O[C@H]5C[C@H](OC)[C@@H](O)[C@H](C)O5)[C@H](C)O4)[C@@H](C)C=CC=C6CO[C@@H]7[C@H](O)C(=C[C@@H](C(=O)O3)[C@@]76O)C)O2	CID:3085416	phase I
BRD-K80451230	C(Cc1ccc2OCOc2c1)N1CCC[C@H](C1)OC(c1ccccc1)c1ccccc1	CID:3086618	phase I
BRD-K49890030	OC(=O)c1[nH]c2cc(Cl)cc(Cl)c2c1C=CC(=O)Nc3ccccc3	CID:3086670	phase I
BRD-K22314899	Cc1cc(ccc1NC(=O)c1ccnn1C)\N=N\c1ccccc1C	CID:3091786	phase I
BRD-K15888437	CCc1cc2c(=O)c(c3nc4ccccc4n3C)c(C)oc2cc1OC(=O)C	CID:3092570	phase I
BRD-K47709646	CCCCC1CCC(CC1)c2ccc(cc2)C(=O)O	CID:3104706	phase I
BRD-K58628167	OCCNC(=O)c1ccc(cc1)N2C(=O)c3ccccc3C2=O	CID:3107687	phase I
BRD-A12633378	Cc1cc(C)c(NC(=O)C2CC3CCC2C3)c(C)c1	CID:3111211	phase I
BRD-K37141476	CCOc1ccc(cc1[N+](=O)[O-])C(=O)Nc2ccc(cc2)c3nc4ccccc4[nH]3	CID:3116236	phase I
BRD-A84238007	CC1CCc2c(C#N)c(NC(=O)c3cc4nc(cc(n4n3)C(F)(F)F)c5ccccc5)sc2C1	CID:3122973	phase I
BRD-K18749194	CC=CCn1c(SCCCc2ccccc2)nc2n(C)c(=O)[nH]c(=O)c12	CID:3123448	phase I
BRD-A93015352	OC(COc1cccc2cccnc12)Cn3c4ccccc4c5ccccc35	CID:3124281	phase I
BRD-K99705204	Cn1c2ccccc2c(Nc2ccc(Cl)cc2)c([N+]([O-])=O)c1=O	CID:3125011	phase I
BRD-A41649729	Cc1ccc(cc1)C2=NNC3(S2)C(=O)Nc4ccccc43	CID:3136666	phase I
BRD-A83255679	Brc1cc2OCOc2cc1C3Nc4ccccc4C5C=CCC53	CID:3136844	phase I
BRD-A71707563	Cc1cc(C)c2C3C=CCC3C(Nc2c1)c4cc5OCOc5cc4Br	CID:3136845	phase I
BRD-K89383912	Cc1cccc(Nc2nc(NCCO)nc(n2)N3CCCC3)c1	CID:3146158	phase I
BRD-A36411721	O=S(=O)(CC(CN1CCCCC1)N2CCCCC2)c3ccccc3	CID:3150672	phase I
BRD-A82628254	CC1CCN(CN2CC(COc3ccccc3C)OC2=O)CC1	CID:3151270	phase I
BRD-K21237738	OCC#CCSc1nnc(o1)c2cccc3ccccc23	CID:3152427	phase I
BRD-A03520402	CC(C)c1ccc(cc1)C2C3CN(C)CC=C3C(C#N)(C#N)C(=C2C#N)N	CID:3156173	phase I
BRD-K24665987	CCOC(=O)N1CCC(CC1)NCCNC(=O)c2ccc(F)cc2	CID:3156884	phase I
BRD-A87455648	CC(C)OCCCNC(=O)c1ccc(cc1)C2SCC(=O)N2Cc3ccco3	CID:3157053	phase I
BRD-K84864079	Cc1ccc(OCCn2c(CCNC(=O)C3CCCCC3)nc3ccccc23)cc1	CID:3159995	phase I
BRD-K91863345	Oc1nc2ccccc2nc1c3ccccc3NC(=O)c4cccs4	CID:3162043	phase I
BRD-K28916077	CCCc1nn(C)c2nc(=O)n(C)c(=O)c2n1	CID:3164059	phase I
BRD-K41652870	COc1ccc(cc1)-c1csc(NC(=O)CSc2nnc3c(C)cc4cc5OCCOc5cc4n23)n1	CID:3190037	phase I
BRD-K06652922	COc1ccc(cc1)-c1csc(NC(=O)CSc2nnc3c(C)cc4cc5OCOc5cc4n23)n1	CID:3190055	phase I
BRD-A11929187	CC1CCc2c(C1)sc3nc(C)nc(N4CCN(CC4)C(=O)c5ccco5)c23	CID:3193014	phase I
BRD-A42969626	CC1CCc2c(C1)sc1nc(C)nc(N3CCN(CC3)C(=O)C3CC3)c21	CID:3193022	phase I
BRD-K98856658	COc1cccc(c1)c2csc(n2)N3CCN(CC3)C(=Nc4cccc(Cl)c4)S	CID:3223669	phase I
BRD-K95807833	COc1ccc(cc1)-c1cc2nc(cc(N3CCN(CC3)C(C)=O)n2n1)-c1ccccc1	CID:3230028	phase I
BRD-K23978082	Cc1ccccc1NC(=O)NCC2CCN(CC2)c3ccc(cc3)S(=O)(=O)N4CCOCC4	CID:3232217	phase I
BRD-K70693222	C(Nc1ncnc2ccc(cc12)c3ccc4OCOc4c3)c5cccs5	CID:3232621	phase I
BRD-K44978960	CN(Cc1ccco1)c2ncnc3ccc(cc23)c4ccc5OCOc5c4	CID:3233012	phase I
BRD-K54168141	COc1cccc(c1)c2ccc3ncnc(N(C)Cc4ccco4)c3c2	CID:3233276	phase I
BRD-K79491139	Cc1cccc(CNc2ncnc3ccc(cc23)c4ccc5OCOc5c4)c1	CID:3234028	phase I
BRD-K73304092	Clc1ccccc1c2ccc3ncnc(NCc4cccnc4)c3c2	CID:3234184	phase I
BRD-K57457519	Cc1cccc(CNc2ncnc3ccc(cc23)c4ccoc4)c1	CID:3234345	phase I
BRD-K28366444	C(Nc1ncnc2ccc(cc12)c3cccnc3)c4cccnc4	CID:3234518	phase I
BRD-K07668032	C(Nc1ncnc2ccc(cc12)c3ccoc3)c4cccs4	CID:3234850	phase I
BRD-K01333970	C(Nc1ccnc(n1)-c1ccc2OCOc2c1)c1cccnc1	CID:3234998	phase I
BRD-K63569039	COc1cccc(c1)c2ccc3ncnc(NCc4cccnc4)c3c2	CID:3235086	phase I
BRD-K25373946	CN(Cc1ccco1)c2ncnc3ccc(cc23)c4ccccc4Cl	CID:3235166	phase I
BRD-K74292317	COc1cccc(c1)c2ccc3ncnc(NCc4cccs4)c3c2	CID:3235398	phase I
BRD-K04779531	C(Nc1ncnc2ccc(cc12)c3ccoc3)c4cccnc4	CID:3235429	phase I
BRD-K78189262	Cc1cccc(CNc2ncnc3ccc(cc23)c4cccnc4)c1	CID:3235537	phase I
BRD-K93229693	COc1cccc(c1)-c1nc(no1)-c1ccc(NC(=O)Cc2ccccc2OC)cc1	CID:3236979	phase I
BRD-A03772856	COc1ccccc1C2N(C(=O)C3CCCN23)c4ccc(Cl)cc4	CID:3237298	phase I
BRD-K92742972	CCOc1ccc(cc1)c2nc(CSCC(=O)NCc3ccco3)c(C)o2	CID:3237327	phase I
BRD-K84203638	Cc1ccnc(NC(=O)CCCOc2cc(=O)n(C)c3ccccc23)c1	CID:3237904	phase I
BRD-K53423944	Clc1cccc(c1)N2CCN(CC2)c3cc(=O)n(C4CCCCC4)c(=O)[nH]3	CID:3238389	phase I
BRD-K60870698	Oc1c(CN2CCCCC2)cc(COCc3ccccc3)c4cccnc14	CID:3238417	phase I
BRD-A98248982	COc1ccc(CCN(C)C(=O)C2CCCN(Cc3ccc(OC)c(OC)c3)C2)cc1OC	CID:3238551	phase I
BRD-K33182644	Cc1cccc(Nc2nn3c(=O)c4ccccc4nc3s2)c1	CID:3238944	phase I
BRD-K18595892	CCCN(CCC)CCNC(=O)C1CCN(Cc2nc(oc2C)c3ccc(Cl)cc3)CC1	CID:3240581	phase I
BRD-A73747855	CC1CCCN(C1)C(C(=O)Nc2ccc3OCCOc3c2)c4ccccc4	CID:3240990	phase I
BRD-K95760042	Cc1cccn2c(=O)c(/C=N/c3ccc(Cl)cc3)c(NCCO)nc12	CID:3241836	phase I
BRD-K95196255	CN1CCN(Cc2cc(COCc3ccccc3)c4cccnc4c2O)CC1	CID:3242434	phase I
BRD-K82747512	O=C(CCNS(=O)(=O)c1cccc2nsnc12)N3CCN(CC3)c4ccccn4	CID:3242997	phase I
BRD-K95149906	C/C(=C\1/SC(=NC1=O)N2CCCC2)/c3ccc(Br)cc3	CID:3243424	phase I
BRD-K45443730	Cc1cccc(c1)n2cnc3cc(ccc23)C(=O)N4CCCCC4	CID:3243760	phase I
BRD-K37150847	COC(=O)Cn1nc(c2ccccc2)c3ccccc13	CID:3243873	phase I
BRD-K23980805	Brc1c[nH]c2nc(SCc3ccccc3C#N)nc2c1	CID:3245059	phase I
BRD-K10833576	CCOc1ccc(NC(=O)CN2CCN(CC(=O)Nc3cc(OC)cc(OC)c3)CC2)cc1	CID:3245746	phase I
BRD-K16233984	Oc1cc(c2cc(ccc2c1N=Nc3ccc4ccccc4c3O)[N+](=O)[O-])S(=O)(=O)O	CID:3246023	phase I
BRD-K61480498	C[C@H](CC[C@@H]1OC1(C)C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:3247059	phase I
BRD-K80639402	COc1ccc(NS(=O)(=O)c2ccc(I)cc2)cc1N1CCN(C)CC1	CID:3248571	phase I
BRD-A53107311	CC(C)OC(=O)C1=C(C)N=c2sc(=Cc3ccc(OCC(=O)O)cc3)c(=O)n2C1c4ccc(Cl)cc4	CID:3266419	phase I
BRD-A08003242	CCC(C)C(=O)c1c(O)c(C)c2oc3c(C)c(O)c(C(=O)C(C)CC)c(O)c3c2c1O	CID:3270699	phase I
BRD-K27141178	O=C(OCCN1CCCCC1)c1c[nH]c2ccccc12	CID:3272300	phase I
BRD-K47717570	NS(=O)(=O)c1cccc2c3nc(O)c(O)nc3cc([N+](=O)[O-])c12	CID:3272524	phase I
BRD-A11609859	CN1CCC2(Cc3nc4ccccc4cc3CC2C1)c5cccc(O)c5	CID:3277599	phase I
BRD-K78883024	Cc1c([n+]2ccccc2n1C)P(=S)(c3ccccc3)c4ccccc4	CID:3278392	phase I
BRD-K68866125	Cc1ccc2[nH]/c(=N\C(=O)C(C)(C)C)/sc2c1	CID:3290072	phase I
BRD-K30867024	COc1ccc(NC(=O)c2ccc(cc2)-c2ccc(cc2C)-c2noc(C)n2)cc1OCCN(C)C	CID:3292447	phase I
BRD-A94675310	CN(C(CN1CCCC1)c2ccccc2)C(=O)Cc3ccccc3	CID:3298213	phase I
BRD-K39522184	Cc1cc(ccc1[N+](=O)[O-])C(=O)Nc2nc[nH]n2	CID:3301126	phase I
BRD-K61220632	COC(=O)c1c(C)c2Oc3c(Cl)c(OC)c(Cl)c(C)c3C(=O)Oc2c(C)c1OC	CID:3310692	phase I
BRD-K06159959	OC(=O)Cc1cc2ccccc2nc1C(O)=O	CID:3337816	phase I
BRD-K97274161	CC(C)N(CCNC(=O)c1ccc(CNS(=O)(=O)c2ccc(C)cc2)cc1)Cc3ccccc3	CID:3342390	phase I
BRD-K37413063	COc1ccc(OC)c(NC(=O)c2ccccc2OC(=O)C)c1	CID:3361211	phase I
BRD-K68102868	CC(=O)Oc1ccccc1C(=O)Nc2ccccc2	CID:3364609	phase I
BRD-K95606637	CSc1nc(nc(n1)c2ccc(C)cc2)C(Cl)Cl	CID:3380841	phase I
BRD-K16664969	c1ccc(cc1)-c1n[nH]c2c1oc1ccccc21	CID:3385203	phase I
BRD-A06352508	O=C1NC(=O)c2c1c1c3ccccc3n3C4CCC(O4)n4c5ccccc5c2c4c13	CID:3387354	phase I
BRD-K48716658	CNc1nc(N)c([N+](=O)[O-])c(Nc2cccc(Cl)c2)n1	CID:3392161	phase I
BRD-A51929314	OC(=O)CCCC=CCC1COC(OC1c2ccccc2O)C(F)(F)F	CID:3392534	phase I
BRD-K96263742	CC(C)(Sc1ccc(CCN(CCCCC2CCCCC2)C(=O)NC2CCCCC2)cc1)C(O)=O	CID:3392731	phase I
BRD-K92726801	C[N+]1=Cc2cc3OCOc3cc2CC1	CID:3397945	phase I
BRD-A71262238	CCCCN1CCCC1CNC(=O)c1cc(C#N)c2ccccc2c1OC	CID:3408722	phase I
BRD-A06664848	CC(Sc1nc2cc(Cl)ccc2s1)C(=O)Nc3cccc(c3)S(=O)(=O)N4CCOCC4	CID:3409332	phase I
BRD-K56115039	C1CN=C(N1)c2cc3ccccc3cn2	CID:3410883	phase I
BRD-K73610817	Oc1c(CN2CCCC2)cc(COCc3ccccc3)c4cccnc14	CID:3426979	phase I
BRD-K10355322	CC(=NOC(=O)c1ccc(F)cc1)c2nccs2	CID:3427192	phase I
BRD-K28167849	COc1cc2OCOc2cc1c3coc4c5C=CC(C)(C)Oc5c(OC)cc4c3=O	CID:3428129	phase I
BRD-K54405293	CNc1nc(N)c(c(Nc2ccccc2)n1)[N+]([O-])=O	CID:3449329	phase I
BRD-K38910949	O=C(Nc1ccccc1)c2cccc(c2)S(=O)(=O)NCCC3(CC4CC5CC(C4)C3)C5	CID:3455588	phase I
BRD-K48112880	Cc1cc(ccc1NS(=O)(=O)c1cc(Cl)ccc1Cl)[N+]([O-])=O	CID:3463933	phase I
BRD-K53445087	CC(=O)NN=C(C)c1ccc(NC(=O)C2CC2)cc1	CID:3464963	phase I
BRD-K06014311	CCCCC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12	CID:3467177	phase I
BRD-K52620403	OC(=O)c1ccc2c3nc4ccccc4n3c(=O)c5cccc1c52	CID:3467590	phase I
BRD-K94919853	Cc1ccc(cc1)C(=O)N2c3ccccc3Sc4ccccc24	CID:3473393	phase I
BRD-A20846977	Cc1ccc(NC(=O)C2CC3CCC2C3)c(C)c1	CID:3473417	phase I
BRD-A75817871	Cc1ccc2N=C3N(CCC3(O)C(=O)c2c1)c1ccccc1	CID:3476986	phase I
BRD-K66224104	Cc1ccc(NCn2c(=O)oc3ccccc23)cc1	CID:3477497	phase I
BRD-A90490067	CC12CCC3C(C2CCC1O)C(CCCCCCCCCS(=O)CCCC(F)(F)C(F)(F)F)Cc4cc(O)ccc34	CID:3478439	phase I
BRD-A55369275	CC(NCC(O)CP(=O)(O)CC1CCCCC1)c2ccc(Cl)c(Cl)c2	CID:3489614	phase I
BRD-A83402799	CN(Cc1ccccc1)C(=O)C2CCCN(Cc3cccc(Cl)c3)C2	CID:3500831	phase I
BRD-A11483079	CC(C)C1COc2cc3oc(=O)ccc3cc2O1	CID:3503044	phase I
BRD-A24054354	CCN1CCN(CC1)C(c2cccnc2)c3cc(Cl)c4cccnc4c3O	CID:3516032	phase I
BRD-K95851186	CC(C)(Cc1cc(c(O)c(c1)C(C)(C)C)C(C)(C)C)C=O	CID:3519541	phase I
BRD-K07161233	CNc1nc(N)c([N+](=O)[O-])c(Nc2cccc(F)c2)n1	CID:3528206	phase I
BRD-K37061750	COc1ccc(cc1NC(=O)c2ccc(cc2)n3nc(C)cc3C)S(=O)(=O)N4CCOCC4	CID:3538139	phase I
BRD-A62890442	CC(CN)CC(O)=O	CID:3539719	phase I
BRD-K96362535	COc1c(ccc2OC(C)(C)CCc12)C(=O)O	CID:3548249	phase I
BRD-K49181186	Fc1cc(F)c(c(F)c1Cl)S(=O)(=O)NNC(=O)C2(CC3CC4CC(C3)C2)C4	CID:3550807	phase I
BRD-A96882008	CC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)OCc3cc(cc(c3)C(F)(F)F)C(F)(F)F	CID:3563638	phase I
BRD-A70155556	CCC(C)C(=O)OC1CC(C)C=C2C=CC(C)C(CCC(O)CC(O)CC(=O)O)C12	CID:3565209	phase I
BRD-K08640512	Cc1c[nH]c(=O)n(CCCN2CCN(CC2)c2ccccc2OCC(F)(F)F)c1=O	CID:3567002	phase I
BRD-K77856555	Cc1ccc2c(Cl)c(sc2c1)C(=O)NCCCN1CCOCC1	CID:3579902	phase I
BRD-A48257147	ON=C1C2CC2(Oc3ccccc13)C(=O)Nc4ccccc4	CID:3579925	phase I
BRD-A74382794	COc1cc(cc(OC)c1OC)C(=O)NCCC(=O)NC2CCCc3ccccc23	CID:3593902	phase I
BRD-K75477256	C(N1CCN(CC1)c1ncnc2sccc12)c1ccccc1	CID:3610226	phase I
BRD-K14232336	Cc1c(N=Cc2cc(Br)cc(Br)c2O)cccc1C(=O)O	CID:3610881	phase I
BRD-A22997170	Cc1[nH]c2ccccc2c1C(Nc1ccccn1)c1ccc(Cl)cc1	CID:3634881	phase I
BRD-K51276371	CCCCc1c([nH]c2nccnc12)c3ccc(OC)cc3	CID:3641059	phase I
BRD-K47761761	Cc1cccc(c1)C(=O)NCN1CCN(CC1)c1ccccc1C#N	CID:3645619	phase I
BRD-A75931230	Cc1[nH]c2ccccc2c1C(Nc3cc(C)ccn3)c4ccc(Cl)cc4	CID:3646984	phase I
BRD-K61106942	Clc1cccc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)c1	CID:3647906	phase I
BRD-K86652643	Cc1ccccc1NS(=O)(=O)c1ccc2NC(=O)CCc2c1	CID:3648364	phase I
BRD-K59556282	Clc1ccccc1C(=O)N(c2ccc3oc(=O)sc3c2)S(=O)(=O)c4ccc(Br)cc4	CID:3650962	phase I
BRD-K20168484	CC(C)c1ccc2n(Cc3ccc(Cl)cc3)c(CC(C)(C)C(=O)O)c(SC(C)(C)C)c2c1	CID:3651377	phase I
BRD-A51829654	OC(CN1CCN(CC1)c1cccc(Cl)c1)C(c1ccccc1)c1ccccc1	CID:3654103	phase I
BRD-K94580036	Cc1ccc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)cc1	CID:3656150	phase I
BRD-K47664560	CC(=O)Nc1ccc(cc1)C(=O)Nc1ccccc1O	CID:3682562	phase I
BRD-K10484463	Cn1c(=NC(=O)CCl)sc2ccccc12	CID:3685735	phase I
BRD-A36275421	COc1ccc(cc1Cl)N(C(C(=O)NCCc2ccccc2)c3cccs3)C(=O)CCl	CID:3689413	phase I
BRD-A39093044	COc1cccc(c1)N(C(C(=O)NCCc2ccccc2)c3cccs3)C(=O)CCl	CID:3689415	phase I
BRD-A72180425	COc1ccc(cc1)N(C(C(=O)NCCc2ccccc2)c3cccs3)C(=O)CCl	CID:3689416	phase I
BRD-K87048468	COc1cc(OC)c(cc1NS(=O)(=O)c1ccc(cc1)C(F)(F)F)C(=O)CCCCN1CCC2(CC1)NC(=O)NC2=O	CID:3693566	phase I
BRD-K07653295	Cc1[n+](C)ccc2ccccc12	CID:3708824	phase I
BRD-A94567954	COc1ccc(cc1OC)C2c3c(Oc4ccc5ccccc5c24)ncn(CCN6CCOCC6)c3=N	CID:3719993	phase I
BRD-K53545112	Oc1nc2cc(C#N)c(cc2nc1O)[N+](=O)[O-]	CID:3721046	phase I
BRD-K24346336	CNc1nc(N)c(c(Nc2ccc(F)cc2)n1)[N+]([O-])=O	CID:3739601	phase I
BRD-K27688565	CN1CCN(CC1)C2=C(NS(=O)(=O)c3ccccc3)C(=O)c4ccccc4C2=O	CID:3763775	phase I
BRD-A42553870	CC1(C)CC(=O)C(C2c3ccccc3OC3=C2C(=O)CC(C)(C)C3)C(=O)C1	CID:3765615	phase I
BRD-A60256353	OC(=O)CC1N=Cc2ccccc12	CID:3780913	phase I
BRD-A25337146	Brc1ccc(cc1)C(=O)C(CN2CCOCC2)c3ccccc3	CID:3816756	phase I
BRD-K28284219	OS(=O)(=O)CCN1C(=S)SC(=Cc2cn(nc2-c2ccc(OCc3ccccc3F)cc2)-c2ccccc2)C1=O	CID:3823393	phase I
BRD-A85648045	CCC1(O)CC2CN(C1)CCc1c([nH]c3ccccc13)C(C2)(C(=O)OC)c1cc2c(cc1OC)N(C)C1C22CCN3CC=CC(CC)(C23)C(OC(C)=O)C1(O)C(=O)OC	CID:3823887	phase I
BRD-K35100517	CC(=NOC(=O)C1CCCCC1)c1nccs1	CID:3830711	phase I
BRD-A81372523	Cc1cccc(NC(=O)C2CC3CCC2C3)c1C	CID:3843095	phase I
BRD-K61323504	Oc1cc(ccc1NC(=O)Nc1ccccc1Br)[N+]([O-])=O	CID:3854666	phase I
BRD-K08115555	Oc1cc(C=C(C#N)C#N)cc([N+](=O)[O-])c1O	CID:3856780	phase I
BRD-A29119732	COc1ccc(cc1OC)C(O)CN	CID:3863978	phase I
BRD-K76840893	CC(C)(Cc1c[nH]c2ccc(Cl)cc12)NCCOc1ccccc1OCC1CC1	CID:3894573	phase I
BRD-K85266041	Oc1nc2cc([N+](=O)[O-])c(cc2nc1O)[N+](=O)[O-]	CID:3899541	phase I
BRD-K36009368	COC(=O)CN1CN(c2ccccc2)C3(CCN(Cc4ccc5ccccc5c4)CC3)C1=O	CID:3906780	phase I
BRD-A39522003	CCCCCCCCC=CCCCCCCCC(=O)NC(CO)Cc1ccc(O)cc1	CID:3906781	phase I
BRD-A62021152	Clc1cc2NC(=O)C3CNCCN3c2cc1Cl	CID:3906894	phase I
BRD-A47832959	CC(Sc1cc(C)c2ccccc2n1)C(=O)Nc3ncc(Cl)cc3Cl	CID:3913264	phase I
BRD-K75302809	Cc1ccc(C=NNC(=O)CCC(=O)Nc2ccc(C)cc2C)o1	CID:3913840	phase I
BRD-A14014306	CC1=NN(C(=O)C1Cc2ccccc2)c3nc4ccccc4[nH]3	CID:3915969	phase I
BRD-K19049172	Cc1cccc(C)c1NC(=O)C2(CCCC2)N(Cc3ccccc3)C(=O)c4ccc(cc4)n5cnnn5	CID:3917094	phase I
BRD-A02176148	CC(=C)C1Cc2c(O1)ccc(C(=O)O)c2O	CID:3919910	phase I
BRD-A03946276	[O-][N+](=O)c1ccc2NC(=O)C3(NNc4ccccc4O3)c2c1	CID:3921071	phase I
BRD-K26997899	COc1ccc2[nH]c(cc2c1)C(=O)c1ccccc1	CID:3921152	phase I
BRD-K98490050	COc1cc(NS(=O)(=O)C)ccc1Cc2c3ccccc3nc4ccccc24	CID:3926765	phase I
BRD-K18678457	CCN(c1ccccc1)c1cc(NC)[n+](C)c(C)n1	CID:3938007	phase I
BRD-K28453807	CCN(CC)CCOC(=O)C1(CCCC1)c1ccc(cc1)[N+]([O-])=O	CID:3941250	phase I
BRD-A74134989	CCC(C)(N(Cc1cccs1)C(=O)c2ccccn2)C(=O)NC3CCCC3	CID:3950572	phase I
BRD-K51973945	O=C(NC1CCCCC1)C2(CCCCC2)N(Cc3ccco3)C(=O)c4ccccn4	CID:3950926	phase I
BRD-K04722205	[O-][N+](=O)c1ccc(N2CCN(CC2)C(=O)c2ccc(Cl)cc2)c2cccnc12	CID:3953303	phase I
BRD-A83802330	CCC(C)(N(Cc1ccco1)C(=O)c2ccccn2)C(=O)NC3CCCCC3	CID:3964693	phase I
BRD-K14355517	Cc1c(c2ccccc2n1C)P(=S)(c1ccccc1)c1ccccc1	CID:3989078	phase I
BRD-K66093087	CCCCCCN(CCCCCC)C(=O)Cc1c([nH]c2ccc(Cl)cc12)-c1ccc(Cl)cc1	CID:3995234	phase I
BRD-A54077041	CC(OC(=O)C1=NNC(=O)CC1)C(=O)c2cc(C)n(c2C)c3ccc(OC(F)F)cc3	CID:4003359	phase I
BRD-A36630025	CCc1c2Cn3c(cc4c(COC(=O)C4(O)CC)c3=O)-c2nc5ccc(O)cc15	CID:4014291	phase I
BRD-A30395175	NC(C(=O)O)c1ccc(O)c(c1)C(=O)O	CID:4014619	phase I
BRD-K89832926	O=C(NC1CCCCC1)C2(CCCCC2)N(Cc3cccs3)C(=O)c4cnccn4	CID:4014737	phase I
BRD-A10715913	CCN1CCC(CNC(=O)c2cc(ccc2OC)S(=O)(=O)N)C1	CID:4018928	phase I
BRD-K05433219	CC(=CCc1c2OC(C)(C)C=Cc2c(O)c3c(=O)c(O)c(oc13)c4ccccc4)C	CID:4020240	phase I
BRD-K63938928	COC(=O)c1cc(OC)c(=O)c2c(OC)c(OC)ccc2c1	CID:4020695	phase I
BRD-K33860217	CCCOc1ccc2[nH]cc(C3=CCNCC3)c2n1	CID:4029677	phase I
BRD-A00267231	CCCCC#Cc1nc(NC)c2ncn(C3OC(CO)C(O)C3O)c2n1	CID:4043357	phase I
BRD-K08174547	OS(=O)(=O)CCN1C(=S)SC(=Cc2cn(nc2-c2ccc(OCc3ccccc3)cc2)-c2ccccc2)C1=O	CID:4050965	phase I
BRD-K40329609	CN1CCc2c(C1)sc(NC(C)=O)c2-c1nc2ccccc2s1	CID:4055306	phase I
BRD-K66555411	Cc1ccc(cc1)-c1nn(cc1C=C1SC(=S)N(CCS(O)(=O)=O)C1=O)-c1ccccc1	CID:4064091	phase I
BRD-A43885598	CCOC(=O)C(C)Oc1cccc2c1ccn(CC(=O)Nc1ccc3OCCOc3c1)c2=O	CID:4076092	phase I
BRD-K15601958	FC(F)(F)c1sc(cc1-c1ccccc1)-c1nc(no1)-c1cccc(c1)C(F)(F)F	CID:4077460	phase I
BRD-A97833537	Fc1ccccc1C(=O)N2CC(=O)Nc3ccc(Cl)cc3C2c4ccccc4	CID:4084010	phase I
BRD-K54070802	OC(=O)c1ccccc1NS(=O)(=O)c2cccc(c2)n3sc4ccccc4c3=O	CID:4089709	phase I
BRD-K59331372	COc1cccc(NC(=O)C=Cc2ccc(Cl)cc2)c1	CID:4099413	phase I
BRD-A32214171	CCN1CCN(CC1)C(c2cccnc2)c3ccc4cccnc4c3O	CID:4124546	phase I
BRD-A17664363	CCOC(=O)C(C)Oc1cccc2c1ccn(CC(=O)Nc1ccc(OC)cc1)c2=O	CID:4131581	phase I
BRD-A05874290	NC(C(OCc1ccccc1)C(=O)O)C(=O)O	CID:4133412	phase I
BRD-K47695085	O=C1CCc2cc(ccc2N1)S(=O)(=O)Nc1ccc2OCCOc2c1	CID:4149969	phase I
BRD-K67550673	CCOc1ccc(cc1)c2nc(CSCC(=O)NC3CC3)c(C)o2	CID:4174238	phase I
BRD-K50234570	[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc2cccc(NC(=O)c3cc(ccc3Cl)[N+](=O)[O-])n2	CID:4183496	phase I
BRD-A46802340	CC1CN(CC(C)O1)S(=O)(=O)c2ccc(cc2)C(=O)/N=c\3/sc4cccc(Cl)c4n3C	CID:4190864	phase I
BRD-A84389091	CCOC(=O)c1ncn-2c1C3CCCN3C(=O)c4cc(OC)ccc42	CID:4203080	phase I
BRD-A03926027	NC1=C(C#N)C(c2ccc(Br)cc2)c3c(N1)c4ccccc4oc3=O	CID:4207396	phase I
BRD-A99518825	COc1ccc(CN2CCCC(C2)C(=O)N3CCCC3)c(OC)c1OC	CID:4207918	phase I
BRD-K76805682	Oc1ccc(NC2=C(C(=O)NC2=O)c2ccccc2[N+]([O-])=O)cc1Cl	CID:4210951	phase I
BRD-A02836799	OCCOc1ccccc1C1N2C(C(C(=O)N3CCCCCCC3)C11C(=O)Nc3ccccc13)C(=O)OC(C2c1ccccc1)c1ccccc1	CID:4211082	phase I
BRD-K63792901	CC#CCOC(=O)C1=CCCN(C)C1	CID:4214594	phase I
BRD-K29622226	Clc1ccc(OCC(=O)NCc2n[nH]c(=S)n2c3cccc(Cl)c3)cc1	CID:4220279	phase I
BRD-A25852922	COC(=O)C1=C(N)N(C2=C(C1c3ccccc3)C(=O)CCC2)c4cccc(c4)C(F)(F)F	CID:4221587	phase I
BRD-A23683907	C(Oc1cccc2C=C(CN3CCOCC3)COc12)C4CNCCO4	CID:4233538	phase I
BRD-K23872647	Cc1cc2C(=O)C(=C(C(=O)c2cc1C)c3ccccc3)NCc4ccccc4	CID:4234918	phase I
BRD-A06276885	Oc1ccc2CC3N(CC4CC4)CCC5(C6Oc1c25)C3(O)Cc7c6n(Cc8ccccc8)c9ccccc79	CID:4257102	phase I
BRD-K58214070	[O-][N+](=O)c1ccc(cc1)N(CCCNC(=O)C(F)(F)F)C(=O)CCl	CID:4257368	phase I
BRD-K17140735	CC(C)c1ccc(Cn2ccc3c2ccc4nc(NC5CC5)nc(N)c34)cc1	CID:4259181	phase I
BRD-A28422058	OC(=O)C1CC(NC(=O)Nc2ccccc2)c3c(Cl)cc(Cl)cc3N1	CID:4267713	phase I
BRD-K17796732	CCCn1c(C)c(C(=O)c2cccc3ccccc23)c4ccccc14	CID:4273754	phase I
BRD-K83023055	COC(=O)Nc1ccc2[nH]cc(CCNC(C)=O)c2c1	CID:4284525	phase I
BRD-A17428743	CC(N)Cc1c[nH]c2ccc(OCc3cccs3)cc12	CID:4284720	phase I
BRD-K78797196	O=C(Nc1cccc(c1)S(=O)(=O)N2CCOCC2)c3ccc(cc3)N4CCCC4=O	CID:4292126	phase I
BRD-A26777759	O=C(Nc1ccc2ccccc2c1)C1CC2CCC1C2	CID:4296446	phase I
BRD-A64850503	CCOC(=O)C1=C(C)N=c2sc(=Cc3ccc(OCC(=O)O)cc3)c(=O)n2C1c4ccc(SC)cc4	CID:4302116	phase I
BRD-K50891186	COc1ccccc1N1CCN(CCCCNC(=O)c2ccc(cc2)-c2ccc(cc2)C(C)=O)CC1	CID:4302960	phase I
BRD-K59419204	Cc1c(nn(c1-c1ccc(I)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCOCC1	CID:4302962	phase I
BRD-K63533170	COc1ccc(cc1)C(=O)c1c(C)n(CCN2CCOCC2)c2cc(I)ccc12	CID:4302963	phase I
BRD-A38747044	CCC1(Cc2ccccc2O1)c1ncc[nH]1	CID:4302964	phase I
BRD-K14767410	COc1ccc(cc1)-n1nc(cc1-c1ccc(Cl)cc1)C(F)(F)F	CID:4306515	phase I
BRD-K80307267	COc1ccc2C(=O)c3cc(OC)c(OC)cc3CC(=O)COc2c1OC	CID:4309557	phase I
BRD-A89208012	OC(=O)CCC=CCC1COC(OC1c2ccccc2O)c3ccccc3Cl	CID:4330476	phase I
BRD-K53913732	CN(C)c1ccc(NC(=O)Nc2cc(C)nc3c(F)cc(F)cc23)cc1	CID:4331799	phase I
BRD-K52512893	CC(=O)NNC(=O)N1Cc2ccccc2Oc2ccc(Cl)cc12	CID:4336830	phase I
BRD-K14939371	CC(=O)Nc1sc2CN(CCc2c1-c1nc2ccccc2s1)C(C)=O	CID:4348310	phase I
BRD-K01648091	CN1CCc2c(Cc3ccccc3CC1)[nH]c4ccccc24	CID:4350931	phase I
BRD-A80641450	CC(C)CC(NC(=O)N1CCCCCC1)C(=O)NC(Cc2cn(C)c3ccccc23)C(=O)NC(Cc4ccccn4)C(=O)O	CID:4353886	phase I
BRD-K33864865	CC(C)Oc1cccc(c1)-n1c(CCc2c[nH]c3ccc(Br)cc23)nc2ccccc2c1=O	CID:4355450	phase I
BRD-K40656405	CCCc1c(O)c(CC=O)ccc1OCCCOc2ccc(OCC(=O)O)cc2	CID:4364841	phase I
BRD-K15402119	C\C=C1/[C@H]2Cc3[nH]c(=O)ccc3[C@]1(N)CC(C)=C2	CID:4369233	phase I
BRD-K18518344	C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@@H](O)CC[C@]34C)[C@@]1(O)CC[C@@H]2C1=CC(=O)OC1	CID:4369270	phase I
BRD-K19416115	N[C@@H](CC(=O)N1CCn2c(C1)nnc2C(F)(F)F)Cc1cc(F)c(F)cc1F	CID:4369359	phase I
BRD-K82823804	Oc1ccc2[nH]c3cc(c4C(=O)NC(=O)c4c3c2c1)-c1ccccc1	CID:4369491	phase I
BRD-A37735495	Fc1ccc(cc1)N(C(C(=O)NC2CCCCC2)c3cccnc3)C(=O)CCl	CID:4380267	phase I
BRD-A76490030	Cc1ccc(cc1C)N(C(C(=O)NC2CCCCC2)c3cccnc3)C(=O)CCl	CID:4381125	phase I
BRD-A58924247	COc1ccc(cc1)N(C(C(=O)NC2CCCCC2)c3cccnc3)C(=O)CCl	CID:4381126	phase I
BRD-A68065211	ClCC(=O)N(C(C(=O)NC1CCCCC1)c2cccnc2)c3cccc(Cl)c3	CID:4381127	phase I
BRD-A90643929	OCCOc1ccccc1C1N2C(C(C(=O)NCC(O)c3ccccc3)C11C(=O)Nc3ccc(cc13)C#CC1=CCCCC1)C(=O)OC(C2c1ccccc1)c1ccccc1	CID:4387699	phase I
BRD-K97019106	CC(=O)N1CC[N+](C)(C)CC1	CID:4392675	phase I
BRD-A33084410	NC(=N)Nc1ccc2[nH]c3C4Oc5c6c(CC7N(CC8CC8)CCC46C7(O)Cc3c2c1)ccc5O	CID:4396344	phase I
BRD-A03816571	CCCCCCC(C)(C)c1ccc(C2CC(O)CCC2CCCO)c(O)c1	CID:4412255	phase I
BRD-A38275906	CCC(=O)NC1CC2C(OC1=O)c3cccc(C)c3NC2=O	CID:4423427	phase I
BRD-A55142378	O=C1C2CC=CCC2C(=O)N1C3CC(=O)C4OCC3O4	CID:4423767	phase I
BRD-K09460252	Nc1nc(Nc2cccc(F)c2)nc(Nc2cccc(F)c2)c1[N+]([O-])=O	CID:4431362	phase I
BRD-K25144184	O=C(CN1C(=O)CCC1=O)Nc2cccc3C(=O)NC(=O)c32	CID:4432160	phase I
BRD-K13725475	CC(C)CC(=O)c1c(O)c(C)c(O)c2c1oc3c(C(=O)CC(C)C)c(O)c(C)c(O)c32	CID:4445621	phase I
BRD-K36591038	Clc1nssc1=Nc2nncs2	CID:4453692	phase I
BRD-A45206415	Cc1noc(C)c1C(c2ccccc2)S(=O)(=O)c3ccc(C)cc3	CID:4460128	phase I
BRD-K54987996	OC(=O)CN1C(=O)c2c(C1=O)c(I)c(I)c(I)c2I	CID:4462449	phase I
BRD-A94570195	Nc1ncnc2Oc3ccc4ccccc4c3C(c5ccccc5)c12	CID:4464266	phase I
BRD-A26595446	Cc1cccc(C)c1NC(=O)C(Cl)C(=O)c2ccccc2	CID:4484064	phase I
BRD-A15415227	CN(CCOc1ccc(CC(Nc2ccccc2C(=O)c2ccccc2)C(O)=O)cc1)c1ccccn1	CID:4516886	phase I
BRD-K37724988	CCc1ccc(C=C2SC(=S)N(CCCC(=O)Nc3ccc(cc3)C(O)=O)C2=O)cc1	CID:4518240	phase I
BRD-A06784547	CCOC(=O)C1=C(C)NC(=C(C1C#Cc2ccccc2)C(=O)OCc3ccc(cc3)[N+](=O)[O-])c4ccccc4	CID:4519822	phase I
BRD-K11696279	C1CN=C(N1)c1cnc2ccccc2n1	CID:4520732	phase I
BRD-K67298865	NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccccn1)-c1ccc2OCOc2c1	CID:4521392	phase I
BRD-K17743697	NC(=N)SCCc1ccc(OCc2ccc(cc2)[N+]([O-])=O)cc1	CID:4534086	phase I
BRD-K77690805	Cc1ccc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)cc1C	CID:4547230	phase I
BRD-K41603276	COC(=O)c1c(C)c2Oc3c(Cl)c(O)c(Cl)c(C)c3C(=O)Oc2cc1OC	CID:4565183	phase I
BRD-K69396629	Cc1cc(C)n2ncc(C(=O)Nc3ccc4CCCc4c3)c2n1	CID:4573811	phase I
BRD-A54029483	CN(C(Cc1ccc(cc1)c2ccccc2)C(=O)NC(Cc3c[nH]c4ccccc34)C(=O)O)C(=O)c5cc(C)cc(C)c5	CID:4574540	phase I
BRD-K21009077	OS(=O)(=O)CCN1C(=S)SC(=Cc2cn(nc2-c2ccc(OCc3ccc(Cl)cc3)cc2)-c2ccccc2)C1=O	CID:4601225	phase I
BRD-K56518176	Nc1ccc(cc1)C(=O)Nc2ccc(cc2N)C(=O)O	CID:4602050	phase I
BRD-A71339955	CCc1sc(nc1c2ccccc2)N3C(=O)C4C5CCC(C4C3=O)C5=C(C)C	CID:4624993	phase I
BRD-A32582647	CCN1CCCC1c1cccnc1	CID:4658388	phase I
BRD-A76463343	Cc1ccc(NC(=O)C2CC3CCC2C3)cc1	CID:4658599	phase I
BRD-K92977333	CCN(CC)C(=O)C(=Cc1cc(O)c(O)c(c1)[N+]([O-])=O)C#N	CID:4659568	phase I
BRD-K10852020	Cc1ccc(cc1)C(=O)c1cc(O)c(O)c(c1)[N+]([O-])=O	CID:4659569	phase I
BRD-K60298136	COC(=O)c1csc(n1)C(=O)c2c[nH]c3ccccc23	CID:4668801	phase I
BRD-K02269790	[O-][N+](=O)c1cc2C(=O)N(C(=O)c2cc1N3CCOCC3)c4cccc5CCCCc45	CID:4671491	phase I
BRD-K77998258	COC(=O)c1c(C)c2Oc3c(Cl)c(OC(=O)C)c(Cl)c(C)c3C(=O)Oc2cc1OC	CID:4673190	phase I
BRD-K11373525	CCc1cc2N(Cc3ccc(cc3)-c3ccccc3-c3nnn[nH]3)C(=O)CCc2c(CC)n1	CID:4673492	phase I
BRD-K00863322	Clc1ccc(cc1)C(=O)OCC#CCSc2nnc(o2)c3cccc4ccccc34	CID:4675130	phase I
BRD-A81772229	CCC(C)(C)C(=O)OC1CC(C)C=C2C=CC(C)C(CCC3CC(O)CC(=O)O3)C12	CID:4677798	phase I
BRD-K83322645	C(N1CCC2(CCc3ccccc23)CC1)c1ccccc1	CID:4687238	phase I
BRD-A14574269	Clc1ccc(cn1)C1=CCCC2CCC1N2	CID:4694339	phase I
BRD-K40941388	COc1ccc(C=C2SC(=S)N(CCCC(=O)Nc3ccc(C(O)=O)c(O)c3)C2=O)cc1OC	CID:4758367	phase I
BRD-K72787121	OC(=O)c1ccc(NC(=O)CCCN2C(=S)SC(=Cc3ccc4OCOc4c3)C2=O)cc1O	CID:4758734	phase I
BRD-K26160061	Cc1ccc(OCCOc2ccc(Cl)cc2Cl)c(n1)[N+](=O)[O-]	CID:4780551	phase I
BRD-K45505681	O=S(=O)(N1CCN(CC1)c1nc(nc2ccccc12)-c1cccs1)c1ccccc1C#N	CID:4787756	phase I
BRD-K23774426	Clc1ccc(cc1Cl)-n1c(SCC(=O)Nc2ccc3CCCc3c2)nc2ccccc2c1=O	CID:4831588	phase I
BRD-K98219271	CN(C)S(=O)(=O)c1ccc(N2CCCC2)c(c1)C(=O)N3CCN(CC3)c4ccc(cc4)[N+](=O)[O-]	CID:4832119	phase I
BRD-A55554369	Oc1nc2SC3C4CCC(C4)C3C(c2s1)c5cccnc5	CID:4870494	phase I
BRD-A84909344	Brc1ccc2NC(=O)C3(NNc4ccccc4O3)c2c1	CID:4879298	phase I
BRD-A06909528	O=C1N(Cc2ccccc2)c2ccccc2C11NNc2ccccc2O1	CID:4879301	phase I
BRD-A60386802	CCN1C(=O)C2(NNc3ccccc3O2)c2ccccc12	CID:4879425	phase I
BRD-A02198599	CC1CC(C)(C)N2C(=O)C3(Nc4ccccc4S3)c5cccc1c25	CID:4898145	phase I
BRD-K16300438	COc1ccc(NC2=C(NC(=O)C)C(=O)c3ccccc3C2=O)cc1	CID:4919237	phase I
BRD-A31227688	NCC(N)C(=O)c1ccccc1	CID:4990100	phase I
BRD-A89337244	CCOC(=O)c1c(C)[nH]c2ccc3OC4N(CCc5cc(OC)ccc45)Cc3c12	CID:4995951	phase I
BRD-A76528577	CCC1(O)CC2CN(C1)CCc3c([nH]c4ccccc34)C(C2)(C(=O)OC)c5cc6c(cc5OC)N(C=O)C7C86CCN9CC=CC(CC)(C98)C(C(=O)OC)C7(O)C(=O)OC	CID:5022426	phase I
BRD-A58157837	CCCCNC(=O)C1Cc2ccccc2N1C(=O)C(N)CC	CID:5023925	phase I
BRD-K65786282	CC(C)(CO)Cc1cc(c(O)c(c1)C(C)(C)C)C(C)(C)C	CID:5024764	phase I
BRD-K46068882	Cc1cc(=O)c2c(O)c(C)c(O)cc2o1	CID:5036604	phase I
BRD-K00312224	CCCc1c(nn(c1-c1ccc(O)cc1)-c1ccc(O)cc1)-c1ccc(O)cc1	CID:5040063	phase I
BRD-K65742362	CN(C)S(=O)(=O)c1cccc(c1)n2sc3ccccc3c2=O	CID:5040456	phase I
BRD-K30647638	CC(C)(C)n1nc(Cc2cccc3ccccc23)c(C#N)c1N	CID:5050726	phase I
BRD-K69852452	Oc1c(Sc2cccc3cccnc23)cc(NS(=O)(=O)c4ccc(Cl)cc4)c5ccccc15	CID:5056826	phase I
BRD-A59193861	CC1CCCCC1NC(=O)c2cnn3c(cc(nc23)c4ccccc4)C(F)(F)F	CID:5065494	phase I
BRD-K81933000	Cc1cc(nc2ccc(NC(=O)C3CCCCC3)cc12)N1CCOCC1	CID:5067281	phase I
BRD-K74305673	Oc1ccc(Cl)cc1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F	CID:5081913	phase I
BRD-A92585442	CCCC1CC2=CC(=O)CCC2(C)C3CCC4(C)C(CCC4(O)CCC(=O)O)C13	CID:5092098	phase I
BRD-A73908300	NC(=O)C1CCCc2c1[nH]c1ccc(Cl)cc21	CID:5113032	phase I
BRD-K37883585	COc1ccc2[nH]cc(CCNCc3ccc(Br)cc3)c2c1	CID:5124753	phase I
BRD-A18202423	CCOC(=O)C12CC2C(=NO)c3ccccc3O1	CID:5126051	phase I
BRD-K25884242	CNc1nc(N)c(c(Nc2ccc(Cl)cc2)n1)[N+]([O-])=O	CID:5132371	phase I
BRD-K69328504	CC(C)(C)C(=O)OCOP(=O)(OCOC(=O)C(C)(C)C)C(C)(Oc1ccc(O)cc1)P(=O)(OCOC(=O)C(C)(C)C)OCOC(=O)C(C)(C)C	CID:5132514	phase I
BRD-A35072120	NC(Cc1ccc(O)cc1N)C(O)=O	CID:5134354	phase I
BRD-K20742498	COc1cc(COc2cc(N)c(Cl)cc2C(=O)CCC2CCN(CCNS(C)(=O)=O)CC2)cc(OC)c1	CID:5145950	phase I
BRD-K81255325	Oc1ccccc1NC(=O)c1cccnc1	CID:5153532	phase I
BRD-K78278890	CC(C)(C)n1nc(Cc2cccc3ccccc23)c4c(N)ncnc14	CID:5154691	phase I
BRD-A10386413	OCC(O)C1OC(=O)C(=O)C1O	CID:5176753	phase I
BRD-A49370193	CC(N)Cn1ccc2cc(F)c(Cl)cc12	CID:5191289	phase I
BRD-K62300190	Cc1c(CCOC(=O)c2ccc(N3CCOCC3)c(c2)[N+](=O)[O-])sc[n+]1CC#N	CID:5197049	phase I
BRD-A32949107	COC(=O)C1=C(C)N(CC#C)C(=C(C1c2cccc(c2)n3oo3)C(=O)CCO)C	CID:5202074	phase I
BRD-K98157055	Cc1ccc(O)c(N=Nc2ccccc2)n1	CID:5218788	phase I
BRD-A06131576	CC(C)C1CCC(C)C(C(O)c2ccc(cc2)c3ccccc3)C1=O	CID:5221400	phase I
BRD-K26925640	OC(=O)c1ccccc1NC(=O)c1cccc(NC(=O)Cc2ccccc2)c1	CID:5221450	phase I
BRD-A52650764	CC1CC2C(C3C=C(COC(=O)c4ccccc4)C(O)C4(O)C(OC(=O)c5ccccc5)C(C)=CC14C3=O)C2(C)C	CID:5225086	phase I
BRD-A23290232	CCCCC(=O)OC1(CCC2C3CCC4=CC(=O)CCC4(C)C3C(O)CC12C)C(=O)CO	CID:5225092	phase I
BRD-A48631911	COCC(=O)OC1(CCN(C)CCCc2nc3ccccc3[nH]2)CCc2cc(F)ccc2C1C(C)C	CID:5230270	phase I
BRD-K28452084	O=C(NC1CCCCC1)C2(CCCCC2)N(Cc3cccs3)C(=O)c4ccccn4	CID:5236771	phase I
BRD-A37347161	Clc1ccc(CC(=O)N2CCCCC2CN2CCCC2)cc1Cl	CID:5244802	phase I
BRD-A68039575	COc1ccc(cc1)C2CC(=O)c3ccc(OC)cc3O2	CID:5271544	phase I
BRD-K76587808	COc1cc2ccc(=O)oc2c(O)c1O	CID:5273569	phase I
BRD-K54472332	COc1cc2n(cc(C(O)=O)c(=O)c2cc1Cc1cccc(Cl)c1F)[C@H](CO)C(C)C	CID:5277135	phase I
BRD-K25311561	O=c1cc(oc(c1)-c1cccc2Sc3ccccc3Sc12)N1CCOCC1	CID:5278396	phase I
BRD-K62959606	CCCCCCCCCCCCC/C=C/[C@@H](O)[C@@H](N)CO	CID:5280335	phase I
BRD-K97399794	Oc1cc(O)c2c(c1)oc(-c1ccc(O)c(O)c1)c(O)c2=O	CID:5280343	phase I
BRD-K26521938	CCCCC[C@H](O)\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1C\C=C/CCCC(O)=O	CID:5280360	phase I
BRD-K07303502	CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)C(F)(F)F	CID:5280436	phase I
BRD-K01493881	Oc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)cc2o1	CID:5280443	phase I
BRD-K05236810	Oc1cc(O)c2c(c1)oc(cc2=O)-c1ccc(O)c(O)c1	CID:5280445	phase I
BRD-K08973992	CCCCC/C=C\C/C=C\CCCCCCCC(=O)O	CID:5280450	phase I
BRD-K27316855	C[C@H](CCCC(C)(C)O)[C@H]1CC[C@@H]2[C@]1(C)CCC\C2=C/C=C1/C[C@@H](O)C[C@H](O)C1=C	CID:5280453	phase I
BRD-A55815733	CC(C)CCCC(C)CCCC(C)CCC/C(=C/CC1=C(C)C(=O)c2ccccc2C1=O)/C	CID:5280483	phase I
BRD-K46424862	Cc1cc(=O)oc2cc(O)ccc12	CID:5280567	phase I
BRD-K61269089	Oc1ccc2ccc(=O)oc2c1O	CID:5280569	phase I
BRD-K20152659	CCCCC\C=C/C\C=C/C\C=C/CCCCCCC(O)=O	CID:5280581	phase I
BRD-K06692906	Oc1ccc(cc1O)c2oc3c(O)c(O)cc(O)c3c(=O)c2O	CID:5280647	phase I
BRD-K13642330	OC[C@H]1O[C@@H](Oc2cc(O)c3c(=O)cc(oc3c2)c4ccc(O)cc4)[C@H](O)[C@@H](O)[C@@H]1O	CID:5280704	phase I
BRD-K52459643	CCCCC[C@H](O)\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(O)=O	CID:5280723	phase I
BRD-A69815203	CCC1NC(=O)C(C(O)C(C)C\C=C\C)N(C)C(=O)C(C(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)C(C)NC(=O)C(C)NC(=O)C(CC(C)C)N(C)C(=O)C(NC(=O)C(CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C	CID:5280754	phase I
BRD-K73991644	OC[C@H]1O[C@@H](Oc2c(oc3cc(O)cc(O)c3c2=O)c4ccc(O)c(O)c4)[C@H](O)[C@@H](O)[C@@H]1O	CID:5280804	phase I
BRD-K20482099	C[C@@H]1O[C@@H](OC[C@H]2O[C@@H](Oc3c(oc4cc(O)cc(O)c4c3=O)-c3ccc(O)c(O)c3)[C@H](O)[C@@H](O)[C@@H]2O)[C@H](O)[C@H](O)[C@H]1O	CID:5280805	phase I
BRD-K12807006	Oc1ccc(cc1)-c1oc2cc(O)cc(O)c2c(=O)c1O	CID:5280863	phase I
BRD-K82865713	CCCCC[C@H](O)/C=C/C1=C(C/C=C\CCCC(=O)O)C(=O)CC1	CID:5280881	phase I
BRD-K18059238	CCCCC\C=C/C\C=C/C\C=C/CCCCC(O)=O	CID:5280933	phase I
BRD-K33396764	CC\C=C/C\C=C/C\C=C/CCCCCCCC(O)=O	CID:5280934	phase I
BRD-K30984264	COc1ccc2c(c1)[nH]c3c(C)nccc23	CID:5280953	phase I
BRD-K52930707	CO[C@H]1[C@@H](C[C@@H]2CN3CCc4c([nH]c5cc(OC)ccc45)[C@H]3C[C@@H]2[C@@H]1C(=O)OC)OC(=O)/C=C/c6cc(OC)c(OC)c(OC)c6	CID:5280954	phase I
BRD-K43797669	Oc1ccc(cc1)-c1coc2cc(O)cc(O)c2c1=O	CID:5280961	phase I
BRD-A34299591	CCCC1O[C@@H]2C[C@H]3[C@@H]4CCC5=CC(=O)C=C[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:5281004	phase I
BRD-K67977190	CCCCc1ncc(\C=C(/Cc2cccs2)C(O)=O)n1Cc1ccc(cc1)C(O)=O	CID:5281037	phase I
BRD-K69470111	CC(C)(O)c1ccccc1CC[C@@H](SCC1(CC(O)=O)CC1)c1cccc(\C=C\c2ccc3ccc(Cl)cc3n2)c1	CID:5281040	phase I
BRD-K67637637	CN(C)CC/C=C\1/c2ccccc2COc3ccc(CC(=O)O)cc13	CID:5281071	phase I
BRD-K92428153	COc1c(C)c2COC(=O)c2c(O)c1C\C=C(/C)CCC(=O)OCCN1CCOCC1	CID:5281078	phase I
BRD-K83636919	CCN(CC)C(=O)C(\C#N)=C\c1cc(O)c(O)c(c1)[N+]([O-])=O	CID:5281081	phase I
BRD-K66019333	CN1CCCN=C1\C=C\c1cccc(O)c1	CID:5281087	phase I
BRD-K17497770	Oc1ccc(C(=O)\C=C\c2ccc(O)c(O)c2)c(O)c1	CID:5281222	phase I
BRD-K95402279	CC(C)=CCC\C(C)=C\CC\C(C)=C\CC\C(C)=C\CO	CID:5281365	phase I
BRD-K87991767	Oc1ccc2ccc(=O)oc2c1	CID:5281426	phase I
BRD-K07996107	C[C@@]1(C[C@@H](O)[C@]2(O)C=CO[C@@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[C@H]12)OC(=O)/C=C/c4ccccc4	CID:5281542	phase I
BRD-K09497549	COC1=CC(=O)O[C@H](C1)/C=C/c2ccccc2	CID:5281565	phase I
BRD-K31023358	Oc1cc2cccc(O)c(=O)c2c(O)c1O	CID:5281571	phase I
BRD-K94436377	COc1ccc(cc1O)-c1cc(=O)c2c(O)cc(O[C@@H]3O[C@H](CO[C@@H]4O[C@@H](C)[C@H](O)[C@@H](O)[C@H]4O)[C@@H](O)[C@H](O)[C@H]3O)cc2o1	CID:5281613	phase I
BRD-K05485208	OC[C@H]1O[C@@H](Oc2c(O)cc(O)c3c2oc(-c2ccc(O)c(O)c2)c(O)c3=O)[C@H](O)[C@@H](O)[C@@H]1O	CID:5281621	phase I
BRD-K84955386	OC[C@H]1O[C@@H](Oc2c(oc3cc(O)cc(O)c3c2=O)c4ccc(O)c(O)c4)[C@H](O)[C@@H](O)[C@H]1O	CID:5281643	phase I
BRD-K97951054	Cc1cc(O)cc2oc3cc(O)cc(O)c3c(=O)c12	CID:5281657	phase I
BRD-K11590034	Oc1ccc(c(O)c1)-c1oc2cc(O)cc(O)c2c(=O)c1O	CID:5281670	phase I
BRD-K43149758	Oc1cc(O)c2c(c1)oc(-c1cc(O)c(O)c(O)c1)c(O)c2=O	CID:5281672	phase I
BRD-K37206356	COc1cc(O)c2c(=O)c(O)c(oc2c1)c3ccc(O)c(O)c3	CID:5281691	phase I
BRD-K97509413	Oc1ccc2c(c1)oc3c2c(=O)oc4cc(O)ccc34	CID:5281707	phase I
BRD-K42095107	Oc1ccc(cc1)-c1coc2cc(O)ccc2c1=O	CID:5281708	phase I
BRD-K43236057	OC[C@H]1O[C@@H](Oc2cc(O)cc(\C=C\c3ccc(O)cc3)c2)[C@H](O)[C@@H](O)[C@@H]1O	CID:5281718	phase I
BRD-K92870997	COc1cc(OC)cc(/C=C/c2ccc(O)cc2)c1	CID:5281727	phase I
BRD-K42142750	C/C=C\1/C[C@@H](C)[C@](O)(CO)C(=O)OCC2=CCN3CC[C@@H](OC1=O)[C@H]32	CID:5281743	phase I
BRD-K38449220	C/C=C\1/CC(=C)[C@@](C)(O)C(=O)OCC2=CCN3CC[C@@H](OC1=O)[C@H]32	CID:5281750	phase I
BRD-K96188950	Oc1ccc(\C=C\C(=O)OCCc2ccccc2)cc1O	CID:5281787	phase I
BRD-K20313525	OC(=O)[C@@H](Cc1ccc(O)c(O)c1)OC(=O)\C=C\c1ccc(O)c(O)c1	CID:5281792	phase I
BRD-K57546357	COc1cc(O)c2c(=O)c(coc2c1)c3ccc(O)cc3	CID:5281804	phase I
BRD-K03816923	CC(=O)c1c(O)c(C)c(O)c(Cc2c(O)c(C(=O)/C=C/c3ccccc3)c4OC(C)(C)C=Cc4c2O)c1O	CID:5281847	phase I
BRD-K30466858	Oc1cc2c3c(oc(=O)c4cc(O)c(O)c(oc2=O)c34)c1O	CID:5281855	phase I
BRD-K70487031	OCCN1CCN(CC\C=C2\c3ccccc3Sc3ccc(cc23)C(F)(F)F)CC1	CID:5281881	phase I
BRD-K56450366	Oc1ccc2c(=O)cc(oc2c1)c3ccccc3	CID:5281894	phase I
BRD-K04010869	CCCCC[C@H](O)/C=C/[C@H]1C=CC(=O)[C@@H]1CCCCCCC(=O)O	CID:5281912	phase I
BRD-K13872703	OS(=O)(=O)c1cc(ccc1\C=C\c1ccc(cc1S(O)(=O)=O)N=C=S)N=C=S	CID:5281951	phase I
BRD-K42352790	CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)NCCO	CID:5281969	phase I
BRD-K52075040	C\C=C\C\C=C\CCC(=O)[C@H]1O[C@H]1C(N)=O	CID:5282054	phase I
BRD-K50384076	Oc1ccc(cc1)-c1cc(=O)c2ccc(O)cc2o1	CID:5282073	phase I
BRD-K17849083	COc1ccc(\C=C\C(=O)Nc2ccccc2C(O)=O)cc1OC	CID:5282230	phase I
BRD-K78280988	CCCCC/C=C\C/C=C\C/C=C\CCCCCCC(=O)NCCO	CID:5282272	phase I
BRD-K76723084	CC(/C=C/C1=C(C)CCCC1(C)C)=C\C=C\C(C)=C/C(O)=O	CID:5282379	phase I
BRD-K53061490	OC(=O)\C=C\c1ccc(Cn2ccnc2)cc1	CID:5282440	phase I
BRD-K11742128	Cc1ccc(cc1)C(=C/CN1CCCC1)\c1ccccn1	CID:5282443	phase I
BRD-K30097969	O[C@H](C[C@H](O)/C=C/c1c(nc2ccccc2c1c3ccc(F)cc3)C4CC4)CC(=O)O[Ca]OC(=O)C[C@H](O)C[C@H](O)/C=C/c5c(nc6ccccc6c5c7ccc(F)cc7)C8CC8	CID:5282451	phase I
BRD-K38003476	C[C@@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]2(C)[C@H]1C(=O)COC(=O)C(C)(C)C	CID:5282493	phase I
BRD-K92301463	CCCCC(C)(C)[C@H](O)\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1C\C=C/CCCC(O)=O	CID:5283066	phase I
BRD-A15914070	CCCCCC(O)/C=C/C=O	CID:5283344	phase I
BRD-K51557114	CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCC(=O)O	CID:5283389	phase I
BRD-K29555132	CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)N	CID:5283393	phase I
BRD-K87905482	CCCCC/C=C\C/C=C\CCCCCCCC(=O)NCCO	CID:5283446	phase I
BRD-K66956375	CCCCCCCC\C=C/CCCCCCCC(=O)NCCO	CID:5283454	phase I
BRD-K77175907	C[C@H](CCCC(C)(C)O)[C@H]1CC[C@@H]2[C@]1(C)CCC\C2=C/C=C1/C[C@@H](O)CCC1=C	CID:5283731	phase I
BRD-K73397362	C1CCC(CC1)n1cnc2c(Nc3ccc(cc3)N3CCOCC3)nc(Oc3cccc4ccccc34)nc12	CID:5284329	phase I
BRD-A60274948	CC(C)C[C@@H]1N2C(=O)[C@](NC(=O)[C@H]3CN(C)C4Cc5c(Br)[nH]c6cccc(C4=C3)c56)(O[C@@]2(O)[C@@H]7CCCN7C1=O)C(C)C	CID:5284353	phase I
BRD-K13533483	CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C/C=C/C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C	CID:5284373	phase I
BRD-K62012036	COc1cc(C)c(\C=C\C(C)=C\C=C\C(C)=C\C(O)=O)c(C)c1C	CID:5284513	phase I
BRD-K48617017	CCN[C@H]1C[C@H](C)S(=O)(=O)c2sc(cc12)S(=O)(=O)N	CID:5284549	phase I
BRD-K54759182	CN(C)CC\C=C1/c2ccccc2CSc2ccccc12	CID:5284550	phase I
BRD-K03981224	C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]1CC[C@@]2(O)C#C	CID:5284557	phase I
BRD-K49404994	CC[C@H](N1CCCC1=O)C(N)=O	CID:5284583	phase I
BRD-K28935038	N[C@@H](C(=O)N[C@H]1[C@H]2CCC(Cl)=C(N2C1=O)C(O)=O)c1ccccc1	CID:5284585	phase I
BRD-A31312900	CC(C)(O)c1ccccc1CCC(SCC1(CC(O)=O)CC1)c1cccc(\C=C\c2ccc3ccc(Cl)cc3n2)c1	CID:5284590	phase I
BRD-K67511046	Oc1ccc2C[C@H]3N(CC=C)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O	CID:5284596	phase I
BRD-K84937637	CO[C@@H]1C[C@H](C[C@@H](C)[C@@H]2CC(=O)[C@H](C)\C=C(C)\[C@@H](O)[C@@H](OC)C(=O)[C@H](C)C[C@H](C)\C=C\C=C\C=C(C)\[C@H](C[C@@H]3CC[C@@H](C)[C@@](O)(O3)C(=O)C(=O)N3CCCC[C@H]3C(=O)O2)OC)CC[C@H]1O	CID:5284616	phase I
BRD-K29653726	CC1(C)O[C@@H]2CO[C@@]3(COS(N)(=O)=O)OC(C)(C)O[C@H]3[C@@H]2O1	CID:5284627	phase I
BRD-A36151937	OCC1OC(Oc2cc(O)c3c(=O)c(coc3c2)c4ccc(O)cc4)C(O)C(O)C1O	CID:5284639	phase I
BRD-A83237092	C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2O)C(CCCCCCCCCS(=O)CCCC(F)(F)C(F)(F)F)Cc1cc(O)ccc31	CID:5284640	phase I
BRD-K03600170	CCOC(=O)CSC1=NC(=O)/C(=C\c2ccc(Cl)cc2)/S1	CID:5286239	phase I
BRD-K66763349	[O-][N+](=O)c1cccc(/C=C(\C#N)/c2nc3ccccc3[nH]2)c1	CID:5286534	phase I
BRD-K47703442	FC(F)(F)c1cccc(NC(=O)CSc2nnc3c4ccccc4[nH]c3n2)c1	CID:5286678	phase I
BRD-K63915849	FC1(F)Oc2ccc(cc2O1)\C=C1/SC(=O)NC1=O	CID:5287855	phase I
BRD-K87909389	CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl	CID:5287969	phase I
BRD-K89085489	CC(/C=C/C1=C(C)CCCC1(C)C)=C\C=C\C(C)=C\C(=O)Nc1ccc(O)cc1	CID:5288209	phase I
BRD-K11528507	CO[C@H]1C[C@H](C)CC2=C(OC)C(=O)C=C(NC(=O)\C(C)=C\C=C/[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)C2=O	CID:5288382	phase I
BRD-K09638361	COc1cc(OC)c(/C=C\2/C(=O)Nc3ccccc23)c(OC)c1	CID:5288600	phase I
BRD-K83988098	CO[C@H]1C[C@H](C)CC2=C(NCCN(C)C)C(=O)C=C(NC(=O)\C(C)=C\C=C/[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)C2=O	CID:5288674	phase I
BRD-K56429665	C[C@H](\C=C\[C@@H](O)C1CC1)[C@H]1CC[C@@H]2[C@]1(C)CCC\C2=C/C=C1/C[C@@H](O)C[C@H](O)C1=C	CID:5288783	phase I
BRD-K76188144	OC(=O)[C@@H](Cc1ccccc1)NC(=O)C(O)=O	CID:5288998	phase I
BRD-K76773351	O=C1NC(=O)\C(S1)=C\c1ccc2nccnc2c1	CID:5289247	phase I
BRD-K49685476	C\C(=C/c1ccc(cc1)C(O)=O)c1ccc2c(c1)C(C)(C)CCC2(C)C	CID:5289501	phase I
BRD-K76052538	C(CN1CCCCC1)Sc2nnc3c4ccccc4[nH]c3n2	CID:5290633	phase I
BRD-A34907681	CC1OC(OCC2OC(Oc3c(oc4cc(O)cc(O)c4c3=O)c5ccc(O)c(O)c5)C(O)C(O)C2O)C(O)C(O)C1O	CID:5293655	phase I
BRD-A49581300	Cc1ccc(cc1)S(=O)(=O)N2C(C3CC2C=C3)C(=O)O	CID:5308776	phase I
BRD-K14048378	CCCc1cc(no1)C(=O)N(C2CCCCC2)C3CCCCC3	CID:5309153	phase I
BRD-K01578344	C/C=C/Cn1c(SCCCc2ccccc2)nc3n(C)c(=O)[nH]c(=O)c13	CID:5310346	phase I
BRD-K95547711	CCn1c2ccccc2c3nnc(SCCCn4c(O)nc5ccccc45)nc13	CID:5310786	phase I
BRD-K18855837	C1[C@H]2CNC[C@@H]1c1cc3nccnc3cc21	CID:5310966	phase I
BRD-A79052425	CN1CCCC1CCSc1ccc(O)cc1	CID:5310968	phase I
BRD-K18722736	Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)\C(C[C@@]35O)=C\c1ccccc1	CID:5310988	phase I
BRD-K63736853	Cc1cnc(c[n+]1[O-])C(O)=O	CID:5310993	phase I
BRD-A36471396	OC(CCN1CCCCC1)(C2C[C@H]3C[C@@H]2C=C3)c4ccccc4	CID:5311030	phase I
BRD-A89672324	C[C@H](NC[C@H](O)CP(O)(=O)Cc1ccccc1)c1ccc(Cl)c(Cl)c1	CID:5311042	phase I
BRD-K59163477	CO[C@@H]1CN(CCCOc2ccc(F)cc2)CC[C@@H]1NC(=O)c3cc(Cl)c(N)cc3OC	CID:5311047	phase I
BRD-K30697463	C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@H]1C(=O)CO	CID:5311067	phase I
BRD-K95899059	CN(C)[C@@H]1CCc2[nH]c3ccc(NC(=O)c4ccc(F)cc4)cc3c2C1	CID:5311097	phase I
BRD-K31611373	O[C@@H](COc1cccc(c1)C(F)(F)F)/C=C/[C@H]2[C@H](O)C[C@H](O)[C@@H]2C/C=C\CCCC(=O)O	CID:5311100	phase I
BRD-A45664787	CC#CCC(C)[C@H](O)\C=C\[C@H]1[C@H](O)C[C@@H]2C\C(C[C@H]12)=C/CCCC(O)=O	CID:5311181	phase I
BRD-K67582595	CCCN1CCc2cccc-3c2[C@@H]1Cc1ccc(O)c(O)c-31	CID:5311191	phase I
BRD-K05528470	Clc1ccc(cc1)N1CCN(Cc2c[nH]c3ncccc23)CC1	CID:5311200	phase I
BRD-K05396879	CCCCC/C=C/C=C/1\[C@@H](C/C=C\CCCC(=O)O)C=CC1=O	CID:5311211	phase I
BRD-K10961822	CC(C)OC(=O)CCC\C=C/C[C@H]1[C@@H](O)C[C@@H](O)[C@@H]1CC[C@@H](O)CCc1ccccc1	CID:5311221	phase I
BRD-K78637815	COc1ccc(cc1)-c1oc2cc(OC)ccc2c1C(=O)c1ccc(cc1)C#N	CID:5311257	phase I
BRD-K18036262	CCCOc1ccc(Br)cc1-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1	CID:5311276	phase I
BRD-K26664453	C[C@H]1[C@H]2[C@H](Cc3ccccc3)NC(=O)[C@]22OC(=O)\C=C\[C@H](O)CCC[C@@H](C)C\C=C\[C@H]2[C@H](O)C1=C	CID:5311281	phase I
BRD-K66404838	O[C@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5O[C@@H]1[C@]2(CCN3CC1CCC1)c45	CID:5311304	phase I
BRD-K17705806	CCc1ccc(OCc2ccccc2C(=O)Nc2ccc3nc(C)cc(N)c3c2)cc1	CID:5311340	phase I
BRD-A39996500	CC1CC2OC2\C=C\C=C\C(=O)Cc2c(Cl)c(O)cc(O)c2C(=O)O1	CID:5311380	phase I
BRD-K32480324	CCOc1ccccc1O[C@H]([C@H]1CNCCO1)c1ccccc1	CID:5311403	phase I
BRD-K31627533	CCC(=O)[C@@]1(C)[C@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@]12C	CID:5311412	phase I
BRD-K91243525	COc1cccc(OC)c1c2cc(nn2c3ccc(cc3C(C)C)C(=O)N(C)CCCN(C)C)C(=O)NC4(C5CC6CC(C5)CC4C6)C(=O)O	CID:5311451	phase I
BRD-K35430135	CCc1ccccc1OC[C@@H](O)CN[C@H]1CCCc2ccccc12	CID:5311452	phase I
BRD-A72441487	CC(C)(C)C(O)/C=C/c1ccc2OCOc2c1	CID:5311454	phase I
BRD-K40167599	C[C@](N)([C@H]1C[C@@H]1C(O)=O)C(O)=O	CID:5311457	phase I
BRD-K49027941	CCCn1c(=O)[nH]c2nc([nH]c2c1=O)-c1ccc(cc1)S(O)(=O)=O	CID:5311479	phase I
BRD-K18757346	CCCCC[C@H](O)/C=C/[C@@H]1[C@@H](C/C=C\CCCC(=O)O)[C@H]2CO[C@@H]1C2	CID:5311493	phase I
BRD-K28761384	OCCN1CCN(CC\C=C2\c3ccccc3Sc3ccc(Cl)cc23)CC1	CID:5311507	phase I
BRD-K97056771	NC(=O)c1cccc(c1)-c1cc(Nc2ccc(OC(F)(F)F)cc2)ncn1	CID:5311510	phase I
BRD-K36324071	OS(=O)(=O)c1ccc(NC(=O)c2cc(NC(=O)Nc3cc(cc(c3)C(=O)Nc3ccc(c(c3)S(O)(=O)=O)S(O)(=O)=O)C(=O)Nc3ccc(c(c3)S(O)(=O)=O)S(O)(=O)=O)cc(c2)C(=O)Nc2ccc(c(c2)S(O)(=O)=O)S(O)(=O)=O)cc1S(O)(=O)=O	CID:5312111	phase I
BRD-K31912990	Nc1nc(NCC2CCC(CNS(=O)(=O)c3cccc4ccccc34)CC2)nc5ccccc15	CID:5312114	phase I
BRD-K93480852	COc1ccc(cc1)S(=O)(=O)N(CCO)c2ccccc2CN(C)C/C=C/c3ccc(Cl)cc3	CID:5312122	phase I
BRD-K97354755	CN(C)S(=O)(=O)c1ccc2NC(=O)/C(=C\c3cc4CCCCc4[nH]3)/c2c1	CID:5312137	phase I
BRD-K43290182	CNc1cc(NS(=O)(=O)c2ccc(N)cc2)nc(NC)n1	CID:5312145	phase I
BRD-K63913457	CC/C=C\C/C=C\C/C=C\CCCCCCCCCC(=O)O	CID:5312529	phase I
BRD-K96144918	CCCCCCCC/C=C\C/C=C\C/C=C\CCCC(=O)O	CID:5312531	phase I
BRD-K01624546	CC/C=C\C/C=C\C/C=C\CCCCCCCCCCCC(=O)O	CID:5312557	phase I
BRD-K14536225	COc1ccc(/C=C/c2cc(O)cc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c2)cc1	CID:5316606	phase I
BRD-A18917088	C[C@]12CCC3C(CCc4cc(O)ccc34)C1CC[C@@H]2O	CID:5317221	phase I
BRD-A18620900	C[C@]12CCC3C(CCc4cc(O)ccc34)C1C[C@@H](O)[C@@H]2O	CID:5317223	phase I
BRD-K05737787	Cc1cc(=O)c2c(O)cc(O)c(C)c2o1	CID:5318562	phase I
BRD-K65639003	COc1ccc(cc1)c2oc3c(CC=C(C)C)c(O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)cc(O)c3c(=O)c2O[C@@H]5O[C@@H](C)[C@H](O)[C@@H](O)[C@H]5O	CID:5318997	phase I
BRD-K99667445	COc1cc(O)c(cc1/C=C/C(=O)c2ccc(O)cc2)C(C)(C)C=C	CID:5318998	phase I
BRD-A75172220	C[C@]12C[C@H](O)C3C(CCC4=CC(=O)CC[C@]34C)C1CC[C@]2(O)C(=O)CO	CID:5320346	phase I
BRD-A72758037	C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CCC4[C@@]5(C)C[C@@H](O)[C@H](O)[C@@](C)(CO)C5CC[C@@]34C)[C@@H]2[C@H]1C)C(O)=O	CID:5320556	phase I
BRD-A67479912	CC(=O)[C@H]1CCC2C3CCC4=CC(=O)CC[C@]4(C)C3CC[C@]12C	CID:5320716	phase I
BRD-K72726508	O=C1NC(=O)c2c1c1c3ccccc3[nH]c1c1[nH]c3ccccc3c21	CID:5327723	phase I
BRD-K33204703	NC(=C(C#N)C#N)/C(=C/c1ccc2[nH]ccc2c1)/C#N	CID:5328748	phase I
BRD-K07888196	Oc1ccc(/C=C(\C#N)/C(=O)c2ccc(O)c(O)c2)cc1O	CID:5328760	phase I
BRD-K60184833	NC(=O)C(=C\c1ccc(O)c(O)c1)\C#N	CID:5328768	phase I
BRD-K17415526	C[C@H](NC(=O)C(=C\c1ccc(O)c(O)c1)\C#N)c1ccccc1	CID:5328769	phase I
BRD-K34533029	Oc1ccc(cc1O)\C=C(/C#N)C(=O)Nc1ccccc1	CID:5328771	phase I
BRD-K43405658	C[C@@H](NC(=O)/C(=C/c1ccc(O)c(O)c1)/C#N)c2ccccc2	CID:5328772	phase I
BRD-K47105409	Oc1ccc(cc1O)\C=C(/C#N)C(=O)NCc1ccccc1	CID:5328779	phase I
BRD-K01192156	NC(=C(C#N)C#N)/C(=C/c1ccc(O)cc1)/C#N	CID:5328804	phase I
BRD-K47943470	NC(=C(C#N)C#N)/C(=C/c1cc(O)c(O)c(O)c1)/C#N	CID:5328807	phase I
BRD-K99964838	COc1cc(Nc2c(cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)C#N)c(Cl)cc1Cl	CID:5328940	phase I
BRD-K41337261	COc1cc2ncnc(Nc3ccc(Cl)cc3F)c2cc1OC	CID:5329006	phase I
BRD-K63504947	Cc1cc(C)c(\C=C2/C(=O)Nc3ccccc23)[nH]1	CID:5329098	phase I
BRD-K55966568	Cc1[nH]c(\C=C2/C(=O)Nc3ccccc23)c(C)c1CCC(O)=O	CID:5329099	phase I
BRD-K60623809	CCN(CC)CCNC(=O)c1c(C)[nH]c(/C=C/2\C(=O)Nc3ccc(Cl)cc23)c1C	CID:5329103	phase I
BRD-K32906660	Oc1ccc(/C=C(\C#N)/C(=O)NCCCNC(=O)\C(=C\c2ccc(O)c(O)c2)\C#N)cc1O	CID:5329255	phase I
BRD-K61737877	COc1ccc(cc1)c2cnc3c(cnn3c2)c4ccsc4	CID:5329468	phase I
BRD-K79930101	CS(=O)(=O)CCNCc1nc(cs1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1	CID:5329480	phase I
BRD-K51313569	CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)N3CCNCC3)nc2n(C2CCCC2)c1=O	CID:5330286	phase I
BRD-K27665173	Oc1ccc2[nH]c(cc2c1)C(=O)c3cc4ccccc4[nH]3	CID:5330535	phase I
BRD-K11636097	Nc1nc(Nc2ccc(cc2)S(N)(=O)=O)nn1C(=O)c1c(F)cccc1F	CID:5330790	phase I
BRD-K09997269	[O-][N+](=O)c1ccc(/C=N/NC(=O)c2ccccn2)s1	CID:5334616	phase I
BRD-K96076993	CC/1=NNC(=O)\C1=C/c2cn(nc2c3ccc(F)cc3)c4ccccc4	CID:5337366	phase I
BRD-K33392208	[O-][N+](=O)c1ccccc1-c1ccc(\C=c2/sc3nc4cc(Br)cnc4n3c2=O)o1	CID:5341934	phase I
BRD-K09191212	Cc1cc(C)c2nc3s\c(=C/c4ccc(o4)-c4ccccc4C(O)=O)c(=O)n3c2c1	CID:5341943	phase I
BRD-K67470788	[O-][N+](=O)c1ccc(/C=N/NC(=O)CN2CCOCC2)o1	CID:5344250	phase I
BRD-A26962727	CCOC(=O)C1=C(C)N=c2s\c(=C\c3cc(Cl)c(OCC(O)=O)c(OC)c3)c(=O)n2C1c1ccccc1Cl	CID:5346285	phase I
BRD-K91047982	Cc1ccc(NC(=O)CCC(=O)N/N=C/c2ccco2)c(C)c1	CID:5349954	phase I
BRD-K32412559	COc1ccc2C[C@H]3N(C)CCc4cc(O)cc(c34)-c2c1O	CID:5351542	phase I
BRD-K76525302	CSc1ccc(\C=C2\C(C)=C(CC(O)=O)c3cc(F)ccc23)cc1	CID:5352624	phase I
BRD-K15025317	Cc1ccc(cc1)S(=O)(=O)\C=C\C#N	CID:5353431	phase I
BRD-A31107743	CC1CCC\C=C/C2CC(O)CC2C(O)\C=C/C(=O)O1	CID:5353446	phase I
BRD-A55946879	CC(\C=C\c1cccc(Oc2ccc(F)cc2)c1)N(O)C(N)=O	CID:5353454	phase I
BRD-A31158127	CC(\C=C\C(O)C1CC1)C1CCC2C1(C)CCC\C2=C/C=C1\CC(O)CC(O)C1=C	CID:5353464	phase I
BRD-K96084870	CN(C)c1ccc(/C=C\2/C(=O)Nc3ccccc23)cc1	CID:5353593	phase I
BRD-K35573744	COC(=O)\C=C\c1cc(O)ccc1O	CID:5353609	phase I
BRD-K63089472	CC(=CCC/C(=C/CC/C(=C/CSCC(=O)O)/C)/C)C	CID:5353623	phase I
BRD-K96402602	CC(=CCC/C(=C/CC/C(=C/CSc1nc[nH]n1)/C)/C)C	CID:5353633	phase I
BRD-K56800335	NC(=N)N\N=C/c1c(Cl)cccc1Cl	CID:5353646	phase I
BRD-K35377380	COc1cc(/C=C(\C#N)/C(=O)c2ccc(O)c(O)c2)cc(I)c1O	CID:5353685	phase I
BRD-A41145729	COC(C)(C)CCCC(C)C/C=C/C(=C/C(=O)O)/C	CID:5353760	phase I
BRD-K46652470	CN\C(NCCSCc1csc(CN(C)C)n1)=C\[N+]([O-])=O	CID:5353831	phase I
BRD-K85318537	CCCCCCCCCCCCCCCCCCc1ccc(cc1)C(=O)/C=C/C(=O)O	CID:5353842	phase I
BRD-K14221870	ONC(=O)/C=C/C#Cc1cccc(NS(=O)(=O)c2ccccc2)c1	CID:5353852	phase I
BRD-K10016611	CN1C=CC=C\C1=C/N=O	CID:5353895	phase I
BRD-K51476772	CCOc1cc(/C=C(/C#N)\C(=O)N)cc(CSc2ccccc2)c1O	CID:5353962	phase I
BRD-A62809825	CCCCCCCC(=O)OC1C(OC(=O)/C(=C/C)/C)C(=C2C3OC(=O)C(C)(O)C3(O)C(CC(C)(OC(=O)C)C12)OC(=O)CCC)C	CID:5353993	phase I
BRD-K91701654	N\C(Sc1ccccc1N)=C(C#N)/C(C#N)=C(/N)Sc1ccccc1N	CID:5354033	phase I
BRD-K30296925	COc1cc(O)c(C(=O)/C=C/c2ccccc2)c(OC)c1	CID:5356121	phase I
BRD-K88172511	Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)CC[C@@]35O	CID:5360515	phase I
BRD-A92651262	O[C@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5OC1[C@]2(CCN3CC1CCC1)c45	CID:5360630	phase I
BRD-K33211335	COc1ccc2C[C@H]3[C@H]4CCCC[C@@]4(CCN3C)c2c1	CID:5360696	phase I
BRD-K88304388	CN1CC[C@]23CCCC[C@@H]3[C@@H]1Cc4ccc(O)cc42	CID:5360697	phase I
BRD-K10207760	CC[C@H]([C@H]1O[C@@](CC)(C[C@@H]1C)[C@H]2CC[C@](O)(CC)[C@H](C)O2)C(=O)[C@@H](C)[C@@H](O)[C@H](C)CCc3ccc(C)c(O)c3C(=O)O	CID:5360807	phase I
BRD-K31534764	COCCCC\C(c1ccc(cc1)C(F)(F)F)=N\OCCN	CID:5361192	phase I
BRD-K63641886	CO/N=C(/C(=O)N[C@H]1[C@H]2SCC(=C(N2C1=O)C(=O)O)COC(=O)N)\c3ccco3	CID:5361202	phase I
BRD-A67981824	CO\N=C(\C(=O)NC1C2SCC(COC(C)=O)=C(N2C1=O)C(O)=O)c1csc(N)n1	CID:5361298	phase I
BRD-K23369905	Clc1ccc(CO\N=C(\Cn2ccnc2)c2ccc(Cl)cc2Cl)c(Cl)c1	CID:5361463	phase I
BRD-K44497846	CCOC(=O)[C@@H](CCc1ccccc1)N[C@@H](C)C(=O)N1CCC[C@H]1C(O)=O	CID:5362032	phase I
BRD-K71059170	Nc1nc(cs1)C(=N\OCC(O)=O)\C(=O)N[C@H]1[C@H]2SCC(C=C)=C(N2C1=O)C(O)=O	CID:5362065	phase I
BRD-K67966701	NCCCC[C@H](N[C@@H](CCc1ccccc1)C(O)=O)C(=O)N1CCC[C@H]1C(O)=O	CID:5362119	phase I
BRD-K49807096	CCOC(=O)[C@H](CCc1ccccc1)N[C@H]1CCc2ccccc2N(CC(O)=O)C1=O	CID:5362124	phase I
BRD-K89348303	CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCC[C@H]2C[C@H]1C(O)=O	CID:5362129	phase I
BRD-K82818427	CNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)[C@H](CSc1cccs1)C(=O)NO	CID:5362422	phase I
BRD-K33226500	CC(C)(C)NC(=O)[C@@H]1CN(Cc2cccnc2)CCN1C[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12	CID:5362440	phase I
BRD-A75455249	COC1=CC(=O)OC(C1)/C=C/c2ccccc2	CID:5369129	phase I
BRD-A26002865	CC1CCOC(=O)\C=C\C=C/C(=O)OC2CC3OC4C=C(C)CCC4(COC(=O)C1O)C2(C)C31CO1	CID:5369716	phase I
BRD-K94304934	O=C1NC(=O)/C(=C/c2ccco2)/N1	CID:5370029	phase I
BRD-K40213712	O=c1[nH]c(=O)c2nc3ccccc3nc2[nH]1	CID:5372720	phase I
BRD-A94796533	CC1CCCC(=O)CCC\C=C\c2cc(O)cc(O)c2C(=O)O1	CID:5375083	phase I
BRD-K33193182	COc1cc(C)c2c(=O)c3c(O)cc(O)cc3oc2c1	CID:5377914	phase I
BRD-K57545991	CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1CCC[C@H]1C(O)=O	CID:5388962	phase I
BRD-K82109576	CC[C@]1(O)C[C@@H]2CN(C1)CCc3c([nH]c4ccccc34)[C@@](C2)(C(=O)OC)c5cc6c(cc5OC)N(C=O)[C@@H]7[C@@]86CCN9CC=C[C@](CC)([C@H]98)[C@@H](OC(=O)C)[C@]7(O)C(=O)OC	CID:5388993	phase I
BRD-K59633395	Oc1ccc2c(c1)oc(cc2=O)-c1ccccc1O	CID:5391149	phase I
BRD-K59851896	CN1CC[C@]23[C@@H]4Nc5ccccc5[C@]3(CCN4C)[C@@H]1Nc6ccccc62	CID:5392245	phase I
BRD-K89784888	O=C(Nc1ccccc1)/C(=C/c2ccccc2)/NC(=O)c3ccccc3	CID:5405270	phase I
BRD-K51320264	CC(C)c1ccc(/C=C/C(=O)NC2=NCCS2)cc1	CID:5416418	phase I
BRD-K81651477	C\C1=C\CC[C@@]2(C)O[C@@H]2[C@H]2OC(=O)C(=C)[C@@H]2CC1	CID:5420804	phase I
BRD-K79092138	NC(=O)N/N=C/c1ccc(o1)[N+](=O)[O-]	CID:5447130	phase I
BRD-K47207162	CN(C)C/C=C(\c1ccc(Br)cc1)/c2cccnc2	CID:5458656	phase I
BRD-K73323637	CC(C)(C)NC[C@@H](O)COc1cccc2C(=O)CCCc12	CID:5460339	phase I
BRD-K99447003	C[C@H](N[C@@H](CCc1ccccc1)C(O)=O)C(=O)N1CCC[C@H]1C(O)=O	CID:5462501	phase I
BRD-A33325795	CC(C)CC(NCc1c(O)ccc2c(C)cc(=O)oc12)C(=O)O	CID:5466054	phase I
BRD-K89930444	Oc1ccc(/C=C(\C#N)/C(=O)NC2CCC(CC3CCC(CC3)NC(=O)\C(=C\c4ccc(O)c(O)c4)\C#N)CC2)cc1O	CID:5467485	phase I
BRD-K82688027	COc1ccc(/C=C(\C#N)/c2cccnc2)cc1OC	CID:5468216	phase I
BRD-K40901640	CN(C)CCCSc1ccccc1NC(=O)\C=C\c1ccccc1	CID:5475158	phase I
BRD-A11007541	O=C1c2ccccc2C(NC2CCCCC2)\C1=C\c1ccccc1	CID:5475586	phase I
BRD-K13571841	CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)C[C@H](O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CC(C)C)C(C)C)C(C)C)[C@@H](O)CC(O)=O	CID:5478883	phase I
BRD-K84639753	C[C@@H](NCc1ccc(OCc2cccc(F)c2)cc1)C(N)=O	CID:5487407	phase I
BRD-K40831222	CO[C@]1(NC(=O)[C@H](C(O)=O)c2ccc(O)cc2)[C@H]2OCC(CSc3nnnn3C)=C(N2C1=O)C(O)=O	CID:5488645	phase I
BRD-K30020243	COCCCOc1cc(C[C@@H](C[C@H](N)[C@@H](O)C[C@@H](C(C)C)C(=O)NCC(C)(C)C(N)=O)C(C)C)ccc1OC	CID:5493444	phase I
BRD-K59369769	CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1	CID:5494449	phase I
BRD-K41707108	CCCCCCCCCCCCC\C=C\[C@@H](O)[C@H](CO)NC(C)=O	CID:5497136	phase I
BRD-K15935639	CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)/C=C/S(=O)(=O)C	CID:5497183	phase I
BRD-K76896292	Cc1ccc(NC(=O)CN2C(=O)N/C(=C\c3ccco3)/C2=O)cc1	CID:5584298	phase I
BRD-A48720949	CCC(=O)O[C@H]1CCC2C3CCC4=CC(=O)CC[C@]4(C)C3CC[C@]12C	CID:5701990	phase I
BRD-K37080523	CO[C@H]1[C@@H](C[C@@H]2CN3CCc4c([nH]c5cc(OC)ccc45)[C@@H]3C[C@@H]2[C@@H]1C(=O)OC)OC(=O)c6cc(OC)c(OC)c(OC)c6	CID:5701996	phase I
BRD-A55393291	C[C@]12CCC3C(CCC4=CC(=O)CC[C@]34C)C1CC[C@@H]2O	CID:5701998	phase I
BRD-A48237631	CO[C@@]12[C@@H]3NC3CN1C1=C([C@@H]2COC(N)=O)C(=O)C(N)=C(C)C1=O	CID:5702003	phase I
BRD-A80151636	CC(C)CC1N2C(=O)[C@](NC(=O)C3CN(C)[C@@H]4Cc5c(Br)[nH]c6cccc(C4=C3)c56)(OC2(O)[C@@H]2CCCN2C1=O)C(C)C	CID:5702015	phase I
BRD-A54487287	CC(=O)OCC(=O)[C@@]1(O)CCC2C3CCC4=CC(=O)CC[C@]4(C)C3C(=O)C[C@]12C	CID:5702028	phase I
BRD-A92537424	C[C@]12CCC3C(CCC4=Cc5oncc5C[C@]34C)C1CC[C@@]2(O)C#C	CID:5702031	phase I
BRD-A75402480	CC(=O)OCC(=O)[C@H]1CCC2C3CCC4=CC(=O)CC[C@]4(C)C3CC[C@]12C	CID:5702034	phase I
BRD-A10188456	C[C@@H]1CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:5702035	phase I
BRD-A93424738	C[C@@H]1CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)COC(C)=O	CID:5702036	phase I
BRD-K24053527	COc1ccc2C[C@H]3[C@@H]4CCCC[C@@]4(CCN3C)c2c1	CID:5702040	phase I
BRD-A93236127	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)O[C@H]1[C@@H](O)C[C@H](O[C@H]2[C@@H](O)C[C@H](O[C@H]3CC[C@@]4(C)[C@H](CCC5C4CC[C@]4(C)[C@H](CC[C@]54O)C4=CC(=O)OC4)C3)O[C@@H]2C)O[C@@H]1C	CID:5702041	phase I
BRD-A94756469	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)O[C@H]1[C@@H](O)C[C@H](O[C@H]2[C@@H](O)C[C@H](O[C@H]3CC[C@@]4(C)[C@H](CCC5C4C[C@@H](O)[C@]4(C)[C@H](CC[C@]54O)C4=CC(=O)OC4)C3)O[C@@H]2C)O[C@@H]1C	CID:5702042	phase I
BRD-A25687296	CC[C@H]1CN2CCc3cc(OC)c(OC)cc3C2C[C@@H]1CC1NCCc2cc(OC)c(OC)cc12	CID:5702048	phase I
BRD-A91452556	C[C@]12CCC3C(CCc4cc(O)ccc34)C1CC[C@@H]2OC(=O)CCC1CCCC1	CID:5702051	phase I
BRD-A13133631	C[C@H]1CC2C3CC[C@](O)(C(C)=O)[C@@]3(C)C[C@H](O)[C@]2(F)C2(C)C=CC(=O)C=C12	CID:5702058	phase I
BRD-K62736196	NC(=N)N\N=C\c1c(Cl)cccc1Cl	CID:5702063	phase I
BRD-A65767837	CC(=O)OCC(=O)[C@@]1(O)CCC2C3CCC4=CC(=O)CC[C@]4(C)C3[C@@H](O)C[C@]12C	CID:5702068	phase I
BRD-A07000685	C[C@]12C[C@H](O)C3C(CCC4=CC(=O)CC[C@]34C)C1CC[C@]2(O)C(=O)COC(=O)CCC(O)=O	CID:5702069	phase I
BRD-A29731977	CCCCCC(=O)O[C@@]1(CCC2C3CCC4=CC(=O)CC[C@]4(C)C3CC[C@]12C)C(C)=O	CID:5702072	phase I
BRD-A16700644	CC(COc1ccccc1)NC(C)[C@H](O)c1ccc(O)cc1	CID:5702076	phase I
BRD-A20126139	C[C@H]1CC2C3CC[C@H](C(C)=O)[C@@]3(C)C[C@H](O)C2[C@@]2(C)CCC(=O)C=C12	CID:5702081	phase I
BRD-A70461345	Oc1ccc2C[C@H]3N(CC=C)CC[C@]4(C5Oc1c24)[C@@]3(O)CCC5=O	CID:5702090	phase I
BRD-A39415247	C[C@]12CCC3C(CCC4=CC(=O)CC[C@H]34)C1CC[C@@]2(O)C#C	CID:5702093	phase I
BRD-A09349126	CC(=O)O[C@]1(CCC2C3CCC4=CC(=O)CC[C@@H]4C3CC[C@@]21C)C#C	CID:5702094	phase I
BRD-A00758722	C[C@]12CCC3C(CCC4=C3CCC(=O)C4)C1CC[C@@]2(O)C#C	CID:5702095	phase I
BRD-A50928468	CC[C@@]12CCC3C(CCC4=CC(=O)CC[C@H]34)C2CC[C@@]1(O)C#C	CID:5702096	phase I
BRD-A27887842	C[C@]12C[C@H](O)C3C(CCC4=CC(=O)C=C[C@]34C)C1CC[C@]2(O)C(=O)CO	CID:5702106	phase I
BRD-A01643550	CC(=O)OCC(=O)[C@@]1(O)CCC2C3CCC4=CC(=O)C=CC4(C)C3[C@@H](O)C[C@]12C	CID:5702107	phase I
BRD-A62525898	C[C@]12CC(=O)C3C(CCC4=CC(=O)C=C[C@]34C)C1CC[C@]2(O)C(=O)CO	CID:5702108	phase I
BRD-A43974575	NC1C[C@H]1c1ccccc1	CID:5702124	phase I
BRD-A37780065	C[C@]12C[C@H](O)[C@@]3(F)C(CCC4=CC(=O)C=C[C@]34C)C1C[C@@H](O)[C@]2(O)C(=O)CO	CID:5702125	phase I
BRD-A92439610	CC1(C)O[C@@H]2CC3C4CCC5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:5702126	phase I
BRD-A30717181	CC(=O)OCC(=O)[C@@]1(O)[C@@H](CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C)OC(=O)C	CID:5702127	phase I
BRD-A09094913	O=C1CC2OCC=C3CN4CC[C@@]56C4C[C@@H]3[C@@H]2C5N1c1ccccc61	CID:5702135	phase I
BRD-A87445400	COC(=O)C1[C@@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12	CID:5702140	phase I
BRD-A60571864	CCCC1O[C@@H]2CC3C4CCC5=CC(=O)C=CC5(C)C4[C@@H](O)CC3(C)[C@@]2(O1)C(=O)CO	CID:5702148	phase I
BRD-K14693417	O[C@@H]([C@H]1C[C@@H]2CC[N@]1C[C@@H]2C=C)c1ccnc2ccccc12	CID:5702153	phase I
BRD-A28970875	COc1ccc(C[C@H](N)C(=O)N[C@@H]2[C@@H](CO)OC([C@@H]2O)n2cnc3c(ncnc23)N(C)C)cc1	CID:5702164	phase I
BRD-A57089740	CO[C@@H]1[C@@H](O)[C@H](C)O[C@H](O[C@H]2CC[C@@]3(C=O)[C@H](CCC4C3CC[C@]5(C)[C@H](CC[C@]45O)C6=CC(=O)OC6)C2)[C@H]1O	CID:5702166	phase I
BRD-A49765801	CC1(C)O[C@@H]2CC3C4C[C@H](F)C5=CC(=O)CC[C@]5(C)C4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:5702172	phase I
BRD-A65449987	CC1(C)O[C@@H]2CC3C4C[C@H](F)C5=CC(=O)C=CC5(C)C4C(O)CC3(C)[C@@]2(O1)C(=O)CO	CID:5702174	phase I
BRD-A01346607	C[C@@H]1CC2C3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:5702178	phase I
BRD-K56001384	CCCCC[C@@H]1[C@@H](OC(=O)CC(C)C)[C@H](C)OC(=O)[C@@H](NC(=O)c2cccc(NC=O)c2O)[C@@H](C)OC1=O	CID:5702199	phase I
BRD-A15931911	CCCC(=O)Nc1ncnc2n(cnc12)C1O[C@@H]2COP(O)(=O)O[C@H]2[C@H]1OC(=O)CCC	CID:5702210	phase I
BRD-A64242993	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O[C@H]1C[C@H](O)[C@H](O[C@H]2C[C@H](OC(C)=O)[C@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[C@@H](C)O2)[C@@H](C)O1)O[C@H]1CC[C@@]2(C)C(CCC3C2C[C@@H](O)[C@]2(C)[C@H](CC[C@]32O)C2=CC(=O)OC2)C1	CID:5702228	phase I
BRD-A66559694	Oc1ccc2C[C@H]3N(CC4CC4)CCC45[C@@H](Oc1c24)C(=O)CC[C@@]35O	CID:5702239	phase I
BRD-A55416093	CC(=O)O[C@H]1[C@@H](O)C2C(C)(C)CC[C@H](O)[C@]2(C)[C@@]2(O)C(=O)C[C@@](C)(O[C@]12C)C=C	CID:5702265	phase I
BRD-A36010170	CC(=O)OCC(=O)[C@@]12OC3(CCCC3)O[C@@H]1CC1C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]21C	CID:5702266	phase I
BRD-A26095496	CCC(=O)O[C@@]1([C@@H](C)CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C)C(=O)CCl	CID:5702274	phase I
BRD-K31412180	CS(=O)(=O)/C(=C/c1cccn1S(=O)(=O)c2ccccc2)/C#N	CID:5703330	phase I
BRD-K64440589	Cc1oc(N)c(c1C)S(=O)(=O)/C(=C/c2cc(Cl)cc(Cl)c2)/C#N	CID:5703601	phase I
BRD-K34332553	CCOC(=O)CSC1=N/C(=C/c2ccc(cc2)n3cncn3)/C(=O)N1C(=O)C	CID:5707818	phase I
BRD-K00910650	COc1cc(\C=C\C(=O)c2ccccc2)cc(OC)c1OC	CID:5712112	phase I
BRD-K85266146	FC(F)(F)c1cc(nc(S/C=C/C(=O)c2ccccc2)c1C#N)c3cccs3	CID:5716606	phase I
BRD-K52678950	N#C/C(=C\c1ccco1)/c2nc3ccccc3[nH]2	CID:5716861	phase I
BRD-A71799696	CC(C)C(N1C(=O)/C(=C/c2ccccc2)/SC1=S)C(=O)O	CID:5717719	phase I
BRD-A38913120	CC(C)C(N1C(=O)/C(=C/c2ccc(Br)cc2)/SC1=S)C(=O)O	CID:5720188	phase I
BRD-K10882151	O=c1n(Cc2ccccc2)c(/C=C/c3cccnc3)nc4ccccc14	CID:5738263	phase I
BRD-K30715099	Oc1cc(OCC(=O)c2ccc(Cl)cc2)cc3oc4ccccc4c(=O)c13	CID:5741425	phase I
BRD-K04986062	C\C(N)=C(\C#N)C(=O)COC(=O)c1cc(C)n(c1C)-c1ccc(F)cc1	CID:5742565	phase I
BRD-K92138166	CC(C)CC(=O)c1c(O)c(CC=C(C)C)c(O)c2c(cc(=O)oc12)c3ccccc3	CID:5748555	phase I
BRD-K98824517	CCn1nc(/C=C/c2ccccc2)nc3c(=O)n(C)c(=O)nc13	CID:5756371	phase I
BRD-A75517195	CCOC(=O)C1=C(C)N=c2s\c(=C/c3cc(Br)c(O)c(Br)c3)c(=O)n2C1c1ccc2OCOc2c1	CID:5758458	phase I
BRD-K05979026	O=C(NCCc1nc2ccccc2n1C\C=C\c1ccccc1)C1CCCCC1	CID:5769809	phase I
BRD-K92015269	C(CN1CCN(C\C=C\c2ccccc2)CC1)OC(c1ccccc1)c1ccccc1	CID:5788723	phase I
BRD-A85025557	OC1c2ccccc2CCC\C1=C/C(O)=O	CID:5875451	phase I
BRD-K06765193	[O-][N+](=O)c1ccc(/C=C(\C#N)/c2nc3ccccc3[nH]2)o1	CID:5904441	phase I
BRD-K51816706	O=C/1Nc2ccccc2\C1=C\c3ccc[nH]3	CID:5908088	phase I
BRD-A47065382	C/C=C/1\C2Cc3[nH]c(=O)ccc3C1(N)CC(=C2)C	CID:5912039	phase I
BRD-A09186529	OC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)/C=C/c3ccccn3	CID:5918561	phase I
BRD-K07859598	Oc1c(Br)cc(cc1Br)\C=C1/C(=O)Nc2ccc(I)cc12	CID:5924208	phase I
BRD-K21853356	Clc1cc(Cl)cc(/C=C(\C#N)/c2cccnc2)c1	CID:5926218	phase I
BRD-K03601405	COc1cc(\C=C\C(=O)n2cnc3ccccc23)cc(OC)c1OC	CID:5929052	phase I
BRD-K76425827	OS(=O)(=O)CCN1C(=S)S\C(=C/c2cn(nc2-c2ccc(OCc3ccccc3F)cc2)-c2ccccc2)C1=O	CID:5932584	phase I
BRD-K91987625	O/N=C(/Cn1nnc(n1)N2CCCC2)\c3ccc(Cl)cc3	CID:5932959	phase I
BRD-K80346834	Cc1ccc2nc([nH]c2c1)/C(=C/c3ccc(o3)[N+](=O)[O-])/C#N	CID:5938151	phase I
BRD-K34995470	CC(C)c1cc(/C=C(\C#N)/C(=O)NCCCc2ccccc2)cc(C(C)C)c1O	CID:5941539	phase I
BRD-K80946661	CC(=O)Oc1ccc(/C=C/c2cc(OC(=O)C)cc(OC(=O)C)c2)cc1	CID:5962587	phase I
BRD-K92577649	Fc1ccc(cc1)C(OCCN1CCN(C\C=C\c2ccccc2)CC1)c1ccc(F)cc1	CID:5974189	phase I
BRD-K91696562	Cc1[nH]c(\C=C2\C(=O)Nc3ccccc23)c(C)c1CCC(O)=O	CID:5995546	phase I
BRD-K95253417	OS(=O)(=O)CCN1C(=S)S\C(=C/c2cn(nc2-c2ccc(OCc3ccccc3)cc2)-c2ccccc2)C1=O	CID:5998084	phase I
BRD-A82913781	CCOC(=O)C1=C(C)N=c2s\c(=C/c3cc(Cl)c(OCC(O)=O)c(Cl)c3)c(=O)n2C1c1cccc(OC)c1	CID:6000533	phase I
BRD-K33586157	Cc1ccc(cc1)-c1nn(cc1\C=C1/SC(=S)N(CCS(O)(=O)=O)C1=O)-c1ccccc1	CID:6001181	phase I
BRD-K49807497	CCCCC(=O)N/N=C(\C)/c1ccc(NC(=O)C(F)(F)F)cc1	CID:6048135	phase I
BRD-K55991774	Cc1ccc(/C=C(\C#N)/c2nc3ccc(C)cc3[nH]2)o1	CID:6070589	phase I
BRD-K87919739	COc1cc(\C=C(/C#N)C(N)=O)cc(CSc2nc3ccccc3s2)c1O	CID:6091659	phase I
BRD-K70515009	C[C@]12CC[C@@H]3[C@@H](CCc4cc(OS(O)(=O)=O)ccc34)[C@H]1CCC2=O	CID:6093179	phase I
BRD-K57174586	CN[C@H]1CC[C@H](c2ccc(Cl)c(Cl)c2)c2ccccc12	CID:6093397	phase I
BRD-K91485395	OS(=O)(=O)CCN1C(=S)S\C(=C/c2cn(nc2-c2ccc(OCc3ccc(Cl)cc3)cc2)-c2ccccc2)C1=O	CID:6161281	phase I
BRD-K11987803	OS(=O)(=O)CCN1C(=S)S\C(=C/c2cn(nc2-c2ccc(cc2)S(=O)(=O)N2CCCCC2)-c2ccccc2)C1=O	CID:6166563	phase I
BRD-K62683350	COC(=O)c1ccc(COc2ccccc2/C=C/C(=O)c3ccc(OCC(=O)O)cc3)cc1	CID:6173479	phase I
BRD-K25375605	COc1ccc(\C=C2/SC(=S)N(CCCC(=O)Nc3ccc(C(O)=O)c(O)c3)C2=O)cc1OC	CID:6202912	phase I
BRD-K87432599	OC(=O)c1ccc(NC(=O)CCCN2C(=S)S\C(=C/c3ccc4OCOc4c3)C2=O)cc1O	CID:6203183	phase I
BRD-K91671201	OS(=O)(=O)CCN1C(=S)S\C(=C/c2cn(nc2-c2ccc(OCc3ccccc3Cl)cc2)-c2ccccc2)C1=O	CID:6274486	phase I
BRD-A05729358	CCOC(=O)C12CC1\C(=N/O)c1ccccc1O2	CID:6278000	phase I
BRD-A01295252	CCCN(C\C=C\I)C1CCc2ccc(O)cc2C1	CID:6305587	phase I
BRD-K04993501	Nc1nc(cs1)/C(=N\OCC(=O)O)/C(=O)N[C@H]2[C@H]3SCC(=C(N3C2=O)C(=O)O)C=C	CID:6321411	phase I
BRD-A87387433	COCC1=C(N2[C@H](SC1)[C@H](NC(=O)C(=N\OC)\c1csc(N)n1)C2=O)C(=O)OC(C)OC(=O)OC(C)C	CID:6321414	phase I
BRD-A60414806	CC[C@]1(O)CC2CN(C1)CCc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C=O)[C@@H]1[C@]22CCN3CC=C[C@](CC)([C@@H]23)[C@@H](OC(C)=O)[C@]1(O)C(=O)OC	CID:6324671	phase I
BRD-K39330046	CN1[C@@H]2CC[C@@H]1C[C@H](C2)OC(=O)[C@H](CO)c1ccccc1	CID:6334600	phase I
BRD-K31168993	CSc1ccc(cc1)[C@H]1CN2CCC[C@H]2c2ccccc12	CID:6336338	phase I
BRD-K08924299	O=C1N(C[C@H]2CCCc3cccc1c23)[C@@H]1CN2CCC1CC2	CID:6337614	phase I
BRD-K23163214	C[C@@]12N[C@@H](Cc3ccccc13)c1ccccc21	CID:6337640	phase I
BRD-A25775766	O=C1OC2(C[C@H]3C=CC2=C1)[C@H]4CCCCN34	CID:6338099	phase I
BRD-A52934756	CCCCC\C=C\C=C1/C(C\C=C\CCCC(O)=O)C=CC1=O	CID:6375741	phase I
BRD-A19037878	CC(\C=C(C)\C=C\C(=O)NO)C(=O)c1ccc(cc1)N(C)C	CID:6376322	phase I
BRD-K03012696	Nc1nc(cs1)C(=NO)C(=O)N[C@H]2[C@H]3SCC(=C(N3C2=O)C(=O)O)C=C	CID:6398970	phase I
BRD-K52735702	Nc1nc(cs1)C(=N/O)\C(=O)N[C@H]1[C@H]2SCC(C=C)=C(N2C1=O)C(O)=O	CID:6399253	phase I
BRD-K94987138	CC1CCN(CC1)c2nnc(c3ccc(C)c(C)c3)c4ccccc24	CID:6401129	phase I
BRD-K37932103	Nc1nc(CSc2nnc3c4ccccc4[nH]c3n2)cs1	CID:6401201	phase I
BRD-K94572506	Cn1c2ccccc2c3nnc(SCC(=O)c4ccc(Cl)cc4)nc13	CID:6403456	phase I
BRD-K93623754	COc1nc(nnc1c2ccccc2)c3ccccc3	CID:6404603	phase I
BRD-K30189597	Cn1cc(/C=C/2\C(=O)Nc3ccc(cc23)S(=O)(=O)N)c4ccccc14	CID:6419747	phase I
BRD-K09132007	NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccccn1)-c1ccc2OCCOc2c1	CID:6419753	phase I
BRD-K89687904	O=C1NC(=O)C(=C1Nc1ccccc1)c1cn(CCCn2ccnc2)c2ccccc12	CID:6419755	phase I
BRD-K08502430	O=C/1Nc2ccccc2\C1=C/c3c[nH]cn3	CID:6419833	phase I
BRD-K56033645	C[C@@H]1NC(=O)NC1=O	CID:6419931	phase I
BRD-A67709388	CCCCCC[C@@H]1[C@@H](OC(=O)CC(C)C)[C@H](C)OC(=O)C(NC(=O)c2cccc(NC=O)c2O)[C@@H](C)OC1=O	CID:6420045	phase I
BRD-K77171813	C(COCc1ccccc1)Cc1cnc[nH]1	CID:6421522	phase I
BRD-K01767299	O=C(C1CC1)c1ccc(OCCCc2c[nH]cn2)cc1	CID:6422124	phase I
BRD-A84134924	CC(=O)OC1C(C[C@H]2C3CC[C@H]4C[C@H](OC(=O)C)C(CC4(C)[C@H]3CCC12C)[N+]5(C)CCCCC5)[N+]6(C)CCCCC6	CID:6426894	phase I
BRD-K76293260	CCCCC/C=C\C/C=C\CCCCCCCC(=O)NCC(=O)O	CID:6433346	phase I
BRD-K85518562	CC1(C)C[C@@H]1C(=O)N/C(=C\CCCCSC[C@H](N)C(=O)O)/C(=O)O	CID:6435415	phase I
BRD-K64044582	CCCCC/C=C\C/C=C\CCCCCCCC(=O)N	CID:6435901	phase I
BRD-A84228258	C[C@H]1CCC\C=C\C2C[C@H](O)C[C@H]2[C@H](O)\C=C\C(=O)O1	CID:6436187	phase I
BRD-K27499107	CCCCC[C@H](O)/C=C/[C@H]1[C@H](O)C[C@@H]2C/C(=C\CCCC(=O)O)/C[C@H]12	CID:6436393	phase I
BRD-K17219111	CCC\C(=C/CC)C(O)=O	CID:6437068	phase I
BRD-K99369265	CC[C@@H]1\C=C(C)/C[C@H](C)C[C@H](OC)[C@H]2O[C@](O)([C@H](C)C[C@@H]2OC)C(=O)C(=O)N2CCCC[C@H]2C(=O)O[C@@H]([C@H](C)[C@@H](O)CC1=O)C(\C)=C\[C@@H]1CC[C@@H](O)[C@@H](C1)OC	CID:6437370	phase I
BRD-K79437791	CC(=O)N[C@@H](CSC\C=C(/C)CC\C=C(/C)CCC=C(C)C)C(O)=O	CID:6438381	phase I
BRD-A96799240	CC(/C=C/C1=C(C)C(O)CCC1(C)C)=C\C=C\C(C)=C\C(O)=O	CID:6438629	phase I
BRD-K38756014	COC(=O)[C@@H](N)CSC/C=C(\C)/CC/C=C(\C)/CCC=C(C)C	CID:6439225	phase I
BRD-K80325895	CCCCC/C=C\C/C=C\CCCCCCCCCC(=O)O	CID:6439848	phase I
BRD-K57139258	C\C=C1\C(=O)C[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:6439929	phase I
BRD-A62025033	COC1CC(CC(C)C2CC(=O)C(C)\C=C(C)\C(O)C(OC)C(=O)C(C)CC(C)\C=C\C=C\C=C(C)\C(CC3CCC(C)C(O)(O3)C(=O)C(=O)N3CCCCC3C(=O)O2)OC)CCC1OC(=O)C(C)(CO)CO	CID:6440033	phase I
BRD-K13514097	CO[C@@H]1C[C@H](C[C@@H](C)[C@@H]2CC(=O)[C@H](C)\C=C(C)\[C@@H](O)[C@@H](OC)C(=O)[C@H](C)C[C@H](C)\C=C\C=C\C=C(C)\[C@H](C[C@@H]3CC[C@@H](C)[C@@](O)(O3)C(=O)C(=O)N3CCCC[C@H]3C(=O)O2)OC)CC[C@H]1OCCO	CID:6442177	phase I
BRD-K86465814	CCCCC[C@H](O)/C=C/C=C\CCCCCCCC(=O)O	CID:6443013	phase I
BRD-K55070890	CN(C)S(=O)(=O)c1ccc2Sc3ccccc3\C(=C\CCN3CCNCC3)c2c1	CID:6444849	phase I
BRD-K56957086	OCCN(CCc1c[nH]c2ccccc12)Cc1ccc(\C=C\C(=O)NO)cc1	CID:6445533	phase I
BRD-K08799216	CCOc1cc2ncc(C#N)c(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C	CID:6445562	phase I
BRD-K83643280	Cc1cccc2nc([nH]c12)/C(=C/c3ccc(o3)[N+](=O)[O-])/C#N	CID:6446335	phase I
BRD-K34092021	CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCc1ccc(O)c(OC)c1	CID:6449767	phase I
BRD-K26674531	C\C=C1/C(=O)C[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:6450278	phase I
BRD-K29905972	CNC(=O)c1ccccc1Sc1ccc2c(\C=C\c3ccccn3)n[nH]c2c1	CID:6450551	phase I
BRD-K20287671	CN(C)c1ccc(cc1)\C=C1/C(=O)Nc2ccccc12	CID:6450842	phase I
BRD-A66794241	CC[C@H](C)[C@@H](COC(Cc1ccccc1)C(=O)N[C@@H](CCS(C)(=O)=O)C(=O)OC(C)C)NC[C@@H](N)CS	CID:6451153	phase I
BRD-K06198550	COc1cc2OC[C@H]3Oc4c(ccc5oc(cc45)C(C)C)C(=O)[C@H]3c2cc1OC	CID:6453092	phase I
BRD-K44094599	CO[C@@H]1C[C@@H](CC[C@H]1O)\C=C(/C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@]2(O)O[C@@H]([C@H](C[C@H]2C)OC)[C@H](C[C@@H](C)C\C(C)=C/[C@@H](CC=C)C(=O)C[C@H](O)[C@H]1C)OC	CID:6473866	phase I
BRD-K98548675	C\C1=C/CC[C@@]2(C)O[C@H]2[C@H]2OC(=O)C(=C)[C@@H]2CC1	CID:6473881	phase I
BRD-K52756523	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(O)C[C@@H](C)[C@@H]2N[C@@H](COCCOC)O[C@H]([C@H]2C)[C@]1(C)O	CID:6473883	phase I
BRD-K63425657	COc1cc(/C=C/2\Oc3cc(O)cc(O)c3C2=O)cc(OC)c1O	CID:6476406	phase I
BRD-K74402642	Cc1ccc(/C=C/2\CNC/C(=C/c3ccc(C)cc3)/C2=O)cc1	CID:6477762	phase I
BRD-K51644197	Fc1ccccc1CCNc2c3CCCCc3nc4ncnn24	CID:6484054	phase I
BRD-K81473043	CO[C@H]1C[C@H](C)CC2=C(NCC=C)C(=O)C=C(NC(=O)\C(C)=C\C=C/[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)C2=O	CID:6505803	phase I
BRD-K99440638	CC[n+]1c(/C=C\2/CC(C)(C)CC(=C2)C)oc3ccccc13	CID:6520352	phase I
BRD-K67174588	CN(C)CCOc1ccc(cc1)C(=C(/CCCl)c1ccccc1)\c1ccccc1	CID:6536897	phase I
BRD-K09991945	Ic1cccc(CSc2nnc(o2)c3ccncc3)c1	CID:6539732	phase I
BRD-K21401044	C[C@]12CC[C@@H]3[C@@H](CCC4=Cc5oncc5C[C@]34C)[C@H]1CC[C@@]2(O)C#C	CID:6540825	phase I
BRD-K22321414	C[C@@H]1CC(=O)NN=C1c1ccc(Cl)cc1	CID:6541041	phase I
BRD-K78062244	COC(=O)[C@@H]1Cc2c([nH]c3ccccc23)C(C)(C)N1C(=O)CCl	CID:6545175	phase I
BRD-K48519456	CC1(C)S[C@H]2[C@H](NC(=O)Cc3ccccc3)C(=O)N2[C@H]1C(O)=O	CID:6560153	phase I
BRD-K73437736	CC1(C)S[C@H]2[C@H](NC(=O)[C@H](NC(=O)N3CCNC3=O)c3ccccc3)C(=O)N2[C@H]1C(O)=O	CID:6560164	phase I
BRD-K54568510	COc1ccc(CN2C(=O)[C@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)cc1	CID:6572379	phase I
BRD-A64125466	C[C@H](CCC(O)=O)[C@H]1CCC2C3C(CC(=O)[C@]12C)[C@@]1(C)CCC(=O)CC1CC3=O	CID:6602440	phase I
BRD-A46186775	CC12C[C@H](O)C3C(CCC4=CC(=O)CCC34C)C1CC[C@]2(O)C(=O)COP(O)(O)=O	CID:6602442	phase I
BRD-A98702003	CC1(C)[C@H](CC[C@@]2(C)C1CC[C@]1(C)C2C(=O)C=C2[C@@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O)OC(=O)CCC(O)=O	CID:6602447	phase I
BRD-A23034328	CCC[C@@H]1C[C@H](N(C)C1)C(=O)N[C@H]([C@H](C)Cl)C1O[C@H](SC)[C@H](O)[C@@H](O)[C@H]1O	CID:6602476	phase I
BRD-K57773246	CC(C)CCCCC(=O)N[C@H](CCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@H](CCN)C(=O)N[C@@H]1CCNC(=O)[C@@H](NC(=O)[C@H](CCN)NC(=O)[C@H](CCN)NC(=O)[C@@H](CNC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CCN)NC1=O)C(C)C)[C@@H](C)O	CID:6602488	phase I
BRD-K14329163	COC(=O)C1=C(C)NC(C)=C([C@H]1c1ccccc1C(F)(F)F)[N+]([O-])=O	CID:6603728	phase I
BRD-K39187410	CN1CCc2cc(O)cc-3c2[C@H]1Cc4ccc(O)c(O)c43	CID:6603797	phase I
BRD-K16604360	CCCN1CCc2cc(O)cc-3c2[C@H]1Cc4ccc(O)c(O)c43	CID:6603798	phase I
BRD-K31471398	Oc1cc2CC[C@H]3NCc4ccccc4[C@@H]3c2cc1O	CID:6603820	phase I
BRD-K41143549	NC(=O)CNCCC(c1ccccc1)c1ccccc1	CID:6603827	phase I
BRD-K28308851	C[C@H](N)Cc1c[nH]cn1	CID:6603865	phase I
BRD-K28806945	Ic1ccc(cc1)N2CCN(Cc3c[nH]c4ncccc34)CC2	CID:6603897	phase I
BRD-K98372770	CCCc1c(OCCCOc2ccc(OCC(O)=O)cc2)ccc(C(C)=O)c1O	CID:6603901	phase I
BRD-K72024482	CCCn1c(=O)n(CCC)c2nc([nH]c2c1=O)c3ccc(OCC(=O)Nc4ccc(C#N)cc4)cc3	CID:6603931	phase I
BRD-K04414442	CC[C@H](NC(=O)c1c(C)c(nc2ccccc12)-c1ccccc1)c1ccccc1	CID:6604009	phase I
BRD-K12567312	CC(=O)O[C@H]1CC[C@]2(C)[C@@H]3CC[C@@]4(C)[C@H](CCC4=O)[C@@H]3CC=C2C1	CID:6604284	phase I
BRD-K46156294	CC(C)(C)CC(C)(C)c1ccc(OCOCCOCCO)c(Cc2cc(cc(Cc3cc(ccc3OCOCCOCCO)C(C)(C)CC(C)(C)C)c2OCOCCOCCO)C(C)(C)CC(C)(C)C)c1	CID:6604381	phase I
BRD-K05111602	CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCC[C@@H]2C[C@H]1C(O)=O	CID:6604446	phase I
BRD-K02764365	COC(=O)Nc1nc2cc(SC(C)C)ccc2[nH]1	CID:6604471	phase I
BRD-K63899271	OC(=O)CCCC[C@@H]1SC[C@H]2NC(=O)N[C@H]12	CID:6604653	phase I
BRD-K74284736	OC(=O)[C@H]1C[C@H](NC(=O)Nc2ccccc2)c2c(Cl)cc(Cl)cc2N1	CID:6604749	phase I
BRD-K48311056	O[C@H](CNCCOc1ccc(OCC(=O)O)cc1)COc2ccccc2	CID:6604779	phase I
BRD-K45296539	COCCNC(=O)COc1ccc(OCCNC[C@@H](O)COc2ccccc2)cc1	CID:6604780	phase I
BRD-K20714604	Cn1cc(C(=O)C(=O)N[C@H]2CN3CCC2CC3)c2ccccc12	CID:6604789	phase I
BRD-K80725821	CC(C)n1cnc2c(cc(Cl)cc12)C(=O)N[C@H]1CN2CCC1CC2	CID:6604794	phase I
BRD-K55462201	CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)Nc1ccc(O)cc1	CID:6604822	phase I
BRD-K61097567	COC(=O)[C@H](NC(=O)c1cc(nc2ccccc12)-c1ccccc1)c1ccccc1	CID:6604858	phase I
BRD-K51541829	C[C@@H](CN1CCC(Cc2ccccc2)CC1)[C@@H](O)c1ccc(O)cc1	CID:6604887	phase I
BRD-K24201553	CC1CCN(CC[C@H]2CCCN2S(=O)(=O)c2cccc(O)c2)CC1	CID:6604889	phase I
BRD-K53979406	CN(CC[C@@H](Oc1ccc(cc1)-c1ccccc1)c1ccc(F)cc1)CC(O)=O	CID:6604909	phase I
BRD-K12932420	CCc1ccc2c(nc(=O)n(CC)c2n1)-c1cccc(Cl)c1	CID:6604918	phase I
BRD-K41567364	Cc1nc2ccc(NC(=O)Nc3ccnc4cccnc34)cc2o1	CID:6604926	phase I
BRD-K75478907	CSc1nc(NC2CCCC2)c(c(NC2CCCC2)n1)[N+]([O-])=O	CID:6604928	phase I
BRD-K07762753	CC(C)[C@H](CO)Nc1nc(Nc2cc(N)cc(Cl)c2)c2ncn(C(C)C)c2n1	CID:6604931	phase I
BRD-K55430733	C1CCc2c(C1)n1CCNCc3cccc2c13	CID:6604933	phase I
BRD-A50737080	[O-][N+](=O)c1cc(NC(=S)NC(NC(=O)C(c2ccccc2)c2ccccc2)C(Cl)(Cl)Cl)ccc1F	CID:6605258	phase I
BRD-K05653692	CCCCCCCCCC(=O)N[C@H](CN1CCOCC1)[C@H](O)c2ccccc2	CID:6610216	phase I
BRD-K09635134	CCCCCCCCCCCCCC(=O)N[C@@H](C)[C@H](O)c1ccccc1	CID:6610217	phase I
BRD-K03842655	CC(=C)[C@H]1O[C@H]2CC[C@]3(C)[C@]4(C)[C@@H](CC[C@@]3(O)[C@@]52O[C@@H]5[C@H]1O)[C@@H]6OC(C)(C)[C@H]7C[C@@H]8C(=C)Cc9c(Cl)cc%10[nH]c4c6c%10c9[C@@]87O	CID:6610243	phase I
BRD-A50934474	CC[C@@H](C)[C@@H](CO[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCS(=O)(=O)C)C(=O)OC(C)C)NCC(N)CS	CID:6610261	phase I
BRD-A74904029	OC[C@H]1O[C@H](C(O)[C@H]1O)n2cnc3cc(Cl)c(Cl)cc23	CID:6610267	phase I
BRD-K50464341	COc1cc2CCN(C)[C@@H]3Cc4ccc(OC(=O)c5ccc(cc5)[N+](=O)[O-])c(Oc6ccc(C[C@@H]7N(C)CCc8cc(OC)c(Oc(c1OC)c32)cc78)cc6)c4	CID:6610268	phase I
BRD-K62910157	CCCCCCCCCCCCCCC[C@@H](O)[C@H](CO)NC(=O)C	CID:6610273	phase I
BRD-K63915987	Nc1nc(N)c(nc1Cl)C(=O)NC(=N)NCc1ccc(Cl)cc1Cl	CID:6610300	phase I
BRD-A82329351	CCOC(=O)CN1C(=O)CC(C[C@@H](O)C2C[C@@H](C)C[C@H](C)C2=O)CC1=O	CID:6610302	phase I
BRD-A96897502	CC12CC=C3C(CCC4=CC(=O)C=CC43C)C2CC[C@@H]1C(=O)CN5CCN(CC5)c6cc(nc(n6)N7CCCC7)N8CCCC8	CID:6610303	phase I
BRD-K64746805	Clc1ccc2ncnc(NCc3ccc4OCOc4c3)c2c1	CID:6610310	phase I
BRD-K69556541	CC(C)[C@]1(O)[C@@H](OC(=O)c2ccc[nH]2)[C@]3(O)[C@]4(O)[C@]1(C)[C@]5(O)C[C@@]3(C)[C@@]6(O)CC[C@H](C)[C@@H](O)[C@]46O5	CID:6610313	phase I
BRD-A42831637	CCCCCc1cc(O)c2C3C=C(CC[C@H]3C(C)(C)Oc2c1)C(=O)O	CID:6610319	phase I
BRD-K93080877	C[C@H](N)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccccc1)C(=O)CCl	CID:6610326	phase I
BRD-K69690935	COc1ccc(C=CC(=O)CC(=O)C=Cc2cccc(O)c2OC)cc1O	CID:6610332	phase I
BRD-K77830450	CC(=O)O[C@H]1[C@@H](O)[C@H]2C(C)(C)CC[C@@H](O)[C@]2(C)[C@@]3(O)C(=O)C[C@@](C)(O[C@]13C)C=C	CID:6610344	phase I
BRD-K95992530	CC(C)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCNC(=N)N)NC1=O	CID:6610347	phase I
BRD-K99291625	CS(=O)(=O)c1ccc(cc1)c2nc(c([nH]2)c3ccncc3)c4ccc(F)cc4	CID:6610350	phase I
BRD-K70549064	CN[C@@H]1C[C@@]2(C)O[C@@H]([C@@H]1OC)n3c4ccccc4c5c6CNC(=O)c6c7c8ccccc8n2c7c35	CID:6610353	phase I
BRD-K71726959	CC(C)n1cnc2c(NCc3ccccc3)nc(NCCO)nc12	CID:6610355	phase I
BRD-K30381384	COc1cc(NC(=O)c2cc(on2)C3CC3)c(OC)cc1Cl	CID:6619100	phase I
BRD-K53331454	O=C(NC1(CCCCC1)C#N)c2cc3ccccc3oc2=O	CID:6620794	phase I
BRD-K38596918	CC(C)(C)c1ccc(OCCCn2c(=O)sc3ccccc23)cc1	CID:6620960	phase I
BRD-K88964386	COc1ccc(CCNC(=O)CSc2nc3ccccc3nc2N4CCCC4)cc1OC	CID:6621011	phase I
BRD-A72837804	CC1CN(CC(C)O1)c2nc3ccccc3nc2SCC(=O)NCCc4ccccc4	CID:6621029	phase I
BRD-A70879086	CC1CN(CC(C)O1)c2nc3ccccc3nc2SCC(=O)Nc4ccccc4	CID:6621039	phase I
BRD-K64780785	CCc1ccc(cc1)c2nc(CSCC(=O)NC3CC3)c(C)o2	CID:6622243	phase I
BRD-K24925364	COc1ccc(cc1NC(=O)C(C)C)c2cn3cccnc3n2	CID:6622773	phase I
BRD-K71701252	CC(=O)N1CCOc2cc(ccc12)S(=O)(=O)NCC3CCC(CC3)C(=O)Nc4cccc(C)c4	CID:6626036	phase I
BRD-K38690464	OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)OCC=C)c3coc4ccccc4c3=O)cc1	CID:6669976	phase I
BRD-K98426715	OCc1ccc(cc1)[C@@H]2C[C@H](CSc3nc(c(o3)c4ccccc4)c5ccccc5)O[C@@H](O2)c6ccc(NC(=O)CCCCCCC(=O)NO)cc6	CID:6675804	phase I
BRD-A72711497	CC[C@H](C1OC(CC)(C[C@@H]1C)C1CC[C@](O)(CC)[C@H](C)O1)C(=O)C(C)[C@@H](O)[C@H](C)CCc1ccc(C)c(O)c1C(O)=O	CID:6708465	phase I
BRD-A51382177	CCC(=O)O[C@@H](OP(=O)(CCCCc1ccccc1)CC(=O)N1C[C@@H](C[C@H]1C(O)=O)C1CCCCC1)C(C)C	CID:6708482	phase I
BRD-A52805806	CC(C)c1c(O)ccc2c1CCC3[C@](C)(CCC[C@@]32C)C=O	CID:6708512	phase I
BRD-A10969569	CO[C@@H]1CC2N3CC(O)C2(C=C1)c4cc5OCOc5c(OC)c4C3	CID:6708518	phase I
BRD-A32349859	COC(=O)CC1C(C)(C)C(=O)C[C@@H]2O[C@@]34CC(=O)O[C@@H](c5ccoc5)[C@]4(C)CCC(C3=C)[C@]12C	CID:6708532	phase I
BRD-K34330170	COc1cc2OC[C@H]3Oc4c(CC=C(C)C)c(O)ccc4C(=O)[C@H]3c2cc1OC	CID:6708539	phase I
BRD-A18932057	CC(=O)Oc1ccc2C3c4cc(OC(=O)C)c(OC(=O)C)c(OC(=O)C)c4CC3(O)COc2c1OC(=O)C	CID:6708558	phase I
BRD-A41112154	CC(=O)O[C@@H]1CC[C@@]2(C)C(CC[C@]3(C)C2CC=C4C5CC(C)(C)CC[C@@]5(CC[C@]43C)C(=O)O)C1(C)C	CID:6708573	phase I
BRD-A58269583	CC1(C)[C@H](O)C=C[C@]2(C)C3CC[C@@]4(C)[C@@H](OC(=O)C=C4[C@]3(C)OC(=O)CC12)c5ccoc5	CID:6708582	phase I
BRD-A52326238	CC(=O)O[C@@H]1CC2C(C)(C)C=CC(=O)[C@]2(C)C3CC[C@@]4(C)[C@@H](OC(=O)C5OC54[C@]13C)c6ccoc6	CID:6708584	phase I
BRD-A89434049	CC12C[C@@H](O)C3C(CCC4CC(O)CCC43C)C2(O)CCC1C5=CC(=O)OC5	CID:6708600	phase I
BRD-A02713983	CC(=O)O[C@@H]1CC2C(C)(C)C(=O)CC[C@]2(C)C3CC[C@@]4(C)[C@@H](OC(=O)C=C4[C@]13C)c5ccoc5	CID:6708636	phase I
BRD-A47144777	CC1(C)C2C[C@@H](O)[C@]3(C)C(CC[C@@]4(C)[C@@H](OC(=O)C=C43)c5ccoc5)[C@@]2(C)CCC1=O	CID:6708643	phase I
BRD-A92161634	CN1[C@H]2CC3CC1C(O)C2O3	CID:6708684	phase I
BRD-K52015643	COc1ccc(C=Cc2cc(O)cc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c2)cc1	CID:6708703	phase I
BRD-K03600606	O=C(O[C@H]1Cc2c(OC(=O)c3ccccc3)cc(OC(=O)c4ccccc4)cc2O[C@@H]1c5ccc(OC(=O)c6ccccc6)c(OC(=O)c7ccccc7)c5)c8ccccc8	CID:6708716	phase I
BRD-A92826379	O=C1CCCC2C3CC(CN12)[C@@H]1CCCCN1C3	CID:6708718	phase I
BRD-A17819071	CC1(C)C=CC(=O)[C@@]2(C)C1CC(=O)[C@]3(C)C2CC[C@@]4(C)[C@@H](OC(=O)C5OC543)c6ccoc6	CID:6708725	phase I
BRD-A66861218	CCC(=O)OCC(=O)[C@@]1(OC(=O)CC)[C@@H](C)CC2C3CCC4=CC(=O)C=C[C@]4(C)C3(F)[C@@H](O)C[C@]12C	CID:6708733	phase I
BRD-A45333398	CO[C@@H]1C[C@H](O[C@H]2CC[C@]3(C)C4CC[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)C6=CC(=O)OC6)O[C@H](C)[C@@H]1O	CID:6708762	phase I
BRD-A71459254	COC1CC(O[C@H]2CC[C@]3(C=O)C4CC[C@]5(C)C(CC[C@]5(O)C4CC[C@]3(O)C2)C6=CC(=O)OC6)OC(C)C1O	CID:6708764	phase I
BRD-K25905511	COc1ccc(cc1)c2cc(=O)c3c(O)cc(O[C@H]4O[C@H](CO[C@@H]5O[C@@H](C)[C@H](O)[C@@H](O)[C@H]5O)[C@@H](O)[C@H](O)[C@H]4O)cc3o2	CID:6708769	phase I
BRD-A35588707	COc1cc(cc(OC)c1O)[C@H]1[C@@H]2C(COC2=O)C(O[C@@H]2O[C@@H]3CO[C@H](OC3[C@H](O)[C@H]2O)c2cccs2)c2cc3OCOc3cc12	CID:6708778	phase I
BRD-K78838262	C[C@H]1[C@H]2[C@H](OC1=O)[C@@H]3C(=CC(=O)C3=C(C)C[C@@H]2O)C	CID:6708801	phase I
BRD-A02180903	C[C@H]1CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:6710614	phase I
BRD-A84205515	COc1ccc2C3CCC4(C)C(O)[C@H](O)CC4C3CCc2c1	CID:6710621	phase I
BRD-A09495397	CN1CCc2cc3OCOc3cc2[C@H]1C4OC(=O)c5c6OCOc6ccc45	CID:6710622	phase I
BRD-A77824596	CC1(C)O[C@@H]2CC3C4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:6710651	phase I
BRD-A98431941	CNC(C)[C@H](O)c1ccccc1	CID:6710657	phase I
BRD-A37959677	C[C@]12CCC3C(CCc4cc(O)ccc34)C1CCC2=O	CID:6710658	phase I
BRD-A38749782	CC(=O)OCC(=O)[C@@]1(O)CCC2C3CCC4=CC(=O)CC[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]12C	CID:6710659	phase I
BRD-A15297126	CC(=O)OCC(=O)[C@@]12OC(C)(C)O[C@@H]1CC1C3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]21C	CID:6710662	phase I
BRD-A95513702	C[C@@]12CCC3C(CCC4=CC(=O)C=C[C@]34C)C2CCC1=O	CID:6710699	phase I
BRD-A41519720	OC(CC[C@@H]1[C@H](N(C1=O)c1ccc(F)cc1)c1ccc(O)cc1)c1ccc(F)cc1	CID:6710700	phase I
BRD-A35989968	CC(=O)O[C@@]1(CCC2C3C=C(C)C4=CC(=O)CCC4(C)C3CCC12C)C(C)=O	CID:6710729	phase I
BRD-K54728231	O[C@@H]1O[C@H](COC(=O)CC[N+](=O)[O-])[C@@H](OC(=O)CC[N+](=O)[O-])[C@H](OC(=O)CC[N+](=O)[O-])[C@H]1OC(=O)CC[N+](=O)[O-]	CID:6710740	phase I
BRD-K40742111	COc1cc(C)c(C(=O)Oc2cc(C)c(O)c(C(=O)O)c2C)c(O)c1C=O	CID:6710741	phase I
BRD-K78329127	COc1cc(OC)c(C(=O)c2ccc(O)cc2)c(OC)c1	CID:6710752	phase I
BRD-K92678294	COc1ccccc1c2coc3cc(OC)c(OC)c(OC)c3c2=O	CID:6710754	phase I
BRD-K08714182	COc1c(oc2c(CC=C(C)C)c3OC(C)(C)C=Cc3c(OC)c2c1=O)c4ccccc4	CID:6710761	phase I
BRD-K47328134	NCCCC[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)O	CID:6710772	phase I
BRD-A09161221	CC(=O)O[C@@H]1CC(=O)OC(C)(C)C2CC(=O)[C@]3(C)C(CC[C@@]4(C)[C@@H](OC(=O)[C@H]5O[C@]543)c6ccoc6)[C@]21C	CID:6710776	phase I
BRD-A01593789	CC(=O)O[C@@]1(CCC2C3C=C(Cl)C4=CC(=O)CC[C@]4(C)C3CC[C@@]21C)C(=O)C	CID:6710779	phase I
BRD-A55594068	CC[C@]1(O)CC2CN(C1)CCc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C)[C@@H]1[C@]22CCN3CC=C[C@](CC)([C@@H]23)[C@@H](OC(C)=O)[C@]1(O)C(=O)OC	CID:6710780	phase I
BRD-K32292990	Fc1ccc(Nc2cc3C(=O)NC(=O)c3cc2Nc2ccc(F)cc2)cc1	CID:6711154	phase I
BRD-K02607075	COc1cc2CC[N+](C)(C)[C@@H]3Cc4ccc(O)c(Oc5cc6[C@H](Cc7cccc(Oc(c1O)c32)c7)N(C)CCc6cc5OC)c4	CID:6713947	phase I
BRD-A41941932	OC[C@H]1OC([C@H](O)[C@@H](O)[C@@H]1O)c2c(O)cc(O)c3c(=O)cc(oc23)c4ccc(O)cc4	CID:6713958	phase I
BRD-K64236792	C[C@H]1[C@H]2[C@H](OC1=O)[C@H]3C(=CC(=O)C3=C(C)C[C@@H]2O)C	CID:6713966	phase I
BRD-A63894585	CCC(=O)OC1([C@@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C)C(=O)CCl	CID:6713978	phase I
BRD-A85424553	S=C(NC1CCCCC1)N2CCC(CC2)C3C=NC=N3	CID:6713984	phase I
BRD-A13650332	Cc1onc(c1C(=O)N[C@H]1[C@H]2SC(C)(C)C(N2C1=O)C(O)=O)-c1c(F)cccc1Cl	CID:6713996	phase I
BRD-K46137903	CCOC(=O)O[C@@]1(CC[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@@]21C)C(=O)COC(=O)CC	CID:6714002	phase I
BRD-A39290993	CC(=O)O[C@@]1(CC[C@H]2[C@@H]3C=C(Cl)C4=CC(=O)C5CC5[C@]4(C)[C@H]3CC[C@@]21C)C(=O)C	CID:6714003	phase I
BRD-A65739223	CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N2C(C[C@@H]3CCC[C@@H]32)C(=O)O	CID:6714009	phase I
BRD-A23712469	CCC(C)C(N)C1=NC(CS1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@H]2CCCCNC(=O)[C@H](CC(=O)N)NC(=O)[C@@H](CC(=O)O)NC(=O)[C@H](Cc3cnc[nH]3)NC(=O)[C@@H](Cc4ccccc4)NC(=O)[C@@H](NC(=O)[C@@H](CCCN)NC2=O)[C@@H](C)CC	CID:6714010	phase I
BRD-A71816415	CCC(C)C(=O)O[C@H]1C[C@H](O)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(O)=O)C12	CID:6728942	phase I
BRD-K55139645	COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1	CID:6729029	phase I
BRD-K87467896	COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1	CID:6729031	phase I
BRD-K14790374	COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1	CID:6729038	phase I
BRD-K66426634	NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1	CID:6729040	phase I
BRD-K92863101	NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8	CID:6729078	phase I
BRD-K12598223	COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1	CID:6729207	phase I
BRD-K60833663	COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC	CID:6729240	phase I
BRD-K71935468	COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC	CID:6729245	phase I
BRD-K70839030	COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC	CID:6729328	phase I
BRD-K29345712	OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9	CID:6729449	phase I
BRD-K95823739	COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1	CID:6729559	phase I
BRD-K01425313	OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9	CID:6729586	phase I
BRD-K41925105	COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC	CID:6729590	phase I
BRD-K32896438	COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC	CID:6729593	phase I
BRD-K19624190	OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9	CID:6729762	phase I
BRD-K81813927	COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccccc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9	CID:6729775	phase I
BRD-K70947604	NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7	CID:6729782	phase I
BRD-K74569352	NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7	CID:6729815	phase I
BRD-K16180117	COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19	CID:6729968	phase I
BRD-K58347372	COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19	CID:6730584	phase I
BRD-K64525051	COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17	CID:6731173	phase I
BRD-K94991378	COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17	CID:6731789	phase I
BRD-K65342895	COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19	CID:6731816	phase I
BRD-K51592837	COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17	CID:6731927	phase I
BRD-K70086257	COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19	CID:6732081	phase I
BRD-A09749088	C[C@]1(CCC[C@]2(C)[C@H]3CC(O)[C@](C)(C=C)C=C3CC[C@@H]12)C(=O)O	CID:6732844	phase I
BRD-K64881305	CC(C)[C@@H](N(CCCN)C(=O)c1ccc(C)cc1)c1nc2cc(Cl)ccc2c(=O)n1Cc1ccccc1	CID:6851740	phase I
BRD-K72381300	Oc1cc2CCNC[C@H](c3ccccc3)c2cc1O	CID:6852376	phase I
BRD-A68202111	C[C@@H]1O[C@@H](O[C@H]2C[C@@H](O)[C@]3(CO)[C@H]4[C@H](O)C[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)C6COC(=O)C6)[C@H](O)[C@H](O)[C@H]1O	CID:6852401	phase I
BRD-A30856524	CC1(C)CC2C1CC[C@]1(C)CCC3C(CC(=O)O[C@]23C1)C(O)=O	CID:6857784	phase I
BRD-K03557653	COc1ccc2C(=O)/C(=C\c3ccc(OC)c(OC)c3)/COc2c1	CID:6857791	phase I
BRD-K73819439	[O-][N+](=O)c1ccc(/C=N/NC(=O)CNc2cccc(c2)[N+](=O)[O-])o1	CID:6872741	phase I
BRD-K02558072	COC(=O)N/N=C/c1ccc(o1)[N+](=O)[O-]	CID:6875617	phase I
BRD-K64970062	Cc1ccc(NC(=O)CCC(=O)N/N=C/c2ccc(o2)[N+](=O)[O-])cc1C	CID:6875690	phase I
BRD-K85660637	[O-][N+](=O)c1ccc(/C=N/NC(=O)CNc2cccc3ccccc23)o1	CID:6884367	phase I
BRD-K81272440	[O-][N+](=O)c1ccc(cc1)-c1ccc(\C=N\N2CC(=O)NC2=O)o1	CID:6914273	phase I
BRD-K58550667	O=C(NCCCCC1CCN(CC1)C(=O)c1ccccc1)\C=C\c1cccnc1	CID:6914657	phase I
BRD-A52530684	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](OC5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(=O)CO	CID:6916127	phase I
BRD-K06895174	CO[C@H]1CN(CCCOc2ccc(F)cc2)CC[C@H]1NC(=O)c1cc(Cl)c(N)cc1OC	CID:6917698	phase I
BRD-K02283807	O[C@H]1C[C@H](OCc2ccc(cc2)c3ccccc3)[C@H](CC/C=C\CCC(=O)O)[C@H]1N4CCCCC4	CID:6918030	phase I
BRD-K19706299	CCCCC[C@H](O)CC[C@H]1[C@H](O)C[C@@H]2Cc3c(C[C@H]12)cccc3OCC(O)=O	CID:6918140	phase I
BRD-K42679050	CC(=O)N(OCc1ccccc1)[C@H]1[C@H](O)C(C)(C)Oc2ccc(cc12)C#N	CID:6918184	phase I
BRD-K55677650	Cc1ccc(CC2(O)CCN(CCOc3ccc(O)cc3)CC2)cc1	CID:6918409	phase I
BRD-K45995181	CCP(CC)(CC)=[Au]S[C@@H]1O[C@H](COC(C)=O)[C@@H](OC(C)=O)[C@H](OC(C)=O)[C@H]1OC(C)=O	CID:6918453	phase I
BRD-K05104363	Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F	CID:6918454	phase I
BRD-K70914287	CN1CCC(CC1)Nc1ncc2ncnc(Nc3ccc(F)c(Cl)c3)c2n1	CID:6918508	phase I
BRD-K18849474	CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1SC(=O)C(C)C	CID:6918540	phase I
BRD-K17743125	ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)Nc1ccccc1	CID:6918638	phase I
BRD-K55187425	COc1cc(OC)c(\C=C\S(=O)(=O)Cc2ccc(OC)c(NCC(O)=O)c2)c(OC)c1	CID:6918736	phase I
BRD-K02130563	Cc1[nH]c2ccccc2c1CCNCc1ccc(\C=C\C(=O)NO)cc1	CID:6918837	phase I
BRD-K04466929	CC(=O)Nc1ccc(cc1)C(=O)Nc2cc(ccc2N)c3cccs3	CID:6918878	phase I
BRD-K26171350	C[C@]12CC(=O)[C@@H]3[C@H](CCC4=CC(=O)CC[C@]34C)[C@@H]1CCC2=O	CID:6927363	phase I
BRD-K52640952	COc1cc(O)c2C(=O)C[C@@H](Oc2c1)c3ccccc3	CID:6950539	phase I
BRD-K07390541	CCOC(=O)C1=C[C@]2(CC)CCCN3CCc4c([C@@H]23)n1c1ccccc41	CID:6978790	phase I
BRD-K76359782	CN1CC[C@]2(C)[C@@H]1N(C)c3ccc(O)cc32	CID:7015679	phase I
BRD-K04431258	CC(C)[C@H](N)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(O)=O	CID:7020214	phase I
BRD-K17113870	CC[C@H](C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@H]12	CID:7048568	phase I
BRD-K24559712	C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@H]34)[C@H]1CC[C@@]2(O)C#C	CID:7048591	phase I
BRD-K52237148	Cc1nnc(SCC2=C(N3[C@H](SC2)[C@@H](NC(=O)Cn2cnnn2)C3=O)C(O)=O)s1	CID:7048624	phase I
BRD-K87116849	CC(=O)OCC1=C(N2[C@H](SC1)[C@@H](NC(=O)Cc1cccs1)C2=O)C(O)=O	CID:7048637	phase I
BRD-K44094313	CC#C[C@]1(O)CC[C@@H]2[C@@H]3CCC4=CC(=O)CCC4=C3[C@H](C[C@]12C)c1ccc(cc1)N(C)C	CID:7048709	phase I
BRD-K70504303	C[C@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)C=C[C@]34C)[C@H]1CC[C@]2(O)C(=O)CO	CID:7048968	phase I
BRD-K69743918	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@H]1CCC2=O	CID:7059423	phase I
BRD-K99712306	COC(=O)[C@H]1[C@@H](O)CC[C@H]2CN3CCc4c([nH]c5ccccc45)[C@H]3C[C@@H]12	CID:7059505	phase I
BRD-K79062806	CO[C@]12C[C@@H](COC(=O)c3cncc(Br)c3)CN(C)[C@H]1Cc1cn(C)c3cccc2c13	CID:7059561	phase I
BRD-K64106162	C[C@@H]1CC(=O)NN=C1c1ccc(N)c(c1)[N+]([O-])=O	CID:7060079	phase I
BRD-K37208476	C[C@]12CC[C@@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@H]1CC[C@@]2(O)C#C	CID:7061041	phase I
BRD-K00885784	C[C@]12CC[C@@H]3[C@@H](C=CC4=CC(=O)CC[C@]34C)[C@H]1CC[C@@]21CCC(=O)O1	CID:7061052	phase I
BRD-K82481048	C[C@H]1C[C@H]2[C@H]3CC[C@](O)(C(=O)CO)[C@@]3(C)C[C@H](O)[C@H]2[C@@]2(C)C=CC(=O)C=C12	CID:7061270	phase I
BRD-K83229621	C[C@]12CC[C@@H]3[C@@H](CCC4=C3CCC(=O)C4)[C@H]1CC[C@@]2(O)C#C	CID:7061273	phase I
BRD-K28892486	Cc1cccc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)c1	CID:7066682	phase I
BRD-K98519396	CC1(C)[C@H](O)CC[C@@]2(C)[C@H](COc3ccc4ccc(=O)oc4c3)C(=C)CC[C@H]12	CID:7067264	phase I
BRD-K47036706	CC(=O)OCC(=O)[C@@]12OC(C)(C)O[C@@H]1C[C@H]1[C@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]21C	CID:7067797	phase I
BRD-K15744901	CCC1=C[C@@H]2CN3CCc4c([nH]c5ccccc45)[C@@](C2)([C@H]13)C(=O)OC	CID:7073234	phase I
BRD-K10481964	COc1ccc2[C@H]3CC[C@@]4(C)[C@H](CC[C@@]4(O)C#C)[C@@H]3CCc2c1	CID:7076513	phase I
BRD-K62586643	CC1(C)N2[C@@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccccc5)C2=O	CID:7079134	phase I
BRD-K35862502	CC(=O)[C@H]1CC[C@H]2[C@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@@H]3CC[C@]12C	CID:7088398	phase I
BRD-K09129322	C[C@H](CCC(O)=O)[C@H]1CC[C@H]2[C@@H]3[C@@H](CC(=O)[C@]12C)[C@@]1(C)CCC(=O)C[C@H]1CC3=O	CID:7091864	phase I
BRD-K37439386	CC(=O)[C@H]1CC[C@H]2[C@H]3CC[C@H]4C[C@H](O)CC[C@]4(C)[C@@H]3C(=O)C[C@]12C	CID:7092517	phase I
BRD-K47244735	CC(=O)[C@H]1CC[C@H]2[C@H]3CCC4=CC(=O)CC[C@]4(C)[C@@H]3CC[C@]12C	CID:7092664	phase I
BRD-K89097220	CCN(CC)c1ccc(cc1[N+]([O-])=O)C1=NNC(=O)C[C@H]1C	CID:7122097	phase I
BRD-K55502647	COc1ccccc1Nc2nc(nc(n2)N3CCOCC3)N4CCOCC4	CID:7192031	phase I
BRD-K45216862	Brc1cccc2sc(NC(=O)c3ccc4OCCOc4c3)nc12	CID:7202911	phase I
BRD-K27074404	Cc1csc(NC(=O)CSc2ccc(nn2)c3ccccc3)n1	CID:7211972	phase I
BRD-K55186349	[O-][N+](=O)c1ccc(cc1)C(=O)Oc1coc(CSc2ncccn2)cc1=O	CID:7217941	phase I
BRD-K74189021	Cc1ccnc(SCc2cc(=O)c(OC(=O)c3ccc(cc3)[N+]([O-])=O)co2)n1	CID:7217942	phase I
BRD-K74126469	Cc1ccc(cc1[N+]([O-])=O)C(=O)Oc1coc(CSc2ncccn2)cc1=O	CID:7217946	phase I
BRD-K52341396	Cc1ccnc(SCc2cc(=O)c(OC(=O)c3ccc(C)c(c3)[N+]([O-])=O)co2)n1	CID:7217947	phase I
BRD-K28120222	C\C1=C/CC[C@@]2(C)O[C@@H]2[C@H]2OC(=O)C(=C)[C@@H]2CC1	CID:7251185	phase I
BRD-K86574132	CC(C)N1C(=O)S/C(=C/c2ccc(Sc3nc4ccccc4[nH]3)o2)/C1=O	CID:7326481	phase I
BRD-K76595177	Cc1ccc(C)c(OCCn2cc(C(=O)O)c3ccccc23)c1	CID:7345532	phase I
BRD-K76357752	CC1CCN(CC1)C(=O)Cn2c3ccc(F)cc3c4nc5SCCCn5c(=O)c24	CID:7693333	phase I
BRD-K67778494	O=C(Cn1c2ccccc2c3nc4SCCn4c(=O)c13)N5CCCC5	CID:7694069	phase I
BRD-K37127624	CC1CCN(CC1)C(=O)Cn2c3ccccc3c4nc5SCCCn5c(=O)c24	CID:7708820	phase I
BRD-K77918867	Oc1ccccc1NC(=O)c1ccncc1	CID:7791937	phase I
BRD-K70500696	Cc1c(NC(=O)/C(=C/c2ccc3ccccc3c2)/C#N)c(=O)n(c4ccccc4)n1C	CID:7972413	phase I
BRD-K85822033	Cc1cccn2cc(COc3ccc(F)cc3Cl)nc12	CID:8005457	phase I
BRD-K19027210	C(c1ccccc1)n1ncc2c(ncnc12)N1CCN(CC1)c1ccccc1	CID:8056641	phase I
BRD-K99582188	Clc1ccc(Cn2ncc3c(ncnc23)N2CCN(CC2)c2ccccc2)cc1	CID:8056691	phase I
BRD-K96194181	CC(=O)Nc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccc(cc1)C(C)=O	CID:8194745	phase I
BRD-K51896917	CC(=O)c1ccc(cc1)N1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)CCc2c1	CID:8460266	phase I
BRD-K23896287	Fc1ccc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)cc1	CID:8512230	phase I
BRD-K92269225	COc1ccc(NC(=O)c2ccccc2SCc2ccccc2)cc1	CID:8796093	phase I
BRD-K66884694	Cn1nnnc1Sc2ncnc3scc(c4ccc(Cl)cc4)c23	CID:9266740	phase I
BRD-K31286015	CCOc1ccc(CCNC(=O)c2ccccn2)cc1OCC	CID:9474030	phase I
BRD-K85563610	O=C(CCc1cccnc1)NCCCCC1CCN(CC1)C(=O)c1ccccc1	CID:9543513	phase I
BRD-K17820047	Nc1ccccc1NC(=O)CCCCCCC(=O)Nc2ccccc2	CID:9543540	phase I
BRD-K63606607	C[C@@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@@H](O)CC[C@@]43C)[C@@]2(O)CC[C@@H]1c5ccc(=O)oc5	CID:9547215	phase I
BRD-K70881766	C[C@H]1[C@H]2[C@H](C[C@H]3[C@@H]4CC=C5C[C@H](CC[C@]5(C)[C@H]4CC[C@]23C)O[C@@H]6O[C@H](CO)[C@H](O)[C@H](O[C@@H]7O[C@H](CO)[C@@H](O)[C@H](O)[C@H]7O)[C@H]6O[C@@H]8O[C@@H](C)[C@H](O)[C@@H](O)[C@H]8O)N9C[C@@H](C)CC[C@H]19	CID:9549171	phase I
BRD-K36529613	CC(C)NCCCn1c(Sc2cc3OCOc3cc2I)nc2c(N)ncnc12	CID:9549213	phase I
BRD-K12244279	N\C(Sc1ccc(N)cc1)=C(\C#N)c1ccccc1C(F)(F)F	CID:9549284	phase I
BRD-K94176593	Nc1cccc(c1)-c1cc2c(Oc3cccc(O)c3)ncnc2[nH]1	CID:9549289	phase I
BRD-K02965346	CN(c1cccc(Cl)c1)S(=O)(=O)c1ccc2NC(=O)\C(=C/c3[nH]c(C)c(C(=O)N4CCN(C)CC4)c3C)c2c1	CID:9549297	phase I
BRD-K14618467	O=C(N1CCC(CC1)N1CCCC1)c1ccc(Nc2nccc(n2)-c2cc3ccccc3s2)cc1	CID:9549298	phase I
BRD-K67537649	COc1ccc(Cl)cc1NC(=O)Nc1cc(C)nc2ccccc12	CID:9549305	phase I
BRD-K45895591	CCOC(=O)N1CCC(CC1)NC(=O)c2ccc3SCCN(Cc4ccc(F)cc4)c3c2	CID:9550235	phase I
BRD-K81397638	O=C(N1CCN(Cc2ccccc2)CC1)c3ccc(CNS(=O)(=O)c4ccccc4)cc3	CID:9550286	phase I
BRD-K16472144	Cc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)N3CCN(Cc4ccccc4)CC3	CID:9551230	phase I
BRD-K49403449	CC(=O)Nc1ccc(/C=N/NC(=O)CC2CCCCC2)cc1	CID:9555025	phase I
BRD-K17119186	O=C(Oc1cccc(\C=N\Nc2nc(Nc3ccccc3)nc(n2)N2CCOCC2)c1)c1ccco1	CID:9592990	phase I
BRD-K53263234	Clc1ccc(cc1)-c1nc2sccn2c1\C=N\OCc1ccc(Cl)c(Cl)c1	CID:9600409	phase I
BRD-K74430258	Clc1cccc(C=NC=Nc2cccc(Cl)c2)c1	CID:9604992	phase I
BRD-K31699485	COc1cccc(C=NC=Nc2cccc(OC)c2)c1	CID:9604993	phase I
BRD-K95986273	Cc1nc2ccccc2n1\N=C\c1ccc(s1)[N+]([O-])=O	CID:9616928	phase I
BRD-K17628612	Cc1ccc(/C=N/NC(=O)CCC(=O)Nc2ccc(C)cc2C)o1	CID:9640748	phase I
BRD-K92991072	Oc1c(CC=C)cccc1\C=N\NC(=O)CN1CCN(Cc2ccccc2)CC1	CID:9675990	phase I
BRD-K28863208	Clc1ccc(cc1)C(=O)N[C@H]1CN2CCC1CC2	CID:9795278	phase I
BRD-A44551378	CC(=O)C(C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1	CID:9795867	phase I
BRD-K79342257	Nc1scc2c(nn(c3ccccc3)c(=O)c12)C(=O)O	CID:9795907	phase I
BRD-K11153516	NC(=O)c1ccc(I)c(c1)[N+]([O-])=O	CID:9796068	phase I
BRD-K40892394	COc1ccnc(NC2CCN(CC2)C(=O)c2ccc(cc2)C#N)c1	CID:9797857	phase I
BRD-K11927976	Cc1ccc2c(c1C)n(CCCN)c1ccccc1c2=O	CID:9799509	phase I
BRD-K42452249	Cc1ccccc1C(=O)c1ccc(Nc2ccc(Br)cc2N)cc1Cl	CID:9801969	phase I
BRD-K14880289	Cc1nc(sc1CSc1ccc(OCC(O)=O)c(C)c1)-c1ccc(cc1)C(F)(F)F	CID:9803963	phase I
BRD-K13810148	CCN(CC)Cc1ccc2cc(COC(=O)Nc3ccc(cc3)C(=O)NO)ccc2c1	CID:9804992	phase I
BRD-A35511923	COC(=O)C(CCCNC(=N)N)NC(=O)CCCc1c([nH]c2c(F)cc(F)cc12)c3ccccc3	CID:9805390	phase I
BRD-K05151076	CCCCCS(=O)(=O)CCCCCCCCCCn1c(c(C)c2cc(O)ccc12)-c1ccc(O)cc1	CID:9806489	phase I
BRD-K56751279	C[C@@H](N)c1ccc(cc1)C(=O)Nc1ccnc2[nH]ccc12	CID:9810884	phase I
BRD-K19669037	COC(=O)[C@H](CC(C)C)NC(=O)c1ccc(NC[C@@H](N)CS)cc1-c1cccc2ccccc12	CID:9811606	phase I
BRD-K13566078	Cc1cnc2c(NCCN)nc3ccc(C)cc3n12	CID:9813758	phase I
BRD-K31460632	C[C@H](N)Cc1cccc(c1)C(F)(F)F	CID:9815618	phase I
BRD-K59650319	CN(C1CCCCC1)C(=O)c1sc2nc3ccc(N)cc3n2c1C	CID:9819432	phase I
BRD-K69763916	N[C@@](CC1c2ccccc2Oc3ccccc13)([C@H]4C[C@@H]4C(=O)O)C(=O)O	CID:9819927	phase I
BRD-K12079898	CC(C)c1ccccc1S(=O)(=O)c1cc(N)c2ncccc2c1[N+]([O-])=O	CID:9820766	phase I
BRD-K26429091	CC(=CCCN1CCC(CC1)NC(=O)[C@@](O)(C2CCCC2)c3ccccc3)C	CID:9821459	phase I
BRD-K82164249	CC(=O)Nc1ccc(OC[C@](C)(O)C(=O)Nc2ccc(c(c2)C(F)(F)F)[N+]([O-])=O)cc1	CID:9824562	phase I
BRD-K90382497	COc1cc2ncn(-c3cc(OCc4ccccc4C(F)(F)F)c(s3)C(N)=O)c2cc1OC	CID:9826308	phase I
BRD-K49865102	OC[C@@H](O)CONC(=O)c1ccc(F)c(F)c1Nc1ccc(I)cc1F	CID:9826528	phase I
BRD-A34806832	C[C@@H]1O[C@@H](O[C@H]2CC[C@]3(C)C4CC[C@]5(C)[C@H](CC[C@]5(O)C4CCC3=C2)c6ccc(=O)oc6)[C@H](O)[C@H](O)[C@H]1O	CID:9828429	phase I
BRD-K13646352	CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1	CID:9829523	phase I
BRD-K36198571	Cc1cc(C)c(N(Cc2ccccc2)S(=O)(=O)c2ccc(OCCNC(=O)c3cc4ccccc4o3)cc2)c(c1)C(=O)NO	CID:9830392	phase I
BRD-K49519144	N[C@]1(CS(=O)(=O)[C@H]2[C@@H]([C@@H]12)C(O)=O)C(O)=O	CID:9834591	phase I
BRD-K30707190	Cc1ccc(\C=N\NC(=O)c2ccccc2Oc2ccccc2)o1	CID:9836739	phase I
BRD-K95655893	CN(C)c1ccc(/C=C/2\C(=O)Nc3ccccc23)c4ccccc14	CID:9839842	phase I
BRD-K00615600	CN(C)Cc1ccc(cc1)-c1nc2cccc3C(=O)NCCn1c23	CID:9840076	phase I
BRD-K32405725	CCOC(=O)[C@@]1(CCCCCCOc2ccc(Cl)cc2)CO1	CID:9840324	phase I
BRD-K07507905	C[C@H](Cc1ccc(OCC(O)=O)cc1)NC[C@H](O)c1cccc(Cl)c1	CID:9841972	phase I
BRD-K64341947	COc1ccc(NC(=O)c2cc(OCCCN(C)C)nn2Cc2ccccc2)cc1	CID:9844347	phase I
BRD-K33312228	C[C@@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C(=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO)Cl	CID:9846332	phase I
BRD-A78391468	C[C@]12C[C@H](O)C3C(CCC4=CC(=O)C=C[C@]34C)C1CC[C@]2(O)C(=O)COC(=O)CCC(O)=O	CID:9847023	phase I
BRD-K09557221	CCc1c(nn(c1-c1ccc(Br)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1	CID:9849616	phase I
BRD-K09537769	O=c1cc(oc2c3ccccc3ccc12)N1CCOCC1	CID:9860529	phase I
BRD-K16485616	Nc1ccccc1NC(=O)c1ccc(CNc2nccc(n2)-c2cccnc2)cc1	CID:9865515	phase I
BRD-K76630978	CN(C)Cc1ccccc1Sc1ccc(I)cc1CO	CID:9865652	phase I
BRD-K63150726	CCCCCOc1c(OC)ccc2cc(C(=O)NCc3ccc4OCOc4c3)c(=O)[nH]c12	CID:9867770	phase I
BRD-K25340465	FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1	CID:9868037	phase I
BRD-K03015355	CN1CCN(CCCC(=O)O[C@H]2[C@@H](O)[C@H]3C(C)(C)CC[C@H](O)[C@]3(C)[C@@]4(O)C(=O)C[C@@](C)(O[C@]24C)C=C)CC1	CID:9871875	phase I
BRD-K72895815	COc1cc2c(C(=O)N(COc3cc(=O)n4cccc(OCCN5CCCCC5)c4n3)S2(=O)=O)c(c1)C(C)C	CID:9872438	phase I
BRD-K70241288	C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc3ccc(cc3)c4ccccc4c5nn[nH]n5)C1=O	CID:9872740	phase I
BRD-K62221994	CC(C)OC(=O)c1cn(Cc2c(F)cccc2F)c3sc(c(CN(C)Cc4ccccc4)c3c1=O)c5ccc(NC(=O)C(C)C)cc5	CID:9874838	phase I
BRD-K76908866	COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1	CID:9874913	phase I
BRD-K37130656	Clc1ccc(s1)C(=O)NC[C@H]1CN(C(=O)O1)c1ccc(cc1)N1CCOCC1=O	CID:9875401	phase I
BRD-K97591839	NCCc1ccc(O)cc1N	CID:9877425	phase I
BRD-A57382968	CN1C(C(=O)Nc2ccccn2)C(=O)c2ccccc2S1(=O)=O	CID:9880620	phase I
BRD-K33445737	BrCC(=O)NCCc1ccccc1	CID:9881279	phase I
BRD-A12409803	CNC(=O)c1ccc2cc(ccc2c1)C1(O)CCn2cncc12	CID:9883029	phase I
BRD-K67868012	Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1	CID:9884685	phase I
BRD-K40578143	OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N[C@H]3CCC[C@@H]3O)ncnc12	CID:9884817	phase I
BRD-K55454768	COc1ccc(cc1)C(=C2C(=O)Nc3ccccc23)c4ccc(OC)cc4	CID:9885087	phase I
BRD-K21672174	CS(=O)(=O)c1ccc(cc1)[C@@H](CC1CCCC1)C(=O)Nc1nccs1	CID:9886086	phase I
BRD-A15010982	CCCCCCC(C)(C)c1cc(O)c2[C@H]3CC(CO)=CCC3C(C)(C)Oc2c1	CID:9886498	phase I
BRD-K92470030	COc1cccc(c1)c2nc(SC)nc3sc(C(=O)NC(C)(C)C)c(N)c23	CID:9887381	phase I
BRD-K89274813	Fc1cc(CC2(Cc3ccnc(F)c3)c3ccccc3C(=O)c3ccccc23)ccn1	CID:9887884	phase I
BRD-K85015012	COc1ccccc1C1(O)CCN(CCCn2c3ccccc3c3ccccc23)CC1	CID:9888030	phase I
BRD-K70511574	COc1ccc(cc1)S(=O)(=O)N(C(C)=O)c1ccccc1\C=C\c1cc[n+]([O-])cc1	CID:9888590	phase I
BRD-K05181084	Clc1cccc(N2CCN(CCCCNC(=O)c3ccc-4c(Cc5ccccc-45)c3)CC2)c1Cl	CID:9891901	phase I
BRD-K88759641	CCCCc1nc2ccn(CC(=O)N(C)C)c(=O)c2n1Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1	CID:9892554	phase I
BRD-K88186167	CC(C)c1onc(c1COc1ccc(\C=C\c2cccc(c2)C(O)=O)c(Cl)c1)-c1c(Cl)cccc1Cl	CID:9893571	phase I
BRD-A43930669	Cc1ccccc1N1CCN(CC1)S(=O)(=O)CC12CCC(C[C@@H]1NC(=O)[C@@H](N)CCS(C)(=O)=O)C2(C)C	CID:9893887	phase I
BRD-K08438429	Clc1ccc(CN(CCCNC(=S)NCCCc2c[nH]cn2)c3ccc(Br)cn3)cc1Cl	CID:9893924	phase I
BRD-K67075780	Cc1ccccc1Oc2cccc3c(=O)cc([nH]c23)N4CCOCC4	CID:9902311	phase I
BRD-A26787626	CC(=O)C1C(=O)C2C3C(Cc4cccc5[nH]cc3c45)C(C)(C)N2C1=O	CID:9902313	phase I
BRD-K54704028	C=C1C[C@@H]2COC(=O)[C@]2(Cc3ccc4ccccc4c3)C1	CID:9903757	phase I
BRD-K51575138	NC(=O)Nc1sc(cc1C(N)=O)-c1ccc(F)cc1	CID:9903786	phase I
BRD-K13927029	CC(=C\CO)\C=C\C=C(C)\C=C\C1=C(C)CCCC1(C)C	CID:9904001	phase I
BRD-K10870738	Oc1ccc(/C=C(/C#N)\C(=O)OC\C=C\c2ccccc2)cc1O	CID:9905190	phase I
BRD-K92033419	COc1c(O)cccc1[C@H](O)C2CCN(CCc3ccc(F)cc3)CC2	CID:9906851	phase I
BRD-A30655177	CC(=O)C(C#N)C(=O)Nc1cc(Br)ccc1Br	CID:9906875	phase I
BRD-A41692738	CC(Nc1ccccc1)c1cc(C)cn2c1nc(cc2=O)N1CCOCC1	CID:9907093	phase I
BRD-K75430629	Cc1ccccc1n2c(Cn3cnc4c(N)ncnc34)nc5cccc(C)c5c2=O	CID:9908783	phase I
BRD-K86600316	CCS(=O)(=O)N1CCC[C@@H]2CN3CCc4cc(OC)ccc4[C@@H]3C[C@H]12	CID:9908992	phase I
BRD-A95096829	Fc1ccc(cc1)N2CCN(CCC3OCCc4ccccc34)CC2	CID:9909648	phase I
BRD-K31553034	COc1nc(C)cnc1NS(=O)(=O)c1cccnc1-c1ccc(cc1)-c1nnco1	CID:9910224	phase I
BRD-K10705233	COc1ccc2n(C(=O)c3cccc(Cl)c3Cl)c(C)c(CCN3CCOCC3)c2c1	CID:9911463	phase I
BRD-K53414658	COc1cc2nccc(Oc3ccc(NC(=O)Nc4cc(C)on4)c(Cl)c3)c2cc1OC	CID:9911830	phase I
BRD-K72703948	COc1cc2c(Nc3ccc(NC(=O)c4ccccc4)cc3)ncnc2cc1OCCCN1CCOCC1	CID:9914412	phase I
BRD-K85606544	CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C	CID:9915743	phase I
BRD-K26619122	COc1c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)cc2CC[C@H](NC(C)=O)c3cc(=O)c(SC)ccc3-c2c1OC	CID:9915886	phase I
BRD-A75478957	CC(C)C(NS(=O)(=O)c1ccc(cc1)c2ccc(Br)cc2)C(=O)O	CID:9918908	phase I
BRD-K31283835	C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N	CID:9926791	phase I
BRD-K87696786	COc1ccc(Nc2ncnc3ccc(OC)cc23)cc1	CID:9926999	phase I
BRD-K04623885	C\C(=C/C(=O)Nc1ccccc1C(O)=O)c1ccc2ccccc2c1	CID:9927531	phase I
BRD-A22844106	CN1C(C(=O)Nc2ccccn2)C(=O)c2sccc2S1(=O)=O	CID:9927768	phase I
BRD-K57391913	CC(C)N(CCCCOCC(O)=O)c1cnc(-c2ccccc2)c(n1)-c1ccccc1	CID:9931891	phase I
BRD-K88560311	CNCc1ccc(cc1)-c1[nH]c2cc(F)cc3C(=O)NCCc1c23	CID:9931954	phase I
BRD-K86930074	COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1	CID:9933475	phase I
BRD-K82983861	Cc1nc(sc1CSc1ccc(OCC(O)=O)c(C)c1)-c1ccc(c(F)c1)C(F)(F)F	CID:9934458	phase I
BRD-K63195589	Cn1cncc1[C@](N)(c1ccc(Cl)cc1)c1ccc2n(C)c(=O)cc(-c3cccc(Cl)c3)c2c1	CID:9935249	phase I
BRD-K04546108	O=C/1Nc2ccc(cc2\C1=C\c3ccc[nH]3)c4cccnc4	CID:9947841	phase I
BRD-K93023739	Clc1cc(NC(=O)c2cccnc2)c2[nH]c3cnccc3c2c1	CID:9949093	phase I
BRD-K99498722	CC(C)(C)c1[nH]cnc1\C=c1/[nH]c(=O)\c(=C\c2ccccc2)[nH]c1=O	CID:9949641	phase I
BRD-K22878149	CN1CC[C@@]2(Cc3nc4ccccc4cc3C[C@H]2C1)c1cccc(O)c1	CID:9950038	phase I
BRD-K12683773	Cc1cncc2cccc(c12)S(=O)(=O)N3CCCNCC3	CID:9951687	phase I
BRD-K74865981	CNc1cc(OC)c(cc1Cl)C(=O)N[C@H]1CCN(Cc2ccccc2)[C@H]1C	CID:9952220	phase I
BRD-K52751261	CCc1nc(c(s1)-c1ccnc(NC(=O)c2ccccc2)c1)-c1cccc(C)c1	CID:9952773	phase I
BRD-A47342814	Oc1ccc2CC3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)c1[nH]c2ccccc2c1C[C@@]35O	CID:9953592	phase I
BRD-K52394958	COC1(C[S@@](=O)c2ccccc2)CCN(CCc2c[nH]c3ccc(F)cc23)CC1	CID:9953599	phase I
BRD-K87510569	Cc1oc(nc1CCN1CCC2(CC1)OC(=O)Nc1ccc(C)cc21)-c1ccccc1	CID:9953769	phase I
BRD-K54708045	OC(=O)c1n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc2c1Sc1ccccc1	CID:9954280	phase I
BRD-K16189898	Cc1c[nH]c(n1)-c1cnc(NCCNc2ccc(cn2)C#N)nc1-c1ccc(Cl)cc1Cl	CID:9956119	phase I
BRD-K16263608	CC(C)C[C@H](NC(=O)c1ccc(NC[C@@H](N)CS)cc1-c1cccc2ccccc12)C(O)=O	CID:9956145	phase I
BRD-K48488978	Nc1ccc(cn1)C(=O)Nc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1	CID:9956222	phase I
BRD-K88677950	Cc1cc(I)ccc1Nc1c(F)c(F)c(F)cc1C(=O)NOCC1CC1	CID:9956637	phase I
BRD-K78122587	CC(C)[C@H]1c2ccc(F)cc2CC[C@@]1(CCN(C)CCCc1nc2ccccc2[nH]1)OC(=O)C1CC1	CID:9957280	phase I
BRD-K39733634	CCCCc1nn(-c2ccccc2C(F)(F)F)c(=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)c1sccc1C	CID:9961192	phase I
BRD-K37720887	Cc1cccc(n1)-c1[nH]c(nc1-c1ccc2nccnc2c1)C(C)(C)C	CID:9967941	phase I
BRD-A94413429	[O-][N+](=O)c1ccccc1S(=O)(=O)NCC2CCC(CNCC3CCc4ccccc4C3)CC2	CID:9982218	phase I
BRD-K49519092	C(c1cnc[nH]1)c1ccncc1	CID:9989505	phase I
BRD-A84423900	CSc1ccc(cc1)C2CN3CCCC3c4ccccc24	CID:9994677	phase I
BRD-K83063356	FC(F)(F)c1ccc(CCN2CCC3(CC2)OC(=O)Nc2ccccc32)cc1	CID:10000456	phase I
BRD-A14969012	Cc1cccc(c1)C2CN(CC=C)CCc3c(Cl)c(O)c(O)cc23	CID:10020353	phase I
BRD-K84987553	OB(O)c1ccc(cc1)C(=O)/C=C/c2ccc(I)cc2	CID:10022508	phase I
BRD-A13964793	OC12C3C4C5C3C(C3C5CC4C13)N2CCc1cccc(F)c1	CID:10040286	phase I
BRD-K92326486	NCCc1cccc2ccc(O)cc12	CID:10058277	phase I
BRD-K64729807	CC(=CCC/C(=C/CSC[C@H](NC(=O)C)C(=O)O)/C)C	CID:10063341	phase I
BRD-K51941867	COC(=O)c1cc2cc(ccc2n1Cc1ccc(Cl)cc1)S(C)(=O)=O	CID:10068193	phase I
BRD-A39255369	CCCCC1(Cc2cc(OCCCC(O)=O)c(Cl)c(Cl)c2C1=O)C1CCCC1	CID:10071166	phase I
BRD-K71035033	CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1	CID:10074640	phase I
BRD-K47983010	Ic1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCCNC(=O)c1cccs1	CID:10077147	phase I
BRD-K68584490	CCC[C@@H]1OC(=O)C(=C)[C@H]1C(O)=O	CID:10081070	phase I
BRD-A53131506	C[C@]12CCC3C(CCC4=CC(=O)CC[C@]34C)C1CC[C@H]2O	CID:10108190	phase I
BRD-K26979635	OC(=O)c1ccc(Cl)cc1NC(=O)Nc2cccc(c2)C(F)(F)F	CID:10109069	phase I
BRD-A60245366	N#CC(c1nc2ccccc2s1)c1ccnc(NCCc2cccnc2)n1	CID:10109823	phase I
BRD-K74514084	CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1	CID:10113978	phase I
BRD-K66707493	O=C1CC(=O)c2ccccc2C1=O	CID:10125107	phase I
BRD-K24681473	COCC[n+]1c(C)n(Cc2cnccn2)c2c1C(=O)c1ccccc1C2=O	CID:10126189	phase I
BRD-K57080016	Cn1cnc2c(F)c(Nc3ccc(Br)cc3Cl)c(cc12)C(=O)NOCCO	CID:10127622	phase I
BRD-K47659338	Cc1[nH]c2ccc(Cl)cc2c1C1=CCNCC1	CID:10131112	phase I
BRD-K56622826	CN(C)c1ccc(cc1)-c1cn2cc(I)ccc2n1	CID:10133297	phase I
BRD-K35307346	CC(C)[C@H](O)CC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:10135759	phase I
BRD-K38615104	Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2c[nH]c3ccccc23)c1	CID:10172943	phase I
BRD-K49810818	CNC(=O)c1cccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)c1	CID:10173949	phase I
BRD-K66175015	CN(C)C\C=C\C(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1O[C@H]1CCOC1	CID:10184653	phase I
BRD-K53281329	COc1ccc(cc1OC)-c1cc2nccn2c(Nc2ncccc2C(N)=O)n1	CID:10200390	phase I
BRD-A50454580	OCC(O)CONC(=O)c1ccc(F)c(F)c1Nc1ccc(I)cc1F	CID:10206158	phase I
BRD-K43330982	CC(C)c1cc(NNC(=O)Nc2cc(Cl)nc(Cl)c2)nc2n(C)nc(C)c12	CID:10223146	phase I
BRD-K65285700	Cc1ccc-2c(Cc3c(nn(c-23)-c2ccc(Cl)cc2Cl)C(=O)NN2CCCCC2)c1	CID:10252734	phase I
BRD-K76108747	CN(C)Cc1ccccc1Sc1ccc(F)cc1N	CID:10265481	phase I
BRD-K49371609	CN(\N=C\c1cnc2ccc(Br)cn12)S(=O)(=O)c1cc(ccc1C)[N+]([O-])=O	CID:10275789	phase I
BRD-A84174393	CN1C(C(=O)Nc2ncc(C)s2)C(=O)c2ccccc2S1(=O)=O	CID:10291556	phase I
BRD-K19540840	CN1CCN(CCOc2cc(OC3CCOCC3)c3c(Nc4c5OCOc5ccc4Cl)ncnc3c2)CC1	CID:10302451	phase I
BRD-K43234716	CCCCCCCCCCCCCCCc1cccc(OCC)c1C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F	CID:10311918	phase I
BRD-K64642496	COc1ccc2c3C[C@@H]4N([C@@H](CC(C)C)c3[nH]c2c1)C(=O)[C@H](CCC(=O)OC(C)(C)C)NC4=O	CID:10322450	phase I
BRD-K62206109	C(CC1CCNCC1)Cc2c[nH]cn2	CID:10330240	phase I
BRD-K13528168	CNCCCN1c2ccccc2Sc2ccc(cc12)C(F)(F)F	CID:10337209	phase I
BRD-K07736136	NC(=O)N(c1ccc(C(N)=O)c(n1)-c1ccc(F)cc1F)c1c(F)cccc1F	CID:10341154	phase I
BRD-K24307074	Nc1cccc(OCC2=NCCN2)c1	CID:10352540	phase I
BRD-K82206012	C[C@]12CC[C@H]3[C@@H](C[C@H](F)C4=CC(=O)CC[C@]34C)[C@@H]1CC[C@@H]2O	CID:10357822	phase I
BRD-A25569250	CC(OC(=O)Nc1c(C)noc1-c1ccc(CSCCC(O)=O)cc1)c1ccccc1Cl	CID:10367662	phase I
BRD-K57011718	C[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCCc1ccc(c(C)c1)-c1ccccc1)CC(=O)NO)C(C)(C)C)c1ccccc1	CID:10370504	phase I
BRD-K41895714	O=C1NC(=O)\C(S1)=C/c1ccc2nccnc2c1	CID:10377751	phase I
BRD-K74733595	Cn1cc(cc1\C=C\C(=O)NO)C(=O)Cc1ccccc1	CID:10379137	phase I
BRD-K19894101	Oc1cccc(C(=O)Nc2cccc(NC(=O)c3cccc(O)c3O)c2)c1O	CID:10385095	phase I
BRD-A87125127	Cc1cc(sc1C(N)C(=O)O)C(=O)O	CID:10398360	phase I
BRD-K84943004	Cc1ccc(cc1)C(=O)c1cc(\C=C\C(=O)NO)n(C)c1	CID:10401611	phase I
BRD-K26669427	Fc1ccc(cc1)C(=O)/C=C/2\C(=O)Nc3ccc(Br)cc23	CID:10405323	phase I
BRD-A15493168	CC1[C@H]2C[C@H]3[C@H](N(C)C)C(=O)C(C(N)=O)C(=O)[C@@]3(O)C(=O)C2C(=O)c2c(O)cccc12	CID:10410310	phase I
BRD-K06593056	CN1c2cc3c(cc2N=C(c2ccc(cc2)C(O)=O)c2ccccc12)C(C)(C)CCC3(C)C	CID:10410894	phase I
BRD-K07888107	C[C@@H](O)[C@H]1O[C@H]1\C=C\[C@H]1O[C@H]1[C@H](O)C=C	CID:10420710	phase I
BRD-K64785675	Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1	CID:10427712	phase I
BRD-A61858259	CCc1ccc(nc1)C(=O)COc1ccc(CC2SC(=O)NC2=O)cc1	CID:10429242	phase I
BRD-K15086322	CN1CCN(CC1)C(=O)c1nc2ccc(Cl)cc2[nH]1	CID:10446295	phase I
BRD-K99257182	COc1ccc2nccc([C@H](O)[C@@H]3C[C@@H]4CCN3C[C@@H]4C=C)c2c1	CID:10448938	phase I
BRD-K60932973	Oc1cc2[C@H](CN(CC=C)CCc2c(Br)c1O)c3ccccc3	CID:10452020	phase I
BRD-K95435023	Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1	CID:10461815	phase I
BRD-K95609758	Oc1ccc(Cl)cc1Cn1nc(oc1=O)-c1ccc(cc1)C(F)(F)F	CID:10474339	phase I
BRD-K18799075	FC(F)(F)CCCS(=O)(=O)Oc1cccc(Oc2cccc(c2C#N)C(F)(F)F)c1	CID:10479060	phase I
BRD-K95138506	Oc1ccc(CCc2ccccc2)c2cccnc12	CID:10490845	phase I
BRD-K70792160	CCN(CC)CCCCN1c2ccccc2Oc2ccc(Cl)cc12	CID:10521421	phase I
BRD-K81633055	CCOC(=O)C1=CN(Cc2ccccc2)C=C(C1c1ccccc1)C(=O)OCC	CID:10620479	phase I
BRD-K46469693	COc1ccc(CCCn2ncc3c4nc(nn4c(N)nc23)c5ccco5)cc1	CID:10668061	phase I
BRD-K15588452	COc1cccc(CCc2ccccc2OCC[C@@H]2C[C@@H](O)CN2C)c1	CID:10668211	phase I
BRD-K86191271	CCCCCCCC(=O)c1c(O)cc(O)cc1CC(=O)OCC	CID:10687292	phase I
BRD-K16297709	C[C@@H]1C[C@H](O[C@@H]2O[C@@H](C)[C@H](O[C@@H]3O[C@H](COC(=O)C)[C@@H](O)[C@H](O)[C@H]3O)[C@@H](O)[C@H]2O)[C@]4(C)[C@H](CCC=C4C)[C@@]1(C)CC[C@](C)(O[C@@H]5O[C@H](C)[C@H](O[C@@H]6O[C@@H](C)[C@H](O)[C@@H](O)[C@H]6O)[C@H](O)[C@H]5O)C=C	CID:10724564	phase I
BRD-A22143024	C[C@]12CCC3C(CCc4cc(OS(O)(=O)=O)ccc34)C1CCC2=O	CID:10861069	phase I
BRD-K08227907	NCCc1cc(O)c(O)cc1[N+]([O-])=O	CID:10932412	phase I
BRD-K19277754	CN1CC[C@H]([C@H](COc2ccc3OCOc3c2)C1)c1ccc(F)cc1	CID:10947895	phase I
BRD-A83081521	CC(C)(C)NC(=O)[C@H]1CCC2C3CCC4NC(=O)C=C[C@]4(C)C3CC[C@]12C	CID:10970751	phase I
BRD-K68873215	CCCCN1C(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@@H](N2C1=O)c5ccc(OC)cc5	CID:11003969	phase I
BRD-K34079378	COc1cc2[nH]c3ccccc3c2cc1C	CID:11052947	phase I
BRD-K26300881	COc1ccc(cc1)-n1sc2ccccc2c1=O	CID:11054313	phase I
BRD-A65076780	CC(C)[C@@]1(NC(=O)[C@@H]2CC3[C@@H](Cc4c[nH]c5cccc3c45)N(C)C2)O[C@@]6(O)[C@@H]7CCCN7C(=O)[C@H](Cc8ccccc8)N6C1=O	CID:11072143	phase I
BRD-K12040459	Clc1ccc(cc1)C1(CCNCC1)c1ccc(cc1)-c1cn[nH]c1	CID:11175137	phase I
BRD-K76568384	Oc1ccc(cc1)-c1c(nn2c(cc(nc12)C(F)(F)F)C(F)(F)F)-c1ccccc1	CID:11201035	phase I
BRD-K64402243	CC(=O)OCCN1C(=O)c2c(C1=O)c3cc(ccc3nc2C)S(=O)(=O)N4CCOCC4	CID:11201705	phase I
BRD-K49119234	CCCCCCC(=O)OC1CC(C)(C)NC(C)(C)C1	CID:11207937	phase I
BRD-K42624714	COc1cccc(c1)c2cc(NCc3ccc4OCOc4c3)nc(N)n2	CID:11210285	phase I
BRD-K20285085	COc1cc(Nc2ncc(F)c(Nc3ccc4OC(C)(C)C(=O)Nc4n3)n2)cc(OC)c1OC	CID:11213558	phase I
BRD-A25004090	CCOc1ccccc1-n1c(=O)c2ccccc2nc1C(C)N1CCN(CC1)C(=O)COc1ccc(Cl)cc1	CID:11214940	phase I
BRD-K52800308	Clc1ccc(cc1)-n1sc2ccccc2c1=O	CID:11219195	phase I
BRD-K94830329	OC(=O)c1cccc(c1)-c1noc(n1)-c1ccccc1F	CID:11219835	phase I
BRD-K56301217	CN(C)CC[C@H](CSc1ccccc1)Nc1ccc(cc1[N+]([O-])=O)S(=O)(=O)NC(=O)c1ccc(cc1)N1CCN(Cc2ccccc2-c2ccc(Cl)cc2)CC1	CID:11228183	phase I
BRD-K28428262	C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C	CID:11234052	phase I
BRD-K73261812	Oc1ccc(C[C@@H]2N3[C@H](CN(Cc4cccc5ccccc45)C2=O)N(CCC3=O)C(=O)NCc2ccccc2)cc1	CID:11238147	phase I
BRD-K02950022	C[C@@H](N(c1cc(F)ccc1F)S(=O)(=O)c1ccc(Cl)cc1)c1ccc(F)cc1CCCC(O)=O	CID:11249248	phase I
BRD-K66538826	S=C(NCc1ccc2OCOc2c1)N1CCN(CC1)c1ncnc2c3ccccc3oc12	CID:11282283	phase I
BRD-K73395020	CC(C)ON([C@H](C(C)C)C(=O)NO)S(=O)(=O)c1ccc(cc1)c2ccccc2	CID:11292680	phase I
BRD-K33272502	Cc1cn(Cc2ccc(Cl)cc2Cl)c2c(\C=C\C(=O)NS(=O)(=O)c3cc(Cl)c(Cl)s3)cc(F)cc12	CID:11296282	phase I
BRD-K83794624	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@H](O[C@@H]6CCCCO6)[C@H](C)O5)c4c(O)c3C(=O)c12)C(=O)CO	CID:11296583	phase I
BRD-K64670467	COC1CCC(CC1)C(=O)c2ccc3nc4OCCCc4cc3c2	CID:11313361	phase I
BRD-K47150025	COc1cc2nccc(Oc3ccc(NC(=O)Nc4ccc(F)cc4F)c(F)c3)c2cc1OC	CID:11317348	phase I
BRD-K00337317	O=c1cc(oc2c(cccc12)-c1cccc2c3ccccc3sc12)N1CCOCC1	CID:11327430	phase I
BRD-K13390322	Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1	CID:11338033	phase I
BRD-K99174507	COc1ccc(Nc2nccc(NCCO)n2)cc1	CID:11345983	phase I
BRD-K23363278	CCC[C@H](Nc1nc(ncc1C)-c1ccc(NC(=O)NCC)c(OC)c1)c1cccnc1	CID:11351021	phase I
BRD-K64890080	CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	CID:11364421	phase I
BRD-A10523515	CC1=C(C(CC(=O)N1)c1ccc(cc1)C(F)(F)F)C(=O)Nc1cc2cn[nH]c2cc1F	CID:11373846	phase I
BRD-K54095730	Oc1ccc(NC(=O)CCCc2ccc(cc2)-c2ccccc2F)cc1	CID:11382492	phase I
BRD-K52522949	CC(C)C(=O)SCCCCCCC(=O)Nc1nc(cs1)-c1ccccc1	CID:11395181	phase I
BRD-A37052580	CNC(=O)Oc1ccc2N(C)C3N(C)CC[C@@]3(C)c2c1	CID:11403114	phase I
BRD-K07881437	CO[C@@H](C(=O)N1Cc2[nH]nc(NC(=O)c3ccc(cc3)N3CCN(C)CC3)c2C1)c1ccccc1	CID:11442891	phase I
BRD-A21584801	CC(O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C	CID:11451527	phase I
BRD-K28360340	CC(C)c1ccccc1Cc1cc(C(=O)Nc2ccc(cc2)S(=O)(=O)c2ccccc2C(C)(C)C)c(O)c(O)c1O	CID:11455910	phase I
BRD-K99749624	Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1	CID:11485656	phase I
BRD-A35153197	OC(=O)[C@@H]1CSC(Cc2c[nH]c3ccc(O)cc23)N1	CID:11492836	phase I
BRD-K68756823	Nc1[nH]nc2nnc(cc12)-c1c(nn2ccccc12)-c1ccccc1	CID:11493598	phase I
BRD-K33379087	O=C1NC(=O)[C@H]([C@@H]1c1c[nH]c2ccccc12)c1cn2CCCc3cccc1c23	CID:11494412	phase I
BRD-K69837166	CCn1c2ccccc2n(C2=C(CO)CN(CC3CCCCCCC3)CC2)c1=O	CID:11494970	phase I
BRD-K37865504	CN(C)C(=O)n1nnnc1Cc1ccc(cc1)-c1ccccc1	CID:11507802	phase I
BRD-K54233340	C(CN1CCCCC1)Oc2ccc(cc2)c3cnc4c(cnn4c3)c5ccncc5	CID:11524144	phase I
BRD-K83837640	Cn1cc(CNCC2CCN(CC2)c2ncc(cn2)C(=O)NO)c2ccccc12	CID:11538455	phase I
BRD-K75181824	CC(=CCC/C(=C/CC/C(=C/CC/C(=C/CSC[C@H](NC(=O)C)C(=O)O)/C)/C)/C)C	CID:11575713	phase I
BRD-K71534238	OC(=O)CCc1ccc(NCc2cccc(Oc3ccccc3)c2)cc1	CID:11595431	phase I
BRD-K93788137	CN(c1ccccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)ncc1C(F)(F)F)S(C)(=O)=O	CID:11598628	phase I
BRD-K60866521	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(F)c2c(=O)n1-c1ccccc1	CID:11625818	phase I
BRD-K78431006	C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl	CID:11626560	phase I
BRD-K51781482	COc1cc2ncn(-c3cc(OCc4ccccc4S(C)(=O)=O)c(s3)C#N)c2cc1OC	CID:11626927	phase I
BRD-K95739795	COc1cc2CCN3C[C@H](CC(C)C)C(=O)C[C@H]3c2cc1OC	CID:11634155	phase I
BRD-K93725829	Cc1cnc(Nc2ccc(F)cc2Cl)nc1-c1c[nH]c(c1)C(=O)N[C@H](CO)c1cccc(Cl)c1	CID:11634725	phase I
BRD-K42500029	Nc1ncnc2[nH]nc(Nc3ccc(F)cc3)c12	CID:11644425	phase I
BRD-K63068307	FC(F)c1nc2ccccc2n1-c1nc(nc(n1)N1CCOCC1)N1CCOCC1	CID:11647372	phase I
BRD-K74325648	C[C@H](CN(C(=O)C1CCCCC1)c1ccccn1)N1CCN(CC1)c1cccc2[nH]ccc12	CID:11647989	phase I
BRD-K99616396	CC1(C)CNc2cc(NC(=O)c3cccnc3NCc3ccncc3)ccc12	CID:11667893	phase I
BRD-A45499626	NC(Cn1ccc(=O)n(Cc2ccccc2C(O)=O)c1=O)C(O)=O	CID:11674376	phase I
BRD-K05804044	Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ccc2ncn(C)c(=O)c2c1	CID:11676786	phase I
BRD-K35723520	C[As](C)SC[C@H](NC(=O)CC[C@H](N)C(O)=O)C(=O)NCC(O)=O	CID:11683005	phase I
BRD-K56403959	OCCOCCN1CCN(Cc2cccc(Oc3ccccc3)c2)CC1	CID:11688990	phase I
BRD-A70407468	CCCCn1c(=O)n(CCCO)c2nc([nH]c2c1=O)C12CC3CC1CC(C2)C3	CID:11689583	phase I
BRD-K12343256	CC(=O)Nc1cccc(c1)-n1c2c(C)c(=O)n(C)c(Nc3ccc(I)cc3F)c2c(=O)n(C2CC2)c1=O	CID:11707110	phase I
BRD-K83963101	OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1	CID:11712649	phase I
BRD-K99545815	CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)ncc1C(F)(F)F)S(C)(=O)=O	CID:11713159	phase I
BRD-K48059230	Cc1c(sc2nc3ccc(N)cc3n12)C(=O)NC1CCCCC1	CID:11716890	phase I
BRD-K67578145	OCCn1cc(c(n1)-c1ccncc1)-c1ccc2c(CC\C2=N/O)c1	CID:11717001	phase I
BRD-K10466330	CC1(C)Oc2ccc3C4=C[C@@]56NC(=O)[C@]7(CCCN7C5=O)C[C@H]6C(C)(C)C4=[N+]([O-])c3c2C=C1	CID:11719255	phase I
BRD-K12867552	CN(C)Cc1c(oc2ccccc12)C(=O)NCCOc1ccc(cc1)C(=O)NO	CID:11749858	phase I
BRD-K49669041	Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1c[nH]cn1	CID:11754511	phase I
BRD-K94832621	CC(C)N1CCN(CC1)c1ccc(cc1)C(=O)c1c(sc2cc(O)ccc12)-c1ccc(O)cc1	CID:11784736	phase I
BRD-K39111395	COc1ccc([N+][O-])c(CCc2cc(OC)ccc2[N+][O-])c1	CID:11822705	phase I
BRD-K50199947	COc1ccc(N(C(=O)Oc2c(C)cccc2C)c2ccnc(Nc3ccc(cc3)N3CCN(C)CC3)n2)c(OC)c1	CID:11844351	phase I
BRD-K25079130	CC1(C)CC(C)(C)C2=[N+]([O-])c3cc4OC(C)(C)C=Cc4cc3C2=C1	CID:11852606	phase I
BRD-K59720958	CC(C)(C)NC(=O)[C@H]1CC[C@H]2[C@H]3CC[C@H]4NC(=O)C=C[C@]4(C)[C@@H]3CC[C@]12C	CID:11865433	phase I
BRD-K80115247	C[C@]12CC[C@@H]3[C@@H](CC[C@H]4C[C@@H](O)CC[C@]34C)[C@H]1CCC2=O	CID:11868648	phase I
BRD-K39168746	C[C@]12CC[C@@H]3[C@@H](CC[C@H]4C[C@H](O)CC[C@]34C)[C@H]1CCC2=O	CID:11868768	phase I
BRD-K67919934	CC(=O)S[C@@H]1CC2=CC(=O)CC[C@]2(C)[C@@H]2CC[C@@]3(C)[C@H](CC[C@@]33CCC(=O)O3)[C@H]12	CID:11869580	phase I
BRD-K23714869	C[C@]12C[C@H](O)[C@@]3(F)[C@H](CCC4=CC(=O)C=C[C@]34C)[C@@H]1C[C@@H](O)[C@]2(O)C(=O)CO	CID:11870426	phase I
BRD-K60132694	CC(=O)O[C@@]1(CC[C@@H]2[C@H]3C=C(C)C4=CC(=O)CC[C@]4(C)[C@@H]3CC[C@]12C)C(C)=O	CID:11872394	phase I
BRD-K11439261	CC(=O)[C@H]1CC[C@@H]2[C@@H]3C=CC4=CC(=O)CC[C@@]4(C)[C@@H]3CC[C@]12C	CID:11875278	phase I
BRD-K60507178	COc1cc(cc(OC)c1OC)[C@H]1[C@@H]2[C@@H](COC2=O)[C@@H](O)c2cc3OCOc3cc12	CID:11892032	phase I
BRD-K44495371	CO[C@H]1[C@@H](C[C@@H]2CN3CCc4c([nH]c5cc(OC)ccc45)[C@@H]3C[C@H]2[C@@H]1C(=O)OC)OC(=O)c1cc(OC)c(OC)c(OC)c1	CID:11908593	phase I
BRD-K41431477	CNc1ccc2oc(C[C@H]3O[C@@]4(CC[C@H]3C)O[C@H]([C@H](C)C(=O)c5ccc[nH]5)[C@H](C)C[C@H]4C)nc2c1C(=O)O	CID:11957499	phase I
BRD-A48809242	CNC(=O)[C@H]1O[C@H](C(O)[C@H]1O)n2cnc3c(NCc4cccc(I)c4)ncnc23	CID:11957586	phase I
BRD-K88871508	CCN(CC)C(=O)N[C@H]1CN(C)[C@@H]2Cc3c[nH]c4cccc(C2=C1)c34	CID:11957615	phase I
BRD-K05901394	CCN(CC)C(=O)N[C@@H]1C[C@H]2[C@@H](Cc3c[nH]c4cccc2c34)N(C)C1	CID:11957722	phase I
BRD-A50364343	CC1(CCCN1)c1nc2c(cccc2[nH]1)C(N)=O	CID:11960528	phase I
BRD-K87142802	C[C@@]1(CCCN1)c1nc2c(cccc2[nH]1)C(N)=O	CID:11960529	phase I
BRD-K09499853	CCN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1	CID:11964036	phase I
BRD-K63265447	CC(=O)O[C@]12CO[C@@H]2C[C@H](O)[C@]3(C)[C@@H]1[C@H](OC(=O)c4ccccc4)[C@@]5(O)C[C@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c6ccccc6)C(=C([C@@H](O)C3=O)C5(C)C)C	CID:11970251	phase I
BRD-K12184916	Cn1c2cnc3ccc(cc3c2n(-c2ccc(cc2)C(C)(C)C#N)c1=O)-c1cnc2ccccc2c1	CID:11977753	phase I
BRD-A18411371	COc1ccc(cc1)C(N(C(=O)CCl)c2cccc(Cl)c2)C(=O)NC3CCCCC3	CID:12004949	phase I
BRD-A18725729	COc1ccc(cc1)C(N(C(=O)CCl)c2ccc(Cl)cc2)C(=O)NC3CCCCC3	CID:12004950	phase I
BRD-K88198340	COC1(OC)C=CC(=O)C=C1NC(=O)c2ccccc2OC(=O)C	CID:12043281	phase I
BRD-K61033289	CCCCC\C=C\C=C1/[C@@H](C\C=C\CCCC(O)=O)C=CC1=O	CID:12068863	phase I
BRD-K71970656	CN(C)S(=O)(=O)c1ccc2CCc3ccc(cc3C(=O)c2c1)S(=O)(=O)N(C)C	CID:12135546	phase I
BRD-K25150581	COc1ccc2nc(sc2c1)c3ccc(F)cc3	CID:12179987	phase I
BRD-A35769934	C\C1=C/CC\C(CO)=C\[C@H]2OC(=O)C(=C)[C@@H]2[C@H](C1)OC(=O)C(=C)C(O)CO	CID:12303703	phase I
BRD-K91966436	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@@H](O[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O	CID:12309103	phase I
BRD-A51393488	COc1ccc2[C@H](OC(=O)c2c1OC)C1N(C)CCc2cc3OCOc3c(OC)c12	CID:12310313	phase I
BRD-K75971499	OCCN1CCN(CCCN2c3cc(Cl)ccc3Sc3cc(O)c(O)cc23)CC1	CID:12333107	phase I
BRD-K98336812	C[N+](C)(C)CCCN1c2ccc(O)cc2Sc2ccc(Cl)cc12	CID:12333113	phase I
BRD-K83161876	CCN1c2ccccc2Sc2ccc(Cl)cc12	CID:12351242	phase I
BRD-K25190777	O=c1n(oc2ccccc12)-c1ccccc1	CID:12385463	phase I
BRD-K73037408	NS(=O)(=O)c1ccc(NC2=CC(=O)c3ccccc3C2=O)cc1	CID:12387471	phase I
BRD-K12238169	Cn1c(N)c(C#N)c(c(C#N)c1=O)c2ccccc2	CID:12425537	phase I
BRD-K35858371	CS(=O)(=O)c1nc(cs1)-c1ccc(Br)cc1	CID:12474112	phase I
BRD-A14798026	COc1ccc2C3CC[C@@]4(C)C(CC[C@@]4(O)C#C)C3CCc2c1	CID:12598376	phase I
BRD-K23933163	Cc1onc(c1C(=O)N[C@H]1[C@@H]2SC(C)(C)[C@@H](N2C1=O)C(O)=O)-c1ccccc1Cl	CID:12625909	phase I
BRD-K53249762	COc1cc2c(CCN(C)C)c[nH]c2c(OC)c1OC	CID:12650292	phase I
BRD-K84421793	Oc1cc2[C@H](CNCCc2c(Cl)c1O)c3ccccc3	CID:12668019	phase I
BRD-K36269259	NCCc1cccc(O)c1O	CID:12707042	phase I
BRD-K76747609	CCC(=O)OCC(=O)[C@@]1(OC(=O)CC)[C@@H](C)C[C@H]2[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]12C	CID:12790158	phase I
BRD-A77144340	CC(C)CCCC(C)[C@H]1CC[C@H]2[C@H]3[C@H](CC[C@]12C)[C@@]1(C)CC[C@H](O)CC1=CC3=O	CID:12791166	phase I
BRD-K39397585	CCN1CCN(C(=O)N[C@@H](C(=O)N[C@H]2[C@@H]3SC(C)(C)[C@@H](N3C2=O)C(O)=O)c2ccccc2)C(=O)C1=O	CID:12799467	phase I
BRD-K42870217	C[C@@H](O)[C@H]1[C@H]2CC(SCCNC=N)=C(N2C1=O)C(O)=O	CID:12801781	phase I
BRD-K21815137	CN(C)CCn1nnnc1SCC1=C(N2[C@H](SC1)[C@@H](NC(=O)Cc1csc(N)n1)C2=O)C(O)=O	CID:12810432	phase I
BRD-K21955335	CC1(C)[C@H](CC[C@@]2(C)[C@H]1CC[C@]1(C)[C@@H]2C(=O)C=C2[C@H]3C[C@](C)(CC[C@]3(C)CC[C@@]12C)C(O)=O)OC(=O)CCC(O)=O	CID:12866477	phase I
BRD-K84252391	C[C@@H](N)Cc1cccc(c1)C(F)(F)F	CID:12895728	phase I
BRD-K37124285	Brc1ccc2CCc3ccccc3C(=O)c2c1	CID:12909391	phase I
BRD-A19500257	COC1CC(C)CC2=C(OC)C(=O)C=C(NC(=O)\C(C)=C\C=C\C(OC)C(OC(N)=O)\C(C)=C\C(C)C1O)C2=O	CID:13017911	phase I
BRD-K31616564	[O-][N+](=O)O[C@@H]1CO[C@H]2[C@H](CO[C@H]12)O[N+]([O-])=O	CID:13019152	phase I
BRD-K18674849	CC1(C)O[C@@H]2C[C@H]3[C@H]4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:13021033	phase I
BRD-A80869209	CC1(C)S[C@H]2[C@H](NC(=O)C(C(O)=O)c3ccsc3)C(=O)N2[C@H]1C(O)=O	CID:13025387	phase I
BRD-A47714657	COc1ccc2C(Cc3ccc(OC)c(O)c3)NCCc2c1	CID:13071436	phase I
BRD-K30682080	CCOc1ccc2ccccc2c1C(=O)N[C@H]1[C@@H]2SC(C)(C)[C@@H](N2C1=O)C(O)=O	CID:13121776	phase I
BRD-K24281017	Clc1cccc(c1)-n1sc2ccccc2c1=O	CID:13186954	phase I
BRD-K97514127	CCC1=C[C@H]2CN(C1)Cc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C)[C@@H]1[C@]22CCN3CC=C[C@](CC)([C@@H]23)[C@@H](OC(C)=O)[C@]1(O)C(=O)OC	CID:13200033	phase I
BRD-K09436313	CCCCC[C@H](O)\C=C\[C@H]1[C@H](C\C=C/CCCC(O)=O)[C@@H](O)CC1=O	CID:13292831	phase I
BRD-A80536908	C[C@H](NC(=O)CCC1CCC(=O)N1)c2ccccc2	CID:13564432	phase I
BRD-K79366068	Nc1c(cc(Nc2ccc(Cl)cc2)c3C(=O)c4ccccc4C(=O)c13)S(=O)(=O)O	CID:13782419	phase I
BRD-K65261396	CO[C@@H]1C[C@@H](CC[C@H]1O)\C=C(/C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@@]2(O)O[C@@H]([C@H](C[C@H]2C)OC)[C@H](C[C@@H](C)C\C(C)=C\[C@@H](CC=C)C(=O)C[C@H](O)[C@H]1C)OC	CID:13819073	phase I
BRD-A80386041	Cc1ccc(cc1)C1CC(=NN1c1ccc(cc1)S(N)(=O)=O)c1ccccc1	CID:13927310	phase I
BRD-A81402010	NS(=O)(=O)c1ccc(cc1)N1N=C(CC1c1ccc(Br)cc1)c1ccccc1	CID:13927312	phase I
BRD-A35825362	CN(C)CC(O)CN1c2ccccc2Sc2ccccc12	CID:13954252	phase I
BRD-K87166736	N[C@@H](CSc1cc(C[C@H](N)C(O)=O)cc(O)c1O)C(O)=O	CID:14178745	phase I
BRD-K84265381	OC(=O)CCc1c[nH]c2ccc(O)cc12	CID:14182642	phase I
BRD-A98888159	COc1cc(CC2COC(C2COC(=O)/C=C/c3ccc(O)cc3)c4ccc(O)c(OC)c4)ccc1O	CID:14205635	phase I
BRD-K77625572	OC(=O)[C@]1(CCCCCCOc2ccc(Cl)cc2)CO1	CID:14249524	phase I
BRD-A08658758	CC1CC(=O)NN=C1c1ccc(F)c(F)c1	CID:14459459	phase I
BRD-K15241725	COc1cc2CCN3C[C@@H](CC(C)C)[C@H](O)C[C@@H]3c2cc1OC	CID:14580381	phase I
BRD-A84280790	CN(CC#CCN1CCCC(CO)C1)C(=O)C	CID:14896501	phase I
BRD-A26333730	Oc1cc(O)c(CC2NC(=O)NC2=O)cc1O	CID:14951773	phase I
BRD-K91904471	NC(=O)c1ccc2[nH]ccc2c1	CID:14973220	phase I
BRD-K61260019	CC[N+](C)(C)CCOC(C)=O	CID:15029196	phase I
BRD-K23342641	CN1CCN(CC(=O)N2c3ccc(cc3C(=O)Nc4cccnc24)S(=O)(=O)NCCNC(=O)OC(C)(C)C)CC1	CID:15050929	phase I
BRD-A82323890	CCCN(CCc1ccc(N)cc1)C1CCc2c(O)cccc2C1	CID:15115512	phase I
BRD-K32043164	[O-][N+](=O)c1ccc2[nH]c(COCc3nc4ccccc4[nH]3)nc2c1	CID:15301607	phase I
BRD-K51073125	NCCCCNCCCN1c2ccccc2Sc2ccc(Cl)cc12	CID:15491403	phase I
BRD-K92241597	CC(C)C[C@H]([C@H](O)C(=O)NO)C(=O)N[C@H](C(=O)OC1CCCC1)c1ccccc1	CID:15547703	phase I
BRD-A99411506	OC[C@H]1OC(Oc2cc3ccc(=O)oc3cc2O)[C@H](O)[C@@H](O)[C@@H]1O	CID:15558439	phase I
BRD-A62200266	CCCCCCCCCCC1C(=O)OC(C(=O)O)C1(O)C(=O)O	CID:15560547	phase I
BRD-K51418664	CO[C@@]12[C@H]3N[C@H]3CN1C1=C([C@H]2COC(N)=O)C(=O)C(N)=C(C)C1=O	CID:15560563	phase I
BRD-A70814879	Clc1ccc(cc1)C12CC3CC(CC(C3)(C1)C(=O)NCc1ccncc1)C2	CID:15604015	phase I
BRD-K52453128	CN1c2ccccc2Sc2ccc(cc12)C(F)(F)F	CID:15692209	phase I
BRD-K99475920	COc1ccc(cc1NC(=O)c2cc3CCCCc3s2)S(=O)(=O)N4CCOCC4	CID:15945391	phase I
BRD-K12393722	Cc1onc(C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4)c1[N+](=O)[O-]	CID:15945539	phase I
BRD-K56851771	CNC(=O)c1ccc(cc1F)N1C(=S)N(C(=O)C1(C)C)c1ccc(C#N)c(c1)C(F)(F)F	CID:15951529	phase I
BRD-K92428232	C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F	CID:15983966	phase I
BRD-K63923597	CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1	CID:16007391	phase I
BRD-K30381304	CC(C)c1nnc(NC(=O)c2nc(ncc2Cl)S(=O)(=O)Cc3ccc(C)cc3)s1	CID:16014341	phase I
BRD-K09661167	CC(C)c1nnc(NC(=O)c2nc(ncc2Cl)S(=O)(=O)Cc3cccc(C)c3)s1	CID:16014494	phase I
BRD-K50140147	COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)N1CCN(C)CC1	CID:16038120	phase I
BRD-K68488863	CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(\C=C\c2ccccc2)n1	CID:16041424	phase I
BRD-A31195449	COc1cc(Br)c(OC)c2CC(CN)c21	CID:16046239	phase I
BRD-A87137733	CCn1c(nc2c(ncc(OCC3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N	CID:16048642	phase I
BRD-K09764130	CCCCCCCC/C=C\C/C=C\C/C=C\CCCC(=O)NCCO	CID:16061185	phase I
BRD-K34608650	Cc1ccc-2c(Cc3c(nn(c-23)-c2ccc(Cl)cc2Cl)C(=O)NC2CCCCC2)c1	CID:16094766	phase I
BRD-K02590140	CC1=CC[C@@H]2[C@@H](C1)c3c(O)cc(CC#CCCCNS(=O)(=O)C)cc3OC2(C)C	CID:16102146	phase I
BRD-K22631935	COc1ccc(cc1)-c1nc([nH]c1-c1ccc(OC)cc1)-c1ccc(o1)-c1cccc(Cl)c1	CID:16112820	phase I
BRD-K11187612	COc1cc2CC[C@H](NC(=O)C)c3cc(ccc3-c2c(OC)c1OC)C(=O)O	CID:16114799	phase I
BRD-A90451247	CC1CN(CC(=O)Nc2ccc3Sc4c(Cc3c2)cccc4-c2cc(=O)cc(o2)N2CCOCC2)CC(C)O1	CID:16117018	phase I
BRD-A35869383	Nc1ncnc2n(nc(-c3ccc(Oc4ccccc4)cc3)c12)C1CCCN(C1)C(=O)C=C	CID:16126651	phase I
BRD-K76698671	ONC(=O)CCCCCCSc1ccc2ccccc2c1	CID:16126782	phase I
BRD-A20697603	CCC(C)C1NC2C=Cc3c(cc(nc3C2O)C(=O)OC(C)C2NC(=O)c3csc(n3)C(NC(=O)C3CSC(=N3)\C(NC(=O)C(NC(=O)c3csc(n3)C3(CCC(=NC3c3csc2n3)c2nc(cs2)C(=O)NC(=C)C(=O)NC(=C)C(N)=O)NC(=O)C(C)NC(=O)C(=C)NC(=O)C(C)NC1=O)C(C)O)=C/C)C(C)(O)C(C)O)C(C)O	CID:16129666	phase I
BRD-K14681867	C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)[C@@H](C)O)C(O)=O)NC(=O)CNC(=O)[C@H](C)N	CID:16129706	phase I
BRD-A06641369	CC(C)Oc1cccc(c1)C(=O)C2CCCN(Cc3cnn(c3)C(C)C)C2	CID:16187238	phase I
BRD-A88878656	CC(C)Oc1cccc(c1)C(=O)C2CCCN(C2)C(=O)Cn3nc(C)cc3C	CID:16190091	phase I
BRD-A12083771	CCCn1ncc(CN2CCCC(C2)C(=O)c3cccc(OC(C)C)c3)c1C	CID:16190867	phase I
BRD-K36031023	CC(C)(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)O	CID:16195819	phase I
BRD-A65327625	CN1C2C[C@@H](O)C1CC(=O)C2	CID:16211224	phase I
BRD-K87555556	CCCCCc1oc2ccccc2c1C(=O)c1cc(I)c(OCCN(CC)CC)c(I)c1	CID:16218975	phase I
BRD-A52886023	CCCCCCC1[C@@H](OC(=O)CC(C)C)[C@H](C)OC(=O)[C@@H](NC(=O)c2cccc(NC=O)c2O)[C@@H](C)OC1=O	CID:16218979	phase I
BRD-A17448384	CC1CC2C3CCC4=CC(=O)C=CC4(C)[C@@]3(Cl)C(O)CC2(C)C1(O)C(=O)CO	CID:16218996	phase I
BRD-K98404142	C[C@@]12CC[C@H]3[C@@H](CC[C@H]4C[C@H](O)CC[C@@]43C)[C@@H]2C[C@H](Br)C1=O	CID:16219061	phase I
BRD-K04146668	Cn1cc(C=C2C(=O)Nc3cccnc23)c4ccccc14	CID:16219401	phase I
BRD-A24643465	COC1=C[C@@]23CCCN3CCc4cc5OCOc5cc4[C@]2(C)C1OC(=O)[C@@](O)(CCCC(C)(C)O)CC(=O)O	CID:16219462	phase I
BRD-A13122391	CC(C)[C@@]12O[C@H]2[C@@H]3O[C@]34[C@]5(O[C@H]5CC6C7=C(CC[C@@]64C)C(=O)OC7)[C@@H]1O	CID:16220015	phase I
BRD-K10573841	CC(C)CCCCCCCC\C=C\C(=O)N[C@H]1[C@H](O[C@@H]2O[C@@H](CO)[C@H](O)[C@@H](O)[C@@H]2NC(C)=O)O[C@H](C[C@@H](O)[C@H]2O[C@H]([C@H](O)[C@@H]2O)n2ccc(=O)[nH]c2=O)[C@H](O)[C@@H]1O	CID:16220051	phase I
BRD-K16051505	Cc1ccc(cc1)-c1csc(NC(=O)CSc2nnc3cc(C)c4ccccc4n23)n1	CID:16253428	phase I
BRD-K83620635	CN(C)S(=O)(=O)c1ccc(Cl)c(c1)C(=O)N1CCN(CC1)c1cccc(C)c1C	CID:16273006	phase I
BRD-A95504714	Brc1ccc(cc1)C(=O)NCCC(=O)NC2CCCc3ccccc23	CID:16273161	phase I
BRD-A35207501	Clc1ccc(cc1)C(=O)NCCC(=O)NC2CCCc3ccccc23	CID:16307489	phase I
BRD-K80368509	COc1ccccc1NC(=O)c2cccc(c2)S(=O)(=O)N3CCN(CC3)c4ccccc4	CID:16330153	phase I
BRD-K95786143	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccccc2C)c1C	CID:16391507	phase I
BRD-A38030642	CCC1NC(=O)C([C@H](O)[C@H](C)C/C=C/C)N(C)C(=O)C(C(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)C(C)NC(=O)C(CC(C)C)N(C)C(=O)C(NC(=O)C(CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C	CID:16404350	phase I
BRD-K29003210	CCc1nnc(NC(=O)c2nc(ncc2Cl)S(=O)(=O)Cc3ccccc3)s1	CID:16446678	phase I
BRD-K60895275	CCSc1nnc(NC(=O)c2nc(ncc2Cl)S(=O)(=O)Cc3ccc(F)cc3)s1	CID:16446868	phase I
BRD-A72498772	CCOC(=O)C1=C(CN2CCc3ccccc23)NC(=O)NC1c1ccc(F)cc1	CID:16654605	phase I
BRD-K42191735	Nc1cc(c(cn1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1)C(F)(F)F	CID:16654980	phase I
BRD-K37687095	Cc1cc(C(=O)NOCCO)c(Nc2ccc(I)cc2F)n(C)c1=O	CID:16666708	phase I
BRD-A73741725	C[C@]12CCC3C(CC(=C)C4=CC(=O)C=C[C@]34C)C1CCC2=O	CID:16667705	phase I
BRD-A90131694	CCC(=O)OCC(=O)[C@@]1(OC(=O)CC)[C@H](C)CC2C3[C@H](Cl)CC4=CC(=O)C=C[C@]4(C)C3[C@@H](O)C[C@@]21C	CID:16667717	phase I
BRD-A95696820	NC(=O)c1ncn(C2O[C@H](CO)[C@@H](O)[C@H]2O)c1N	CID:16667722	phase I
BRD-A93426597	OC(C(=O)N1CCC(CC1)Nc1ccc2[nH]ncc2c1)c1ccc(Br)cc1	CID:16681732	phase I
BRD-K67844266	NS(=O)(=O)OC[C@@H]1C[C@H](C[C@@H]1O)n1ccc2c(N[C@H]3CCc4ccccc34)ncnc12	CID:16720766	phase I
BRD-K12502280	Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C	CID:16722836	phase I
BRD-K51967704	COc1c(C)cnc(Cn2cnc3c(Cl)nc(N)nc23)c1C	CID:16736529	phase I
BRD-K67566344	COc1ccc(cc1CO)-c1ccc2c(nc(nc2n1)N1C[C@H](C)O[C@H](C)C1)N1CCOCC1	CID:16736978	phase I
BRD-K52836380	CN(C)C(=O)c1ccc(cc1)S(=O)(=O)c1ccc(NC(=O)[C@@](C)(O)C(F)(F)F)c(Cl)c1	CID:16741245	phase I
BRD-A16934955	OC1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5OC1[C@]2(CCN3CC6CCC6)c54	CID:16741281	phase I
BRD-A75769826	CC(=C)CN1CC[C@@]23[C@H]4Oc5c2c(CC1[C@]3(O)Cc1c4[nH]c2ccccc12)ccc5O	CID:16741282	phase I
BRD-A11731846	CC(OC1OC(CO)C(O)C(O)C1O)/C=C/C2(O)C(C)CC(O)CC2(C)C	CID:16745401	phase I
BRD-A00626522	COc1ccc(cc1)C(CC(=O)N2CCCC(C)C2)c3c(O)cc(OC)cc3OC	CID:16746329	phase I
BRD-A32917072	COc1cc(O)c(C(CC(=O)N2CCCC(C)C2)c3ccc4OCOc4c3)c(OC)c1	CID:16746402	phase I
BRD-K72414522	CC(C)n1c(C)ncc1-c1ccnc(Nc2ccc(cc2)S(C)(=O)=O)n1	CID:16747683	phase I
BRD-K43620258	COc1ccc(cc1NS(=O)(=O)c1cc(Cl)cc(Cl)c1O)-c1ccccc1	CID:16747776	phase I
BRD-K19922318	CN(C)C(=O)c1cccc(c1)-n1sc2ccccc2c1=O	CID:16749996	phase I
BRD-K15475572	O=C(NCc1ccccc1)c1cccc(c1)-n1sc2ccccc2c1=O	CID:16749997	phase I
BRD-K37323001	OC(=O)[C@@H](Cc1cccc2ccccc12)N1C(=O)c2ccc(cc2C1=O)C(O)=O	CID:16752640	phase I
BRD-K29983336	COc1ccc2c(Oc3ccc(NC(=O)c4c(C)n(CC(C)(C)O)n(-c5ccccc5)c4=O)cc3F)ccnc2c1	CID:16757524	phase I
BRD-A11706664	Cn1nc(N)c2cn([C@@H]3O[C@H](CO)C(O)[C@@H]3O)c3ncnc1c23	CID:16759157	phase I
BRD-K21064560	CCCCCCCCCCCCCCCC(=O)NCCc1ccc(O)c(O)c1	CID:16759163	phase I
BRD-K68633617	CN(C)c1nc(N)c(nc1Cl)C(=O)Nc1cccnc1	CID:16759169	phase I
BRD-K79684402	Cc1ncc(CN2CCC(=CC2)c2ccccc2)c(N)n1	CID:16759175	phase I
BRD-A91866971	OC(=O)CCC/C=C\CC1C(CNNC(=O)Nc2ccccc2)C3CCC1O3	CID:16759359	phase I
BRD-K67831364	Cc1cc(F)c(Nc2ncnc3cc(OCc4ccccc4)ccc23)cc1O	CID:16759369	phase I
BRD-A17757596	COc1ccc(cc1COc1ccc(NC(C)=O)cc1)C1Nc2ccccc2C(=O)N1Cc1ccccc1	CID:16759579	phase I
BRD-K14696368	Cc1ccc2c(c1)-c1ccc3cccnc3c1NS2(=O)=O	CID:16759925	phase I
BRD-K52405437	C[C@]12[C@@H](CC[C@@]3(O)[C@@]45O[C@@H]4[C@@H](O)[C@H](O[C@H]5CC[C@]13C)C(O)=O)[C@@H]1OC(C)(C)[C@H]3C[C@@H]4C(=C)Cc5c(Cl)cc6[nH]c2c1c6c5[C@]34O	CID:16759989	phase I
BRD-K40965114	CC(C)(C)NC[C@H](O)COc1cccc2[nH]c(C#N)cc12	CID:16759997	phase I
BRD-K71799778	CC(C)c1cnc(NC(=O)Cc2ccccc2)s1	CID:16760027	phase I
BRD-A41301928	COC(C/C=C/C=C/CC\C=C/CC(C)\C=C/C(=C\C(=O)O)/CC(=O)O)/C(=C\C=C(/C)\C(=O)O)/C	CID:16760034	phase I
BRD-A47513740	COC[C@H]([C@@H](O)[C@@H](O)C(=O)NCC[C@@H](C)c1nc(/C=C/C[C@H]2OC3(C[C@H](O)[C@H]2C)OC([C@@H](C[C@@H](O)[C@@H](C)[C@@H](O)[C@@H](C)/C=C(\C)/C(=C/C=C/C(=C\C#N)/C)/C)OC)[C@@H](OP(=O)(O)O)C3(C)C)co1)N(C)C	CID:16760037	phase I
BRD-K74148702	COc1ccc(/C=C/C(=O)CC(=O)\C=C\c2cccc(O)c2OC)cc1O	CID:16760039	phase I
BRD-K25504083	C[C@H]1[C@H]2[C@H](Cc3ccccc3)NC(=O)[C@@]22[C@@H](\C=C\C[C@H](C)C(=O)[C@@](C)(O)\C=C\[C@H]2OC(C)=O)[C@H](O)C1=C	CID:16760041	phase I
BRD-K53792571	N[C@H](CSCCB(O)O)C(=O)O	CID:16760312	phase I
BRD-K51018020	Oc1cc(ccc1C(=O)c2ccccc2)N3CCOCC3	CID:16760391	phase I
BRD-K83354763	Cc1ccc(NCCCc2ccccc2)c(N)c1	CID:16760588	phase I
BRD-K46678324	Clc1cc(Cl)c(NC(=O)Nc2ccncc2)c(Cl)c1	CID:16760634	phase I
BRD-K10136726	Cc1ccc(cc1)S(=O)(=O)N[C@H](CCCCN)C(=O)CCl	CID:16760682	phase I
BRD-K48427617	CS/C(=C(\C#N)/C(=C(\N)/SC)/[N+]#[C-])/N	CID:16760692	phase I
BRD-K27756844	Nc1ccccc1NC(=O)c1cnccn1	CID:16773791	phase I
BRD-K08856548	Cc1ccc(cn1)C(=O)Nc1ccccc1N	CID:16793302	phase I
BRD-K32827536	COc1ccc(Cl)cc1NC(=O)c1cc(on1)C1CC1	CID:17253222	phase I
BRD-K21005091	Clc1ccccc1C(=O)NNC(=O)c2csc(n2)N3CCOCC3	CID:17400499	phase I
BRD-K22129929	COc1ccccc1C(=O)NNC(=O)c2csc(n2)N3CCOCC3	CID:17400500	phase I
BRD-K25774147	COc1ccc(C)cc1n2nnnc2SCc3nc(N)nc(n3)N(C)C	CID:17425317	phase I
BRD-K40094191	CN(C)c1nc(N)nc(CSc2nnnn2c3c(C)cccc3C)n1	CID:17452347	phase I
BRD-K69516039	O=C(Nc1cc(ccc1N1CCCC1)S(=O)(=O)N1CCOCC1)c1cc2CCCCc2s1	CID:17460708	phase I
BRD-K95337198	Fc1cccc(F)c1C(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:17540423	phase I
BRD-K31553917	CC(C)c1ccc(cc1)n2nnnc2SCc3nc(N)nc(N)n3	CID:17562110	phase I
BRD-K55630727	CN(C)c1nc(N)nc(CSc2nnnn2c3ccc(Cl)cc3)n1	CID:17564913	phase I
BRD-K05510762	CN1[C@H]2CCC[C@H]1C[C@H](C2)NC(=O)c1nn(C)c2ccccc12	CID:17572266	phase I
BRD-K53923665	COc1ccc2n(CC(=O)N3CCC(Cc4ccccc4)CC3)c3c(nc4SCCn4c3=O)c2c1	CID:17581348	phase I
BRD-K76132250	Clc1ccc(CCNC(=O)Cn2c3ccccc3c3nc4SCCn4c(=O)c23)cc1	CID:17581618	phase I
BRD-K73319509	OCCn1cc(cn1)-c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1	CID:17754438	phase I
BRD-K52911425	CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1	CID:17755052	phase I
BRD-A75368507	CN(C)C1C2CC3C(O)c4c(Cl)ccc(O)c4C(=O)C3C(=O)C2(O)C(=O)C(C(N)=O)C1=O	CID:17756785	phase I
BRD-K00486786	Cc1cc2nc3c(nc(=O)[nH]c3=O)n(C)c2cc1C=O	CID:17756791	phase I
BRD-K49294207	CCN(CC)CC1CCN(CC1)c1ncc2ncnc(Nc3ccc(F)c(Cl)c3)c2n1	CID:17756796	phase I
BRD-K23412959	COc1cccc(CNc2ncnc3ccc(cc23)c4c(C)noc4C)c1	CID:17757075	phase I
BRD-K88622704	CCOc1ccccc1CNc2ncnc3ccc(cc23)c4c(C)noc4C	CID:17757080	phase I
BRD-K10361096	CC(=O)Nc1ccc(CNc2ncnc3ccc(cc23)c4c(C)noc4C)cc1	CID:17757086	phase I
BRD-A98444709	CN1CCCCC1CNc2ncnc3ccc(cc23)c4c(C)noc4C	CID:17757092	phase I
BRD-A11087911	CC(Nc1ncnc2ccc(cc12)c3c(C)noc3C)c4ccco4	CID:17757094	phase I
BRD-K52163391	Cc1ccsc1CNc2ncnc3ccc(cc23)c4c(C)noc4C	CID:17757095	phase I
BRD-A05831822	COc1ccc(cc1COc1ccc(NC(C)=O)cc1)C1NC(=O)c2ccccc2N1	CID:17757109	phase I
BRD-A81045722	CCCCN1C(Nc2ccccc2C1=O)c1ccc(OC)c(COc2ccc(NC(C)=O)cc2)c1	CID:17757110	phase I
BRD-K05402890	COc1ccc(OC)c(c1)c2nnc3SCC(=Nn23)c4ccc(OC)c(OC)c4	CID:17757146	phase I
BRD-K91691979	CC(C)(C)Oc1ccccc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:17757274	phase I
BRD-A32449311	Oc1ccc(Cl)cc1Nc2nc(NCC3CCCO3)c4ccccc4n2	CID:17757275	phase I
BRD-A81416315	COc1ccc(cc1COc1ccc(NC(C)=O)cc1)C1Nc2ccccc2C(=O)N1Cc1ccncc1	CID:17757294	phase I
BRD-K92202821	COc1ccc(cc1COc1ccc(NC(C)=O)cc1)-c1nc2ccccc2c(=O)n1Cc1ccccc1	CID:17757314	phase I
BRD-K00088062	Fc1ccc(Nc2c(cnc3c(Cl)cc(NCc4cnc[nH]4)cc23)C#N)cc1Cl	CID:17759555	phase I
BRD-K05861053	CNC(=O)CCc1nc(no1)-c1ccc(cc1)C(C)C	CID:18148563	phase I
BRD-K71917235	NC(=O)c1ccc(O)c2ncccc12	CID:18378031	phase I
BRD-A71356100	CCC(C)C(NC(=O)C(N)Cc1c[nH]cn1)C(=O)NC(CCCNC(N)=N)C(=O)NC(CC(C)C)C(O)=O	CID:18496254	phase I
BRD-A44244100	CNC(=O)C(=O)NCCC1CCCCN1S(=O)(=O)c2ccc(F)cc2C	CID:18574628	phase I
BRD-A31007383	COC1C(O)C(CO)OC1n2cnc3c(NC4CCCCC4)ncnc23	CID:18755269	phase I
BRD-A41986761	CNCCC(Oc1ccccc1I)c1ccccc1	CID:19102988	phase I
BRD-A93206962	CCCCCCNC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(CCNCC(O)COc3ccc(O)cc3)cc2	CID:19385000	phase I
BRD-K53903639	O=C(NC1CC1)c2cc(on2)c3cccs3	CID:19582717	phase I
BRD-K78984681	Cc1cc(C)n2ncc(C(=O)Nc3ccc4OCCOc4c3)c2n1	CID:19585362	phase I
BRD-K25210139	CCN(CC)CCn1c2[C@H]3C[C@H]4[C@H](C[C@@H](OC(=O)c5cc(OC)c(OC)c(OC)c5)[C@H](OC)[C@H]4C(=O)OC)CN3CCc2c2ccc(OC)cc12	CID:20054848	phase I
BRD-K06209536	CN(C)CCCNc1ccc(O)cc1	CID:20283862	phase I
BRD-A14795281	CC(N)C(O)c1ccccc1Cl	CID:20348787	phase I
BRD-K99554241	COc1cc2c(CCNC(C)=O)c(C)[nH]c2cc1Cl	CID:20355585	phase I
BRD-A75552914	CN1C(C(=O)Nc2cc(C)on2)C(=O)c2ccccc2S1(=O)=O	CID:20507134	phase I
BRD-A29901043	COc1cc(C)c(Sc2cnc(NC(=O)c3ccc(CNC(C)C(C)C)cc3)s2)cc1C(=O)N1CCN(CC1)C(C)=O	CID:20635522	phase I
BRD-K33495169	COc1ccc(cc1)S(=O)(=O)NCc1ccc(cc1)C(=O)NCCN(C)Cc1ccccc1	CID:20854195	phase I
BRD-K43782924	COc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)N3CCN(Cc4ccccc4)CC3	CID:20854208	phase I
BRD-K14402394	CN(CCNC(=O)c1ccc(CNS(=O)(=O)c2ccc(NC(C)=O)cc2)cc1)Cc1ccccc1	CID:20854254	phase I
BRD-A73558769	CCOc1ccccc1C1N2CCCC2C(=O)N1c1ccc(Cl)cc1	CID:20856774	phase I
BRD-K89009594	Cn1c2ccccc2c(OCCCC(=O)Nc2cccc(Cl)c2)cc1=O	CID:20862013	phase I
BRD-K69676861	Cc1cc(Br)ccc1NC(=O)CCCOc1cc(=O)n(C)c2ccccc12	CID:20862025	phase I
BRD-K13277629	COC(=O)c1ccccc1NC(=O)CCCOc1cc(=O)n(C)c2ccccc12	CID:20862034	phase I
BRD-K75641083	CCc1ccc(NC(=O)CCCOc2cc(=O)n(C)c3ccccc23)cc1	CID:20862056	phase I
BRD-K73334721	CSc1cccc(NC(=O)CCCOc2cc(=O)n(C)c3ccccc23)c1	CID:20862086	phase I
BRD-K75308990	COc1ccc(OC)c(CCNC(=O)c2ccc3SCCN(Cc4ccc(F)cc4)c3c2)c1	CID:20876331	phase I
BRD-K25094947	COc1cc(NC(=O)c2cnn3c(C)cc(C)nc23)cc(OC)c1OC	CID:20952848	phase I
BRD-K44575778	CN1CCN(CC1)C(=O)c1cc2cc3cc(C)ccc3nc2s1	CID:20966339	phase I
BRD-K83589469	CC(=O)c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc4NC(=O)Cc4c3	CID:20969430	phase I
BRD-K84874839	CCOc1ccccc1/C=C/c2onc(C)c2S(=O)(=O)N3CCC(CC3)C(=O)NC(C)(C)C	CID:20969756	phase I
BRD-K80062189	COc1ccc2N(CCCN(C)C)c3cc(Cl)ccc3Sc2c1	CID:21115409	phase I
BRD-A66229260	CC(CCCC(C)(C)O)C1CCC2C1(C)CCC\C2=C/C=C1/CC(O)CC(O)C1=C	CID:21158442	phase I
BRD-K28180706	OC(c1ccc(NC(=O)c2ccc(Cl)cc2)cc1)(C(F)(F)F)C(F)(F)F	CID:21179063	phase I
BRD-K99922388	CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1P(=O)(c1ccccc1)c1ccccc1	CID:21678144	phase I
BRD-K02458594	Cc1ccccc1N1Cc2ccccc2C1=O	CID:21785456	phase I
BRD-A39969961	COC(=O)C1CC2=CC(=O)CCC2(C)C34OC4CC5(C)C(CCC65CCC(=O)O6)C13	CID:21865526	phase I
BRD-K55242988	Oc1ccc2cccc(CCNC(=O)CBr)c2c1	CID:21917176	phase I
BRD-K89626439	CO[C@@H]1C[C@H](C[C@@H](C)[C@@H]2CC(=O)[C@H](C)\C=C(C)\[C@@H](O)[C@@H](OC)C(=O)[C@H](C)C[C@H](C)\C=C/C=C/C=C(C)/[C@H](C[C@@H]3CC[C@@H](C)[C@@](O)(O3)C(=O)C(=O)N3CCCC[C@H]3C(=O)O2)OC)CC[C@H]1O	CID:21944094	phase I
BRD-A57905915	CNCCCC1(OCc2cc(ccc12)[N+]#[C-])c1ccc(F)cc1	CID:22094941	phase I
BRD-A05581237	NCCCC1(OCc2cc(ccc12)[N+]#[C-])c1ccc(F)cc1	CID:22094944	phase I
BRD-K09085930	CCc1cncc2cccc(c12)S(=O)(=O)N3CCCNCC3	CID:22121918	phase I
BRD-A58767537	CN(C)C\C=C\C(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1OC1CCOC1	CID:22225683	phase I
BRD-K28178212	Cn1cc(\C=C2\C(=O)Nc3cccnc23)c2ccccc12	CID:22228376	phase I
BRD-A42610307	NC(Cc1ccc(O)c(O)c1O)C(O)=O	CID:22326275	phase I
BRD-A81472640	NC(Cc1ccc(O)c(O)c1Cl)C(O)=O	CID:22326433	phase I
BRD-K32656671	Fc1ccc2sn(c3ccccc3)c(=O)c2c1	CID:22416235	phase I
BRD-K38483076	Fc1ccccc1-n1sc2ccccc2c1=O	CID:22416236	phase I
BRD-K53579868	Clc1ccc(c(Cl)c1)-n1sc2ccccc2c1=O	CID:22416251	phase I
BRD-K19609011	[O-][N+](=O)c1ccc2sn(-c3ccccc3)c(=O)c2c1	CID:22416272	phase I
BRD-K06748700	Fc1ccc(cc1)n2sc3ccccc3c2=O	CID:22416276	phase I
BRD-K51774655	COc1ccc2cc3cc(sc3nc2c1)C(=O)Nc1ccc(F)cc1	CID:22434552	phase I
BRD-K04930762	Cc1ccc(NS(=O)(=O)c2cc3OCC(=O)Nc3cc2Cl)cc1C	CID:22548477	phase I
BRD-K50493736	CCCN(CCC)c1nc(Cl)nc2ccccc12	CID:22693263	phase I
BRD-K25841245	CC[C@H](C)C(=O)O[C@H]1C[C@H](O)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(O)=O)[C@H]12	CID:22833647	phase I
BRD-K95048846	OC(C1CCN(CCCOc2ccccc2)CC1)(c1ccccc1)c1ccccc1	CID:23036271	phase I
BRD-A55317422	CC(N(Cc1ccccc1)Cc1ccccc1)C(=O)c1ccc(OCc2ccccc2)cc1	CID:23212022	phase I
BRD-K69458799	CNCCCN1c2ccccc2S(=O)c2ccccc12	CID:23275476	phase I
BRD-K33551950	C[C@@H]1C[C@@H]2O[C@H]2\C=C\C=C\C(=O)Cc2c(Cl)c(O)cc(O)c2C(=O)O1	CID:23351218	phase I
BRD-K52431530	CO[C@H]1[C@@H](CC(=O)O[C@H](C)CC=CC=C[C@H](O)[C@H](C)C[C@H](CC=O)[C@@H]1O[C@@H]2O[C@H](C)[C@@H](O[C@H]3C[C@@](C)(OC(=O)CC(C)C)[C@@H](O)[C@H](C)O3)[C@@H]([C@H]2O)N(C)C)OC(=O)C	CID:23581794	phase I
BRD-A62434282	CC(C)CC(NC(=O)C(COC(C)(C)C)NC(=O)C(Cc1ccc(O)cc1)NC(=O)C(CO)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C(Cc1c[nH]cn1)NC(=O)C1CCC(=O)N1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCCC1C(=O)NNC(N)=O	CID:23581805	phase I
BRD-A73929928	OC[C@H]1O[C@H]([C@@H](O)C1O)n1cnc2c(N[C@H]3CCC[C@@H]3O)ncnc12	CID:23581828	phase I
BRD-K06750613	O=C1NC(=O)\C(S1)=C\c1ccc2nccc(-c3ccncc3)c2c1	CID:23582824	phase I
BRD-A80788753	CCCCC(O)(C(CN1CCOCC1)c2ccc(Cl)cc2)c3ccc(F)cc3	CID:23606608	phase I
BRD-K91028164	O=C(N1CCC(CC1)n1nc(oc1=O)-c1ccccc1)C1(CCCC1)c1ccccc1	CID:23612543	phase I
BRD-K73315009	O=C(Cc1ccc2OCOc2c1)N1CCC(CC1)n1nc(oc1=O)-c1ccccc1	CID:23612548	phase I
BRD-K25460880	COc1ccc(cc1)C2(CC2)C(=O)N3CCC(CC3)n4nc(oc4=O)c5ccccc5	CID:23612550	phase I
BRD-K89412978	Cc1ccc(cc1)C2(CC2)C(=O)N3CCC(CC3)n4nc(oc4=O)c5ccccc5	CID:23612552	phase I
BRD-K58846134	O=C(N1CCC(CC1)n2nc(oc2=O)c3ccccc3)C4(CC4)c5ccccc5	CID:23612554	phase I
BRD-K86108784	Clc1ccc(cc1)C2(CC2)C(=O)N3CCC(CC3)n4nc(oc4=O)c5ccccc5	CID:23612567	phase I
BRD-K30553817	BrCC(=O)NCCc1ccc2ccccc2c1	CID:23626931	phase I
BRD-K83194053	Oc1ccc(CCNc2ncnc3ccc(Cl)cc23)cc1	CID:23631972	phase I
BRD-K06319591	NCc1ccccc1CC(=O)N[C@@H]1[C@H]2SCC(CSc3nnnn3CC(O)=O)=C(N2C1=O)C(O)=O	CID:23637804	phase I
BRD-K75644678	CCCCOc1cccc2c1ccn(CC(=O)Nc1ccc3OCCOc3c1)c2=O	CID:23640021	phase I
BRD-K12811596	OC(=O)COc1c(Br)c(sc1C(O)=O)-c1ccc(NC(=O)c2cccnc2)cc1	CID:23646672	phase I
BRD-K41284916	COc1ccc(Cl)cc1Nc2nc(NCCO)nc(n2)N3CCCCC3	CID:23648012	phase I
BRD-K35389996	Cc1ccc(Nc2nc(NCCO)nc(n2)N3CCCC3)cc1	CID:23648018	phase I
BRD-K35920785	OCCNc1nc(Nc2ccccc2Cl)nc(n1)N3CCCC3	CID:23648019	phase I
BRD-K12540328	COc1ccccc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:23648021	phase I
BRD-K13604076	COc1cccc(Nc2nc(NCCO)nc(n2)N3CCCC3)c1	CID:23648022	phase I
BRD-K19117583	COc1ccc(Nc2nc(NCCO)nc(n2)N3CCCC3)cc1	CID:23648023	phase I
BRD-K45355657	OCCNc1nc(Nc2ccccc2O)nc(n1)N3CCCC3	CID:23648024	phase I
BRD-K55966666	OCCNc1nc(Nc2ccccc2Oc3ccccc3)nc(n1)N4CCCC4	CID:23648026	phase I
BRD-K67941506	OCCNc1nc(Nc2ccccc2OC(F)(F)F)nc(n1)N3CCCC3	CID:23648028	phase I
BRD-K53653395	CCOc1ccc(Cl)cc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:23648036	phase I
BRD-K58519325	CC(C)Oc1ccc(Cl)cc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:23648037	phase I
BRD-K02708799	O=C1NC(=O)\C(S1)=C/c1ccc2nccc(-c3ccncc3)c2c1	CID:23658330	phase I
BRD-K02113016	Fc1ccc(Cc2n[nH]c(=O)c3ccccc23)cc1C(=O)N1CCN(CC1)C(=O)C1CC1	CID:23725625	phase I
BRD-K05452595	OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5	CID:23747926	phase I
BRD-K37194137	CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6	CID:23748511	phase I
BRD-K95202259	C[S+](O)c1ccc(CSc2nc(c([nH]2)c3ccc(F)cc3)c4ccncc4)cc1	CID:23748533	phase I
BRD-K90697054	NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O	CID:23748550	phase I
BRD-K31706415	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78	CID:23748696	phase I
BRD-K84106030	COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78	CID:23748755	phase I
BRD-K87730440	OCc1ccc(/C=N/NC(=O)CCCCCCC(=O)O)o1	CID:23749418	phase I
BRD-A59728941	CC(=O)OC[C@@]12CCC(=CC2O[C@@H]3[C@H](O)[C@@H](O[C@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)[C@@]1(C)C53CO5)C	CID:23757080	phase I
BRD-K60685007	COc1cc(O)c(CC=C(C)C)cc1C(=O)/C=C/c2ccc(O)c(CC=C(C)C)c2	CID:23757123	phase I
BRD-A43188678	CC(C)CCCC/C=C\CCCCCCCC(=O)OCC(O)CO	CID:23757164	phase I
BRD-A04172077	COc1ccc2ccc(=O)oc2c1CC(O)C(C)(C)OC	CID:23757203	phase I
BRD-A99879977	COc1ccc(CN2C(C)Cc3cc(OC)c(OC)cc3C2C=C)cc1	CID:23757372	phase I
BRD-K12266212	COC(=O)c1cn(nn1)c2cccc(N)c2	CID:23760093	phase I
BRD-K56392985	C/C=C/C#CC#C[C@@H](O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@H](O)\C=C\CCCO	CID:23760109	phase I
BRD-A96820077	CO[C@H]1C=C2CCN(C)[C@H]2C3[C@@H]1OC(=O)c4cc5OCOc5cc34	CID:23760135	phase I
BRD-A11263757	Nc1ncn(C2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1	CID:23760137	phase I
BRD-K96659869	CC(=O)N[C@@H](CC(=O)N[C@H](CCC(=O)O)C(=O)O)C(=O)O	CID:23760140	phase I
BRD-A56020723	CCCNC(=O)[C@H]1O[C@@H]1C(=O)N[C@@H](C(C)CC)C(=O)N2CCC[C@H]2C(=O)OC	CID:23760717	phase I
BRD-K24102129	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCOC5=O)c6ccccc63	CID:23777110	phase I
BRD-A89907244	NC(=O)N1C(=O)C2C(C3C(C4CC4)N(Cc5sc6ccccc6c5Cl)C2C=C3c7ccc(CO)cc7)C1=O	CID:23777133	phase I
BRD-K37340241	CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS	CID:23777578	phase I
BRD-K05520923	OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCCN6CCOCC6)c7ccc(cc7)[N+](=O)[O-])c(I)c1	CID:23777600	phase I
BRD-K00944562	OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5	CID:23777636	phase I
BRD-A70591769	COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)c4ccc(CN5CCCC5)cc4	CID:23777637	phase I
BRD-K16541732	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73	CID:23777756	phase I
BRD-A71171460	CC1CC\C=C/[C@H]2OC34C=CCN(C(=O)[C@H]3N(CCCO)C(=O)[C@@H]4C2C(=O)O1)C(C)(C)C	CID:23777784	phase I
BRD-K08799950	OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCCCC2)c3cccs3	CID:23778527	phase I
BRD-K16057611	C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccc(cc3)N4CCCCC4=O)c5ccccc52)[Si](C)(C)F	CID:23778539	phase I
BRD-A81282034	C[C@H]1[C@H]2[C@@H](CC1=O)C(=C)C[C@@H](OC(=O)/C(=C/CO)/COC(=O)/C(=C/CO)/C)C3[C@@H]2OC(=O)C3=C	CID:23786279	phase I
BRD-A70633932	CCCCCC1OC2=C(C(O)C1(C)O)C(=O)N(OC)C2CSCC(O)C(=O)O	CID:23786305	phase I
BRD-A94546435	CC1(C)CC[C@@]2(CC[C@]3(C)C(=CCC4[C@@]5(C)CC[C@H](O)[C@](C)(C5CC[C@]43C)C(=O)O)C2C1)C(=O)O[C@@H]6O[C@H](CO[C@@H]7O[C@H](CO)[C@@H](O)[C@H](O)[C@H]7O)[C@@H](O)[C@H](O[C@@H]8O[C@H](CO)[C@@H](O)[C@H](O)[C@H]8O)[C@H]6O	CID:23786410	phase I
BRD-K28925416	CC(C)(O)CCc1c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)cc(O)c3C(=O)[C@H](O)[C@H](Oc13)c4ccc(O)cc4	CID:23786458	phase I
BRD-A50796384	OC(CSc1nc(c(o1)c2ccccc2)c3ccccc3)CC(O)c4ccc(cc4)[N+](=O)[O-]	CID:23786513	phase I
BRD-A39903068	CN[C@H]1[C@@H](O)[C@H](O[C@@H]2[C@@H](N)C[C@@H](N)[C@H](OC3OC(=CCC3N)CN)[C@@H]2O)OC[C@@]1(C)O	CID:23789067	phase I
BRD-A60583491	C1CN[C@H]2[C@@H](C1)C3CCC2[C@H]4N3CCc5c4[nH]c6ccccc56	CID:23789069	phase I
BRD-K73418978	CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O	CID:23806106	phase I
BRD-K55071917	COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4	CID:23806752	phase I
BRD-K86110682	COC(=O)CCCCCCC(=O)N/N=C/c1cc2OCOc2cc1Br	CID:23807491	phase I
BRD-K90430314	COC(=O)CCCCCCC(=O)N/N=C/c1ccccc1C(=O)O	CID:23807495	phase I
BRD-K27630390	C[C@H](O)C(=O)Nc1ccc2N(CC=C)C(=O)[C@]3(O[C@H](CCO)[C@H]([C@@H]3C)[Si](C)(C)F)c2c1	CID:23807536	phase I
BRD-A75471153	C[C@@H]1CCC2C(C)(C)[C@H](O)CC[C@]2(C)[C@]31Cc4c(O3)c5CN([C@@H](CCC(=O)O)C(=O)O)C(=O)c5cc4O	CID:23815265	phase I
BRD-K85565420	CCCCC[C@@H]1OC2=C([C@H](O)[C@]1(C)O)C(=O)N(OC)C2=C	CID:23815293	phase I
BRD-A94381689	CO[C@H]1C(O[C@@H]2C[C@H]3O[C@@H]([C@@H](O)[C@H](O)[C@]3(O)O[C@H]12)C(=O)OC)n4cnc5c(N)ncnc45	CID:23815298	phase I
BRD-A77722753	N/N=C/1\N=NC=C2C=CC=CC12	CID:23817956	phase I
BRD-A17535965	CN1C[C@@]2(C=C)C3CC4OC[C@@H]3[C@@H]1[C@H]2[C@@]45C(=O)Nc6ccccc65	CID:23817963	phase I
BRD-A95944315	OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCC(O)CO	CID:23834891	phase I
BRD-K86901264	OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(CC=C)C3=O	CID:23834901	phase I
BRD-K75234292	COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3	CID:23834916	phase I
BRD-K90849765	OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5	CID:23835417	phase I
BRD-K47764688	NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4	CID:23835472	phase I
BRD-K83998179	COC(=O)CCCCCCC(=O)N/N=C/c1cc(Br)ccc1OC	CID:23836178	phase I
BRD-K55536701	C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccc(cc32)N4C(=O)c5ccccc5Oc6ccccc46)[Si](C)(C)F	CID:23836210	phase I
BRD-A64811980	CN(CC(O)CC(O)c1ccccc1)Cc2ccccc2	CID:23844163	phase I
BRD-K54573313	C/C(=C/CC[C@@H](CO)[C@H]1CC[C@@]2(C)[C@@H]3CC[C@@H]4[C@]5(C[C@@]35CC[C@]12C)[C@@H](O)C[C@H](O[C@@H]6O[C@H](CO)[C@@H](O)[C@H](O)[C@H]6O)C4(C)C)/CO	CID:23846550	phase I
BRD-A63998256	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)OC2CC[C@]3(C=O)[C@H]4CC[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)C6=CC(=O)OC6	CID:23846563	phase I
BRD-A83029311	NCCC(O)C(=O)N[C@@H]1C[C@H](N)[C@@H](OC2O[C@H](CN)[C@@H](O)[C@H](O)[C@H]2N)[C@H](OC3O[C@H](CO)C(O)[C@H]3O)[C@H]1O	CID:23846564	phase I
BRD-K28789065	Oc1ccccc1N2C(=O)/C(=C/c3ccc(Br)cc3)/C=C2c4ccccc4	CID:23863188	phase I
BRD-K48016779	CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCCCC4	CID:23863215	phase I
BRD-K24031526	CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCC[N+](C)(C)C	CID:23863733	phase I
BRD-K71292008	CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10	CID:23863734	phase I
BRD-K84677391	C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O	CID:23863739	phase I
BRD-K96752129	COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6	CID:23863760	phase I
BRD-K16290432	OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5	CID:23863781	phase I
BRD-A13914662	COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(c4cccs4)c2cc1O	CID:23863790	phase I
BRD-K63549648	COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(C(=O)c3ccccc32)c4ccc(C)cn4)c5ccc(CO)cc5)cc1	CID:23863791	phase I
BRD-A89333723	NC(=O)N1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5ccc(CN6CCCC6)cc5)C1=O	CID:23863814	phase I
BRD-A30083233	C[C@@H]1O[C@@H](O[C@H]2[C@H](O[C@H]3CC[C@@]4(C)C(CC[C@]5(C)C4CC[C@@H]6C7[C@@](C)(O)[C@@H](CC=C(C)C)O[C@@]7(O)[C@H](O)[C@]65C)C3(C)C)O[C@H](CO)[C@H](O)[C@@H]2O[C@@H]8O[C@H](CO)[C@@H](O)[C@H](O)[C@H]8O)[C@H](O)[C@H](O)[C@H]1O	CID:23872142	phase I
BRD-A77704559	COC1OC(=O)C(CCC2(C)C(C)CCC3(C)C2CC(O)C(O)C43CO4)C1O	CID:23874489	phase I
BRD-A13461302	CC1CC(=O)C2C(O)(C1)CC(O)C34OC4c5c(O)cccc5C(=O)C23O	CID:23874505	phase I
BRD-A15070535	CCCC(=O)Nc1ncnc2n(cnc12)[C@@H]3O[C@@H]4OP(=O)(O)OC[C@H]4[C@H]3OC(=O)CCC	CID:23874512	phase I
BRD-A66199457	C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)C[C@@H](O)[C@H](O)[C@@](C)(CO)C5CC[C@]43C)[C@@H]2[C@H]1C)C(=O)O[C@@H]6O[C@H](COC7O[C@H](CO)[C@@H](OC8O[C@@H](C)[C@H](O)[C@@H](O)[C@H]8O)[C@H](O)[C@H]7O)[C@@H](O)[C@H](O)[C@H]6O	CID:23874513	phase I
BRD-K16533489	CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]2OC(=O)Nc5ccccc5c6ccccc6)c1	CID:23891056	phase I
BRD-K67010098	CN(C)CCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4	CID:23891087	phase I
BRD-K77877933	CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7	CID:23891514	phase I
BRD-K58279162	COCCCNC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3	CID:23891538	phase I
BRD-K89558221	OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O	CID:23891542	phase I
BRD-K74109131	OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F	CID:23891544	phase I
BRD-K16331660	COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CC(F)(F)F)C4=O)c6ccccc6C2=O	CID:23891545	phase I
BRD-K81314178	COCCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4	CID:23891566	phase I
BRD-K95080859	Cc1ccccc1/C=N/NC(=O)CCCCCC(=O)O	CID:23892245	phase I
BRD-K35568648	COC(=O)CCCCCCC(=O)N/N=C/c1ccc(Sc2nnc(C)n2C)o1	CID:23892254	phase I
BRD-K25731886	COC(=O)CCCCCCC(=O)N/N=C/[C@@H](O)[C@H](O)[C@H](O)CO	CID:23892255	phase I
BRD-A57300602	C/C=C(\C)/C(=O)OC1CCC(=O)OC1\C=C\C(O)C(C)O	CID:23900051	phase I
BRD-A41997916	COc1ccc(cc1)c2coc3c(OC)c(OC)cc(OC4OC(CO)C(O)C(O)C4OC5OCC(O)C(O)C5O)c3c2=O	CID:23900084	phase I
BRD-A38878059	CC(=O)C1CC[C@H]2[C@@H]3CC[C@@H]4CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:23902994	phase I
BRD-K11158509	C[C@@H](NC(=O)/C(=C\c1ccc(O)c(O)c1)/C#N)c2ccccc2	CID:23919058	phase I
BRD-K33164466	OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)N4CCOCC4	CID:23919109	phase I
BRD-K72161580	C[C@@H]1ON([C@@H]([C@H]1C(=O)O)c2ccccc2)c3ccccc3	CID:23919667	phase I
BRD-A26097136	CCN1C[C@]2(COC)CCC(OC)[C@]3(C4C[C@@]5(O)[C@H](OC(=O)c6ccc(OC)cc6)C4[C@](C[C@H]5OC)(OC(=O)C)[C@H]7[C@H](OC)C32)[C@@H]71	CID:23919696	phase I
BRD-K07850148	OCCOc1cccc(CN2CCC(CN3C(=O)c4ccccc4C3=O)CC2)c1	CID:23920343	phase I
BRD-K94493764	COC(=O)c1ccc(O)c2oc3cc(CO)cc(O)c3c(=O)c12	CID:23928086	phase I
BRD-K28293491	O[C@@H]1[C@@H](O)[C@H](Oc2ccc(cc2)c3coc4cc(O)ccc4c3=O)O[C@@H]([C@H]1O)C(=O)O	CID:23930394	phase I
BRD-A08709697	CO[C@H](C)C(O)(C(C)C)C(=O)OCC1=CCN2CC[C@H](O)[C@H]21	CID:23930397	phase I
BRD-K44812652	CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS	CID:23946995	phase I
BRD-K80981391	CCOC(=O)[C@H]1C\C=C\C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccc(OC)cc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O	CID:23947034	phase I
BRD-A81530502	COc1ccc(cc1)/C(=N/N2C(Nc3ccccc3C2=O)c4ccccc4O)/C	CID:23947494	phase I
BRD-A80502530	C[C@@H]1C[C@H]2[C@@H](CC[C@@H]3C[C@@H](O)CC[C@@]32C)[C@]45O[C@@H]5[C@H](OC(=O)C)[C@@H](C14)c6ccc(=O)oc6	CID:23947601	phase I
BRD-A78909648	COCC#CC1N(Cc2ccc(o2)[N+](=O)[O-])CCc3cc(OC)c(O)cc13	CID:23948194	phase I
BRD-A68274214	CC1=CCC2[C@](C)(CCC[C@]2(C)[C@H]1CCc3ccoc3)C(=O)O	CID:23955883	phase I
BRD-K63697730	CC(=CCc1c(O[C@@H]2O[C@H](COC(=O)CC(=O)O)[C@@H](O)[C@H](O)[C@H]2O)cc(O)c3C(=O)C[C@H](Oc13)c4ccc(O)cc4)C	CID:23955913	phase I
BRD-K30958640	CC(C)(O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@@H](O)COc2c3ccoc3cc4oc(=O)ccc24	CID:23958168	phase I
BRD-A61486721	CN[C@H]1[C@@H](O)C2O[C@H](O[C@@H]3[C@@H](N)C[C@@H](N)[C@H](O)[C@H]3O)[C@H](N)C[C@@H]2OC1O[C@H]4O[C@H](CO)[C@@H](N)[C@H](O)[C@H]4O	CID:23958199	phase I
BRD-K94173926	CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4	CID:23975549	phase I
BRD-K88569143	OC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O	CID:23975571	phase I
BRD-K93215584	COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCCCN(C)C)c5ccccc5C2=O	CID:23975579	phase I
BRD-K93296644	CC(C)NC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5	CID:23975589	phase I
BRD-K94137285	CCCC[C@H]1OB(O)C[C@H]2C1=C(COC)Cn3n2c(=O)n(c4ccccc4)c3=O	CID:23976270	phase I
BRD-A13367427	CC1OC(OC2CCC3(C)C(CCC4(C)C3CC=C5C6CC(C)(C)CCC6(CCC54C)C(=O)OC7OC(CO)C(OC8OCC(OC9OC(CO)C(O)C(O)C9O)C(OC%10OCC(O)C(O)C%10O)C8O)C(O)C7O)C2(C)C)C(O)C(O)C1OC%11OCC(O)C(O)C%11O	CID:23983744	phase I
BRD-A14178283	C[C@H]1O[C@@H](O[C@H]2CC[C@@]3(C)C(CC[C@]4(C)C3C=C[C@@]56OC[C@@]7(CCC(C)(C)C[C@H]76)[C@@H](O)C[C@]54C)[C@]2(C)CO)[C@H](O[C@@H]8O[C@H](CO)[C@@H](O)[C@H](O)[C@H]8O)[C@@H](O[C@@H]9O[C@H](CO)[C@@H](O[C@@H]%10O[C@H](CO)[C@@H](O)[C@H](O)[C@H]%10O)[C@H](O)[C@H]9O)[C@H]1O	CID:23986040	phase I
BRD-A37501891	C[C@@H]1CC[C@@]2(CC[C@]3(C(=O)O)C(=CCC4[C@@]5(C)CC[C@H](O[C@@H]6O[C@@H](C)[C@H](O)[C@@H](O)[C@H]6O)C(C)(C)C5CC[C@]43C)[C@@H]2[C@H]1C)C(=O)O	CID:23986044	phase I
BRD-A43849199	CCN1C[C@]2(C)CC[C@H](O)[C@]3([C@@H]4C[C@H]5C(O)[C@@H]4[C@](O)(C[C@@H]5OC)[C@H]6C[C@@H]32)C61	CID:23986045	phase I
BRD-K83982653	O=C(Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)Nc4ccon4	CID:23986308	phase I
BRD-K51674646	CCCSC1=N/C(=C/c2cccs2)/C(=O)N1c3ccc(F)c(Cl)c3	CID:24002878	phase I
BRD-K18163752	CC(=CCN([C@H](CO)c1ccccc1)C(=O)C#Cc2ccccc2)C	CID:24030598	phase I
BRD-K54159704	CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N	CID:24031038	phase I
BRD-K89156937	NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4	CID:24031043	phase I
BRD-A84102390	CS(=O)(=O)CCOC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)c3ccc(CN4CCCC4)cc3	CID:24031075	phase I
BRD-K69501658	COC(=O)CCCCCCC(=O)N/N=C/c1ccccc1Cl	CID:24031702	phase I
BRD-A95820578	C/C=C/C1OC2=C(C(O)C1O)C(=O)OC2=C	CID:24039271	phase I
BRD-A37817666	CC(=C)[C@H]1[C@H]2OC(=O)C1[C@]3(O)CC4O[C@]45C(=O)O[C@H]2[C@@]53C	CID:24041599	phase I
BRD-K74793820	CC[C@]1(O)C[C@H]2C[N@@](C1)CCc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C=O)[C@@H]1[C@]22CCN3CC=C[C@@](CC)([C@@H]23)[C@@H](OC(C)=O)[C@]1(O)C(=O)OC	CID:24058669	phase I
BRD-K00486725	CC(C)CNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-]	CID:24058689	phase I
BRD-K82971429	C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(CC=C)c3ccc(cc32)N4CCCCC4=O)[Si](C)(C)F	CID:24059344	phase I
BRD-A22272113	CCCC1=C(/C=C/C(=O)O)C(=O)C(O1)C(C)(C)C2OC(=C(/C=C/C(=O)O)C2=O)CCC	CID:24069148	phase I
BRD-K86761848	CCOC(=O)[C@H]1C\C=C\C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccc(Br)cc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O	CID:24086306	phase I
BRD-K61192129	COC(=O)CCCCCCC(=O)N/N=C/CCCC1OCC(C)(C)CO1	CID:24086889	phase I
BRD-K15419449	CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Br)cc2)[C@@H]2OC(=O)[C@H](Cc3cccc(Br)c3)C\C=C\C[C@@H](Cc3cccc(Br)c3)C(=O)O[C@@H]12	CID:24094067	phase I
BRD-K96274284	OCc1c(Cl)cccc1N2[C@@H](C(=O)NCc3ccccc3)[C@]4(O[C@H]5C=C4)[C@H]([C@@H]5C(=O)O)C2=O	CID:24094187	phase I
BRD-K09790412	NCCNCc1cccc2cnccc12	CID:24113957	phase I
BRD-K09977233	Cc1cc(O)c(O)c(c1)C(=O)C(=O)c2c(O)cc(O)cc2O	CID:24123440	phase I
BRD-K08845546	CO[C@@H]1C[C@@H](CC[C@H]1O)\C=C(/C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@]2(O)O[C@H](C[C@H](C[C@@H](C)C\C(C)=C/[C@@H](CC=C)C(=O)C[C@H](O)[C@H]1C)OC)[C@H](C[C@H]2C)OC	CID:24140138	phase I
BRD-K72541103	OCc1cc2ncnc(Nc3ccc(O)cc3)c2cc1CO	CID:24140566	phase I
BRD-K01800709	COC(=O)C1(CCCCC1)N2CC3=CCCC=C[C@H]3[C@@H]2[C@@H](O)Cc4ccccc4	CID:24148563	phase I
BRD-A41114263	OCCCCC/C=C\C/C=C\C(O)CC1CCC(CC(=O)O)O1	CID:24150636	phase I
BRD-A74771556	CC(C(C)c1ccc(O)cn1)C(N)C(=O)NC([C@H]2O[C@H]([C@@H](O)[C@H]2O)N3C=CC(=O)CC3=O)C(=O)O	CID:24151277	phase I
BRD-K44540157	Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCCN6CCOCC6)cc1	CID:24167050	phase I
BRD-A20488704	CC1(C)C(CCC2(C)C3CC(O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)C(C)(C=C)C=C3CCC12)O[C@@H]5O[C@@H](CO)[C@H](O)[C@H]5O	CID:24177547	phase I
BRD-K54331210	OCCNC(=O)c1cc(n[nH]1)-c1ccc(Cl)c(Cl)c1Cl	CID:24178170	phase I
BRD-K16478699	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F	CID:24180719	phase I
BRD-K64877338	O=C(N1CCc2ccccc2C1)C1=CC=CN2CCS(=O)(=O)N=C12	CID:24239644	phase I
BRD-A95937159	CCC1CCc2sc(cc2C1)C(=O)Nc1cc(ccc1OC)S(=O)(=O)N1CCOCC1	CID:24242928	phase I
BRD-K70229243	CCOC(=O)C(Cc1cc(OC)cc(OC)c1)(Cc2cc(OC)cc(OC)c2)C#N	CID:24747148	phase I
BRD-K91184774	Cc1nc(N)c2c(Cc3cccc4ccccc34)nn(c2n1)C(C)(C)C	CID:24747149	phase I
BRD-A74983348	CC(=O)OC1CCC2C3CCC4=CC(=O)CCC4(C)C3CCC2(C)[C@]1(C)O	CID:24747150	phase I
BRD-K45308677	Nc1c(C#N)c(Cc2cccc3ccccc23)nn1CCC#N	CID:24747151	phase I
BRD-K32132269	COc1c(O)cccc1[C@@H](O)C2CCN(CCc3ccc(F)cc3)CC2	CID:24747152	phase I
BRD-K67306351	Nc1c(C#N)c(Cc2cccc3ccccc23)nn1CCO	CID:24747153	phase I
BRD-K62716919	CC(C)n1nc(Cc2cccc3ccccc23)c(C#N)c1N	CID:24747154	phase I
BRD-K11671649	CCn1nc(Cc2cccc3ccccc23)c(C#N)c1N	CID:24747155	phase I
BRD-K01602319	NC(=O)c1ccccc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:24747156	phase I
BRD-K37372998	Cn1c(=O)c([N+][O-])c(N)n(Cc2ccccc2)c1=S	CID:24747160	phase I
BRD-K44652183	Cn1c(=O)c2nc(CCCC(=O)O)[nH]c2n(Cc3ccccc3)c1=S	CID:24747161	phase I
BRD-K49749421	COc1cc(/C=C\2/N=C(OC2=O)c3ccccc3)c(F)cc1OCc4ccccc4	CID:24747162	phase I
BRD-K79522882	COc1cccc(CN2C(=O)[C@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)c1	CID:24747169	phase I
BRD-K97666802	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccccc5F)C2=O	CID:24747172	phase I
BRD-K16947188	CCOc1ccccc1Nc2nc(nc(n2)N3CCOCC3)N4CCCC4	CID:24747173	phase I
BRD-K22546959	Cc1cc(Nc2cc(Cl)nc(Sc3ccc(NC(=O)C4CC4)cc3)n2)[nH]n1	CID:24747174	phase I
BRD-K66438357	OCCNc1nc(Nc2ccccc2C(F)(F)F)nc(n1)N3CCCC3	CID:24747175	phase I
BRD-K59429476	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccccc5Cl)C2=O	CID:24747176	phase I
BRD-K70415218	CCCCOc1ccc(Cl)cc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:24747177	phase I
BRD-K97926541	COc1ccccc1Nc2nc(NCCCCO)nc(n2)N3CCCC3	CID:24747178	phase I
BRD-K61923775	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccccc5)C2=O	CID:24747179	phase I
BRD-K54503842	CC1(C)N2[C@@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccc(F)cc5)C2=O	CID:24747180	phase I
BRD-K91264756	CCCOc1ccc(Cl)cc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:24747181	phase I
BRD-K27630941	COc1ccccc1Nc2nc(nc(n2)N3CCOCC3)N4CCCC4	CID:24747182	phase I
BRD-K99494806	CC1(C)N2[C@@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccccc5F)C2=O	CID:24747183	phase I
BRD-K71671265	Cc1ccccc1CN2C(=O)[C@@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O	CID:24747188	phase I
BRD-K17915279	Cc1ccc(CN2C(=O)[C@@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)cc1	CID:24747189	phase I
BRD-K93875449	Cn1nc(Cc2cccc3ccccc23)c(C#N)c1N	CID:24747191	phase I
BRD-K78481586	Nc1[nH]nc(Cc2cccc3ccccc23)c1C#N	CID:24747192	phase I
BRD-K44929916	COc1ccccc1CN2C(=O)[C@@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O	CID:24747193	phase I
BRD-K65741250	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(C2=O)c5cc(F)ccc5F	CID:24747194	phase I
BRD-K82566177	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccco5)C2=O	CID:24747195	phase I
BRD-K84284996	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5ccc(F)cc5)C2=O	CID:24747196	phase I
BRD-K02113384	Cc1ccccc1CN2C(=O)[C@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O	CID:24747209	phase I
BRD-K67880862	CC1(C)N2[C@H](Cc3c1[nH]c4ccccc34)C(=O)N(C2=O)c5ccc(F)cc5F	CID:24747210	phase I
BRD-A24225650	CC(C)c1cn(C2OC(COC(=O)c3ccccc3)C(OC(=O)c4ccccc4)C2OC(=O)c5ccccc5)c(=O)[nH]c1=O	CID:24747211	phase I
BRD-K22006123	C1CCN(C1)c2nc(Nc3ccccc3)nc(n2)N4CCOCC4	CID:24747212	phase I
BRD-K90207583	Cc1ccc(CN2C(=O)[C@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)cc1	CID:24747213	phase I
BRD-K57480017	OC(=O)c1ccc(cc1)c2noc(n2)c3ccc(F)cc3	CID:24747214	phase I
BRD-K33086940	COc1cccc(CN2C(=O)[C@@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)c1	CID:24747215	phase I
BRD-K91818252	OC(=O)c1ccc(cc1)c2noc(n2)c3ccccc3Cl	CID:24747216	phase I
BRD-K56977905	COc1ccc(cc1O)C2(CCN(CC2)C(=O)C)c3cccc(O)c3OC	CID:24747217	phase I
BRD-K11260407	COc1cc(F)c(cc1OC)C(=O)NC(C)(C)CO	CID:24747218	phase I
BRD-K45675241	COc1cc(ccc1O)c2cc[n+](C)cc2	CID:24747220	phase I
BRD-K23623013	COC(=O)C1=C(C[C@@H]2CC[C@H]1N2C(=O)NC3CCCCC3)c4cc5ccccc5s4	CID:24747230	phase I
BRD-K62493605	CC1(C)N2[C@@H](Cc3c1[nH]c4ccccc34)C(=O)N(Cc5cccc(F)c5)C2=O	CID:24747231	phase I
BRD-K44878494	Cc1c(CCCC(=O)O)sc(N)c1C(=O)c2cccc(c2)C(F)(F)F	CID:24747232	phase I
BRD-K37021324	OCCNc1nc(Nc2cc(Cl)ccc2OC3CCCC3)nc(n1)N4CCCC4	CID:24747241	phase I
BRD-K92419424	COc1ccc(cc1)c2nc(no2)c3ccc(cc3)C(=O)O	CID:24747242	phase I
BRD-K71172276	COc1ccc(Nc2nc(nc(n2)N3CCOCC3)N4CCCC4)cc1	CID:24747245	phase I
BRD-K49967178	OC(=O)c1ccc(cc1)c2noc(n2)c3ccccc3C(F)(F)F	CID:24747246	phase I
BRD-K53142391	COc1cccc(c1)c2nc(no2)c3ccc(cc3)C(=O)O	CID:24747270	phase I
BRD-K72676786	CSc1ncc(CNc2cc(ccc2C)[N+](=O)[O-])c(N)n1	CID:24747271	phase I
BRD-K95934080	Cc1cccc(CN2C(=O)[C@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)c1	CID:24747272	phase I
BRD-K82115270	COc1ccccc1CN2C(=O)[C@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O	CID:24747273	phase I
BRD-K29198371	Cc1cccc(CN2C(=O)[C@@H]3Cc4c([nH]c5ccccc45)C(C)(C)N3C2=O)c1	CID:24747274	phase I
BRD-K13046565	CC(C)(C)OC(=O)N[C@@H](Cc1ccc(cc1)C(=O)c2ccccc2)C(=O)NCC#C	CID:24747275	phase I
BRD-K60202068	CC(=O)Nc1ccccc1Nc2nc(NCCO)nc(n2)N3CCCC3	CID:24747276	phase I
BRD-A21481508	COc1ccc(CC2NCCC3=CC(=O)CCC23)cc1O	CID:24747278	phase I
BRD-K72883421	OC(=O)c1ccc(cc1)c2noc(n2)c3cccc(c3)C(F)(F)F	CID:24747338	phase I
BRD-K63157263	COc1ccccc1c2nc(no2)c3ccc(cc3)C(=O)O	CID:24747339	phase I
BRD-K18761689	OC(=O)c1ccc(cc1)c2noc(n2)c3cccc(F)c3	CID:24747340	phase I
BRD-K22831754	OC(=O)c1ccc(cc1)c2noc(n2)c3ccccc3F	CID:24747341	phase I
BRD-K86231656	CN(C(=O)OC(C)(C)C)c1ccc(cc1)c2nc3ccccc3s2	CID:24747342	phase I
BRD-K88742110	COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1	CID:24753719	phase I
BRD-K10405667	CCC(=O)N1CCc2cc(ccc12)c3csc(NC(=O)c4ccco4)n3	CID:24761960	phase I
BRD-K58033748	O=C(CCNS(=O)(=O)c1cccc2nsnc12)N1CCN(CC1)c1ccncc1	CID:24768606	phase I
BRD-K48923948	CCS(=O)(=O)N[C@@H]1C[C@@]2(C)O[C@]1(C)[C@H]1[C@@H]2C(=O)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F	CID:24768935	phase I
BRD-K75295174	COc1cc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2OC)ccc1C(O)=O	CID:24771867	phase I
BRD-K19796430	C[C@H]1CN(C[C@@H](C)O1)c1ccc(NC(=O)c2cccc(-c3ccc(OC(F)(F)F)cc3)c2C)cn1	CID:24775005	phase I
BRD-K19477839	Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1	CID:24779724	phase I
BRD-K13049116	C[C@]1(CCCN1c1nc(Nc2cc(n[nH]2)C2CC2)c2cccn2n1)C(=O)Nc1ccc(F)nc1	CID:24785538	phase I
BRD-K40738845	CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc(N)c2Cl)c(F)c1	CID:24794418	phase I
BRD-K81783531	CC1CCC(CC1)C(=O)N(C1CCC(O)CC1)c1cc(sc1C(O)=O)C#CC(C)(C)C	CID:24798764	phase I
BRD-A70311631	Cc1cc(C)n(CC(=O)NC2CCCc3c2cnn3c4ccc(C)c(C)c4)n1	CID:24820091	phase I
BRD-K44227013	CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1	CID:24826799	phase I
BRD-K61248029	COC(=O)N1N(C(=O)OC)[C@](CC(C)C)(C1=O)c2ccccc2	CID:24856224	phase I
BRD-K25662647	COC(=O)N1N(C(=O)OC)[C@](C(C)C)(C1=O)c2ccc(OC)cc2	CID:24856237	phase I
BRD-K92895207	COC(=O)N1N(C(=O)OC)[C@](C(C)C)(C1=O)c2ccccc2	CID:24856238	phase I
BRD-K34452916	COC(=O)N1N(C(=O)OC)[C@](C2CCCC2)(C1=O)c3ccccc3	CID:24856313	phase I
BRD-K54256913	CN1CCN(CC1)c1ccc(Nc2ncc3c(n2)n(-c2cccc(n2)C(C)(C)O)n(CC=C)c3=O)cc1	CID:24856436	phase I
BRD-K16554956	OP(O)(=O)C(F)(F)c1cc2cc(ccc2cc1Br)C#N	CID:24857885	phase I
BRD-K97447442	ONC(=O)CCCCCCC(=O)Nc1ccc(F)cc1	CID:24861442	phase I
BRD-K25737009	OC(=O)c1ccc(cc1)c2ccc3cc(c(O)cc3c2)C4(CC5CC6CC(C5)C4)C6	CID:24868309	phase I
BRD-A20968261	NC(CC(=O)Nc1ccc(Oc2cc(F)c(F)cc2Br)cc1)C(=O)O	CID:24868316	phase I
BRD-K50325075	C(NC(c1ccccc1)(c1ccccc1)c1ccccc1)c1cccnc1	CID:24868317	phase I
BRD-K71670746	OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O	CID:24868572	phase I
BRD-K51683034	CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(CC=C)C1=O)c4ccc(OCCCO)cc4	CID:24868580	phase I
BRD-K06405410	OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O	CID:24868581	phase I
BRD-K72451865	CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5	CID:24868588	phase I
BRD-K33606495	OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCCN3CCOCC3	CID:24868685	phase I
BRD-K62169556	OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(C(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6	CID:24868692	phase I
BRD-K00816165	C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4	CID:24868992	phase I
BRD-K96167523	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(NC(=O)C)cc43	CID:24869058	phase I
BRD-K07023879	COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(I)cc43	CID:24869062	phase I
BRD-K01614657	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(C)c4c3cc(C)cc4Br	CID:24869085	phase I
BRD-K73155123	COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(C)c5c3cc(C)cc5Br	CID:24869094	phase I
BRD-A56702968	C[C@H]1O[C@@H](OC2CC(O)C(C(O)CC(=O)CC(O)C(O)CCC(O)CC(O)CC(O)CC(=O)OC(C)C(C)C(O)C(C)C=CC=CCCC=CC=CC=CC=C2)C(=O)O)[C@@H](O)[C@@H](N)[C@@H]1O	CID:24871028	phase I
BRD-K22096725	Cc1ccc(cc1Nc1cncc(c1)C(N)=O)C(=O)Nc1cccc(c1)C(F)(F)F	CID:24875320	phase I
BRD-K68191783	Cc1cn(cn1)-c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(NC(=O)c2ccno2)c1	CID:24880028	phase I
BRD-K93918653	CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1	CID:24889392	phase I
BRD-K56277358	Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1	CID:24901704	phase I
BRD-K03618428	CC(C)n1nc(-c2ccc3cn[nH]c3c2)c2c(N)ncnc12	CID:24905203	phase I
BRD-K69840642	CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO	CID:24951314	phase I
BRD-K68065987	NC1(CCC1)c1ccc(cc1)-c1nc2ccn3c(n[nH]c3=O)c2cc1-c1ccccc1	CID:24964624	phase I
BRD-K82746043	CC1(C)CCC(=C(CN2CCN(CC2)c2ccc(cc2)C(=O)NS(=O)(=O)c2ccc(N[C@H](CCN3CCOCC3)CSc3ccccc3)c(c2)S(=O)(=O)C(F)(F)F)C1)c1ccc(Cl)cc1	CID:24978538	phase I
BRD-K28774715	[O-][N+](=O)c1ccccc1C(=O)NNC(=O)c2csc(n2)N3CCOCC3	CID:24980924	phase I
BRD-K71512533	Clc1cccc(NC(=O)Nc2ncc(CCNc3ncnc4ccsc34)s2)c1	CID:24995524	phase I
BRD-K27520107	CCOC(=O)N1CCC(CC1)NCCNC(=O)c2cccc(F)c2	CID:25010829	phase I
BRD-K69231968	CCOC(=O)N1CCC(CC1)NCCNC(=O)c2ccc(F)c(F)c2	CID:25010835	phase I
BRD-K45446451	OC(C1CCN(CC1)C(=O)Oc1ccc(cc1)[N+]([O-])=O)(c1ccc2OCOc2c1)c1ccc2OCOc2c1	CID:25021165	phase I
BRD-K14991967	OC(=O)c1ccc(cc1C1CCCC1)-c1c[nH]c2ncc(cc12)-c1ccccc1	CID:25022668	phase I
BRD-K02581333	CC(C)(c1ccc(NS(=O)(=O)C(F)(F)F)cc1)c2ccc(cc2)C(C)(C)c3cccc(NS(=O)(=O)C(F)(F)F)c3	CID:25035942	phase I
BRD-K41220170	COC(=O)CCCCCCC(=O)N/N=C/c1ccc(o1)S(=O)(=O)O	CID:25042413	phase I
BRD-K50311478	Cc1ccc(cc1)S(=O)(=O)N[C@H](Cc2ccccc2)C(=O)CCl	CID:25044204	phase I
BRD-K23353440	Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc4[nH]ccc4c3)C2	CID:25044703	phase I
BRD-K65464785	Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCn3cc(CN4[C@@H](COCC4=O)c5ccccc5)nn3	CID:25047668	phase I
BRD-K87737963	O=C(NCC#N)c1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1	CID:25062766	phase I
BRD-K90705745	CN(C(=O)CSc1ccc(nn1)-c1ccccc1)c1nc(C)cs1	CID:25067404	phase I
BRD-K59470558	CCc1nccn1CC(=O)c1ccc(O)c(O)c1	CID:25067484	phase I
BRD-K89190195	Cc1nccn1CC(=O)c2ccc(O)c(O)c2	CID:25067492	phase I
BRD-K59794046	Cc1nc2ccccc2n1CC(=O)c3ccc(O)c(O)c3	CID:25067496	phase I
BRD-A77349281	CCCCCCCCCCCCCCCC(=O)C1C(=O)OC(CO)C1=O	CID:25067890	phase I
BRD-A28412351	COc1cccc2c1O[C@H]3C(=O)CC[C@H]4CN(C)CCC342	CID:25079076	phase I
BRD-K61662457	O=C(NCCN1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc2ccccc2c1	CID:25105715	phase I
BRD-K94287906	O=C(NCc1cccc2ccsc12)c3cccs3	CID:25105719	phase I
BRD-K99605820	O=C(NCc1cccc2ccccc12)c3cccs3	CID:25105722	phase I
BRD-A89494828	COc1cccc(c1)C1c2c(Oc3ncn(-c4ccccc4)c(=N)c13)ccc1ccccc21	CID:25109888	phase I
BRD-A42737819	COc1ccccc1C1c2c(Oc3ncn(-c4ccccc4)c(=N)c13)ccc1ccccc21	CID:25109893	phase I
BRD-A86792397	COc1cccc(C2c3c(Oc4ncn(-c5ccccc5)c(=N)c24)ccc2ccccc32)c1OC	CID:25109896	phase I
BRD-A75301702	N=c1c2C(c3ccccc3)c3c(Oc2ccn1Cc1ccccc1)ccc1ccccc31	CID:25109904	phase I
BRD-A85891951	O=C(Cc1ccccc1)Nc2ncnc3Oc4ccc5ccccc5c4C(c6ccccc6)c23	CID:25109906	phase I
BRD-A82197375	CCOC(=O)CCC(=O)Nc1ncnc2Oc3ccc4ccccc4c3C(c5ccccc5)c12	CID:25109908	phase I
BRD-A08610364	CCOC(=O)CCCC(=O)Nc1ncnc2Oc3ccc4ccccc4c3C(c5ccccc5)c12	CID:25109909	phase I
BRD-A60784279	O=C(Nc1ncnc2Oc3ccc4ccccc4c3C(c5ccccc5)c12)c6ccccc6	CID:25109910	phase I
BRD-A11095214	O=C(N(C(=O)c1ccccc1)c2ncnc3Oc4ccc5ccccc5c4C(c6ccccc6)c23)c7ccccc7	CID:25109911	phase I
BRD-A11512624	CCOC(=O)CC(=O)Nc1ncnc2Oc3ccc4ccccc4c3C(c5ccccc5)c12	CID:25109912	phase I
BRD-K65111630	Clc1ccc(CNC(=O)C[C@@H]2C\C=C\CCC(=O)O[C@@H](CNC2=O)c2ccccc2)cc1	CID:25109985	phase I
BRD-K35010406	ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)c2ccccc2	CID:25118059	phase I
BRD-K04833372	CCc1cc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2ccc(OC)c(c2)C(=O)Nc2c(F)cccc2F)c(OC)cc1N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O	CID:25124816	phase I
BRD-K71266197	Nc1c2C(=O)c3ccccc3C(=O)c2c(Nc2cccc3ccccc23)cc1S(O)(=O)=O	CID:25124826	phase I
BRD-K53972329	N#CC[C@H](C1CCCC1)n1cc(cn1)-c1ncnc2[nH]ccc12	CID:25126798	phase I
BRD-K20697946	CCc1ccc(cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1)S(=O)(=O)c1ccccc1	CID:25147679	phase I
BRD-K26818574	COc1cc2nc(nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC)N1CCCN(C)CC1	CID:25150857	phase I
BRD-K68997413	FC(F)(F)c1ccc(Oc2cccc(CC3CCN(CC3)C(=O)Nc3cccnc3)c2)nc1	CID:25154867	phase I
BRD-K83213911	O=C(Nc1ccccc1)N2CCC(Cc3cnc4ccccc4c3)CC2	CID:25154868	phase I
BRD-K26257340	Cc1c(cccc1[N+](=O)[O-])C(=O)NNC(=O)c2csc(n2)N3CCOCC3	CID:25161537	phase I
BRD-K97365803	Nc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1	CID:25181195	phase I
BRD-K37160541	[O-][N+](=O)c1c(Br)cccc1\N=c1\ssnc1Cl	CID:25181240	phase I
BRD-K78659596	CC(C)C[C@H](NC(=O)CNC(=O)c1cc(Cl)ccc1Cl)B(O)O	CID:25183872	phase I
BRD-K08451418	COc1cc2ncn(-c3cc(OCc4ccc(cc4)S(C)(=O)=O)c(s3)C(N)=O)c2cc1OC	CID:25190912	phase I
BRD-K04853698	C1CN(CCN1)c1ccc(cc1)-c1cnc2c(cnn2c1)-c1ccnc2ccccc12	CID:25195294	phase I
BRD-K32330832	Nc1ncnc2n([C@@H]3O[C@H](COCc4ccc(cc4)C#N)[C@@H](O)[C@H]3O)c(NCc3ccc(Cl)c(Cl)c3)nc12	CID:25195348	phase I
BRD-K37885773	NCC1CCN(CC1)c1nccc(n1)-c1ccc2ccccc2c1	CID:25199517	phase I
BRD-K13146765	CSc1nc(nc(n1)c2ccccc2)C(C)C	CID:25199536	phase I
BRD-K23027438	Cc1cnn(CC(=O)c2ccc(O)c(O)c2)c1	CID:25199538	phase I
BRD-K69241845	CN1C(=O)C(NCCc2ccc(F)cc2)=C(C1=O)c1c(C)[nH]c2ccccc12	CID:25209788	phase I
BRD-K57044355	Fc1cccc(F)c1S(=O)(=O)N1CCN(CC1)S(=O)(=O)c1ccc2OCCOc2c1	CID:25210493	phase I
BRD-K06569345	COc1cc(ccc1Nc1nc(N)c(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)C(N)=O	CID:25226117	phase I
BRD-K16621777	C[C@@](O)(COc1ccc(cc1)C#N)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F	CID:25226380	phase I
BRD-K93747373	CNC(=O)c1ccc(Nc2cc(Nc3ccccc3S(=O)(=O)C(C)C)c3cc[nH]c3n2)nc1	CID:25226483	phase I
BRD-K61053657	CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1CCC[C@H]1C(=O)Nc1cccc2ncccc12	CID:25241666	phase I
BRD-K90736214	O=S(=O)(N1CCN(CC1)S(=O)(=O)c1ccc2OCCOc2c1)c1ccccc1	CID:25243713	phase I
BRD-K50746423	Fc1ccc(cc1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243714	phase I
BRD-K30779094	Cn1ccc2cc(ccc12)S(=O)(=O)N1CCN(CC1)S(=O)(=O)c1c(F)cccc1F	CID:25243719	phase I
BRD-K89786160	Fc1cccc(F)c1S(=O)(=O)N1CCN(CC1)S(=O)(=O)c1ccc2OCCCOc2c1	CID:25243721	phase I
BRD-K00430421	Fc1cccc(F)c1S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3	CID:25243723	phase I
BRD-K12579869	C[C@@H]1CN(CCN1S(=O)(=O)c2ccc3OCCOc3c2)S(=O)(=O)c4c(F)cccc4F	CID:25243728	phase I
BRD-K71169984	Fc1cccc(F)c1S(=O)(=O)N2CCN(CC2)C(=O)c3ccc4OCCOc4c3	CID:25243729	phase I
BRD-K99423120	C[C@@H]1CN(CCN1S(=O)(=O)c2c(F)cccc2F)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243730	phase I
BRD-K68826049	C[C@H]1CN(CCN1S(=O)(=O)c2ccc3OCCOc3c2)S(=O)(=O)c4c(F)cccc4F	CID:25243735	phase I
BRD-K46869836	C[C@H]1CN(CCN1S(=O)(=O)c2c(F)cccc2F)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243736	phase I
BRD-K94381355	Fc1cccc(F)c1S(=O)(=O)C2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243744	phase I
BRD-K04279026	O=S(=O)(N1CCN(CC1)S(=O)(=O)c2ccccn2)c3ccc4OCCOc4c3	CID:25243746	phase I
BRD-K69834151	Cc1cc2n(C)c3c(cnn(Cc4ccc(F)cc4F)c3=O)c2s1	CID:25243750	phase I
BRD-K39507792	Fc1cccc(F)c1S(=O)(=O)N2CCC(CC2)NS(=O)(=O)c3ccc4OCCOc4c3	CID:25243774	phase I
BRD-K59024967	Fc1cccc(F)c1S(=O)(=O)N2CCCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243775	phase I
BRD-K69304050	FC(F)(F)c1cccc(c1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243777	phase I
BRD-K95168667	Fc1cccc(F)c1S(=O)(=O)NCC2CN(C2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243778	phase I
BRD-K40175949	Fc1cccc(F)c1S(=O)(=O)N2CC(CNS(=O)(=O)c3ccc4OCCOc4c3)C2	CID:25243779	phase I
BRD-A81389811	Fc1cccc(F)c1S(=O)(=O)NC2CCN(C2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25243780	phase I
BRD-K90692502	Fc1cccc(F)c1S(=O)(=O)NCCCNS(=O)(=O)c2ccc3OCCOc3c2	CID:25243781	phase I
BRD-K77032321	Fc1cccc(F)c1S(=O)(=O)NCCCCCNS(=O)(=O)c2ccc3OCCOc3c2	CID:25243782	phase I
BRD-K20923001	Fc1cccc(F)c1S(=O)(=O)NCCCCCCNS(=O)(=O)c2ccc3OCCOc3c2	CID:25243783	phase I
BRD-K26906367	Fc1cccc(F)c1S(=O)(=O)NCCNS(=O)(=O)c2ccc3OCCOc3c2	CID:25243784	phase I
BRD-A83993876	Fc1cccc(F)c1S(=O)(=O)N2CCC(C2)NS(=O)(=O)c3ccc4OCCOc4c3	CID:25243785	phase I
BRD-K77762110	Fc1cccc(F)c1S(=O)(=O)NCCCCNS(=O)(=O)c2ccc3OCCOc3c2	CID:25243786	phase I
BRD-K54674709	Cc1cc2n(C)c3c(=O)n(ncc3c2s1)c4ccccc4	CID:25243787	phase I
BRD-K45256078	Cn1c2ccsc2c3ncn(Cc4ccccc4F)c(=O)c13	CID:25243788	phase I
BRD-A02241946	CC(O)c1cc2n(C)c3c(=O)n(Cc4ccccc4F)ncc3c2s1	CID:25243794	phase I
BRD-A89049230	COc1ccc(cc1COc1ccc(NC(C)=O)cc1)C1Nc2cccc(O)c2C(=O)N1Cc1ccccc1	CID:25246343	phase I
BRD-A45498368	CNC(=O)Nc1ccc(cc1)-c1nc(N2CC3CCC(C2)O3)c2cnn(C3CCC4(CC3)OCCO4)c2n1	CID:25260757	phase I
BRD-K69932463	COc1ccc(cc1CO)-c1ccc2c(nc(nc2n1)N1CCOC[C@@H]1C)N1CCOC[C@@H]1C	CID:25262965	phase I
BRD-K11469942	CCC(=O)O[C@@]1([C@H](C)C[C@@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]12C)C(=O)SCF	CID:25320895	phase I
BRD-K65971331	COc1cccc(CN(C)C(=O)c2ccc(OCc3cn4cccc(C)c4n3)cc2)c1OC	CID:25330436	phase I
BRD-K13077924	COc1cc(\C=C\C)ccc1OCc1cn2cccc(C)c2n1	CID:25405916	phase I
BRD-K53325797	Cc1cccn2cc(COc3ccc(cc3)C#N)nc12	CID:25529404	phase I
BRD-K20032655	O=C(NNC(=O)c1ccccc1)c2csc(n2)c3ccccc3	CID:25668960	phase I
BRD-K34495954	[O-][N+](=O)c1ccccc1S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:25886838	phase I
BRD-K48654774	COc1ccc(cc1)C(=O)C1CCN(CC1)c1ncnc2sccc12	CID:26043913	phase I
BRD-K73709114	Cc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1nc(nc2ccccc12)-c1cccs1	CID:26450846	phase I
BRD-K42489623	COc1ccc(cc1)c2csc3ncnc(Sc4nnnn4C)c23	CID:26471808	phase I
BRD-K92310201	C[C@@H]1C[C@H]2[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]2(C)[C@@]1(OC(=O)c1ccco1)C(=O)CCl	CID:26849680	phase I
BRD-K40758391	C/C(=N\NC(=O)C1CCCC1)/c2ccc(NC(=O)C(F)(F)F)cc2	CID:26871482	phase I
BRD-A23637604	C[C@]1(O)CC[C@H]2[C@@H]3CC[C@H]4CC(=O)C(C[C@]4(C)[C@H]3CC[C@]12C)C=O	CID:27806705	phase I
BRD-K31374463	CC(=O)O[C@H]1[C@H](C[C@H]2[C@H]3CC[C@H]4C[C@H](OC(C)=O)[C@H](C[C@]4(C)[C@@H]3CC[C@]12C)N1CCCCC1)[N+]1(C)CCCCC1	CID:28280238	phase I
BRD-K08229828	CC[C@H](C)C(=O)O[C@H]1CCC=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CCO3)[C@@H]12	CID:29922189	phase I
BRD-K71552035	CC(=O)O[C@@]1(CC[C@@H]2[C@@H]3C=C(C)C4=CC(=O)CC[C@@H]4[C@@H]3CC[C@]12C)C(C)=O	CID:29926609	phase I
BRD-K74741811	CC[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@H]34)[C@H]1CC[C@@]2(O)C#C	CID:29985980	phase I
BRD-K77547920	Cn1nnnc1Sc2ncnc3scc(c4ccc(Br)cc4)c23	CID:31055126	phase I
BRD-K07403598	Nc1ccc2NCN=C(NCCc3ccc(Oc4ccccc4)cc3)c2c1	CID:35026803	phase I
BRD-K88551539	COC(=O)c1ccc(O)c(NC(=O)COc2ccc(cc2)C2C3CC4CC(C3)CC2C4)c1	CID:35028748	phase I
BRD-K56446541	FC(F)(F)c1ccc(Cl)c(NC(=O)COC(=O)CNC(=O)C2CCCCC2)c1	CID:35647030	phase I
BRD-K90177246	OC1C(=O)C(=O)C(O)C(=O)C1=O	CID:36689751	phase I
BRD-K60965159	Cc1ccc(NS(=O)(=O)c2cc3OCC(=O)Nc3cc2Br)cc1C	CID:38888103	phase I
BRD-K05926469	Nc1cccc2C(=O)N(Cc12)[C@@H]1CCC(=O)NC1=O	CID:40461270	phase I
BRD-K84443303	CCC(=O)O[C@@]1([C@@H](C)C[C@H]2[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]12C)C(=O)CCl	CID:40469415	phase I
BRD-K45149020	CC(=O)OCC(=O)[C@@]12OC3(CCCC3)O[C@@H]1C[C@H]1[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]21C	CID:40469418	phase I
BRD-K38159897	C[C@H](CCC(O)=O)[C@H]1CC[C@H]2[C@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@@H]3CC[C@]12C	CID:40469454	phase I
BRD-K54264597	C[C@]12CC[C@@H]3[C@@H](C=CC4=CC(=O)CC[C@]34C)[C@H]1CC[C@@]2(O)CCC(O)=O	CID:40469463	phase I
BRD-K82624463	C[C@]12CC(=O)[C@@H]3[C@H](CCC4=CC(=O)C=C[C@]34C)[C@@H]1CC[C@]2(O)C(=O)CO	CID:40469477	phase I
BRD-K13027675	C[C@H]1C[C@H]2[C@H]3CC[C@](O)(C(C)=O)[C@@]3(C)C[C@H](O)[C@]2(F)[C@@]2(C)C=CC(=O)C=C12	CID:40469506	phase I
BRD-K34817515	CC1(C)O[C@@H]2C[C@H]3[C@H]4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:40469508	phase I
BRD-K30207000	C[C@@H]1C[C@H]2[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)COC(C)=O	CID:40469526	phase I
BRD-K00835182	C[C@H]1C[C@H]2[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:40469540	phase I
BRD-K81774264	C[C@@H]1C[C@@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO	CID:40469854	phase I
BRD-K18316707	COc1cc(C)cc(OC)c1[C@@H]1C=C(C)CC[C@H]1C(C)=C	CID:40469923	phase I
BRD-K93367411	OC(=O)[C@@H]1CCCC[C@@H]1C(=O)N1CCc2ccccc2[C@H]1CN1C(=O)c2ccccc2C1=O	CID:40482356	phase I
BRD-K32403583	CC[C@H](C)C(=O)O[C@H]1CCC=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@H]12	CID:40488233	phase I
BRD-K32793530	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@H]1C[C@@H](O)[C@@H]2O	CID:40488277	phase I
BRD-K18739469	CC(=O)N/N=C(\C)/c1ccc(NC(=O)C2CC2)cc1	CID:40532013	phase I
BRD-K90241462	CC(=O)O[C@@]1(CC[C@@H]2[C@H]3C=C(Cl)C4=CC(=O)CC[C@]4(C)[C@@H]3CC[C@]12C)C(C)=O	CID:40532410	phase I
BRD-K56411643	COC(=O)[C@@H]1Cc2c([nH]c3ccccc23)[C@H](N1C(=O)CCl)c4ccc(cc4)C(=O)OC	CID:40911229	phase I
BRD-K89059493	O=C(C1CCN(CC1)c1ncnc2sccc12)c1ccccc1	CID:41724711	phase I
BRD-K46212057	C[C@@H](c1ncncc1F)[C@@](O)(Cn1cncn1)c1ccc(F)cc1F	CID:42052020	phase I
BRD-K36665199	Fc1ccc(c(F)c1)-n1ncc2[C@H](CCCc12)NC(=O)c1ccccn1	CID:42288155	phase I
BRD-K98439022	Fc1ccc(c(F)c1)-n1ncc2[C@@H](CCCc12)NC(=O)c1ccccn1	CID:42288156	phase I
BRD-K05323277	COc1cc(ccc1Nc2ncc3N(C)C(=O)CCN(C4CCC(O)CC4)c3n2)C(=O)NC5CCN(C)CC5	CID:42601363	phase I
BRD-K56343971	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F	CID:42611257	phase I
BRD-K87634564	COc1ccc(Br)c(/C=N/NC(=O)CCCCCC(=O)NO)c1	CID:42618298	phase I
BRD-K02526760	OC[C@H](Cc1ccccc1)Nc1nc(Oc2ccc3CCCc3c2)nc2n(Cc3ccc(cc3)-c3ccccc3)cnc12	CID:42623900	phase I
BRD-K83151319	Oc1ccc(-c2csc(Nc3ccc4OCOc4c3)n2)c(O)c1	CID:42626479	phase I
BRD-K34294489	COc1ccccc1NCc1nc2ccccc2n1C	CID:42628057	phase I
BRD-K46805185	COc1cc(ccc1Nc1ncc2N(C(C)C)C(=O)CCN(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	CID:42628535	phase I
BRD-K19056367	Cc1cc(-c2ccc(F)cc2)n2ncc(-c3ccccc3)c2n1	CID:42640807	phase I
BRD-K97936712	Fc1ccc(CC2CCN(CC2)c2ncnc3sccc23)cc1	CID:42640808	phase I
BRD-K33680967	Fc1ccc(cc1)C(=O)C1CCN(CC1)c1ncnc2sccc12	CID:42640809	phase I
BRD-K01089529	Cc1cc(-c2ccncc2)n2ncc(-c3ccccc3)c2n1	CID:42640811	phase I
BRD-K03449891	COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)ccnc2cc1OCCCN1CCOCC1	CID:42642645	phase I
BRD-A00763758	COc1cc(ccc1O)C(O)C(C)N	CID:43209100	phase I
BRD-A02333338	CC1C2NC[C@@H](C)C[C@H]2O[C@@]31CC[C@H]4[C@@H]5CC=C6C[C@@H](O)CC[C@]6(C)[C@H]5CC4=C3C	CID:44118238	phase I
BRD-K13605477	Cc1cc(NC(=O)CS(=O)(=O)c2cn(Cc3cccc(Cl)c3)c3ccccc23)no1	CID:44129591	phase I
BRD-K58772419	C[C@@H](Nc1ccccc1C(O)=O)c1cc(C)cn2c1nc(cc2=O)N1CCOCC1	CID:44137675	phase I
BRD-K53561341	CCN1CCN(CC1)C(=O)Cc1ccc(Nc2ncc(F)c(Nc3ccc(cc3)C(=O)Nc3ccccc3Cl)n2)cc1	CID:44139710	phase I
BRD-K24705176	COc1cc(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c(OC)cc1Cl	CID:44141936	phase I
BRD-K42021584	COc1ccc(CC2CCN(CC2)c2ncnc3sccc23)cc1	CID:44141937	phase I
BRD-K82580504	Clc1ccc(cc1)C(=O)C1CCN(CC1)c1ncnc2sccc12	CID:44141938	phase I
BRD-K63550534	OC(=O)CN1C(=O)N/C(=C\c2cccn2c3ccc(cc3)P(=O)(O)O)/C1=O	CID:44142042	phase I
BRD-K26767475	CN(Cc1ccco1)c2ncnc3ccc(cc23)c4ccc5n(C)ccc5c4	CID:44142043	phase I
BRD-K07101857	Cc1cccc(CNc2ncnc3ccc(cc23)c4ccccc4Cl)c1	CID:44142044	phase I
BRD-K76933066	COc1cccc(c1)c2ccc3ncnc(NCc4cccc(C)c4)c3c2	CID:44142045	phase I
BRD-K00028814	Cc1cccc(CNc2ncnc3ccc(cc23)c4ccc5OCCOc5c4)c1	CID:44142046	phase I
BRD-K41797142	Clc1ccccc1c2ccc3ncnc(NCc4cccs4)c3c2	CID:44142047	phase I
BRD-K58318000	Clc1cccc(c1)c2ccc3ncnc(NCc4cccs4)c3c2	CID:44142048	phase I
BRD-K92932331	C(Nc1ncnc2ccc(cc12)c3cccnc3)c4cccs4	CID:44142049	phase I
BRD-K70977695	Cc1cccc(c1)c2ccc3ncnc(NCc4cccs4)c3c2	CID:44142050	phase I
BRD-K49630153	Cn1ccc2cc(ccc12)c3ccc4ncnc(NCc5cccs5)c4c3	CID:44142051	phase I
BRD-K51140856	C(Nc1ncnc2ccc(cc12)c3ccc4OCCOc4c3)c5cccs5	CID:44142052	phase I
BRD-K46645809	C(Nc1ncnc2ccc(cc12)c3ccc4OCCOc4c3)c5ccc6OCOc6c5	CID:44142053	phase I
BRD-K50532160	C(Nc1ncnc2ccc(cc12)c3ccc4OCCOc4c3)c5cccnc5	CID:44142054	phase I
BRD-K92458042	Fc1cccc(CNc2ncnc3ccc(cc23)c4ccc5OCOc5c4)c1	CID:44142055	phase I
BRD-K82140622	Clc1cccc(c1)c2ccc3ncnc(NCc4cccnc4)c3c2	CID:44142056	phase I
BRD-K63181962	Cc1cccc(c1)c2ccc3ncnc(NCc4cccnc4)c3c2	CID:44142057	phase I
BRD-K81751891	C(Nc1ncnc2ccc(cc12)c3ccc4OCOc4c3)c5cccnc5	CID:44142058	phase I
BRD-K88269385	Clc1ccccc1c2ccc3ncnc(NCc4ccc5OCOc5c4)c3c2	CID:44142059	phase I
BRD-K56024573	COc1cccc(c1)c2ccc3ncnc(NCc4ccc5OCOc5c4)c3c2	CID:44142060	phase I
BRD-K80126354	C(Nc1ncnc2ccc(cc12)c3cccnc3)c4ccc5OCOc5c4	CID:44142061	phase I
BRD-K30443205	C(Nc1ncnc2ccc(cc12)c3ccoc3)c4ccc5OCOc5c4	CID:44142062	phase I
BRD-K13842623	Cc1csc(CNc2ncnc3ccc(cc23)c4ccccc4Cl)c1	CID:44142063	phase I
BRD-K27440500	Cc1csc(CNc2ncnc3ccc(cc23)c4cccc(Cl)c4)c1	CID:44142064	phase I
BRD-K93975822	COc1cccc(c1)c2ccc3ncnc(NCc4cc(C)cs4)c3c2	CID:44142065	phase I
BRD-K15054362	Cc1csc(CNc2ncnc3ccc(cc23)c4cccnc4)c1	CID:44142066	phase I
BRD-K70503895	Cc1csc(CNc2ncnc3ccc(cc23)c4ccc5OCOc5c4)c1	CID:44142067	phase I
BRD-K70646792	Cc1csc(CNc2ncnc3ccc(cc23)c4ccc5OCCOc5c4)c1	CID:44142068	phase I
BRD-K57037351	Cc1csc(CNc2ncnc3ccc(cc23)c4ccoc4)c1	CID:44142069	phase I
BRD-K45763312	CN1CCN(CC1)C2CCN(Cc3ccc(O)c4ncccc34)CC2	CID:44142070	phase I
BRD-K08857385	CC(=O)Nc1oc(nc1C#N)c2cccc3ccccc23	CID:44142073	phase I
BRD-K86565213	C=CCNc1oc(nc1C#N)C2CCCC2	CID:44142074	phase I
BRD-K00541156	Cc1ccc(CSc2nnc(o2)c3cccc4ccccc34)cc1	CID:44142075	phase I
BRD-K68158690	Nc1oc(nc1C#N)c2cccc3ccccc23	CID:44142076	phase I
BRD-A21812217	ON1C(Nc2ccccc2C1=O)c3ccc(o3)c4ccc(C#N)cc4	CID:44142077	phase I
BRD-A56831909	ON1C(Nc2ccccc2C1=O)c3ccc(o3)c4ccccc4F	CID:44142078	phase I
BRD-A68820570	ON1C(Nc2ccccc2C1=O)c3ccc(o3)c4cccs4	CID:44142079	phase I
BRD-A99911370	ON1C(Nc2ccccc2C1=O)c3ccc(o3)c4cccc(F)c4	CID:44142080	phase I
BRD-A61825514	ON1C(Nc2ccccc2C1=O)c3ccc(o3)c4ccc(cc4)C(F)(F)F	CID:44142081	phase I
BRD-K95080525	CN(C)c1ccc(cc1)C(=O)OCC#CCSc2nnc(o2)c3cccc4ccccc34	CID:44142082	phase I
BRD-K81300454	COc1ccccc1C(=O)OCC#CCSc2nnc(o2)c3cccc4ccccc34	CID:44142083	phase I
BRD-K40577058	O=C(OCC#CCSc1nnc(o1)c2cccc3ccccc23)c4ccc5ccccc5c4	CID:44142084	phase I
BRD-K88511582	O=C(OCC#CCSc1nnc(o1)c2cccc3ccccc23)c4c[nH]cn4	CID:44142085	phase I
BRD-K35790918	O=C(OCC#CCSc1nnc(o1)c2cccc3ccccc23)c4cccc5[nH]ccc45	CID:44142086	phase I
BRD-K95037415	COc1ccc(cc1OC2CCCC2)C3=Nn4c(nnc4SC3)c5ccccc5OC	CID:44142087	phase I
BRD-K96704648	COc1ccc(cc1OC2CCCC2)C3=Nn4c(nnc4SC3)c5ccccc5Cl	CID:44142088	phase I
BRD-K57238941	COc1ccc(OC)c(c1)c2nnc3SCC(=Nn23)c4ccc(OC)c(OC5CCCC5)c4	CID:44142090	phase I
BRD-K49712247	COc1ccc(cc1OCC2CC2)C3=Nn4c(nnc4SC3)c5ccccc5OC	CID:44142091	phase I
BRD-K18861610	COc1ccc(cc1OCC2CC2)C3=Nn4c(nnc4SC3)c5ccccc5F	CID:44142092	phase I
BRD-K65242613	COc1ccc(cc1OCC2CC2)C3=Nn4c(nnc4SC3)c5ccccc5Cl	CID:44142093	phase I
BRD-K97534490	COc1ccc(OC)c(c1)c2nnc3SCC(=Nn23)c4ccc(OC)c(OCC5CC5)c4	CID:44142094	phase I
BRD-K96456313	COc1ccccc1c2nnc3SCC(=Nn23)c4ccc(OC(F)F)c(OCC5CC5)c4	CID:44142095	phase I
BRD-K39318886	FC(F)Oc1ccc(cc1OCC2CC2)C3=Nn4c(nnc4SC3)c5ccccc5Cl	CID:44142096	phase I
BRD-K39866321	FC(F)Oc1ccc(cc1OCC2CC2)C3=Nn4c(nnc4SC3)c5ccccc5F	CID:44142097	phase I
BRD-K55127335	COc1ccc(OC)c(c1)c2nnc3SCC(=Nn23)c4ccc(OC(F)F)c(OCC5CC5)c4	CID:44142098	phase I
BRD-A93975555	COc1ccc(cc1OC2CCOC2)C3=Nn4c(nnc4SC3)c5ccccc5OC	CID:44142099	phase I
BRD-A38936397	COc1ccc(cc1OC2CCOC2)C3=Nn4c(nnc4SC3)c5ccccc5Cl	CID:44142100	phase I
BRD-A43640821	COc1ccc(cc1OC2CCOC2)C3=Nn4c(nnc4SC3)c5ccccc5F	CID:44142101	phase I
BRD-A01999384	COc1ccc(cc1OC2CCOC2)C3=Nn4c(nnc4SC3)c5ccccc5C(F)(F)F	CID:44142102	phase I
BRD-A16820783	COc1ccc(OC)c(c1)c2nnc3SCC(=Nn23)c4ccc(OC)c(OC5CCOC5)c4	CID:44142103	phase I
BRD-K41059137	Clc1cccc(c1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:44142104	phase I
BRD-K60729220	Brc1cccc(c1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:44142105	phase I
BRD-K50985433	O=S(=O)(N1CCN(CC1)S(=O)(=O)c2ccc3OCCOc3c2)c4ccco4	CID:44142106	phase I
BRD-K95117060	Cc1ccc(F)c(Cn2cnc3n(ncc3c2=O)C(C)(C)C)c1Cl	CID:44142107	phase I
BRD-K85670329	CC(C)(C)n1ncc2c(=O)n(Cc3ccccc3Br)cnc12	CID:44142108	phase I
BRD-K04676863	Cc1cc(F)cc(C)c1Cn2cnc3n(ncc3c2=O)C(C)(C)C	CID:44142109	phase I
BRD-K80822897	CC(C)(C)n1ncc2c(=O)n(Cc3cccc(Cn4cnc5n(ncc5c4=O)C(C)(C)C)c3F)cnc12	CID:44142110	phase I
BRD-K35737468	CC(C)(C)n1ncc2c(=O)n(Cc3cc(F)c(Cl)cc3Cl)cnc12	CID:44142111	phase I
BRD-K33159591	Cc1ccc(Cl)c(Cn2cnc3n(ncc3c2=O)C(C)(C)C)c1F	CID:44142112	phase I
BRD-K89563433	CC(C)(C)n1ncc2c(=O)n(Cc3c(Cl)cccc3Br)cnc12	CID:44142113	phase I
BRD-K13580623	CNS(=O)(=O)c1ccc2CCc3ccc(cc3C(=O)c2c1)S(=O)(=O)NC	CID:44142114	phase I
BRD-K24051260	Fc1cc(F)cc(Nc2nc(Cl)nc(NC3CCCC3)n2)c1	CID:44142115	phase I
BRD-K22210218	FC(F)CNc1nc(Nc2cc(F)cc(F)c2)nc(C#N)n1	CID:44142116	phase I
BRD-K77239206	FC(F)(F)c1ccc(Cl)c(NC(=O)Cn2cc(CNC(=O)C3CCCCC3)nn2)c1	CID:44142117	phase I
BRD-K46170844	Clc1ccccc1NC(=O)COC(=O)CNC(=O)c2ccccc2Cl	CID:44142118	phase I
BRD-K32580836	FC(F)(F)c1ccc(Cl)c(NC(=O)COC(=O)CNC(=O)c2ccccc2Cl)c1	CID:44142119	phase I
BRD-K73567619	O=C(NNC(=O)c1cc2ccccc2[nH]1)OCc3ccccc3	CID:44142120	phase I
BRD-K11611839	O=C(NNC(=O)c1nc2ccccc2[nH]1)OCc3ccccc3	CID:44142121	phase I
BRD-A04392722	CC(C)(C)OC(=O)NCC(=O)NNC(=O)C(C(=O)OCc1ccccc1)c2ccccc2	CID:44142123	phase I
BRD-K29140223	Clc1cccc(Nc2nc(C#N)nc3n(cnc23)C4CCCC4)c1	CID:44142124	phase I
BRD-A99218607	OC1c2ccccc2CCc3ccc(cc13)S(=O)(=O)C(F)(F)F	CID:44142125	phase I
BRD-K47490989	Fc1cccc(F)c1S(=O)(=O)N2C[C@@H]3C[C@H]2CN3S(=O)(=O)c4ccc5OCCOc5c4	CID:44142126	phase I
BRD-K46555875	CCOC(=O)c1cccc(c1)n2cccc2/C=C/3\NC(=O)N(CC(=O)O)C3=O	CID:44142127	phase I
BRD-K62412498	CCOC(=O)c1ccc(cc1)n2cccc2/C=C/3\NC(=O)NC3=O	CID:44142128	phase I
BRD-K19735876	COc1ccccc1c2csc3ncnc(Sc4nnnn4C)c23	CID:44142129	phase I
BRD-K56593336	COc1cccc(c1)c2csc3ncnc(Sc4nnnn4C)c23	CID:44142130	phase I
BRD-K75999307	Cn1nnnc1Sc2ncnc3scc(c4cccc(F)c4)c23	CID:44142131	phase I
BRD-K51377689	Cn1nnnc1Sc2ncnc3scc(c4ccccc4C(F)(F)F)c23	CID:44142132	phase I
BRD-K36354764	Cn1nnnc1Sc2ncnc3scc(c4cccc(c4)C(F)(F)F)c23	CID:44142133	phase I
BRD-K28366633	Cn1nnnc1Sc2ncnc3scc(c4ccc(cc4)C(F)(F)F)c23	CID:44142134	phase I
BRD-K61718261	Cn1nnnc1Sc2ncnc3scc(c4ccccc4Br)c23	CID:44142135	phase I
BRD-K07259155	Cn1nnnc1Sc2ncnc3scc(c4cccc(Br)c4)c23	CID:44142136	phase I
BRD-K55487965	Cn1nnnc1Sc2ncnc3scc(c4ccccc4Cl)c23	CID:44142137	phase I
BRD-K82732294	Cn1nnnc1Sc2ncnc3scc(c4ccc(C#N)cc4)c23	CID:44142138	phase I
BRD-K44366801	Cn1nnnc1Sc2ncnc3scc(c4ccc(cc4)[N+](=O)[O-])c23	CID:44142139	phase I
BRD-K88707333	Cn1nnnc1Sc2ncnc3scc(c4ccc(cc4)c5ccccc5)c23	CID:44142140	phase I
BRD-K42455570	Cn1nnnc1Sc2ncnc3scc(c4ccc5OCOc5c4)c23	CID:44142141	phase I
BRD-K87726525	Cn1nnnc1Sc2ncnc3scc(c4ccsc4)c23	CID:44142143	phase I
BRD-K24156250	Cn1nnnc1Sc2ncnc3scc(c4cc5ccccc5o4)c23	CID:44142144	phase I
BRD-K42499654	Cn1nnnc1Sc2ncnc3scc(c4cccc5c6ccccc6sc45)c23	CID:44142145	phase I
BRD-K89224880	Cn1nnnc1Sc2ncnc3scc(c4ccc[nH]4)c23	CID:44142146	phase I
BRD-K62466453	CC(=O)c1ccccc1c2csc3ncnc(Sc4nnnn4C)c23	CID:44142147	phase I
BRD-K66037923	Cn1nnnc1Sc2ncnc3scc(c4cccc(c4)S(=O)(=O)C)c23	CID:44142148	phase I
BRD-K01834163	Cn1nnnc1Sc2ncnc3scc(c4cccc5ccccc45)c23	CID:44142149	phase I
BRD-K05359840	Cn1nnnc1Sc2ncnc3scc(Br)c23	CID:44142150	phase I
BRD-K44417704	CC(=O)N1CCN(CC1)c2ccc(NCc3ccco3)cc2	CID:44142151	phase I
BRD-K96740880	CC(=O)N1CCN(CC1)c2ccc(NCc3cccc(C)c3)cc2	CID:44142152	phase I
BRD-K47324077	CC(=O)N1CCN(CC1)c2ccc(NCc3ccc(Br)o3)cc2	CID:44142155	phase I
BRD-K74348865	Fc1cc(F)c(c(F)c1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3ccc4OCCOc4c3	CID:44142157	phase I
BRD-K57562268	CCn1cnc2c(NCCc3cccnc3)nc(C#N)nc12	CID:44142159	phase I
BRD-A03436432	COc1cccc(c1)S(=O)(=O)NC2CCN(C2)C#N	CID:44142160	phase I
BRD-A85712510	FC(F)(F)c1ccc(cc1)S(=O)(=O)NC2CCN(C2)C#N	CID:44142161	phase I
BRD-K96621343	FC(F)(F)c1ccc(cc1)S(=O)(=O)NC2CCN(CC2)C#N	CID:44142162	phase I
BRD-K12814321	C/C(=C\c1cc2ccccc2o1)/C3Nc4cccc5cccc(N3)c45	CID:44142164	phase I
BRD-K11928012	COc1cccc(Nc2ccc(cc2)N3CCCCC3)c1OC	CID:44142168	phase I
BRD-A43126523	CC(=O)NC(C1CC1)c2cc(Cl)c3cccnc3c2O	CID:44142346	phase I
BRD-A24021119	CC(=O)NC(c1cccs1)c2cc(F)c3cccnc3c2O	CID:44142351	phase I
BRD-K35254025	OC(=O)c1ccc(cc1)c2noc(n2)c3cccc(Cl)c3	CID:44142416	phase I
BRD-K24468827	CCn1cnc2c(Nc3cc(F)cc(F)c3)nc(C#N)nc12	CID:44143088	phase I
BRD-K39010473	FC(F)Cn1cnc2c(Nc3cc(F)cc(F)c3)nc(C#N)nc12	CID:44143089	phase I
BRD-K80070306	CCn1cnc2c(Nc3cccc(Cl)c3)nc(C#N)nc12	CID:44143090	phase I
BRD-K95789946	CCNc1nc(C#N)nc2n(cnc12)c3cc(F)cc(F)c3	CID:44143091	phase I
BRD-A62496920	O=C(CNC(=O)C1CCCCC1)OC(C(=O)c2ccccc2)c3ccccc3	CID:44143092	phase I
BRD-K56477805	Cc1nnc(N=c2ssnc2Cl)o1	CID:44143153	phase I
BRD-A74608937	CNC(C)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)Nc2ccc3ncccc3c2	CID:44143236	phase I
BRD-A97035593	CNC(C)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)NNc2ccccc2	CID:44143238	phase I
BRD-A05680309	CNC(C)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)NC2CCCc3ccccc23	CID:44143240	phase I
BRD-A69429454	CCC(NC(=O)C(C)NC)C(=O)N1CCCC1C(=O)NC2CCCc3ccccc23	CID:44143242	phase I
BRD-A69470004	CC(C)C(NC(=O)C(C)N)C(=O)N1CCCC1C(=O)NC(c2ccccc2)c3ccccc3	CID:44143244	phase I
BRD-K49468759	CCN1CCC(CC1)n1cc(CNc2cc(Cl)c3ncc(C#N)c(Nc4ccc(F)c(Cl)c4)c3c2)nn1	CID:44143370	phase I
BRD-A71009679	COc1ccc(cc1)C1CC(=NN1c1ccc(cc1)S(N)(=O)=O)c1cccc(OC)c1	CID:44143698	phase I
BRD-A86990971	Cc1cccc(c1)C1CC(=NN1c1ccc(cc1)S(N)(=O)=O)c1ccccc1	CID:44143700	phase I
BRD-A82096673	NS(=O)(=O)c1ccc(cc1)N1N=C(CC1c1cccc(Br)c1)c1ccccc1	CID:44143703	phase I
BRD-K50297939	COc1ccc(cc1OC)[C@H]2CC(=O)C=C(C2)c3cccc4c5ccccc5sc34	CID:44143772	phase I
BRD-K71427192	CC(C)[C@H](NC(=O)[C@H](C)N)C(=O)N[C@@H](C)C(=O)Nc1cccc2ccccc12	CID:44176347	phase I
BRD-K89014967	OC[C@@H](O)CNC(=O)c1ccncc1Nc1ccc(I)cc1F	CID:44187362	phase I
BRD-K78223772	Cc1ccc(C)n1-c1cccc(c1)-c1nn[nH]n1	CID:44197159	phase I
BRD-K30064966	Oc1cccc2cc(C(=O)Nc3cccc(c3)-c3cn4ccccc4n3)c(=O)oc12	CID:44197249	phase I
BRD-K46255814	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44202057	phase I
BRD-K45582470	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44202276	phase I
BRD-K98113345	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44202300	phase I
BRD-K52914903	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44202433	phase I
BRD-K85763971	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44202444	phase I
BRD-K77845911	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44202483	phase I
BRD-K02920722	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44202487	phase I
BRD-K07472106	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C	CID:44202494	phase I
BRD-K20138758	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44202501	phase I
BRD-K41775742	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44202529	phase I
BRD-K84293326	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44202569	phase I
BRD-K11778372	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44202572	phase I
BRD-K81068628	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44202599	phase I
BRD-K69791739	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44202600	phase I
BRD-K52801121	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44202691	phase I
BRD-K82137294	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44202729	phase I
BRD-K38698447	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44202744	phase I
BRD-K01229043	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44202844	phase I
BRD-K11612251	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44202876	phase I
BRD-K42161310	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44202878	phase I
BRD-K58141791	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)C(=O)Nc4ccccc4)[C@H](C)CN([C@H](C)CO)C(=O)Cc3c2)cc1	CID:44202935	phase I
BRD-K06476055	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44202943	phase I
BRD-K55179756	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44202980	phase I
BRD-A82590476	CN(Cc1ccccc1)C(=O)C(Cc2ccc3ccccc3c2)NC(=O)C4CCCN4C(=O)Nc5ccccc5[N+](=O)[O-]	CID:44208964	phase I
BRD-K77008974	COC(=O)Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cnn(C3CCN(CC3)C(=O)OC)c2n1	CID:44219749	phase I
BRD-K68783079	Cc1nc(CNc2ncnc3ccc(cc23)-c2ccc3OCOc3c2)cs1	CID:44223952	phase I
BRD-A96746500	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)C1CCCO1	CID:44223955	phase I
BRD-K58999277	C(Cc1ccco1)Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1	CID:44223965	phase I
BRD-K06217810	CN(Cc1csc(C)n1)c1ncnc2ccc(cc12)-c1ccc2OCOc2c1	CID:44223970	phase I
BRD-K59222562	CN(Cc1cccs1)c1ncnc2ccc(cc12)-c1ccc2OCOc2c1	CID:44223973	phase I
BRD-K86905031	Cc1occc1CNc1ncnc2ccc(cc12)-c1ccc2OCOc2c1	CID:44223974	phase I
BRD-K59705555	C1CN(CCC1Oc1ccccc1)c1ncnc2sccc12	CID:44224142	phase I
BRD-K10114046	OC1(Cc2ccccc2)CCN(CC1)c1ncnc2sccc12	CID:44224143	phase I
BRD-K74690444	O=C(C1CCN(CC1)c1ncnc2sccc12)c1cccs1	CID:44224144	phase I
BRD-K07398339	COc1ccc(cc1)S(=O)(=O)n1c(N)nc2ccccc12	CID:44229066	phase I
BRD-K87657228	Cc1ccc(cc1)S(=O)(=O)n1c(N)nc2cc(C)c(C)cc12	CID:44229067	phase I
BRD-K28610502	CCCN(CCC)c1nc(nc2ccccc12)N3CCCC3	CID:44229302	phase I
BRD-K30804015	CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F	CID:44237404	phase I
BRD-K04136539	OC(c1ccc(NS(=O)(=O)c2cccc3cccnc23)cc1)(C(F)(F)F)C(F)(F)F	CID:44237405	phase I
BRD-K71879957	COC(=O)c1sccc1S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F	CID:44237406	phase I
BRD-K53335770	COc1cccc(c1)S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F	CID:44237407	phase I
BRD-K63129749	OC(c1ccc(NS(=O)(=O)c2cccc3ccccc23)cc1)(C(F)(F)F)C(F)(F)F	CID:44237408	phase I
BRD-K99633092	OC(c1ccc(NS(=O)(=O)c2ccc(Cl)c3nonc23)cc1)(C(F)(F)F)C(F)(F)F	CID:44237409	phase I
BRD-K53855319	O=C(Nc1cc(CN2CCNCC2)cc(c1)-c1nc2ccccc2[nH]1)c1cnc2ccccc2n1	CID:44240264	phase I
BRD-K02735834	CSc1nccc(n1)-c1ccc(s1)S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F	CID:44241374	phase I
BRD-K67619794	OC(c1ccc(NC(=O)c2c(F)cccc2F)cc1)(C(F)(F)F)C(F)(F)F	CID:44241382	phase I
BRD-K40441731	OC(c1ccc(NC(=O)c2ccccc2C(F)(F)F)cc1)(C(F)(F)F)C(F)(F)F	CID:44241404	phase I
BRD-K98676510	OC(c1ccc(NS(=O)(=O)c2ccc(s2)-c2ccccn2)cc1)(C(F)(F)F)C(F)(F)F	CID:44241405	phase I
BRD-K82768082	OC(c1ccc(NS(=O)(=O)c2ccc(s2)-c2ccccc2)cc1)(C(F)(F)F)C(F)(F)F	CID:44241408	phase I
BRD-K74777906	COc1ccsc1S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F	CID:44241411	phase I
BRD-K40378749	OC(c1ccc(NC(=O)c2ccc(F)cc2Cl)cc1)(C(F)(F)F)C(F)(F)F	CID:44241416	phase I
BRD-K98079119	OC(c1ccc(NC(=O)c2ccc(F)cc2F)cc1)(C(F)(F)F)C(F)(F)F	CID:44241432	phase I
BRD-K68863575	OC(c1ccc(NS(=O)(=O)c2ccc(s2)S(=O)(=O)c2ccccc2)cc1)(C(F)(F)F)C(F)(F)F	CID:44241444	phase I
BRD-K82983587	Cc1cc(NC(=O)CS(=O)(=O)c2cn(Cc3cccc(c3)C(F)(F)F)c3ccccc23)no1	CID:44241483	phase I
BRD-K92020737	CCCN1CNc2c(C1)c(=O)[nH]c(=S)n2CCc1c(Cl)cccc1Cl	CID:44246374	phase I
BRD-K68833544	CCCN1CNc2c(C1)c(=O)[nH]c(=S)n2CCc1cccc(Cl)c1Cl	CID:44246394	phase I
BRD-K88761633	CCOC(=O)c1ccccc1S(=O)(=O)N1CCN(CC1)c1nc(nc2ccccc12)-c1cccs1	CID:44246455	phase I
BRD-K19973744	Cc1cc(C)cc(c1)S(=O)(=O)N1CCN(CC1)c1nc(nc2ccccc12)-c1cccs1	CID:44246456	phase I
BRD-K55972177	Cc1ccc(cc1)S(=O)(=O)C1CCN(CC1)c1nc(nc2ccccc12)-c1cccs1	CID:44246457	phase I
BRD-A11968133	COc1cccc(Cn2ncc3c4sc(cc4n(C)c3c2=O)S(C)=O)c1	CID:44246498	phase I
BRD-A18279961	Cn1c2cc(sc2c2cnn(Cc3cccc(N)c3)c(=O)c12)S(C)=O	CID:44246499	phase I
BRD-K91273791	Cn1c2cc(Br)sc2c3cnn(Cc4c(F)cccc4Cl)c(=O)c13	CID:44246512	phase I
BRD-K73004613	Cn1c2cc(Br)sc2c3cnn(Cc4ccc(F)cc4F)c(=O)c13	CID:44246514	phase I
BRD-K49562544	Cn1c2ccsc2c3ncn(Cc4ccc(F)cc4)c(=O)c13	CID:44246515	phase I
BRD-K69795440	CN(Cc1ccco1)Cc2ccc(O)c3ncccc23	CID:44246520	phase I
BRD-K04124609	CNC[C@H]1Oc2c(NS(=O)(=O)c3ccc(OC)cc3)cccc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44246547	phase I
BRD-A41020680	CN(C)[C@@H]1C2CC3Cc4c(ccc(O)c4C(=O)C3C(=O)[C@@]2(O)C(=O)C(C(=O)N)C1=O)N(C)C	CID:44246708	phase I
BRD-A49035384	CN(C)[C@H]1[C@@H]2[C@@H](O)[C@H]3C(C(=O)c4c(O)cccc4C3=C)C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O	CID:44246715	phase I
BRD-A88208128	CN(C)C1C2CC3C(C(=O)c4c(O)cccc4C3(C)O)C(=O)C2(O)C(=O)C(C(=O)N)C1=O	CID:44247471	phase I
BRD-K01926222	Cc1cc(NC(=O)CS(=O)(=O)c2cn(Cc3cccc(Br)c3)c3ccccc23)no1	CID:44247542	phase I
BRD-A84475555	Cc1cc(NC(=O)CS(=O)c2cn(Cc3cccc(Cl)c3)c3ccccc23)no1	CID:44247543	phase I
BRD-K20151898	COc1cc2CCN3C[C@H](CC(C)C)[C@@H](O)C[C@H]3c2cc1OC	CID:44249892	phase I
BRD-K55938002	Fc1ccc(OCC(=O)Nc2nnc(o2)-c2ccc(F)c(F)c2)c(Cl)c1	CID:44251479	phase I
BRD-K42140106	Cc1ccc(cc1C)-c1nnc(NC(=O)COc2ccc(F)cc2Cl)o1	CID:44251485	phase I
BRD-K18573821	NC(=O)CN1CC[C@@H](NC(=O)[C@@H]2CCCN2)C1=O	CID:44281634	phase I
BRD-A64489120	NCC(O)c1cc(O)c(O)cc1[N+]([O-])=O	CID:44287635	phase I
BRD-A25037258	COC(=O)C1C2CC[C@H](C[C@@H]1c1ccc(I)cc1)N2C	CID:44295709	phase I
BRD-A77098556	CNC(=O)[C@H]1O[C@H]([C@@H](O)C1O)n1cnc2c(NCc3cccc(I)c3)nc(Cl)nc12	CID:44348677	phase I
BRD-A55484088	Oc1ccc2CC3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C(=O)\C(C[C@@]35O)=C\c1ccccc1	CID:44369694	phase I
BRD-K72561299	CC(C)[C@H]1NC(=O)[C@@H](NC(=O)c2ccc(C)c3oc4c(C)c(=O)c(N)c(C(=O)N[C@H]5[C@H](C)OC(=O)[C@H](C(C)C)N(C)C(=O)CN(C)C(=O)[C@@H]6CCCN6C(=O)[C@H](NC5=O)C(C)C)c4nc23)[C@H](C)OC(=O)[C@H](C(C)C)N(C)C(=O)CN(C)C(=O)[C@@H]2CCCN2C1=O	CID:44415057	phase I
BRD-K08417745	CCc1ccccc1NC(=O)CSC(=O)NNC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C	CID:44456237	phase I
BRD-K35191571	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)c1csc2ccccc12	CID:44460110	phase I
BRD-K47147974	Clc1ccsc1C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460111	phase I
BRD-K35133769	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)c1ccsc1	CID:44460112	phase I
BRD-K58674774	Fc1cc(cc(F)c1F)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460113	phase I
BRD-K07872006	Fc1ccc(cc1F)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460114	phase I
BRD-K90996982	Fc1ccc(C(=O)OCC#CCSc2nnc(o2)-c2cccc3ccccc23)c(F)c1	CID:44460115	phase I
BRD-K29500995	Fc1ccccc1C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460116	phase I
BRD-K59139557	CS(=O)(=O)c1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460117	phase I
BRD-K89546934	Fc1ccc(cn1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460118	phase I
BRD-K95561591	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)c1ccncc1	CID:44460119	phase I
BRD-K79381128	FC(F)(F)Sc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460120	phase I
BRD-K76612204	FC(F)Oc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460121	phase I
BRD-K60218670	FC(F)(F)Oc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460122	phase I
BRD-K73285375	FC(F)(F)c1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460123	phase I
BRD-K24461445	FC(F)(F)c1cc(ccc1Cl)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460124	phase I
BRD-K01806521	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)C1CC1	CID:44460125	phase I
BRD-K14975149	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)C1CCC1	CID:44460126	phase I
BRD-K96083840	O=C(OCC#CCSc1nnc(o1)-c1cccc2ccccc12)C1CCCC1	CID:44460127	phase I
BRD-K24127443	Fc1cccc(c1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460128	phase I
BRD-K42681396	FC(F)(F)c1cccc(c1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ccccc12	CID:44460129	phase I
BRD-K54657957	O=C(OCC#CCSc1nnc(o1)-c1ccc2ccccc2c1)c1cccs1	CID:44460131	phase I
BRD-K56307118	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1ccco1	CID:44460132	phase I
BRD-K41666683	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccs1	CID:44460133	phase I
BRD-K78206606	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1ccccc1F	CID:44460134	phase I
BRD-K66448556	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1ccccc1Cl	CID:44460135	phase I
BRD-K26211296	COc1ccccc1-c1nnc(SCC#CCOC(=O)c2ccc(F)cc2)o1	CID:44460136	phase I
BRD-K98288062	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc(F)c1	CID:44460137	phase I
BRD-K74596421	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1ccc(F)cc1	CID:44460138	phase I
BRD-K64314806	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1ccc(Cl)cc1	CID:44460139	phase I
BRD-K47917680	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1cccc2ncccc12	CID:44460141	phase I
BRD-K04516579	Oc1ccc(Nc2ccccc2F)c2cccnc12	CID:44460156	phase I
BRD-K82024442	Oc1ccc(NS(=O)(=O)c2ccccc2F)c2cccnc12	CID:44460157	phase I
BRD-K49094915	Oc1ccc(CNc2ccc(cc2F)C(F)(F)F)c2cccnc12	CID:44460159	phase I
BRD-K93155496	Oc1ccc(CNc2cccnc2)c2cccnc12	CID:44460164	phase I
BRD-K55722623	Oc1ccc(-c2ccccc2F)c2cccnc12	CID:44460166	phase I
BRD-A01973626	CCC(=O)NC(c1ccco1)c1cc(Br)c2cccnc2c1O	CID:44460172	phase I
BRD-A54632525	CC(=O)NC(c1cccs1)c1cc(Br)c2cccnc2c1O	CID:44460175	phase I
BRD-A95795120	CCC(=O)NC(c1cccs1)c1cc([N+]([O-])=O)c2cccnc2c1OC	CID:44460176	phase I
BRD-K14027855	Oc1ccc(\C=C\c2ccccc2F)c2cccnc12	CID:44460186	phase I
BRD-K52321331	Oc1ccc(\C=C\c2c(F)cccc2F)c2cccnc12	CID:44460187	phase I
BRD-K14788918	Oc1ccc(CCc2c(F)cccc2F)c2cccnc12	CID:44460189	phase I
BRD-K39757396	Oc1ccc(Oc2ccccc2F)c2cccnc12	CID:44460190	phase I
BRD-A89047717	Fc1cccc(c1)-n1c(=O)c2ccccc2s1=O	CID:44462705	phase I
BRD-K09951645	CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F	CID:44462760	phase I
BRD-K46872340	Cc1cc(C)c2c(ccn(CC(=O)N3CCN(CC3)c3ccccc3)c2=O)n1	CID:44473128	phase I
BRD-A35020550	CC1CN(CCN1c1cccc(C)c1)C(=O)COc1noc2nc(C)cc(C)c12	CID:44473132	phase I
BRD-K61314889	O=C(Nc1cccc2cccnc12)c1ccc(cc1)N1C(=O)[C@H]2[C@@H]3C[C@@H](C=C3)[C@H]2C1=O	CID:44483163	phase I
BRD-K65369159	Cc1ccc(c(C)c1)-n1sc2cc(F)ccc2c1=O	CID:44483164	phase I
BRD-A64228451	CC1C(=O)[C@H]2O[C@H]2C(=O)C1=O	CID:44483234	phase I
BRD-A10420615	CC(=O)C1C(=O)[C@@H]2[C@@H]3[C@@H](Cc4cccc5[nH]cc3c45)C(C)(C)N2C1=O	CID:44483253	phase I
BRD-K78599730	CCCC[C@@H](C)/C=C(\C)/C=C(\C)/C(=O)NC1=C[C@@](O)(\C=C\C=C\C=C\C(=O)NC2C(=O)CCC2=O)[C@@H]3O[C@@H]3C1=O	CID:44483259	phase I
BRD-A18419789	COc1cc(cc(OC)c1O)[C@H]2[C@@H]3C(OCC3=O)C(OC4OC5COC(C)OC5C(O)C4O)c6cc7OCOc7cc26	CID:44483274	phase I
BRD-K64245000	CC(C)c1onc(c1COc2ccc(C=Cc3cccc(c3)C(=O)O)c(Cl)c2)c4c(Cl)cccc4Cl	CID:44483281	phase I
BRD-K67352070	CCOc1cncc(C=CCCNC)c1	CID:44483287	phase I
BRD-A49680073	CC(C)(O)/C=C/C(=O)[C@](C)(O)C1[C@H](O)C[C@@]2(C)[C@@H]3CC=C4C(CC(=O)C(=O)C4(C)C)[C@]3(C)C(=O)C[C@@]12C	CID:44483311	phase I
BRD-K08890269	NC(=O)NN=Cc1ccc(Oc2ccc(F)cc2)cc1	CID:44483319	phase I
BRD-K38477985	CC(C)(C)c1cc(C=C(C#N)[N+]#[C-])cc(c1O)C(C)(C)C	CID:44483329	phase I
BRD-K06024458	CCCCCC=CCC=CCC=CCC=CCCCC(=O)NCCCC(=O)O	CID:44483333	phase I
BRD-A38898897	CC(C)C1[C@H]2[C@@H](CCN2C(=O)/C=C/CN3CCCCC3)N(C1=O)S(=O)(=O)C	CID:44483335	phase I
BRD-A59943784	CC1CC2C3CC(F)C4=CC(=O)C=CC4(C)C3(F)C(O)CC2(C)C1(CC(=O)CO)C(=O)SCF	CID:44483336	phase I
BRD-A22713669	CC1(C)C2C(=NC1=O)c3ccccc3C(=O)C2=O	CID:44483339	phase I
BRD-A72596465	CCOC(=O)NCC(Cc1ccc(OCCc2nc(oc2C)c3ccccc3)cc1)NC(=CC(=O)c4ccc(cc4)C(F)(F)F)C	CID:44483340	phase I
BRD-K86727142	CCCCCCCCCCCC1C(=O)C(=O)CC(=O)C1=O	CID:44483355	phase I
BRD-K96041033	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44483393	phase I
BRD-K00801367	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44483418	phase I
BRD-K19322034	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44483434	phase I
BRD-K72449498	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44483436	phase I
BRD-K50558304	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44483439	phase I
BRD-K03644600	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44483449	phase I
BRD-K76559855	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44483463	phase I
BRD-K80058142	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44483487	phase I
BRD-K46604793	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44483515	phase I
BRD-K36895979	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44483523	phase I
BRD-K70115829	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44483532	phase I
BRD-K64255844	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44483541	phase I
BRD-K58946638	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44483542	phase I
BRD-K10232869	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44483562	phase I
BRD-K81574109	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44483569	phase I
BRD-K70638773	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44483604	phase I
BRD-K81131579	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44483616	phase I
BRD-K88488723	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44483643	phase I
BRD-K06898969	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44483658	phase I
BRD-K25835363	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44483661	phase I
BRD-K74767048	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44483690	phase I
BRD-K02315366	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44483698	phase I
BRD-K71138616	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44483723	phase I
BRD-K50777342	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44483742	phase I
BRD-K54925167	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44483750	phase I
BRD-K72587701	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@@H](C)[C@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@H](C)CO	CID:44483758	phase I
BRD-K32021722	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44483763	phase I
BRD-K20824632	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44483794	phase I
BRD-K40692824	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44483801	phase I
BRD-K80602561	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44483807	phase I
BRD-K66952385	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44483817	phase I
BRD-K24565544	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44483821	phase I
BRD-K49923618	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44483826	phase I
BRD-K67519589	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44483827	phase I
BRD-K12402761	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44483832	phase I
BRD-K55630970	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44483837	phase I
BRD-K53946803	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)c4ccncc4)cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44483849	phase I
BRD-K81941590	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44483863	phase I
BRD-K55216557	CNC[C@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44483865	phase I
BRD-K03486902	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)c4ccncc4)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44483875	phase I
BRD-K53594827	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44483876	phase I
BRD-K33010769	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44483885	phase I
BRD-K29335396	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44483907	phase I
BRD-K85736239	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44483908	phase I
BRD-K31569005	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44483910	phase I
BRD-K09253654	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44483914	phase I
BRD-K42054363	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44483917	phase I
BRD-K04733502	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44483925	phase I
BRD-K56726453	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Cc3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44483932	phase I
BRD-K78009480	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44483933	phase I
BRD-K53359044	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc(F)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44483938	phase I
BRD-K68765796	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44483939	phase I
BRD-K92047490	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44483940	phase I
BRD-K84091085	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44483944	phase I
BRD-K11759662	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44483946	phase I
BRD-K90256762	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44483952	phase I
BRD-K26849279	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44483957	phase I
BRD-K80718156	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44483963	phase I
BRD-K81592585	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44483977	phase I
BRD-K46692335	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44483980	phase I
BRD-K48036219	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44483993	phase I
BRD-K99465084	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44484005	phase I
BRD-K63385089	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44484010	phase I
BRD-K12411950	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44484018	phase I
BRD-K57119046	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44484034	phase I
BRD-K20718732	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44484048	phase I
BRD-K39758243	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44484052	phase I
BRD-K48863671	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44484062	phase I
BRD-K06397242	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44484065	phase I
BRD-K73832524	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44484081	phase I
BRD-K25608435	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44484104	phase I
BRD-K20597651	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44484129	phase I
BRD-K80723690	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)Cc4ccc5OCOc5c4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44484185	phase I
BRD-K76925500	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44484201	phase I
BRD-K09327126	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44484206	phase I
BRD-K59788643	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44484212	phase I
BRD-K40439253	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44484220	phase I
BRD-K21636276	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc(cc4)c5ccccc5)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:44484222	phase I
BRD-K37083752	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc(cc4)c5ccccc5)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44484225	phase I
BRD-K20824593	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44484239	phase I
BRD-K34130171	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44484245	phase I
BRD-K32568627	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44484267	phase I
BRD-K42197878	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44484270	phase I
BRD-K52208857	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44484274	phase I
BRD-K82210103	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44484277	phase I
BRD-K51849212	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:44484281	phase I
BRD-K28184645	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44484287	phase I
BRD-K34094942	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44484295	phase I
BRD-K36490574	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44484296	phase I
BRD-K40623364	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44484297	phase I
BRD-K12601591	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44484302	phase I
BRD-K35628245	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44484331	phase I
BRD-K43111300	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44484332	phase I
BRD-K63077891	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44484343	phase I
BRD-K68989144	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44484345	phase I
BRD-K79259004	COc1ccc(CN(C)C[C@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44484364	phase I
BRD-K42968246	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44484382	phase I
BRD-K20863480	COc1ccc(CN(C)C[C@@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44484391	phase I
BRD-K82504171	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44484438	phase I
BRD-K81060234	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44484464	phase I
BRD-K19729690	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44484466	phase I
BRD-K65160467	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44484478	phase I
BRD-K39624960	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44484483	phase I
BRD-K59024795	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)Oc3ccc(cc3CC1=O)N(C)C	CID:44484501	phase I
BRD-K02811477	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44484511	phase I
BRD-K84876223	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3cn(CCCC1=O)nn3	CID:44484512	phase I
BRD-K12584650	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44484513	phase I
BRD-K66555134	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44484515	phase I
BRD-K58034811	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44484516	phase I
BRD-K40241713	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)OCc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44484522	phase I
BRD-K51740186	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44484523	phase I
BRD-K72773058	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44484525	phase I
BRD-K67314051	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44484526	phase I
BRD-K52540534	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44484528	phase I
BRD-K50605719	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44484531	phase I
BRD-K91899208	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44484534	phase I
BRD-K29279625	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc3OCCCOc23)OCc4cn(CCCC1=O)nn4	CID:44484536	phase I
BRD-K00863274	COc1ccccc1CN(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3	CID:44484538	phase I
BRD-K20037743	COc1ccccc1CN(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3	CID:44484539	phase I
BRD-K49335566	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44484543	phase I
BRD-K08121566	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ncc(cc4C1=O)c5cc6ccccc6o5	CID:44484545	phase I
BRD-K53868452	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)C(=O)Nc4c(C)noc4C)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1OC	CID:44484551	phase I
BRD-K93303857	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44484555	phase I
BRD-K21152218	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44484568	phase I
BRD-K18794550	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44484569	phase I
BRD-K64668459	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44484570	phase I
BRD-K95891443	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44484579	phase I
BRD-K81249836	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44484589	phase I
BRD-K57589644	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44484591	phase I
BRD-K13306582	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44484592	phase I
BRD-K84139072	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44484605	phase I
BRD-K78800374	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44484616	phase I
BRD-K44261129	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44484675	phase I
BRD-K02150184	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44484705	phase I
BRD-K14875361	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44484708	phase I
BRD-K87430974	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44484712	phase I
BRD-K43298786	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44484733	phase I
BRD-K46625537	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44484785	phase I
BRD-K34182570	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44484793	phase I
BRD-K55683015	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44484798	phase I
BRD-K39151050	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44484862	phase I
BRD-K65134192	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44484881	phase I
BRD-K01737880	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc5OCOc5c4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44484893	phase I
BRD-K38891183	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44484911	phase I
BRD-K80818838	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44484916	phase I
BRD-K55322029	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44484927	phase I
BRD-K21458727	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44484946	phase I
BRD-K15219339	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44484956	phase I
BRD-K84128874	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44484959	phase I
BRD-K79426639	COc1ccc(CN(C)C[C@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44485018	phase I
BRD-K27622376	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44485030	phase I
BRD-K82524003	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44485039	phase I
BRD-K80819715	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44485047	phase I
BRD-K61900762	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3cn(CCCC1=O)nn3	CID:44485049	phase I
BRD-K94672699	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3cn(CCCC1=O)nn3	CID:44485050	phase I
BRD-K52371706	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44485051	phase I
BRD-K59870400	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44485055	phase I
BRD-K45028867	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44485056	phase I
BRD-K33832590	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44485057	phase I
BRD-K55035262	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44485058	phase I
BRD-K40199965	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44485059	phase I
BRD-K66035321	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44485060	phase I
BRD-K45663104	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44485061	phase I
BRD-K95805172	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)OCc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44485063	phase I
BRD-K84505894	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44485065	phase I
BRD-K16671107	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44485068	phase I
BRD-K20013327	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44485069	phase I
BRD-K13765840	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44485070	phase I
BRD-K22482035	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44485072	phase I
BRD-K12497208	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44485074	phase I
BRD-K85979978	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cn(CCCC1=O)nn3	CID:44485075	phase I
BRD-K22033912	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cn(CCCC1=O)nn3	CID:44485076	phase I
BRD-K02229102	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44485077	phase I
BRD-K37545156	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44485078	phase I
BRD-K61485275	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44485079	phase I
BRD-K65147077	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44485080	phase I
BRD-K95323941	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44485081	phase I
BRD-K67155745	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc3OCCCOc23)OCc4cn(CCCC1=O)nn4	CID:44485082	phase I
BRD-K22790182	CNC[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@H](C)CO)nn2	CID:44485085	phase I
BRD-K16561280	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44485087	phase I
BRD-K39599822	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485098	phase I
BRD-K61465460	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44485108	phase I
BRD-K34394296	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44485109	phase I
BRD-K38103660	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44485114	phase I
BRD-K30523950	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485115	phase I
BRD-K59248078	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44485117	phase I
BRD-K80954162	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485120	phase I
BRD-K31260488	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44485125	phase I
BRD-K45695271	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44485135	phase I
BRD-K11006288	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44485140	phase I
BRD-K31788299	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCCCC[C@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44485144	phase I
BRD-K73059376	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44485145	phase I
BRD-K31367750	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44485146	phase I
BRD-K77987635	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44485164	phase I
BRD-K05917849	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44485165	phase I
BRD-K40734828	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44485174	phase I
BRD-K46284961	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:44485175	phase I
BRD-K36620425	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4CC1=O	CID:44485177	phase I
BRD-K25436320	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44485182	phase I
BRD-K20479120	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO)N(C)C	CID:44485200	phase I
BRD-K62242359	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44485233	phase I
BRD-K16127898	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44485243	phase I
BRD-K48058738	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44485269	phase I
BRD-K61442593	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44485283	phase I
BRD-K48672996	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc(cc4)C(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:44485289	phase I
BRD-K37557400	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44485312	phase I
BRD-K63368502	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485319	phase I
BRD-K84860580	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44485323	phase I
BRD-K50280607	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44485340	phase I
BRD-K60239116	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44485343	phase I
BRD-K57180092	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C1=O	CID:44485355	phase I
BRD-K11480730	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44485360	phase I
BRD-K58421169	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44485423	phase I
BRD-K99017327	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44485456	phase I
BRD-K47786739	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485465	phase I
BRD-K71742078	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44485525	phase I
BRD-K35719087	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44485530	phase I
BRD-K03634222	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44485537	phase I
BRD-K09729851	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44485547	phase I
BRD-K51400578	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44485559	phase I
BRD-K06388802	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44485563	phase I
BRD-K96433222	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44485578	phase I
BRD-K10055851	COc1ccc(CN(C)C[C@@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44485596	phase I
BRD-K21421563	COc1ccc(CN(C)C[C@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44485610	phase I
BRD-K79532217	CNC[C@H]1Oc2c(NS(=O)(=O)c3ccc(OC)cc3)cccc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44485612	phase I
BRD-K91124206	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44485650	phase I
BRD-K57293132	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44485655	phase I
BRD-K83725960	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44485683	phase I
BRD-K89361242	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44485687	phase I
BRD-K83399162	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44485690	phase I
BRD-K31752292	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(cc2CC(=O)N(C[C@@H]1C)[C@@H](C)CO)N(C)C	CID:44485716	phase I
BRD-K08123827	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44485733	phase I
BRD-K63017817	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44485739	phase I
BRD-K17360472	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44485743	phase I
BRD-K75291656	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44485745	phase I
BRD-K47380281	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44485746	phase I
BRD-K73170797	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44485747	phase I
BRD-K91201009	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44485748	phase I
BRD-K15505145	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44485749	phase I
BRD-K44843438	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)OCc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44485750	phase I
BRD-K95323755	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44485753	phase I
BRD-K75707803	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4cn(CCCC1=O)nn4	CID:44485754	phase I
BRD-K25631986	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44485755	phase I
BRD-K21709199	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44485756	phase I
BRD-K16120913	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44485757	phase I
BRD-K39654705	CC(C)NC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@H](C)CO)nn2	CID:44485758	phase I
BRD-K60520051	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cn(CCCC1=O)nn3	CID:44485761	phase I
BRD-K39464795	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44485763	phase I
BRD-K37407046	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44485764	phase I
BRD-K06260900	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44485765	phase I
BRD-K93061078	CNC[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@@H](C)CO)nn2	CID:44485768	phase I
BRD-K67269534	CNC[C@@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@H](C)CO)nn2	CID:44485769	phase I
BRD-K21827358	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44485773	phase I
BRD-K30645599	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485775	phase I
BRD-K43609604	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44485777	phase I
BRD-K51454562	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485781	phase I
BRD-K04832618	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485790	phase I
BRD-K27198330	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44485796	phase I
BRD-K77006185	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44485797	phase I
BRD-K85694079	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44485799	phase I
BRD-K46512834	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44485803	phase I
BRD-K51877340	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44485804	phase I
BRD-K71240454	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:44485809	phase I
BRD-K90700939	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44485816	phase I
BRD-K93577185	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44485822	phase I
BRD-K97860318	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44485828	phase I
BRD-K08266813	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44485834	phase I
BRD-K80832371	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44485842	phase I
BRD-K06170455	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc5OCOc5c4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44485855	phase I
BRD-K34960081	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44485890	phase I
BRD-K72516992	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44485914	phase I
BRD-K67271639	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44485929	phase I
BRD-K51823671	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:44485930	phase I
BRD-K73804145	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44485978	phase I
BRD-K97972722	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44485990	phase I
BRD-K83940002	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44486010	phase I
BRD-K71555338	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44486037	phase I
BRD-K75972810	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44486060	phase I
BRD-K39294074	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44486095	phase I
BRD-K05197946	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44486126	phase I
BRD-K64523453	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44486132	phase I
BRD-K04117492	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44486138	phase I
BRD-K14533651	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44486156	phase I
BRD-K14374193	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44486164	phase I
BRD-K62748479	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44486180	phase I
BRD-K42056004	COc1ccc(CN(C)C[C@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44486182	phase I
BRD-K38553273	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44486194	phase I
BRD-K73888531	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44486204	phase I
BRD-K43231198	CNC[C@H]1Oc2c(NS(=O)(=O)c3ccc(OC)cc3)cccc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44486217	phase I
BRD-K60569491	CNC[C@@H]1Oc2c(NS(=O)(=O)c3ccc(OC)cc3)cccc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44486225	phase I
BRD-K90143908	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44486244	phase I
BRD-K39880131	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44486267	phase I
BRD-K97888290	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44486277	phase I
BRD-K99179945	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44486299	phase I
BRD-K71006848	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44486300	phase I
BRD-K00991320	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44486305	phase I
BRD-K81313903	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44486306	phase I
BRD-K23211153	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(cc2CC(=O)N(C[C@H]1C)[C@H](C)CO)N(C)C	CID:44486324	phase I
BRD-K69930474	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44486341	phase I
BRD-K13879491	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44486342	phase I
BRD-K44890352	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3cn(CCCC1=O)nn3	CID:44486345	phase I
BRD-K87010407	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44486348	phase I
BRD-K56304906	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44486349	phase I
BRD-K31039264	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44486352	phase I
BRD-K31788208	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44486354	phase I
BRD-K37563991	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44486355	phase I
BRD-K54885483	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)OCc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44486356	phase I
BRD-K23038591	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44486358	phase I
BRD-K57627685	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44486364	phase I
BRD-K08043024	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cn(CCCC1=O)nn3	CID:44486366	phase I
BRD-K82521114	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44486367	phase I
BRD-K12165191	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44486368	phase I
BRD-K00846846	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44486369	phase I
BRD-K19960610	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44486370	phase I
BRD-K54455139	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4cn(CCCC1=O)nn4	CID:44486371	phase I
BRD-K43792870	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4cn(CCCC1=O)nn4	CID:44486372	phase I
BRD-K53488735	COc1ccccc1CN(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3	CID:44486373	phase I
BRD-K70940447	CNC[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@H](C)CO)nn2	CID:44486374	phase I
BRD-K61529775	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44486379	phase I
BRD-K75296800	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486382	phase I
BRD-K65540587	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44486384	phase I
BRD-K25991572	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44486386	phase I
BRD-K57901680	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486389	phase I
BRD-K47825575	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)C)cc2C1=O	CID:44486390	phase I
BRD-K68455755	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44486391	phase I
BRD-K50204028	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44486395	phase I
BRD-K58070753	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44486400	phase I
BRD-K85946956	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44486401	phase I
BRD-K84528570	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486404	phase I
BRD-K66805710	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44486405	phase I
BRD-K33215066	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44486406	phase I
BRD-K51189903	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486410	phase I
BRD-K41931739	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44486411	phase I
BRD-K56884102	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44486424	phase I
BRD-K60093216	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44486428	phase I
BRD-K99756483	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44486455	phase I
BRD-K01877724	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44486502	phase I
BRD-K95482240	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44486602	phase I
BRD-K63375110	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44486621	phase I
BRD-K94109647	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44486640	phase I
BRD-K72460946	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44486643	phase I
BRD-K28573311	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44486680	phase I
BRD-K30066603	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44486706	phase I
BRD-K36928611	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44486720	phase I
BRD-K69347381	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486732	phase I
BRD-K75265238	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44486740	phase I
BRD-K01595245	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44486749	phase I
BRD-K91076377	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44486767	phase I
BRD-K04632192	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44486770	phase I
BRD-K09973807	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44486786	phase I
BRD-K66681850	CNC[C@@H]1Oc2c(NS(=O)(=O)c3ccc(OC)cc3)cccc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44486795	phase I
BRD-K68061938	COc1ccc(CN(C)C[C@@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44486798	phase I
BRD-K23073505	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3c(NC(=O)c4ccc(cc4)c5nccs5)cccc3C1=O	CID:44486806	phase I
BRD-K38455110	COc1ccc(cc1)S(=O)(=O)Nc2cccc3C(=O)N(C[C@@H](C)[C@H](CN(C)Cc4ccc(cc4)C(F)(F)F)Oc23)[C@H](C)CO	CID:44486809	phase I
BRD-K37852224	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44486811	phase I
BRD-K57856779	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3c(cccc3C1=O)N(C)C	CID:44486845	phase I
BRD-K58175397	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44486870	phase I
BRD-K55666799	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44486888	phase I
BRD-K14801883	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44486893	phase I
BRD-K23905744	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(cc2CC(=O)N(C[C@H]1C)[C@H](C)CO)N(C)C	CID:44486903	phase I
BRD-K76882924	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44486917	phase I
BRD-K28312904	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44486924	phase I
BRD-K83533725	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44486935	phase I
BRD-K18048820	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(cc2CC(=O)N(C[C@@H]1C)[C@@H](C)CO)N(C)C	CID:44486939	phase I
BRD-K17976466	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3cn(CCCC1=O)nn3	CID:44486949	phase I
BRD-K65790118	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44486951	phase I
BRD-K03817886	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44486954	phase I
BRD-K13207999	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44486955	phase I
BRD-K42420111	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44486956	phase I
BRD-K77517292	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44486957	phase I
BRD-K08023754	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44486958	phase I
BRD-K85398522	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44486959	phase I
BRD-K04749191	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44486960	phase I
BRD-K15923694	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)OCc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44486961	phase I
BRD-K26273696	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44486963	phase I
BRD-K55025062	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44486964	phase I
BRD-K32294814	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44486966	phase I
BRD-K46205969	CC(C)NC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@@H](C)CO)nn2	CID:44486967	phase I
BRD-K06568278	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44486968	phase I
BRD-K39245862	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44486969	phase I
BRD-K79876173	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44486972	phase I
BRD-K94817443	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44486973	phase I
BRD-K47497589	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44486974	phase I
BRD-K88495921	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4cn(CCCC1=O)nn4	CID:44486975	phase I
BRD-K94263505	COc1ccccc1CN(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44486976	phase I
BRD-K61045425	CNC[C@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@H](C)CO)nn2	CID:44486977	phase I
BRD-K34516743	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44486983	phase I
BRD-K99433267	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44486984	phase I
BRD-K76266174	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44486986	phase I
BRD-K76042595	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486991	phase I
BRD-K74659851	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:44486992	phase I
BRD-K46666779	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)Cc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44486993	phase I
BRD-K21994180	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44486994	phase I
BRD-K95616928	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486995	phase I
BRD-K41513229	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44486997	phase I
BRD-K47630323	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44486998	phase I
BRD-K73939795	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44487002	phase I
BRD-K76005220	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44487007	phase I
BRD-K62719675	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44487010	phase I
BRD-K03111155	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44487018	phase I
BRD-K90970920	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44487024	phase I
BRD-K52831896	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)S(=O)(=O)c3c(C)noc3C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487025	phase I
BRD-K05174693	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44487030	phase I
BRD-K83732250	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C1=O	CID:44487031	phase I
BRD-K47802551	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44487032	phase I
BRD-K89020690	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44487083	phase I
BRD-K46445327	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44487119	phase I
BRD-K65000194	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)Cc4ccc5OCOc5c4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44487159	phase I
BRD-K77264557	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44487168	phase I
BRD-K68565044	CNC[C@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44487195	phase I
BRD-K06623064	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44487206	phase I
BRD-K17238328	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487252	phase I
BRD-K21232697	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487262	phase I
BRD-K45749103	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44487268	phase I
BRD-K42687792	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)S(=O)(=O)c4ccc(C)cc4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44487293	phase I
BRD-K29423519	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487297	phase I
BRD-K64304398	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44487321	phase I
BRD-K95057125	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44487333	phase I
BRD-K52726129	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)c5cccs5)cc4C1=O	CID:44487334	phase I
BRD-K07063907	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44487338	phase I
BRD-K77658626	CNC[C@@H]1Oc2c(NS(=O)(=O)c3ccc(OC)cc3)cccc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44487363	phase I
BRD-K54916924	COc1ccc(CN(C)C[C@@H]2Oc3c(NS(=O)(=O)C)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44487378	phase I
BRD-K54323133	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44487397	phase I
BRD-K66185150	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44487401	phase I
BRD-K55010869	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44487402	phase I
BRD-K18391257	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44487405	phase I
BRD-K01676918	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3cn(CCCC1=O)nn3	CID:44487406	phase I
BRD-K60129749	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44487409	phase I
BRD-K15845256	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44487410	phase I
BRD-K02707544	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44487411	phase I
BRD-K23349860	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44487412	phase I
BRD-K30312461	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44487414	phase I
BRD-K03937518	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44487415	phase I
BRD-K03795299	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cn(CCCC1=O)nn3	CID:44487420	phase I
BRD-K61541549	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44487422	phase I
BRD-K34730083	CNC[C@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44487425	phase I
BRD-K82435102	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487426	phase I
BRD-K42091312	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44487436	phase I
BRD-K97149069	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)Cc3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487439	phase I
BRD-K38986089	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487442	phase I
BRD-K59563627	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487451	phase I
BRD-K81461172	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44487458	phase I
BRD-K52657367	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487460	phase I
BRD-K40846327	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44487461	phase I
BRD-K63383460	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487464	phase I
BRD-K30194621	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3c(C)noc3C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44487465	phase I
BRD-K51981081	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487471	phase I
BRD-K05672354	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)Cc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44487472	phase I
BRD-K82651890	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44487474	phase I
BRD-K22854900	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44487478	phase I
BRD-K89005359	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487483	phase I
BRD-K52099002	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44487484	phase I
BRD-K50368246	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44487490	phase I
BRD-K75666689	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487498	phase I
BRD-K91034707	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487502	phase I
BRD-K65983740	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44487505	phase I
BRD-K76138094	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44487519	phase I
BRD-K91755384	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)Cc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487524	phase I
BRD-K25070860	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487526	phase I
BRD-K56269643	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44487531	phase I
BRD-K99020117	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44487540	phase I
BRD-K55588166	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487544	phase I
BRD-K72429558	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44487546	phase I
BRD-K22828548	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44487555	phase I
BRD-K79131428	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487559	phase I
BRD-K32101742	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44487561	phase I
BRD-K77705921	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487562	phase I
BRD-K34547533	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487564	phase I
BRD-K30640165	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44487568	phase I
BRD-K58191509	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44487571	phase I
BRD-K10839108	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44487576	phase I
BRD-K35418438	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487580	phase I
BRD-K27411973	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccccc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44487588	phase I
BRD-K50277523	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44487589	phase I
BRD-K47394228	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44487592	phase I
BRD-K55971699	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:44487597	phase I
BRD-K59488055	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4CC1=O	CID:44487599	phase I
BRD-K46707574	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44487605	phase I
BRD-K92232855	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(cc2CC(=O)N(C[C@H]1C)[C@@H](C)CO)N(C)C	CID:44487610	phase I
BRD-K98150670	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44487620	phase I
BRD-K10609180	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)Oc3ccc(cc3CC1=O)N(C)C	CID:44487621	phase I
BRD-K15146741	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44487636	phase I
BRD-K22754681	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2C1=O	CID:44487652	phase I
BRD-K33095226	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44487665	phase I
BRD-K54674054	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44487667	phase I
BRD-K26362026	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44487676	phase I
BRD-K25743534	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44487692	phase I
BRD-K78904620	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44487694	phase I
BRD-K09641113	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44487708	phase I
BRD-K80988607	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44487713	phase I
BRD-K34412705	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44487718	phase I
BRD-K76418961	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44487739	phase I
BRD-K59805090	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44487761	phase I
BRD-K20792495	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44487764	phase I
BRD-K86617991	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44487775	phase I
BRD-K14503950	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44487780	phase I
BRD-K82761903	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:44487794	phase I
BRD-K17773477	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44487821	phase I
BRD-K91662540	CNC[C@@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44487844	phase I
BRD-K90310644	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44487847	phase I
BRD-K36134449	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc5OCOc5c4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44487856	phase I
BRD-K38087837	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44487877	phase I
BRD-K72490684	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)Cc4ccc5OCOc5c4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44487879	phase I
BRD-K76583861	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44487884	phase I
BRD-K41129770	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44487898	phase I
BRD-K74010885	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44487900	phase I
BRD-K65715788	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44487905	phase I
BRD-K64368934	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44487909	phase I
BRD-K06417531	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44487912	phase I
BRD-K49687221	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44487922	phase I
BRD-K03957451	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44487927	phase I
BRD-K08311783	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44487934	phase I
BRD-K03228992	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44487954	phase I
BRD-K33326988	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44487971	phase I
BRD-K01048110	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44487978	phase I
BRD-K20197062	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44488016	phase I
BRD-K89144371	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@H](C)[C@@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@@H](C)CO	CID:44488022	phase I
BRD-K69841970	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@H](C)[C@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@H](C)CO	CID:44488050	phase I
BRD-K32670473	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44488053	phase I
BRD-K27014041	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44488065	phase I
BRD-K88307956	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44488069	phase I
BRD-K69021489	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44488070	phase I
BRD-K86894445	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44488084	phase I
BRD-K41726296	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44488092	phase I
BRD-K38149517	CNC[C@@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44488094	phase I
BRD-K22853292	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)c4ccncc4)cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44488113	phase I
BRD-K34673904	CNC[C@@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44488132	phase I
BRD-K51296348	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44488151	phase I
BRD-K39299017	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44488152	phase I
BRD-K18699770	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44488153	phase I
BRD-K31538032	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44488155	phase I
BRD-K46807184	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44488156	phase I
BRD-K96218183	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44488158	phase I
BRD-K78633583	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cn(CCCC1=O)nn4	CID:44488159	phase I
BRD-K15953261	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cn(CCCC1=O)nn4	CID:44488160	phase I
BRD-K60644933	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44488162	phase I
BRD-K30937833	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44488163	phase I
BRD-K87438596	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44488165	phase I
BRD-K50580743	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44488166	phase I
BRD-K33933950	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2cnnn2CCCC1=O	CID:44488167	phase I
BRD-K40750649	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3N(C)CCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44488168	phase I
BRD-K92803302	COc1ccccc1CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44488170	phase I
BRD-K32162364	COc1ccccc1CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44488171	phase I
BRD-K66866270	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44488175	phase I
BRD-K04411796	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44488177	phase I
BRD-K18293432	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)N(C)C	CID:44488184	phase I
BRD-K95842463	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44488188	phase I
BRD-K30459086	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44488191	phase I
BRD-K48465004	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCCCC[C@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44488192	phase I
BRD-K11989708	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)Cc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44488194	phase I
BRD-K44890999	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C1=O	CID:44488199	phase I
BRD-K07026322	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCCN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44488201	phase I
BRD-K53327986	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44488204	phase I
BRD-K81440797	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)N(C)C	CID:44488205	phase I
BRD-K32582686	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44488207	phase I
BRD-K31688005	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44488210	phase I
BRD-K16535949	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44488211	phase I
BRD-K80972048	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44488215	phase I
BRD-K29745382	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44488232	phase I
BRD-K40185230	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44488237	phase I
BRD-K91194707	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44488264	phase I
BRD-K36317223	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44488287	phase I
BRD-K19982400	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44488299	phase I
BRD-K63388446	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44488301	phase I
BRD-K12249810	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44488307	phase I
BRD-K34310783	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44488320	phase I
BRD-K79242575	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)C5CC5)cc4C1=O	CID:44488330	phase I
BRD-K30468800	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44488349	phase I
BRD-K44316554	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44488358	phase I
BRD-K53120552	CNC[C@@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44488361	phase I
BRD-K97919576	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44488374	phase I
BRD-K68657207	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44488420	phase I
BRD-K72193580	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44488424	phase I
BRD-K90135241	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44488429	phase I
BRD-K02354331	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44488432	phase I
BRD-K21259057	CNC[C@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44488434	phase I
BRD-K51595563	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44488451	phase I
BRD-K40078199	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44488469	phase I
BRD-K09821933	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:44488475	phase I
BRD-K36094929	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44488484	phase I
BRD-K49377740	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44488495	phase I
BRD-K65257681	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44488509	phase I
BRD-K37160016	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44488511	phase I
BRD-K77789137	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44488519	phase I
BRD-K20126873	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2C1=O	CID:44488524	phase I
BRD-K20740790	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44488540	phase I
BRD-K48804356	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3CC(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44488623	phase I
BRD-K61543740	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3CC1=O	CID:44488629	phase I
BRD-K44200196	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:44488634	phase I
BRD-K69218883	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO)N(C)C	CID:44488642	phase I
BRD-K36906780	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(cc2CC(=O)N(C[C@H]1C)[C@@H](C)CO)N(C)C	CID:44488670	phase I
BRD-K34898990	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44488673	phase I
BRD-K42737417	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44488685	phase I
BRD-K35290760	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44488687	phase I
BRD-K58377762	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44488690	phase I
BRD-K52574175	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cn(CCCC1=O)nn4	CID:44488691	phase I
BRD-K53174909	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44488693	phase I
BRD-K05662507	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cn(CCCC1=O)nn4	CID:44488694	phase I
BRD-K88872152	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44488697	phase I
BRD-K62191543	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44488698	phase I
BRD-K19471718	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44488699	phase I
BRD-K36718717	CC(C)NC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44488700	phase I
BRD-K54628954	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44488703	phase I
BRD-K78352220	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cn(CCCC1=O)nn3	CID:44488704	phase I
BRD-K06162576	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44488707	phase I
BRD-K66186977	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3cccnc3c2)OCc4cn(CCCC1=O)nn4	CID:44488708	phase I
BRD-K58790952	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2cn(CCCC1=O)nn2	CID:44488709	phase I
BRD-K54671386	CNC[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44488711	phase I
BRD-K92732825	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)Oc3ncccc3C1=O	CID:44488717	phase I
BRD-K78603235	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccccc3	CID:44488725	phase I
BRD-K91339294	CCCN(C)C[C@@H]1Oc2ncc(C#CCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44488728	phase I
BRD-K63828515	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44488739	phase I
BRD-K03463440	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44488749	phase I
BRD-K60558220	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44488751	phase I
BRD-K24992843	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44488752	phase I
BRD-K18249495	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44488755	phase I
BRD-K73592400	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44488757	phase I
BRD-K46080444	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44488769	phase I
BRD-K10170503	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44488775	phase I
BRD-K44696931	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44488783	phase I
BRD-K23931216	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44488800	phase I
BRD-K34206396	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44488817	phase I
BRD-K51633576	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44488837	phase I
BRD-K54350452	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44488848	phase I
BRD-K14833463	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44488849	phase I
BRD-K15221219	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)c5ccc(Cl)cc5)cc4C1=O	CID:44488857	phase I
BRD-K12182524	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44488863	phase I
BRD-K67258928	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3C(=O)N(C[C@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44488905	phase I
BRD-K88822846	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44488910	phase I
BRD-K78025571	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44488942	phase I
BRD-K78738487	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44488951	phase I
BRD-K94127894	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44488994	phase I
BRD-K97423351	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44489025	phase I
BRD-K55077180	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44489027	phase I
BRD-K80728817	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44489063	phase I
BRD-K57759884	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44489073	phase I
BRD-K36290066	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44489091	phase I
BRD-K79102010	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44489122	phase I
BRD-K25708438	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44489132	phase I
BRD-K82558986	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44489135	phase I
BRD-K39732687	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44489173	phase I
BRD-K74864389	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44489177	phase I
BRD-K90417362	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44489186	phase I
BRD-K89338967	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44489213	phase I
BRD-K58698092	CNC[C@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44489216	phase I
BRD-K88624856	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44489228	phase I
BRD-K01008530	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44489265	phase I
BRD-K78921480	COC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@H](C)CO)nn2	CID:44489267	phase I
BRD-K86033856	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44489268	phase I
BRD-K76964118	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cn(CCCC1=O)nn4	CID:44489269	phase I
BRD-K07473223	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44489270	phase I
BRD-K14744524	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44489271	phase I
BRD-K42435091	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44489272	phase I
BRD-K09757845	COc1ccccc1CN(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44489280	phase I
BRD-K62102996	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44489298	phase I
BRD-K60212338	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44489301	phase I
BRD-K23370299	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)N(C)C	CID:44489316	phase I
BRD-K62019540	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44489318	phase I
BRD-K50521229	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44489319	phase I
BRD-K91662172	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44489323	phase I
BRD-K75090653	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44489329	phase I
BRD-K89675250	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489335	phase I
BRD-K28001518	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)N(C)C	CID:44489337	phase I
BRD-K05756698	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)Cc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489338	phase I
BRD-K52043480	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)Cc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44489343	phase I
BRD-K32431994	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44489352	phase I
BRD-K38024133	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44489353	phase I
BRD-K88672507	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44489368	phase I
BRD-K93720819	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44489378	phase I
BRD-K01605959	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44489401	phase I
BRD-K79651181	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44489421	phase I
BRD-K46362951	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44489430	phase I
BRD-K35334027	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44489441	phase I
BRD-K93971872	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44489454	phase I
BRD-K24885102	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44489456	phase I
BRD-K70108530	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44489463	phase I
BRD-K46849403	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44489465	phase I
BRD-K76812993	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44489466	phase I
BRD-K91945291	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44489468	phase I
BRD-K22789789	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44489490	phase I
BRD-K49482378	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44489492	phase I
BRD-K03981069	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44489497	phase I
BRD-K49939055	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44489512	phase I
BRD-K93445052	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44489515	phase I
BRD-K46171293	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44489516	phase I
BRD-K59423635	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44489520	phase I
BRD-K85879095	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44489551	phase I
BRD-K59683187	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44489558	phase I
BRD-K42438139	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44489566	phase I
BRD-K45949967	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44489570	phase I
BRD-K92807185	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44489577	phase I
BRD-K24744176	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44489582	phase I
BRD-K74271701	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44489593	phase I
BRD-K37613339	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3C(=O)N(C[C@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44489606	phase I
BRD-K30365815	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44489649	phase I
BRD-K14475668	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44489655	phase I
BRD-K49596872	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@H](C)[C@@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@H](C)CO	CID:44489669	phase I
BRD-K18100239	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44489672	phase I
BRD-K64610608	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44489675	phase I
BRD-K58273050	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44489681	phase I
BRD-K64754843	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44489685	phase I
BRD-K58381953	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44489694	phase I
BRD-K74046820	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489703	phase I
BRD-K16046246	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44489706	phase I
BRD-K73737710	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489717	phase I
BRD-K51922621	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489719	phase I
BRD-K56904155	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489720	phase I
BRD-K27475558	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489726	phase I
BRD-K88059273	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489738	phase I
BRD-K90734091	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489743	phase I
BRD-K75426909	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489749	phase I
BRD-K06899423	CNC[C@@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44489756	phase I
BRD-K18641148	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)c4ccncc4)cc3CC(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44489766	phase I
BRD-K38760240	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(cc4CC1=O)N(C)C	CID:44489795	phase I
BRD-K57882732	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44489805	phase I
BRD-K82494568	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Oc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44489806	phase I
BRD-K94479191	COC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@@H](C)CO)nn2	CID:44489808	phase I
BRD-K63180587	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2cnnn2CCCC1=O	CID:44489814	phase I
BRD-K15234779	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3N(C)CCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44489816	phase I
BRD-K82899766	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccc(F)cc3	CID:44489821	phase I
BRD-K98832554	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)Oc3ncccc3C1=O	CID:44489824	phase I
BRD-K76999748	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44489837	phase I
BRD-K06574200	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44489842	phase I
BRD-K84157702	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)N(C)C	CID:44489843	phase I
BRD-K47539505	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44489845	phase I
BRD-K07008972	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44489847	phase I
BRD-K03814443	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44489854	phase I
BRD-K41418105	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44489855	phase I
BRD-K00664012	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44489862	phase I
BRD-K43682718	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44489864	phase I
BRD-K40301427	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489870	phase I
BRD-K41649460	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489878	phase I
BRD-K76047634	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44489897	phase I
BRD-K17565092	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44489904	phase I
BRD-K05395601	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:44489941	phase I
BRD-K18271121	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44489947	phase I
BRD-K25990552	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490005	phase I
BRD-K42134801	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490013	phase I
BRD-K86596187	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44490029	phase I
BRD-K38611276	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44490066	phase I
BRD-K14262667	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44490074	phase I
BRD-K61359353	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44490082	phase I
BRD-K58918780	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44490089	phase I
BRD-K57786095	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44490110	phase I
BRD-K57321627	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490131	phase I
BRD-K37856394	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44490159	phase I
BRD-K97727250	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44490160	phase I
BRD-K18772888	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44490187	phase I
BRD-K60487596	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44490190	phase I
BRD-K37788266	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@H](C)[C@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@@H](C)CO	CID:44490221	phase I
BRD-K91180076	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490222	phase I
BRD-K43283261	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44490224	phase I
BRD-K02502363	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490226	phase I
BRD-K27622534	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490229	phase I
BRD-K28497936	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44490230	phase I
BRD-K56951539	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490232	phase I
BRD-K62659735	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44490236	phase I
BRD-K77983109	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)Cc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490239	phase I
BRD-K06592610	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490241	phase I
BRD-K18170480	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc(F)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44490243	phase I
BRD-K28649955	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)N(C)C	CID:44490250	phase I
BRD-K20859359	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44490251	phase I
BRD-K16633354	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Cc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490257	phase I
BRD-K25719068	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490262	phase I
BRD-K06187854	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490265	phase I
BRD-K55208094	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44490269	phase I
BRD-K59472400	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490270	phase I
BRD-K69206710	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(cc2C1=O)N(C)C	CID:44490276	phase I
BRD-K85592362	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44490284	phase I
BRD-K57732441	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490285	phase I
BRD-K74446951	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)N(C)C	CID:44490286	phase I
BRD-K51083659	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)[C@@H](C)CN([C@H](C)CO)C(=O)Cc3c2	CID:44490299	phase I
BRD-K49373277	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44490301	phase I
BRD-K26048698	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cn(CCCC1=O)nn4	CID:44490304	phase I
BRD-K45630356	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44490306	phase I
BRD-K07064094	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44490321	phase I
BRD-K93107794	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490325	phase I
BRD-K73388067	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)N(C)C	CID:44490327	phase I
BRD-K71599932	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490330	phase I
BRD-K46594703	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490336	phase I
BRD-K42543304	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490342	phase I
BRD-K69747917	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)N(C)C	CID:44490348	phase I
BRD-K40829514	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490349	phase I
BRD-K26822808	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490354	phase I
BRD-K16930636	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)N(C)C	CID:44490361	phase I
BRD-K93605482	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490363	phase I
BRD-K19534956	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490364	phase I
BRD-K87779450	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490365	phase I
BRD-K02248910	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44490368	phase I
BRD-K38144109	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490371	phase I
BRD-K72381041	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C1=O	CID:44490380	phase I
BRD-K65572849	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490381	phase I
BRD-K82633701	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)CCCN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490385	phase I
BRD-K14340046	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490392	phase I
BRD-K66221011	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCCN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490393	phase I
BRD-K38546320	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490399	phase I
BRD-K31877241	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)N(C)C	CID:44490402	phase I
BRD-K08777248	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44490403	phase I
BRD-K88616704	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44490406	phase I
BRD-K81927853	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490407	phase I
BRD-K63117650	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44490413	phase I
BRD-K18059480	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490415	phase I
BRD-K82226238	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C1=O	CID:44490427	phase I
BRD-K03725349	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44490429	phase I
BRD-K54385541	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)N(C)C	CID:44490432	phase I
BRD-K38965110	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490435	phase I
BRD-K74163137	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490437	phase I
BRD-K36022244	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44490445	phase I
BRD-K89554882	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCCN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490452	phase I
BRD-K48775333	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44490457	phase I
BRD-K60272788	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490460	phase I
BRD-K46499837	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490464	phase I
BRD-K72269288	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Cc3ccccc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490467	phase I
BRD-K20192397	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490468	phase I
BRD-K62687522	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44490483	phase I
BRD-K64508546	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490497	phase I
BRD-K71672862	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44490511	phase I
BRD-K47774969	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44490520	phase I
BRD-K24214483	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44490530	phase I
BRD-K37048848	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44490552	phase I
BRD-K16010201	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44490584	phase I
BRD-K35024477	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44490586	phase I
BRD-K97073065	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44490600	phase I
BRD-K01140360	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490608	phase I
BRD-K78627754	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44490613	phase I
BRD-K53501402	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44490616	phase I
BRD-K74965436	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44490620	phase I
BRD-K34974324	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44490640	phase I
BRD-K00064929	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44490664	phase I
BRD-K49180909	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44490674	phase I
BRD-K63406873	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44490694	phase I
BRD-K41887163	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44490771	phase I
BRD-K14636731	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44490782	phase I
BRD-K54822214	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44490807	phase I
BRD-K82769855	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44490823	phase I
BRD-K75912549	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44490824	phase I
BRD-K63979920	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44490830	phase I
BRD-K14502067	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44490846	phase I
BRD-K70748405	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44490857	phase I
BRD-K57073585	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44490858	phase I
BRD-K67669478	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44490869	phase I
BRD-K74504761	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44490870	phase I
BRD-K57873755	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44490872	phase I
BRD-K07912534	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44490873	phase I
BRD-K64968742	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490883	phase I
BRD-K64247367	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)N(C)C	CID:44490884	phase I
BRD-K19764902	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490887	phase I
BRD-K05886700	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44490891	phase I
BRD-K24754728	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44490897	phase I
BRD-K28667054	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)N(C)C	CID:44490899	phase I
BRD-K14370088	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C1=O	CID:44490904	phase I
BRD-K98437249	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490906	phase I
BRD-K94352392	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44490907	phase I
BRD-K80553643	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44490909	phase I
BRD-K47611269	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44490912	phase I
BRD-K38571337	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44490916	phase I
BRD-K20761826	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44490918	phase I
BRD-K00429057	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44490923	phase I
BRD-K76073118	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44490929	phase I
BRD-K36177038	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Cc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44490936	phase I
BRD-K19189705	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44490946	phase I
BRD-K10087454	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)N(C)C	CID:44490957	phase I
BRD-K47690943	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44490959	phase I
BRD-K41129365	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44490968	phase I
BRD-K09459434	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44490995	phase I
BRD-K17689300	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44491002	phase I
BRD-K25565604	CNC[C@@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44491029	phase I
BRD-K46428287	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44491032	phase I
BRD-K89257372	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44491059	phase I
BRD-K19596098	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44491071	phase I
BRD-K06809080	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44491094	phase I
BRD-K18067885	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44491103	phase I
BRD-K03302289	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44491110	phase I
BRD-K11224669	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44491123	phase I
BRD-K81904610	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44491139	phase I
BRD-K63399564	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44491148	phase I
BRD-K63435718	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44491171	phase I
BRD-K81554246	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:44491217	phase I
BRD-K49092745	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44491244	phase I
BRD-K51164721	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44491334	phase I
BRD-K39587434	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@@H](C)[C@@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@@H](C)CO	CID:44491340	phase I
BRD-K30802967	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44491342	phase I
BRD-K09033315	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44491378	phase I
BRD-K10499894	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)C4CCOCC4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44491382	phase I
BRD-K15814728	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@@H](C)[C@@H](CN(C)Cc3ccc(Cl)c(Cl)c3)Oc12)[C@H](C)CO	CID:44491385	phase I
BRD-K44510578	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44491394	phase I
BRD-K00270349	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44491404	phase I
BRD-K82666260	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)c4ccncc4)cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44491409	phase I
BRD-K76150323	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44491416	phase I
BRD-K15960830	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44491421	phase I
BRD-K97399889	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44491445	phase I
BRD-K10486333	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44491446	phase I
BRD-K62771544	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44491447	phase I
BRD-K86956630	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44491448	phase I
BRD-K00913793	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44491450	phase I
BRD-K09615275	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44491455	phase I
BRD-K72801689	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44491456	phase I
BRD-K64249376	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44491457	phase I
BRD-K33394674	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44491458	phase I
BRD-K71283713	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44491459	phase I
BRD-K48241951	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2cnnn2CCCC1=O	CID:44491463	phase I
BRD-K22177912	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2cnnn2CCCC1=O	CID:44491464	phase I
BRD-K24053449	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44491467	phase I
BRD-K41763112	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)N(C)C	CID:44491470	phase I
BRD-K79459005	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44491473	phase I
BRD-K78099132	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44491477	phase I
BRD-K49553303	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44491481	phase I
BRD-K91850687	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44491487	phase I
BRD-K47808476	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44491490	phase I
BRD-K81514393	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44491491	phase I
BRD-K84109969	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44491494	phase I
BRD-K83509924	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44491495	phase I
BRD-K54285697	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44491503	phase I
BRD-K61855818	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)Cc3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44491506	phase I
BRD-K57443339	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44491509	phase I
BRD-K90816807	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)Cc3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44491516	phase I
BRD-K95425654	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44491522	phase I
BRD-K35892797	CNC[C@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44491540	phase I
BRD-K77644833	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44491589	phase I
BRD-K70901996	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44491614	phase I
BRD-K49460772	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44491615	phase I
BRD-K89941546	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44491639	phase I
BRD-K99597257	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44491662	phase I
BRD-K91416305	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44491672	phase I
BRD-K73205140	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44491711	phase I
BRD-K18976419	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44491717	phase I
BRD-K50177987	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44491736	phase I
BRD-K81141085	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44491737	phase I
BRD-K71498541	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44491776	phase I
BRD-K15998522	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44491778	phase I
BRD-K68689263	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44491852	phase I
BRD-K89696951	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44491888	phase I
BRD-K04695623	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44491899	phase I
BRD-K99050286	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44491908	phase I
BRD-K50112803	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44491909	phase I
BRD-K96933023	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44491922	phase I
BRD-K17169073	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44491936	phase I
BRD-K12683703	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44491938	phase I
BRD-K33116223	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44491953	phase I
BRD-K46911271	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44491956	phase I
BRD-K28154645	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44491957	phase I
BRD-K00835201	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2ccc(NC(=O)C3CC3)cc2CC1=O	CID:44491974	phase I
BRD-K29648963	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)c4ccncc4)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44491979	phase I
BRD-K24045217	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:44491985	phase I
BRD-K06759695	CNC[C@H]1Oc2ccc(NS(=O)(=O)c3ccccc3)cc2CC(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44492046	phase I
BRD-K17663841	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2cn(CCCC1=O)nn2	CID:44492051	phase I
BRD-K75580081	COC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44492053	phase I
BRD-K37306329	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44492055	phase I
BRD-K19712135	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cn(CCCC1=O)nn4	CID:44492056	phase I
BRD-K02291788	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cn(CCCC1=O)nn4	CID:44492057	phase I
BRD-K48222931	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44492062	phase I
BRD-K36048022	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492067	phase I
BRD-K10143126	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44492069	phase I
BRD-K76437403	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492077	phase I
BRD-K82777549	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44492080	phase I
BRD-K13969067	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44492083	phase I
BRD-K03394322	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44492086	phase I
BRD-K05415698	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44492088	phase I
BRD-K09824708	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)Cc3ccccc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44492090	phase I
BRD-K16118047	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cccs3)cc2C1=O	CID:44492098	phase I
BRD-K60996261	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44492101	phase I
BRD-K18337230	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44492103	phase I
BRD-K31830662	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCCN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44492109	phase I
BRD-K04617562	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44492116	phase I
BRD-K93086630	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44492152	phase I
BRD-K93774845	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44492156	phase I
BRD-K72960152	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44492157	phase I
BRD-K82899116	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44492158	phase I
BRD-K34230554	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44492192	phase I
BRD-K11672064	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44492198	phase I
BRD-K97233756	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44492216	phase I
BRD-K78687850	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44492218	phase I
BRD-K70284064	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492229	phase I
BRD-K85367959	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492244	phase I
BRD-K38659247	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44492265	phase I
BRD-K09540583	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44492274	phase I
BRD-K15507118	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44492308	phase I
BRD-K64751695	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44492321	phase I
BRD-K95193599	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492326	phase I
BRD-K66295580	CNC[C@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44492330	phase I
BRD-K64099269	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44492383	phase I
BRD-K23564441	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44492397	phase I
BRD-K60558601	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44492436	phase I
BRD-K83929831	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44492440	phase I
BRD-K64366758	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44492448	phase I
BRD-K30704475	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44492451	phase I
BRD-K75128590	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)C4CCOCC4)cccc3C1=O	CID:44492456	phase I
BRD-K68437527	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44492462	phase I
BRD-K38468651	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NC(=O)Nc5cccc6ccccc56)cccc4C1=O	CID:44492490	phase I
BRD-K78559095	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)Oc3c(NC(=O)c4cnccn4)cccc3C1=O	CID:44492502	phase I
BRD-K99303177	CNC[C@@H]1Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44492509	phase I
BRD-K96611781	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44492524	phase I
BRD-K52111234	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)[C@H](C)CN([C@@H](C)CO)C(=O)Cc3c2	CID:44492530	phase I
BRD-K86409742	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44492542	phase I
BRD-K25050358	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3cn(CCCC1=O)nn3	CID:44492573	phase I
BRD-K89796490	COC(=O)N(C)C[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44492578	phase I
BRD-K87400432	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3cnnn3CCCC1=O	CID:44492581	phase I
BRD-K95044179	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44492583	phase I
BRD-K52718919	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44492585	phase I
BRD-K57104759	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44492608	phase I
BRD-K30371494	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44492633	phase I
BRD-K11883928	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccccc3)cc2C1=O	CID:44492634	phase I
BRD-K94193354	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44492636	phase I
BRD-K08339178	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44492639	phase I
BRD-K78276903	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44492670	phase I
BRD-K46555627	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44492673	phase I
BRD-K75832278	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:44492693	phase I
BRD-K47378397	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492700	phase I
BRD-K83790954	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44492738	phase I
BRD-K85101781	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44492739	phase I
BRD-K13660244	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44492755	phase I
BRD-K50325722	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44492775	phase I
BRD-K30183231	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44492789	phase I
BRD-K34755514	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44492791	phase I
BRD-K31138070	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44492810	phase I
BRD-K40566034	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44492840	phase I
BRD-K32138919	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44492894	phase I
BRD-K27449529	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3C1=O)N(C)C	CID:44492909	phase I
BRD-K03631605	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44492912	phase I
BRD-K14230553	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CC4)cc3C1=O	CID:44492913	phase I
BRD-K59076458	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44492946	phase I
BRD-K17746689	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44492954	phase I
BRD-K28947191	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44493058	phase I
BRD-K43145106	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3cnnn3CCCC1=O	CID:44493064	phase I
BRD-K02063190	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44493065	phase I
BRD-K45307499	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3N(C)CCOc3c2)OCc4cnnn4CCCC1=O	CID:44493077	phase I
BRD-K57250790	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44493078	phase I
BRD-K02420864	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44493079	phase I
BRD-K68988758	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44493080	phase I
BRD-K81224183	CNC[C@@H]1Oc2ncc(C#CCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44493090	phase I
BRD-K21165668	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ncc(C#Cc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44493094	phase I
BRD-K17817744	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44493105	phase I
BRD-K58284322	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44493119	phase I
BRD-K85144746	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44493124	phase I
BRD-K45758869	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493137	phase I
BRD-K14614387	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44493156	phase I
BRD-K54381041	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44493228	phase I
BRD-K89712338	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493229	phase I
BRD-K59862677	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44493243	phase I
BRD-K75725000	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44493247	phase I
BRD-K00117639	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44493261	phase I
BRD-K20352452	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44493263	phase I
BRD-K39947788	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44493294	phase I
BRD-K59468384	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44493322	phase I
BRD-K91617567	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44493338	phase I
BRD-K43581698	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NS(=O)(=O)c5ccccc5)cc4C1=O	CID:44493344	phase I
BRD-K50634134	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44493347	phase I
BRD-K79779816	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5c(C)noc5C)cc4C1=O	CID:44493356	phase I
BRD-K34359283	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44493368	phase I
BRD-K20178228	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)c5ccncc5)cc4C1=O	CID:44493374	phase I
BRD-K51350137	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCN5CCOCC5)cc4C1=O	CID:44493394	phase I
BRD-K82092559	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44493436	phase I
BRD-K67414432	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44493466	phase I
BRD-K80197532	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NC(=O)Nc5cccc6ccccc56)cccc4C1=O	CID:44493495	phase I
BRD-K76325726	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44493554	phase I
BRD-K15923759	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)[C@H](C)CN([C@H](C)CO)C(=O)Cc3c2	CID:44493556	phase I
BRD-K40918107	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3cnnn3CCCC1=O	CID:44493572	phase I
BRD-K94435288	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44493581	phase I
BRD-K67896259	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44493583	phase I
BRD-K55231301	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44493585	phase I
BRD-K79355010	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44493589	phase I
BRD-K96157570	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44493596	phase I
BRD-K01822243	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44493597	phase I
BRD-K42740486	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44493615	phase I
BRD-K44638353	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44493625	phase I
BRD-K16950565	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44493627	phase I
BRD-K22847783	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44493635	phase I
BRD-K80574047	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493694	phase I
BRD-K63442512	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493722	phase I
BRD-K36031516	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44493759	phase I
BRD-K18127951	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493766	phase I
BRD-K76959261	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44493785	phase I
BRD-K16625384	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44493807	phase I
BRD-K23856550	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44493826	phase I
BRD-K72699596	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493831	phase I
BRD-K95241801	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44493837	phase I
BRD-K14127078	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44493841	phase I
BRD-K13028566	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44493847	phase I
BRD-K60927153	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44493850	phase I
BRD-K44791058	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44493867	phase I
BRD-K40087764	CNC[C@@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44493877	phase I
BRD-K32015301	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)Cn4cnnn4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44493879	phase I
BRD-K69423345	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44493884	phase I
BRD-K42006476	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44493914	phase I
BRD-K56596360	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44493915	phase I
BRD-K28578807	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44493918	phase I
BRD-K87113270	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44493933	phase I
BRD-K24894325	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44493967	phase I
BRD-K16912444	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NC(=O)Nc5cccc6ccccc56)cccc4C1=O	CID:44493984	phase I
BRD-K22375775	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ccc(cc3CC1=O)N(C)C	CID:44494000	phase I
BRD-K93302072	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)[C@H](C)CN([C@H](C)CO)C(=O)Cc3c2	CID:44494036	phase I
BRD-K38519699	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44494043	phase I
BRD-K13618800	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44494044	phase I
BRD-K77995433	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44494067	phase I
BRD-K00480552	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44494071	phase I
BRD-K73532097	COC(=O)N(C)C[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44494074	phase I
BRD-K72195772	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCc3cnnn3CCCC1=O	CID:44494078	phase I
BRD-K02612980	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44494079	phase I
BRD-K01876557	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44494080	phase I
BRD-K01591707	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44494083	phase I
BRD-K93061442	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44494084	phase I
BRD-K21389281	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494086	phase I
BRD-K92865756	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494096	phase I
BRD-K15916856	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494120	phase I
BRD-K31042955	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44494121	phase I
BRD-K56208365	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44494129	phase I
BRD-K59446585	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2C1=O	CID:44494142	phase I
BRD-K35088115	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)N(C)C	CID:44494165	phase I
BRD-K38599483	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:44494258	phase I
BRD-K74931283	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44494269	phase I
BRD-K47897830	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)N(C)C	CID:44494274	phase I
BRD-K38205437	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NS(=O)(=O)c4c(C)noc4C)cccc3C1=O	CID:44494334	phase I
BRD-K07395346	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44494352	phase I
BRD-K33762302	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44494360	phase I
BRD-K72732164	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494372	phase I
BRD-K89505656	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494377	phase I
BRD-K83548510	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44494388	phase I
BRD-K28282432	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44494405	phase I
BRD-K98624380	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494414	phase I
BRD-K41862560	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494417	phase I
BRD-K79768170	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44494423	phase I
BRD-K02590376	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:44494424	phase I
BRD-K01282863	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494440	phase I
BRD-K29360016	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494441	phase I
BRD-K92455082	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494446	phase I
BRD-K32975941	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)CC3CC3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44494463	phase I
BRD-K64366478	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)CC3CC3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44494477	phase I
BRD-K62624932	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44494482	phase I
BRD-K70905242	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(O)cc2)OCc3cnnn3CCCC1=O	CID:44494487	phase I
BRD-K03026470	CCCN(C)C[C@@H]1Oc2ncc(C#Cc3ccc(OC)c(OC)c3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494498	phase I
BRD-K12559526	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44494504	phase I
BRD-K67069164	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44494521	phase I
BRD-K59980440	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44494528	phase I
BRD-K08856690	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494545	phase I
BRD-K22211348	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44494556	phase I
BRD-K66598898	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494563	phase I
BRD-K46505016	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494573	phase I
BRD-K16993590	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494580	phase I
BRD-K40635448	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44494592	phase I
BRD-K86621086	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44494594	phase I
BRD-K74507776	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494597	phase I
BRD-K41520544	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494602	phase I
BRD-K66643665	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44494607	phase I
BRD-K33676730	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44494622	phase I
BRD-K12837223	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2C1=O	CID:44494623	phase I
BRD-K70508482	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:44494628	phase I
BRD-K14270906	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44494645	phase I
BRD-K51954117	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44494652	phase I
BRD-K06311439	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44494668	phase I
BRD-K06905668	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44494694	phase I
BRD-K95838867	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44494748	phase I
BRD-K74305285	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44494782	phase I
BRD-K78691413	CC(C)NC(=O)N(C)C[C@H]1Oc2c(NC(=O)Nc3cccc4ccccc34)cccc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44494796	phase I
BRD-K80883001	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44494800	phase I
BRD-K29792001	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@H](C)[C@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@@H](C)CO)cc1	CID:44494818	phase I
BRD-K80230516	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44494822	phase I
BRD-K27151060	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44494839	phase I
BRD-K72837898	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5nc6ccccc6s5)cccc4C1=O	CID:44494853	phase I
BRD-K28800414	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44494873	phase I
BRD-K53198520	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44494878	phase I
BRD-K71746288	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44494883	phase I
BRD-K86303874	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494904	phase I
BRD-K22657795	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494905	phase I
BRD-K10323659	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44494915	phase I
BRD-K04238564	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494921	phase I
BRD-K93980445	CC(C)NC(=O)N(C)C[C@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44494936	phase I
BRD-K14997413	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44494941	phase I
BRD-K31315646	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44494947	phase I
BRD-K66866904	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44494948	phase I
BRD-K73297432	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44494956	phase I
BRD-K18364651	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494982	phase I
BRD-K01389427	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44494984	phase I
BRD-K06071925	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44494986	phase I
BRD-K41431262	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44494999	phase I
BRD-K26258603	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44495000	phase I
BRD-K08891029	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44495003	phase I
BRD-K69603398	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44495013	phase I
BRD-K60391804	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44495028	phase I
BRD-K37977610	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44495037	phase I
BRD-K47533800	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2C1=O	CID:44495043	phase I
BRD-K84653575	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44495045	phase I
BRD-K06314140	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44495074	phase I
BRD-K32569202	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)c3c(C)noc3C)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44495084	phase I
BRD-K48986374	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44495095	phase I
BRD-K04650027	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc(cc4)C(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)Cc3c2	CID:44495105	phase I
BRD-K74155249	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44495181	phase I
BRD-K89409550	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@@H](C)[C@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@H](C)CO)cc1	CID:44495186	phase I
BRD-K51267267	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44495291	phase I
BRD-K45232279	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:44495329	phase I
BRD-K40056507	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44495340	phase I
BRD-K46532897	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44495351	phase I
BRD-K31088139	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44495355	phase I
BRD-K24861700	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44495386	phase I
BRD-K58532728	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44495414	phase I
BRD-K23620459	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3cnnn3CCCC1=O	CID:44495431	phase I
BRD-K42800143	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCc3cnnn3CCCC1=O	CID:44495438	phase I
BRD-K66363099	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCc3cnnn3CCCC1=O	CID:44495439	phase I
BRD-K71741980	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44495441	phase I
BRD-K54647996	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44495442	phase I
BRD-K47156219	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44495443	phase I
BRD-K33968993	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44495444	phase I
BRD-K05967016	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44495451	phase I
BRD-K49164596	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44495470	phase I
BRD-K46295497	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44495475	phase I
BRD-K68097207	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44495476	phase I
BRD-K51413232	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44495482	phase I
BRD-K90329522	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44495492	phase I
BRD-K06145650	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44495514	phase I
BRD-K78778188	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2C1=O	CID:44495520	phase I
BRD-K71489464	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44495539	phase I
BRD-K91836367	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)[C@@H](C)CN([C@H](C)CO)C(=O)Cc3c2	CID:44495549	phase I
BRD-K53816294	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44495615	phase I
BRD-K82196068	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44495699	phase I
BRD-K51047687	COc1ccc(CN(C)C[C@H]2Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44495717	phase I
BRD-K94616516	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)C)cccc3C1=O	CID:44495742	phase I
BRD-K60757524	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44495777	phase I
BRD-K18000410	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44495824	phase I
BRD-K67798612	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccncc5)cccc4C1=O	CID:44495835	phase I
BRD-K39431601	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44495841	phase I
BRD-K71915010	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4cccs4)cccc3C1=O	CID:44495852	phase I
BRD-K85273981	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NS(=O)(=O)C)cccc4C1=O	CID:44495870	phase I
BRD-K27855499	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc3c2	CID:44495953	phase I
BRD-K05098996	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44495957	phase I
BRD-K96698997	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44495958	phase I
BRD-K80281472	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3cnnn3CCCC1=O	CID:44495964	phase I
BRD-K37081092	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44495966	phase I
BRD-K67197636	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44495967	phase I
BRD-K94643104	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3N(C)CCOc3c2)OCc4cnnn4CCCC1=O	CID:44495968	phase I
BRD-K09584843	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44495970	phase I
BRD-K83829186	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44495971	phase I
BRD-K31883841	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44495973	phase I
BRD-K52827598	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44495977	phase I
BRD-K27597389	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Cc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44495992	phase I
BRD-K93994036	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44495995	phase I
BRD-K65455015	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44496000	phase I
BRD-K39271757	CNC[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44496012	phase I
BRD-K87779281	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44496020	phase I
BRD-K83448671	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44496032	phase I
BRD-K47301880	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44496035	phase I
BRD-K98995789	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@H](C)[C@@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@H](C)CO)cc1	CID:44496046	phase I
BRD-K18323006	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44496122	phase I
BRD-K08887444	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44496174	phase I
BRD-K14340219	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44496217	phase I
BRD-K28377013	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44496236	phase I
BRD-K44781077	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44496255	phase I
BRD-K76691125	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44496299	phase I
BRD-K06589444	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@H](C)[C@H](CN(C)C)Oc12)[C@H](C)CO	CID:44496306	phase I
BRD-K98988337	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@@H](C)[C@@H](CN(C)C)Oc12)[C@@H](C)CO	CID:44496311	phase I
BRD-K38294617	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44496321	phase I
BRD-K20497962	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44496324	phase I
BRD-K12450081	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3CC1=O	CID:44496328	phase I
BRD-K52572235	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44496339	phase I
BRD-K93189515	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:44496342	phase I
BRD-K55640612	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)c3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44496350	phase I
BRD-K43111958	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44496353	phase I
BRD-K04905339	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(cc3CC1=O)N(C)C	CID:44496365	phase I
BRD-K72505722	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)CC3CC3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44496386	phase I
BRD-K11022796	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3	CID:44496389	phase I
BRD-K18273607	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44496391	phase I
BRD-K87904079	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44496392	phase I
BRD-K97186212	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(C)(C)C)OCc3cn(CCCC1=O)nn3	CID:44496399	phase I
BRD-K08209559	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(C)(C)C)OCc3cn(CCCC1=O)nn3	CID:44496400	phase I
BRD-K54522558	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3	CID:44496401	phase I
BRD-K09926293	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(O)cc2)OCc3cn(CCCC1=O)nn3	CID:44496405	phase I
BRD-K53425819	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(O)cc2)OCc3cnnn3CCCC1=O	CID:44496406	phase I
BRD-K37167897	CNC[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44496407	phase I
BRD-K31826120	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44496416	phase I
BRD-K19689423	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44496430	phase I
BRD-K76512739	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44496432	phase I
BRD-K40170731	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44496436	phase I
BRD-K02490064	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44496446	phase I
BRD-K93779718	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)C3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44496449	phase I
BRD-K21387011	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44496450	phase I
BRD-K24391905	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44496454	phase I
BRD-K65124508	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44496471	phase I
BRD-K79732306	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44496473	phase I
BRD-K25997353	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44496475	phase I
BRD-K43806450	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44496612	phase I
BRD-K52044217	CNC[C@@H]1Oc2c(NC(=O)NC(C)C)cccc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44496658	phase I
BRD-K02598395	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44496732	phase I
BRD-K89451495	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@H](C)[C@@H](CN(C)C)Oc12)[C@@H](C)CO	CID:44496738	phase I
BRD-K08519668	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44496756	phase I
BRD-K78780288	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44496758	phase I
BRD-K24149610	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44496769	phase I
BRD-K34447376	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44496773	phase I
BRD-K41296766	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:44496776	phase I
BRD-K30962405	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)c3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44496792	phase I
BRD-K40988761	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44496819	phase I
BRD-K41779994	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44496822	phase I
BRD-K81778946	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44496827	phase I
BRD-K76825413	COc1ccccc1NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3	CID:44496828	phase I
BRD-K45231869	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44496832	phase I
BRD-K95761590	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(O)cc2)OCc3cn(CCCC1=O)nn3	CID:44496833	phase I
BRD-K92125320	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44496834	phase I
BRD-K28480589	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ncc(cc4C1=O)c5ccc(F)cc5	CID:44496843	phase I
BRD-K79826210	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C#N)cc2)Oc3ncc(C#Cc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44496852	phase I
BRD-K05209891	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)Oc3ncc(C#Cc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44496854	phase I
BRD-K89344180	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44496867	phase I
BRD-K62019457	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44496876	phase I
BRD-K93672499	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44496893	phase I
BRD-K08922114	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44496894	phase I
BRD-K24026396	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44496896	phase I
BRD-K00643888	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44496898	phase I
BRD-K87063901	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:44496903	phase I
BRD-K09186736	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44496918	phase I
BRD-K37618507	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)Nc4c(C)noc4C)cccc3C1=O	CID:44496991	phase I
BRD-K95673125	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44497048	phase I
BRD-K75845944	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44497076	phase I
BRD-K85102293	COc1ccc(cc1)S(=O)(=O)Nc2cccc3C(=O)N(C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c4ccc(OC)cc4)Oc23)[C@H](C)CO	CID:44497120	phase I
BRD-K04289865	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44497175	phase I
BRD-K57280824	CNC[C@H]1Oc2c(NC(=O)NC(C)C)cccc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44497178	phase I
BRD-K41866979	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44497202	phase I
BRD-K69492024	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44497244	phase I
BRD-K98758861	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44497248	phase I
BRD-K92978552	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44497250	phase I
BRD-K51106788	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44497251	phase I
BRD-K85967137	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44497252	phase I
BRD-K74472944	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44497254	phase I
BRD-K70345064	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44497255	phase I
BRD-K29285912	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44497256	phase I
BRD-K50079182	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44497267	phase I
BRD-K46558254	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44497281	phase I
BRD-K70711508	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44497291	phase I
BRD-K72913684	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44497297	phase I
BRD-K02314198	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44497303	phase I
BRD-K57200229	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44497312	phase I
BRD-K89144439	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44497318	phase I
BRD-K86191692	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44497321	phase I
BRD-K25902954	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44497328	phase I
BRD-K22630935	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44497341	phase I
BRD-K02772785	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44497349	phase I
BRD-K34174785	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44497365	phase I
BRD-K89966732	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44497370	phase I
BRD-K64577556	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3CC1=O	CID:44497382	phase I
BRD-K24014699	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)Nc5cccc6ccccc56)cc4CC1=O	CID:44497383	phase I
BRD-K37073485	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44497398	phase I
BRD-K43256821	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)Nc4ccccc4)cccc3C1=O	CID:44497409	phase I
BRD-K27367875	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(cccc4C1=O)N(C)C	CID:44497424	phase I
BRD-K53592093	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NS(=O)(=O)c4ccc(F)cc4)cccc3C1=O	CID:44497469	phase I
BRD-K78013650	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44497470	phase I
BRD-K30941218	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C	CID:44497476	phase I
BRD-K23103632	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44497484	phase I
BRD-K46176518	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3c(NC(=O)c4cnccn4)cccc3C1=O	CID:44497487	phase I
BRD-K61158263	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@@H](C)[C@@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@@H](C)CO)cc1	CID:44497517	phase I
BRD-K39958166	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44497527	phase I
BRD-K82004360	CNC[C@H]1Oc2c(NC(=O)NC(C)C)cccc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44497542	phase I
BRD-K70974948	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)C4CC4)cccc3C1=O	CID:44497549	phase I
BRD-K31290665	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)CCCN(C)C)cc2C1=O	CID:44497608	phase I
BRD-K30882656	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44497639	phase I
BRD-K40956802	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44497649	phase I
BRD-K71459980	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCCN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44497655	phase I
BRD-K34556006	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44497710	phase I
BRD-K93104606	COc1ccc(CN(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44497719	phase I
BRD-K60379529	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44497778	phase I
BRD-K85123403	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44497793	phase I
BRD-K09231502	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:44497811	phase I
BRD-K26381032	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44497835	phase I
BRD-K01987080	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@H](C)[C@@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@@H](C)CO)cc1	CID:44497876	phase I
BRD-K68038686	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44497912	phase I
BRD-K24139908	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44497969	phase I
BRD-K69760878	CC(C)NC(=O)Nc1cccc2C(=O)N(C[C@@H](C)[C@@H](CN(C)C)Oc12)[C@H](C)CO	CID:44497988	phase I
BRD-K33619512	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:44498007	phase I
BRD-K02924457	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44498015	phase I
BRD-K49738502	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5ccccc5)cc4C1=O	CID:44498046	phase I
BRD-K09517037	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44498086	phase I
BRD-K86947329	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44498109	phase I
BRD-K26188625	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCC2)OCc3cn(CCCC1=O)nn3	CID:44498140	phase I
BRD-K01121544	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44498144	phase I
BRD-K43160803	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44498145	phase I
BRD-K56379049	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3cccnc3c2)OCc4cnnn4CCCC1=O	CID:44498146	phase I
BRD-K41303952	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44498151	phase I
BRD-K67433402	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44498166	phase I
BRD-K15233676	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44498170	phase I
BRD-K99380810	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44498186	phase I
BRD-K17449871	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44498208	phase I
BRD-K34387287	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44498225	phase I
BRD-K21691498	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44498235	phase I
BRD-K78596368	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44498245	phase I
BRD-K30511626	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc(F)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44498246	phase I
BRD-K99395085	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44498248	phase I
BRD-K58784778	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44498255	phase I
BRD-K99381377	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44498441	phase I
BRD-K07951922	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44498472	phase I
BRD-K09703570	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44498525	phase I
BRD-K01700755	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCc2cn(CCCC1=O)nn2	CID:44498541	phase I
BRD-K77229048	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44498543	phase I
BRD-K48066866	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44498546	phase I
BRD-K60002786	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)c(OC)c1	CID:44498548	phase I
BRD-K78173425	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)c1	CID:44498549	phase I
BRD-K88299492	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44498550	phase I
BRD-K36959991	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44498557	phase I
BRD-K36289461	COc1cccc(CN(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)c1	CID:44498558	phase I
BRD-K42790744	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44498559	phase I
BRD-K35836352	COc1ccc(CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44498560	phase I
BRD-K75023015	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)OCc4cn(CCCC1=O)nn4	CID:44498562	phase I
BRD-K23060602	CCCN(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44498581	phase I
BRD-K45818044	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44498587	phase I
BRD-K48243375	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44498598	phase I
BRD-K61001510	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44498600	phase I
BRD-K55612480	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44498603	phase I
BRD-K11795542	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44498604	phase I
BRD-K36654803	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44498613	phase I
BRD-K46171503	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:44498621	phase I
BRD-K21516480	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44498628	phase I
BRD-K82161520	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44498639	phase I
BRD-K96539190	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44498644	phase I
BRD-K19181733	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44498648	phase I
BRD-K65165610	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44498654	phase I
BRD-K25029498	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44498665	phase I
BRD-K51511759	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44498675	phase I
BRD-K96477379	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44498677	phase I
BRD-K09404347	CNC[C@H]1Oc2c(NC(=O)NC(C)C)cccc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44498703	phase I
BRD-K51216807	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44498722	phase I
BRD-K14328427	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44498818	phase I
BRD-K29916225	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44498824	phase I
BRD-K16984096	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44498906	phase I
BRD-K59728381	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NS(=O)(=O)c4ccc(Cl)cc4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44498994	phase I
BRD-K32485462	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44499001	phase I
BRD-K88714443	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)Nc4ccc(cc4)C(F)(F)F)cccc3C1=O	CID:44499061	phase I
BRD-K74949371	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3c(NC(=O)c4ccc(cc4)c5nccs5)cccc3C1=O	CID:44499123	phase I
BRD-K03203188	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@H](C)[C@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@H](C)CO)cc1	CID:44499176	phase I
BRD-K04046003	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)c4nc5ccccc5s4)cccc3C1=O	CID:44499177	phase I
BRD-K74506886	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3c(NC(=O)c4cnccn4)cccc3C1=O	CID:44499215	phase I
BRD-K31755488	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(cccc4C1=O)N(C)C	CID:44499268	phase I
BRD-K68191033	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3c(NC(=O)Nc4ccc5OCOc5c4)cccc3C1=O	CID:44499430	phase I
BRD-K78603557	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44499449	phase I
BRD-K14600622	COc1ccc(NC(=O)N(C)C[C@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44499486	phase I
BRD-K22828860	COc1ccc(cc1)S(=O)(=O)Nc2cccc3C(=O)N(C[C@H](C)[C@H](CN(C)C(=O)NC4CCCCC4)Oc23)[C@H](C)CO	CID:44499516	phase I
BRD-K96787835	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44499520	phase I
BRD-K69159985	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:44499548	phase I
BRD-K88217904	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)Nc4ccc(F)cc4)cccc3C1=O	CID:44499565	phase I
BRD-K78524708	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44499583	phase I
BRD-K36767861	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)Oc3c(NC(=O)C4CC4)cccc3C1=O	CID:44499704	phase I
BRD-K29138830	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44499735	phase I
BRD-K44302407	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO)N(C)C	CID:44499743	phase I
BRD-K18074178	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)Nc4ccccc4)cccc3C1=O	CID:44499857	phase I
BRD-K21786893	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)c4ccncc4)cccc3C1=O	CID:44499873	phase I
BRD-K88556033	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3c(NC(=O)NC4CCCCC4)cccc3C1=O	CID:44499885	phase I
BRD-K27818252	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(cccc4C1=O)N(C)C	CID:44499947	phase I
BRD-K64058329	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44500012	phase I
BRD-K37262906	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@@H](C)[C@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@@H](C)CO)cc1	CID:44500041	phase I
BRD-K19418153	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(cccc4C1=O)N(C)C	CID:44500046	phase I
BRD-K39289507	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:44500050	phase I
BRD-K14345135	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44500080	phase I
BRD-K65536202	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(cccc4C1=O)N(C)C	CID:44500117	phase I
BRD-K93138145	COc1ccc(NC(=O)Nc2cccc3C(=O)N(C[C@@H](C)[C@@H](CN(C)Cc4ccc5OCOc5c4)Oc23)[C@H](C)CO)cc1	CID:44500128	phase I
BRD-K16969565	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)c4cc(C)nn4C)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44500152	phase I
BRD-K31746020	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3c(NC(=O)NC4CCCCC4)cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44500181	phase I
BRD-K95564984	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44500202	phase I
BRD-K30548766	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2C1=O	CID:44500224	phase I
BRD-K63154426	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(cc3CC1=O)N(C)C	CID:44500308	phase I
BRD-K89915754	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:44500334	phase I
BRD-K86071888	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44500335	phase I
BRD-K15987804	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44500358	phase I
BRD-K44999613	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44500384	phase I
BRD-K19593010	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44500394	phase I
BRD-K41429297	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44500411	phase I
BRD-K29251608	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3C1=O	CID:44500434	phase I
BRD-K15672523	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:44500453	phase I
BRD-K15030062	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(cccc3C(=O)N(C[C@H]2C)[C@H](C)CO)N(C)C	CID:44500461	phase I
BRD-K66191602	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc4OCOc4c3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44500488	phase I
BRD-K68945047	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44500591	phase I
BRD-K35429092	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44500631	phase I
BRD-K36489877	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44500658	phase I
BRD-K19131810	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:44500663	phase I
BRD-K14868367	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3c(NC(=O)Nc4ccccc4)cccc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44500706	phase I
BRD-K44766290	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44500741	phase I
BRD-K14799717	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44500754	phase I
BRD-K36754064	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44500828	phase I
BRD-K16370162	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44500836	phase I
BRD-K80848948	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44500840	phase I
BRD-K46098747	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C	CID:44500855	phase I
BRD-K99958302	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44500857	phase I
BRD-K24991044	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44500869	phase I
BRD-K86312065	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44500947	phase I
BRD-K23657553	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)C5CCCCC5)cc4CC1=O	CID:44500949	phase I
BRD-K93610587	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc4OCOc4c3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44500987	phase I
BRD-K89682702	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)CC3CC3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44500998	phase I
BRD-K76381171	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44501031	phase I
BRD-K89493095	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44501062	phase I
BRD-K11169037	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44501089	phase I
BRD-K47163377	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44501097	phase I
BRD-K20501513	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44501118	phase I
BRD-K95392673	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44501121	phase I
BRD-K90446118	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4C1=O	CID:44501122	phase I
BRD-K60588371	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44501123	phase I
BRD-K02279849	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc4OCOc4c3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44501153	phase I
BRD-K93285993	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44501220	phase I
BRD-K07907451	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44501237	phase I
BRD-K58096890	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44501313	phase I
BRD-K67559633	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3CC1=O	CID:44501373	phase I
BRD-K10062203	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:44501417	phase I
BRD-K24217168	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44501445	phase I
BRD-K68597821	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44501475	phase I
BRD-K91063002	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44501482	phase I
BRD-K90281509	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44501519	phase I
BRD-K55210983	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44501521	phase I
BRD-K02008913	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44501522	phase I
BRD-K33005877	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44501523	phase I
BRD-K30509186	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44501547	phase I
BRD-K96659448	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44501577	phase I
BRD-K62222886	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44501586	phase I
BRD-K27064849	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44501750	phase I
BRD-K51846078	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44501759	phase I
BRD-K07881060	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44501775	phase I
BRD-K61606206	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44501786	phase I
BRD-K50846154	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44501789	phase I
BRD-K41526317	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44501790	phase I
BRD-K66888355	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44501791	phase I
BRD-K73674426	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)CC4CC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44501793	phase I
BRD-K42694358	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44501797	phase I
BRD-K55073475	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44501798	phase I
BRD-K68937023	COc1ccc(NC(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44501811	phase I
BRD-K98714523	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:44501814	phase I
BRD-K72042177	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44501831	phase I
BRD-K30795336	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)Cc4ccc(cc4)C(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)Cc3c2)cc1	CID:44501884	phase I
BRD-K81332148	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44501897	phase I
BRD-K87072268	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44501933	phase I
BRD-K48835133	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc4OCOc4c3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44501978	phase I
BRD-K23117210	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44501994	phase I
BRD-K03358980	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44502032	phase I
BRD-K81218586	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44502164	phase I
BRD-K58536094	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44502184	phase I
BRD-K82729346	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:44502203	phase I
BRD-K07270511	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44502210	phase I
BRD-K80439608	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44502213	phase I
BRD-K03707297	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44502215	phase I
BRD-K30940328	COc1ccc(NC(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44502225	phase I
BRD-K91395443	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44502236	phase I
BRD-K70647219	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44502244	phase I
BRD-K73602693	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44502292	phase I
BRD-K33597548	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:44502348	phase I
BRD-K51530321	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44502358	phase I
BRD-K19198293	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44502376	phase I
BRD-K04458934	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44502400	phase I
BRD-K86043715	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44502461	phase I
BRD-K37669227	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44502466	phase I
BRD-K12117859	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44502468	phase I
BRD-K36864553	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44502476	phase I
BRD-K00547540	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44502485	phase I
BRD-K30854557	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44502556	phase I
BRD-K89406814	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44502578	phase I
BRD-K45092764	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44502612	phase I
BRD-K38885465	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44502654	phase I
BRD-K29162128	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44502673	phase I
BRD-K50916779	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44502688	phase I
BRD-K90646778	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44502701	phase I
BRD-K42427050	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44502708	phase I
BRD-K60144416	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44502715	phase I
BRD-K18396390	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:44502737	phase I
BRD-K73664775	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44502750	phase I
BRD-K23535251	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:44502756	phase I
BRD-K62970326	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44502813	phase I
BRD-K95090559	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44502836	phase I
BRD-K47558670	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:44502838	phase I
BRD-K85886293	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44502845	phase I
BRD-K65148580	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44502929	phase I
BRD-K90234489	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NC(=O)Nc5ccccc5)cc4C1=O	CID:44502951	phase I
BRD-K66608846	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44502953	phase I
BRD-K21658057	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44502964	phase I
BRD-K71404640	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44502971	phase I
BRD-K05677905	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:44502986	phase I
BRD-K46769156	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44502996	phase I
BRD-K77144489	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)Cc4ccc(cc4)C(F)(F)F)[C@H](C)CN([C@H](C)CO)C(=O)Cc3c2)cc1	CID:44503006	phase I
BRD-K08043379	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44503014	phase I
BRD-K00689442	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44503065	phase I
BRD-K10709111	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44503071	phase I
BRD-K15672359	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)CC3CC3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44503093	phase I
BRD-K17730221	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44503122	phase I
BRD-K59939374	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44503125	phase I
BRD-K08130208	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)Cc3ccc(Cl)c(Cl)c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44503128	phase I
BRD-K81417919	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44503145	phase I
BRD-K87063646	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44503185	phase I
BRD-K28288650	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(cc3CC1=O)N(C)C	CID:44503242	phase I
BRD-K30409687	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc4OCOc4c3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44503248	phase I
BRD-K34255700	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)c3ccccc3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44503301	phase I
BRD-K18294324	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44503309	phase I
BRD-K74711637	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)C(=O)Nc4ccccc4)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc3c2)cc1	CID:44503361	phase I
BRD-K97440728	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44503363	phase I
BRD-K65514600	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44503376	phase I
BRD-K87520488	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44503391	phase I
BRD-K91813753	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44503445	phase I
BRD-K69286267	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:44503471	phase I
BRD-K24528445	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44503480	phase I
BRD-K89401337	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44503492	phase I
BRD-K23607904	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44503517	phase I
BRD-K42057752	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44503549	phase I
BRD-K82015643	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)c3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44503579	phase I
BRD-K76712687	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:44503602	phase I
BRD-K36910796	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44503610	phase I
BRD-K68326515	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44503616	phase I
BRD-K18415753	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44503624	phase I
BRD-K61776140	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](C)CCCCO[C@H](CN(C)Cc4ccc(Cl)c(Cl)c4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44503649	phase I
BRD-K67829818	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44503657	phase I
BRD-K91257617	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44503658	phase I
BRD-K08221563	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44503684	phase I
BRD-K57487331	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44503688	phase I
BRD-K02109522	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44503689	phase I
BRD-K17660756	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44503697	phase I
BRD-K00586388	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44503699	phase I
BRD-K07666543	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44503705	phase I
BRD-K28945051	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3CC(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44503722	phase I
BRD-K64790987	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44503776	phase I
BRD-K40249559	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:44503840	phase I
BRD-K78432605	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44503844	phase I
BRD-K32320888	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44503848	phase I
BRD-K80848452	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44503867	phase I
BRD-K31562577	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3ccc(cc3CC1=O)N(C)C	CID:44503931	phase I
BRD-K58808184	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:44503987	phase I
BRD-K46496627	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44503990	phase I
BRD-K17197507	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44504011	phase I
BRD-K31593084	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:44504018	phase I
BRD-K88243749	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44504025	phase I
BRD-K76352008	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:44504031	phase I
BRD-K98004941	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44504041	phase I
BRD-K23263381	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44504058	phase I
BRD-K08293924	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44504059	phase I
BRD-K82882781	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)c3ccccc3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44504109	phase I
BRD-K25980346	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:44504116	phase I
BRD-K60454961	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44504286	phase I
BRD-K27472340	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44504293	phase I
BRD-K56621049	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44504295	phase I
BRD-K75669394	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCCCC[C@@H](C)Oc2ccc(cc2C1=O)N(C)C	CID:44504316	phase I
BRD-K36165258	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44504318	phase I
BRD-K91579227	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@@H](C)Oc4ccc(NS(=O)(=O)c5cccs5)cc4C1=O	CID:44504326	phase I
BRD-K24523081	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44504331	phase I
BRD-K02575886	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44504336	phase I
BRD-K20278954	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:44504350	phase I
BRD-K48673964	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3CC(=O)N(C[C@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44504411	phase I
BRD-K36864604	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:44504418	phase I
BRD-K67192456	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44504449	phase I
BRD-K70272514	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C1=O	CID:44504533	phase I
BRD-K40471847	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44504553	phase I
BRD-K86845397	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:44504576	phase I
BRD-K98168655	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:44504594	phase I
BRD-K83216232	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:44504601	phase I
BRD-K52306726	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:44504636	phase I
BRD-K65158783	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44504669	phase I
BRD-K68253248	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44504736	phase I
BRD-K37495811	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44504748	phase I
BRD-K18727181	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44504802	phase I
BRD-K34051200	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc4OCOc4c3)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44504807	phase I
BRD-K85540993	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44504839	phase I
BRD-K60554389	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)c3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44504873	phase I
BRD-K96403486	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)C(=O)Nc4ccc(OC)cc4)[C@H](C)CN([C@H](C)CO)C(=O)Cc3c2)cc1	CID:44504880	phase I
BRD-K86981922	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:44504912	phase I
BRD-K34522271	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44504916	phase I
BRD-K66809950	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44504919	phase I
BRD-K55910052	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44504920	phase I
BRD-K61044449	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44504923	phase I
BRD-K49123127	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cnnn3CCCC1=O	CID:44504924	phase I
BRD-K08460070	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44504925	phase I
BRD-K87004592	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cnnn3CCCC1=O	CID:44504928	phase I
BRD-K34966059	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44504930	phase I
BRD-K10232830	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44504931	phase I
BRD-K86569253	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cnnn3CCCC1=O	CID:44504932	phase I
BRD-K55860636	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44504933	phase I
BRD-K86390887	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44504934	phase I
BRD-K46033477	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3	CID:44504935	phase I
BRD-K52240583	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cnnn3CCCC1=O	CID:44504937	phase I
BRD-K23108726	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44504943	phase I
BRD-K65548588	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44504944	phase I
BRD-K86895142	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44504945	phase I
BRD-K48336086	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)OCc2cnnn2CCCC1=O	CID:44504950	phase I
BRD-K56654013	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCc2cn(CCCC1=O)nn2	CID:44504954	phase I
BRD-K86466947	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44504955	phase I
BRD-K00468432	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3	CID:44504957	phase I
BRD-K68246261	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44504958	phase I
BRD-K54395291	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3	CID:44504960	phase I
BRD-K77140830	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2cn(CCCC1=O)nn2	CID:44504963	phase I
BRD-K08212968	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44504965	phase I
BRD-K66848791	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cnnn3CCCC1=O	CID:44504967	phase I
BRD-K36674158	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44504971	phase I
BRD-K62875000	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44504973	phase I
BRD-K51569524	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44504979	phase I
BRD-K00977230	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44504982	phase I
BRD-K16769896	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44504984	phase I
BRD-K26087938	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44504985	phase I
BRD-K16079243	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44504986	phase I
BRD-K29128208	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44504987	phase I
BRD-K45937204	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44504988	phase I
BRD-K03321770	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Oc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44504989	phase I
BRD-K57987292	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44504990	phase I
BRD-K02257023	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44504994	phase I
BRD-K61823824	CC(C)OC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@@H](C)CO)nn2	CID:44504998	phase I
BRD-K37487131	COc1ccc(OC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)cc1	CID:44504999	phase I
BRD-K96743424	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505000	phase I
BRD-K63989441	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44505001	phase I
BRD-K57339160	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44505002	phase I
BRD-K26581628	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505004	phase I
BRD-K52947657	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C)OCc3cnnn3CCCC1=O	CID:44505017	phase I
BRD-K77901830	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44505019	phase I
BRD-K12957211	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44505020	phase I
BRD-K33755346	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3cn(CCCC1=O)nn3	CID:44505023	phase I
BRD-K31704218	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505027	phase I
BRD-K92841050	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505028	phase I
BRD-K71254735	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(C)c2)OCc3cn(CCCC1=O)nn3	CID:44505032	phase I
BRD-K39767907	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3cnnn3CCCC1=O	CID:44505033	phase I
BRD-K12057275	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44505035	phase I
BRD-K51762600	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505038	phase I
BRD-K01795516	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(O)c2)OCc3cn(CCCC1=O)nn3	CID:44505039	phase I
BRD-K25348850	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(O)c2)OCc3cn(CCCC1=O)nn3	CID:44505040	phase I
BRD-K32040163	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3cn(CCCC1=O)nn3	CID:44505041	phase I
BRD-K45740917	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505043	phase I
BRD-K14396623	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505045	phase I
BRD-K45735142	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505046	phase I
BRD-K45843042	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505047	phase I
BRD-K51197994	COc1cccc(CN(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3)c1	CID:44505052	phase I
BRD-K36217065	COc1cccc(CN(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:44505053	phase I
BRD-K81821583	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCc3cnnn3CCCC1=O	CID:44505056	phase I
BRD-K60047946	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44505060	phase I
BRD-K49510739	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44505061	phase I
BRD-K63733272	COc1cccc(CN(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)c1	CID:44505062	phase I
BRD-K14738608	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4cnnn4CCCC1=O	CID:44505065	phase I
BRD-K10991887	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505066	phase I
BRD-K56987347	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505070	phase I
BRD-K78824440	CNC[C@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44505071	phase I
BRD-K80995081	CNC[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44505072	phase I
BRD-K52199185	CNC[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44505073	phase I
BRD-K39685923	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ncc(cc3C1=O)c4cc5ccccc5o4	CID:44505076	phase I
BRD-K83879237	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4ncc(cc4C1=O)c5cccc(c5)C(F)(F)F	CID:44505087	phase I
BRD-K54558492	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:44505109	phase I
BRD-K14989228	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505113	phase I
BRD-K07278381	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505118	phase I
BRD-K19973268	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cn(CCCC1=O)nn3	CID:44505119	phase I
BRD-K42269438	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cnnn3CCCC1=O	CID:44505120	phase I
BRD-K28907425	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cnnn3CCCC1=O	CID:44505122	phase I
BRD-K24396417	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc3OCCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505124	phase I
BRD-K83481956	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44505130	phase I
BRD-K77323800	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44505133	phase I
BRD-K07833219	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3	CID:44505136	phase I
BRD-K92135892	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505137	phase I
BRD-K40099330	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3	CID:44505139	phase I
BRD-K21153751	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44505142	phase I
BRD-K60659225	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44505148	phase I
BRD-K75965029	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C)c2)OCc3cn(CCCC1=O)nn3	CID:44505149	phase I
BRD-K74055572	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44505153	phase I
BRD-K91443444	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3	CID:44505159	phase I
BRD-K42466986	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44505160	phase I
BRD-K41880142	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44505163	phase I
BRD-K02724364	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3	CID:44505164	phase I
BRD-K48005659	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44505171	phase I
BRD-K70274124	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCc3cnnn3CCCC1=O	CID:44505175	phase I
BRD-K02960110	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44505177	phase I
BRD-K47247219	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505180	phase I
BRD-K52862624	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3cnnn3CCCC1=O	CID:44505181	phase I
BRD-K25660189	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccccc2)OCc3cnnn3CCCC1=O	CID:44505183	phase I
BRD-K27371551	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505188	phase I
BRD-K17266676	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cnnn4CCCC1=O	CID:44505189	phase I
BRD-K49457424	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccccc2)OCc3cnnn3CCCC1=O	CID:44505195	phase I
BRD-K37556799	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44505198	phase I
BRD-K56242781	CC(C)OC(=O)N(C)C[C@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44505199	phase I
BRD-K18942395	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cnnn4CCCC1=O	CID:44505202	phase I
BRD-K64100337	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cnnn4CCCC1=O	CID:44505203	phase I
BRD-K41005527	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505204	phase I
BRD-K61872587	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cnnn3CCCC1=O	CID:44505208	phase I
BRD-K07417570	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCc4cnnn4CCCC1=O	CID:44505210	phase I
BRD-K59995645	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44505213	phase I
BRD-K92186740	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)OCc3cn(CCCC1=O)nn3	CID:44505219	phase I
BRD-K68359762	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C)OCc3cnnn3CCCC1=O	CID:44505225	phase I
BRD-K82396235	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44505227	phase I
BRD-K63270352	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(C)c2)OCc3cn(CCCC1=O)nn3	CID:44505228	phase I
BRD-K28638920	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3cn(CCCC1=O)nn3	CID:44505229	phase I
BRD-K04518829	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44505231	phase I
BRD-K27986637	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505237	phase I
BRD-K33384411	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505239	phase I
BRD-K08995965	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505242	phase I
BRD-K15428056	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505243	phase I
BRD-K07452532	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505244	phase I
BRD-K48279074	COc1cccc(CN(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:44505245	phase I
BRD-K58134288	COc1cccc(CN(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)c1	CID:44505250	phase I
BRD-K08185175	COc1cccc(CN(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:44505252	phase I
BRD-K54834493	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505257	phase I
BRD-K69158405	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505258	phase I
BRD-K33407589	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505259	phase I
BRD-K61998715	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505262	phase I
BRD-K92959281	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)Oc3ncc(cc3C1=O)c4cc5ccccc5o4	CID:44505298	phase I
BRD-A08778300	CCCC(O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3ccc4OCOc4c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44505316	phase I
BRD-K86770334	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505325	phase I
BRD-K52117630	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cnnn3CCCC1=O	CID:44505326	phase I
BRD-K12331173	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505327	phase I
BRD-K76100122	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cn(CCCC1=O)nn3	CID:44505328	phase I
BRD-K33760789	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44505336	phase I
BRD-K72391864	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3cnnn3CCCC1=O	CID:44505337	phase I
BRD-K03155021	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44505339	phase I
BRD-K83437201	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCc3cnnn3CCCC1=O	CID:44505344	phase I
BRD-K26733240	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3cnnn3CCCC1=O	CID:44505347	phase I
BRD-K25595086	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44505356	phase I
BRD-K62980388	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44505363	phase I
BRD-K65067638	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3ccccc3c2)OCc4cn(CCCC1=O)nn4	CID:44505365	phase I
BRD-K82906409	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2cnnn2CCCC1=O	CID:44505368	phase I
BRD-K57341983	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3	CID:44505378	phase I
BRD-K31866446	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44505379	phase I
BRD-K46370825	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505383	phase I
BRD-K75755028	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505387	phase I
BRD-K28055782	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(cc2)N3CCN(C)CC3)OCc4cnnn4CCCC1=O	CID:44505394	phase I
BRD-K65837806	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44505398	phase I
BRD-K94834134	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505401	phase I
BRD-K01916633	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44505404	phase I
BRD-K19016577	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505406	phase I
BRD-K61953981	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44505407	phase I
BRD-K80564983	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCC2)OCc3cn(CCCC1=O)nn3	CID:44505413	phase I
BRD-K77873562	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cnnn4CCCC1=O	CID:44505414	phase I
BRD-K53839527	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4cnnn4CCCC1=O	CID:44505415	phase I
BRD-K68458302	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cnnn4CCCC1=O	CID:44505421	phase I
BRD-K60679910	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCC2)OCc3cnnn3CCCC1=O	CID:44505423	phase I
BRD-K12682252	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4cnnn4CCCC1=O	CID:44505424	phase I
BRD-K49676673	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cnnn4CCCC1=O	CID:44505428	phase I
BRD-K61553312	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)c(OC)c1	CID:44505436	phase I
BRD-K72783054	COc1ccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3)c(OC)c1	CID:44505438	phase I
BRD-K16670827	COc1ccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)c(OC)c1	CID:44505441	phase I
BRD-K50754265	COc1cccc(NC(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:44505459	phase I
BRD-K62853937	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505460	phase I
BRD-K31045868	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3	CID:44505465	phase I
BRD-K30658064	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505473	phase I
BRD-K11582139	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3cn(CCCC1=O)nn3	CID:44505474	phase I
BRD-K50146767	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3cnnn3CCCC1=O	CID:44505476	phase I
BRD-K62427254	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3cn(CCCC1=O)nn3	CID:44505478	phase I
BRD-K59490275	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505479	phase I
BRD-K09407750	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(O)cc2)OCc3cnnn3CCCC1=O	CID:44505480	phase I
BRD-K98339888	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(O)cc2)OCc3cnnn3CCCC1=O	CID:44505490	phase I
BRD-K68350686	COc1ccc(CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44505498	phase I
BRD-K62567808	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505500	phase I
BRD-K49313348	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ncc(cc4C1=O)c5cccc(F)c5	CID:44505502	phase I
BRD-K13205342	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505531	phase I
BRD-K84277608	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cn(CCCC1=O)nn3	CID:44505532	phase I
BRD-K69343050	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3cnnn3CCCC1=O	CID:44505534	phase I
BRD-K85449516	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44505537	phase I
BRD-K43852369	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505542	phase I
BRD-K78513625	COc1ccc(OC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)cc1	CID:44505550	phase I
BRD-K68741898	CC(C)COC(=O)N(C)C[C@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44505553	phase I
BRD-K56349799	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505555	phase I
BRD-K99470298	COc1ccc(OC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)cc1	CID:44505558	phase I
BRD-K35964632	CCOC(=O)N(C)C[C@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44505560	phase I
BRD-K60840479	CC(C)OC(=O)N(C)C[C@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44505564	phase I
BRD-K60321290	COc1ccc(OC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)cc1	CID:44505571	phase I
BRD-K75710654	CCOC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@H](C)CO)nn2	CID:44505572	phase I
BRD-K39963927	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2ccc3ccccc3c2)OCc4cnnn4CCCC1=O	CID:44505575	phase I
BRD-K04648846	CC(C)OC(=O)N(C)C[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44505579	phase I
BRD-K95105171	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505581	phase I
BRD-K22865069	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cnnn4CCCC1=O	CID:44505584	phase I
BRD-K19845538	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505585	phase I
BRD-K19969618	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cnnn4CCCC1=O	CID:44505586	phase I
BRD-K60002680	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)OCc2ccccc2)OCc3cnnn3CCCC1=O	CID:44505587	phase I
BRD-K80185984	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cnnn4CCCC1=O	CID:44505588	phase I
BRD-K47571551	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505593	phase I
BRD-K12440008	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3cn(CCCC1=O)nn3	CID:44505594	phase I
BRD-K68746558	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3cn(CCCC1=O)nn3	CID:44505596	phase I
BRD-K76703685	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505597	phase I
BRD-K38618007	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3cn(CCCC1=O)nn3	CID:44505599	phase I
BRD-K40294449	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505602	phase I
BRD-K67217705	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)N3CCCCC3)OCc4cnnn4CCCC1=O	CID:44505603	phase I
BRD-K35103917	COc1ccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)cc1	CID:44505604	phase I
BRD-K44746563	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505605	phase I
BRD-K20617704	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505606	phase I
BRD-K18236913	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cnnn4CCCC1=O	CID:44505607	phase I
BRD-K55775078	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505608	phase I
BRD-K48211485	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505614	phase I
BRD-K86194107	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505615	phase I
BRD-K62528537	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505616	phase I
BRD-K59453031	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505619	phase I
BRD-K20931972	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505621	phase I
BRD-K69011607	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505622	phase I
BRD-K64560329	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cnnn3CCCC1=O	CID:44505623	phase I
BRD-K21305828	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cnnn3CCCC1=O	CID:44505624	phase I
BRD-K26653603	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505625	phase I
BRD-K62558637	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505627	phase I
BRD-K58010565	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505628	phase I
BRD-K83456424	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3	CID:44505631	phase I
BRD-K27835062	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)c1	CID:44505633	phase I
BRD-K46322935	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505634	phase I
BRD-K14214369	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cnnn3CCCC1=O	CID:44505636	phase I
BRD-K04465546	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505642	phase I
BRD-K71625503	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(C)c2)OCc3cnnn3CCCC1=O	CID:44505643	phase I
BRD-K10046096	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3cccnc3c2)OCc4cnnn4CCCC1=O	CID:44505646	phase I
BRD-K44541805	CCCN(C)C[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44505649	phase I
BRD-K89063992	COc1cccc(CN(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)c1	CID:44505652	phase I
BRD-K51106827	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505659	phase I
BRD-K71353148	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505660	phase I
BRD-K27772696	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505661	phase I
BRD-K81042289	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505665	phase I
BRD-K14213456	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)c4cccc(c4)C(F)(F)F	CID:44505678	phase I
BRD-K82067034	COc1ccc(cc1)c2cnc3O[C@@H](CN(C)Cc4cccc(C)c4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44505680	phase I
BRD-K83893121	COc1ccc(cc1)c2cnc3O[C@@H](CN(C)Cc4ccccc4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44505681	phase I
BRD-K86236946	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2ncc(C#Cc3ccccc3)cc2C1=O	CID:44505696	phase I
BRD-K10017294	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:44505702	phase I
BRD-K57406954	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(C)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:44505703	phase I
BRD-A18477699	CCCC(O)C#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)c3ccc(C)cc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44505711	phase I
BRD-K69817449	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3ncc(C#Cc4cccc(F)c4)cc3C1=O	CID:44505716	phase I
BRD-K91743203	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505725	phase I
BRD-K40060703	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3	CID:44505727	phase I
BRD-K94157828	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44505728	phase I
BRD-K70681322	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2cn(CCCC1=O)nn2	CID:44505740	phase I
BRD-K02419152	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44505747	phase I
BRD-K45656768	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cnnn4CCCC1=O	CID:44505750	phase I
BRD-K38587340	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCc3cnnn3CCCC1=O	CID:44505751	phase I
BRD-K70102743	CC(C)COC(=O)N(C)C[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44505755	phase I
BRD-K49594309	CC(C)COC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@H](C)CO)nn2	CID:44505756	phase I
BRD-K42982250	COc1ccc(OC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3)cc1	CID:44505757	phase I
BRD-K58747666	CC(C)COC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@H](C)CO)nn2	CID:44505759	phase I
BRD-K61984373	COc1ccc(OC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)cc1	CID:44505760	phase I
BRD-K47520858	COc1ccc(OC(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44505761	phase I
BRD-K69431670	CC(C)COC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44505762	phase I
BRD-K88876691	CCOC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@H](C)CO)nn2	CID:44505764	phase I
BRD-K53241640	CC(C)OC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@H](C)CO)nn2	CID:44505765	phase I
BRD-K04882719	CCOC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@@H](C)CO)nn2	CID:44505766	phase I
BRD-K77836949	CC(C)COC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@@H](C)CO)nn2	CID:44505768	phase I
BRD-K86546828	COc1ccc(OC(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44505769	phase I
BRD-K01594666	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Oc2cccc3ccccc23)OCc4cn(CCCC1=O)nn4	CID:44505773	phase I
BRD-K06492185	CC(C)OC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@H]1C)[C@H](C)CO)nn2	CID:44505778	phase I
BRD-K93473872	CC(C)OC(=O)N(C)C[C@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44505780	phase I
BRD-K79676802	CCOC(=O)N(C)C[C@@H]1OCc2cn(CCCC(=O)N(C[C@@H]1C)[C@@H](C)CO)nn2	CID:44505782	phase I
BRD-K33961669	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505787	phase I
BRD-K29555302	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4cnnn4CCCC1=O	CID:44505790	phase I
BRD-K21682170	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3cn(CCCC1=O)nn3	CID:44505792	phase I
BRD-K08754235	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3cn(CCCC1=O)nn3	CID:44505796	phase I
BRD-K01187795	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3cnnn3CCCC1=O	CID:44505798	phase I
BRD-K19526326	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3cn(CCCC1=O)nn3	CID:44505800	phase I
BRD-K28927944	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505802	phase I
BRD-K27117623	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4cnnn4CCCC1=O	CID:44505803	phase I
BRD-K22609494	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)cc1	CID:44505807	phase I
BRD-K24075340	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505809	phase I
BRD-K60734771	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505810	phase I
BRD-K96839270	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)cc1	CID:44505811	phase I
BRD-K44900726	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505813	phase I
BRD-K93972090	COc1ccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3)cc1	CID:44505814	phase I
BRD-K42989496	COc1ccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)cc1	CID:44505815	phase I
BRD-K15713006	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505818	phase I
BRD-K48805168	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505827	phase I
BRD-K65064082	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505828	phase I
BRD-K11957311	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505829	phase I
BRD-K09324395	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505831	phase I
BRD-K15713104	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505833	phase I
BRD-K31147195	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3cnnn3CCCC1=O	CID:44505834	phase I
BRD-K62447749	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505835	phase I
BRD-K77053712	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505836	phase I
BRD-K10722141	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(C)(C)C)OCc3cn(CCCC1=O)nn3	CID:44505840	phase I
BRD-K27675859	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505841	phase I
BRD-K24321898	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505844	phase I
BRD-K36726271	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505846	phase I
BRD-K52159901	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(F)c2)OCc3cn(CCCC1=O)nn3	CID:44505849	phase I
BRD-K54864501	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCc4cnnn4CCCC1=O	CID:44505850	phase I
BRD-K48140215	COc1cccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)nn3)c1	CID:44505851	phase I
BRD-K80711156	COc1cccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3)c1	CID:44505852	phase I
BRD-K64788035	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505853	phase I
BRD-K64649802	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cnnn3CCCC1=O	CID:44505856	phase I
BRD-K30398452	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505857	phase I
BRD-K45788890	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505858	phase I
BRD-K26682747	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505859	phase I
BRD-K80112796	COc1ccccc1NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44505860	phase I
BRD-K13614235	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)c1	CID:44505861	phase I
BRD-K63473855	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505862	phase I
BRD-K40958081	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cnnn3CCCC1=O	CID:44505863	phase I
BRD-K89364593	COc1cccc(NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@H](C)CO)nn3)c1	CID:44505864	phase I
BRD-K96708215	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCc3cnnn3CCCC1=O	CID:44505865	phase I
BRD-K37513668	COc1ccccc1NC(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3	CID:44505866	phase I
BRD-K23001296	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3cnnn3CCCC1=O	CID:44505871	phase I
BRD-K05671817	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3cnnn3CCCC1=O	CID:44505872	phase I
BRD-K79561347	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3cn(CCCC1=O)nn3	CID:44505876	phase I
BRD-K72915114	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3cnnn3CCCC1=O	CID:44505879	phase I
BRD-K34800739	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3cnnn3CCCC1=O	CID:44505880	phase I
BRD-K33480200	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)OCc3cnnn3CCCC1=O	CID:44505881	phase I
BRD-K48053776	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(O)c2)OCc3cn(CCCC1=O)nn3	CID:44505883	phase I
BRD-K75869048	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505885	phase I
BRD-K84836616	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505888	phase I
BRD-K14721042	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505889	phase I
BRD-K05684908	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44505891	phase I
BRD-K59501784	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cnnn4CCCC1=O	CID:44505892	phase I
BRD-K28185108	COc1cccc(CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:44505896	phase I
BRD-K99681782	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(O)cc2)OCc3cn(CCCC1=O)nn3	CID:44505898	phase I
BRD-K86573519	COc1cccc(CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:44505899	phase I
BRD-K85807048	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505901	phase I
BRD-K81858438	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44505902	phase I
BRD-K09069264	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505904	phase I
BRD-K53193506	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44505905	phase I
BRD-K33576455	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(C)cc2)OCc3cnnn3CCCC1=O	CID:44505906	phase I
BRD-K96390133	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(C)cc2)OCc3cn(CCCC1=O)nn3	CID:44505909	phase I
BRD-K02885102	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ncc(cc3C1=O)c4cc5ccccc5o4	CID:44505929	phase I
BRD-K75152103	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44505935	phase I
BRD-K64418254	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44505943	phase I
BRD-K09300252	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Oc3ccccc3)cc2)OCc4cnnn4CCCC1=O	CID:44505946	phase I
BRD-K84992272	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505949	phase I
BRD-K50325214	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cnnn3CCCC1=O	CID:44505958	phase I
BRD-K30653168	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2cn(CCCC1=O)nn2	CID:44505961	phase I
BRD-K18793708	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCc3cnnn3CCCC1=O	CID:44505963	phase I
BRD-K75090853	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3cn(CCCC1=O)nn3	CID:44505965	phase I
BRD-K58310742	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3cnnn3CCCC(=O)N(C[C@H]2C)[C@H](C)CO	CID:44505966	phase I
BRD-K07381195	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@@H]2C)[C@H](C)CO)nn3	CID:44505971	phase I
BRD-K92541860	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3cnnn3CCCC1=O	CID:44505973	phase I
BRD-K89595887	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44505974	phase I
BRD-K90534988	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505975	phase I
BRD-K92953664	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44505976	phase I
BRD-K78395012	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44505978	phase I
BRD-K68665543	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(on2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44505980	phase I
BRD-K10580927	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3cn(CCCC1=O)nn3	CID:44505983	phase I
BRD-K92266998	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccccc2)OCc3cn(CCCC1=O)nn3	CID:44505985	phase I
BRD-K69565703	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3ccn(C)c3c2)OCc4cnnn4CCCC1=O	CID:44505995	phase I
BRD-K36691793	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Oc2ccccc2)OCc3cnnn3CCCC1=O	CID:44505996	phase I
BRD-K38706806	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCc3cnnn3CCCC1=O	CID:44505997	phase I
BRD-K39158408	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505998	phase I
BRD-K56711030	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCc3cn(CCCC1=O)nn3	CID:44505999	phase I
BRD-K15489726	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(Oc3ccccn3)c2)OCc4cnnn4CCCC1=O	CID:44506006	phase I
BRD-K97207863	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCC2)OCc3cn(CCCC1=O)nn3	CID:44506011	phase I
BRD-K41574893	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCC2)OCc3cn(CCCC1=O)nn3	CID:44506013	phase I
BRD-K68421632	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44506015	phase I
BRD-K21991827	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44506038	phase I
BRD-K08464293	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCc3cnnn3CCCC1=O	CID:44506039	phase I
BRD-K22598343	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3cnnn3CCCC1=O	CID:44506045	phase I
BRD-K65466135	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cnnn4CCCC1=O	CID:44506046	phase I
BRD-K59578981	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3cn(CCCC1=O)nn3	CID:44506048	phase I
BRD-K02563170	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)OCc4cn(CCCC1=O)nn4	CID:44506052	phase I
BRD-K25180881	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44506054	phase I
BRD-K88628885	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(C)c2)OCc3cn(CCCC1=O)nn3	CID:44506055	phase I
BRD-K03373081	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44506058	phase I
BRD-K03354008	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(O)c2)OCc3cnnn3CCCC1=O	CID:44506060	phase I
BRD-K91424547	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44506061	phase I
BRD-K69511939	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44506064	phase I
BRD-K75990826	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(C)c2)OCc3cn(CCCC1=O)nn3	CID:44506065	phase I
BRD-K50510764	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cn(CCCC1=O)nn3	CID:44506066	phase I
BRD-K32854531	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44506067	phase I
BRD-K74109371	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(C)c2)OCc3cn(CCCC1=O)nn3	CID:44506070	phase I
BRD-K66001964	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(F)(F)F)OCc3cnnn3CCCC1=O	CID:44506071	phase I
BRD-K95798815	CCCN(C)C[C@H]1OCc2cnnn2CCCC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44506074	phase I
BRD-K38594532	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCCOc3c2)OCc4cn(CCCC1=O)nn4	CID:44506075	phase I
BRD-K40458025	COc1cccc(CN(C)C[C@@H]2OCc3cnnn3CCCC(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:44506083	phase I
BRD-K37526858	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44506084	phase I
BRD-K76086682	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44506089	phase I
BRD-K08585415	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)OCc4cn(CCCC1=O)nn4	CID:44506090	phase I
BRD-K64825005	COc1cccc(CN(C)C[C@H]2OCc3cn(CCCC(=O)N(C[C@H]2C)[C@@H](C)CO)nn3)c1	CID:44506091	phase I
BRD-K69792860	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4cnnn4CCCC1=O	CID:44506093	phase I
BRD-K28179362	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc3OCCCOc23)OCc4cnnn4CCCC1=O	CID:44506094	phase I
BRD-K45882653	CNC[C@@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44506095	phase I
BRD-K21363211	CNC[C@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@H](C)CO	CID:44506096	phase I
BRD-K33889536	CNC[C@H]1OCc2cnnn2CCCC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44506097	phase I
BRD-K33903208	COc1cccc(c1)c2cnc3O[C@@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44506100	phase I
BRD-K14678536	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)c4cc5ccccc5o4	CID:44506101	phase I
BRD-K34351329	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44506162	phase I
BRD-K13648806	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4C1=O	CID:44506174	phase I
BRD-K31856043	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44506216	phase I
BRD-K72425572	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44506224	phase I
BRD-K37043259	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4C1=O)N(C)C	CID:44506240	phase I
BRD-K74998149	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4C1=O	CID:44506347	phase I
BRD-K18096819	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4C1=O)N(C)C	CID:44506406	phase I
BRD-K23282736	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4C1=O)N(C)C	CID:44506420	phase I
BRD-K86027709	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4C1=O)N(C)C	CID:44506424	phase I
BRD-K48006774	ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)c2ccccc2	CID:44506448	phase I
BRD-K05204496	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4C1=O	CID:44506549	phase I
BRD-K76938712	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44506577	phase I
BRD-K60297835	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506579	phase I
BRD-K69888333	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44506582	phase I
BRD-K28995283	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)OCCCC[C@@H](C)Oc4ccc(NC(=O)Nc5ccc(F)cc5)cc4C1=O	CID:44506617	phase I
BRD-K20000640	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44506630	phase I
BRD-K02969269	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4CC1=O	CID:44506632	phase I
BRD-K23802982	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44506638	phase I
BRD-K67874737	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)CCN5CCOCC5)cc4CC1=O	CID:44506644	phase I
BRD-K51556300	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44506645	phase I
BRD-K14666757	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44506647	phase I
BRD-K86899078	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44506648	phase I
BRD-K09613355	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44506659	phase I
BRD-K70714754	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4CC1=O	CID:44506661	phase I
BRD-K30094073	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44506671	phase I
BRD-K85818861	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44506674	phase I
BRD-K08725721	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506678	phase I
BRD-K33045404	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44506685	phase I
BRD-K76236182	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44506700	phase I
BRD-K67090983	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44506705	phase I
BRD-K84959002	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(NC(=O)CCCCCC(=O)Nc5ccccc5N)cccc4C1=O	CID:44506712	phase I
BRD-K55827386	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506722	phase I
BRD-K99502566	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44506727	phase I
BRD-K73945663	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506745	phase I
BRD-K89451433	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506765	phase I
BRD-K98739056	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44506777	phase I
BRD-K34092011	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44506804	phase I
BRD-K35638681	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44506808	phase I
BRD-K65904652	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506810	phase I
BRD-K74486276	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506811	phase I
BRD-K48803730	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506823	phase I
BRD-K06009608	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44506826	phase I
BRD-K93127801	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44506841	phase I
BRD-K46373671	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44506860	phase I
BRD-K51791390	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44506865	phase I
BRD-K17968366	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3c(cccc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)N(C)C	CID:44506868	phase I
BRD-K28004127	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44506877	phase I
BRD-K65959597	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44506886	phase I
BRD-K87387614	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44506893	phase I
BRD-K74842589	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44506899	phase I
BRD-K02562327	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44506906	phase I
BRD-K60774644	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)CCC(F)(F)F)cc4CC1=O	CID:44506922	phase I
BRD-K46814258	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44506924	phase I
BRD-K23582869	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44506926	phase I
BRD-K53610452	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4CC1=O	CID:44506930	phase I
BRD-K10010115	Cn1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c3ccccc13	CID:44506989	phase I
BRD-K07005393	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44507045	phase I
BRD-K56196992	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44507063	phase I
BRD-K43579410	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507078	phase I
BRD-K00007652	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44507092	phase I
BRD-K13960193	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507093	phase I
BRD-K30231186	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507103	phase I
BRD-K83816656	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:44507111	phase I
BRD-K48950795	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44507118	phase I
BRD-K55116708	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44507138	phase I
BRD-K88426506	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44507140	phase I
BRD-K80094086	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44507145	phase I
BRD-K93578426	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)c5ccc(cc5)c6nccs6)cccc4C1=O	CID:44507158	phase I
BRD-K78915806	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44507165	phase I
BRD-K98834634	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507216	phase I
BRD-K94412749	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507239	phase I
BRD-K24205443	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507242	phase I
BRD-K53308430	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44507247	phase I
BRD-K39921295	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507250	phase I
BRD-K58479490	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4CC1=O	CID:44507255	phase I
BRD-K49010888	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507260	phase I
BRD-K63801873	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507262	phase I
BRD-K94544211	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507263	phase I
BRD-K14482023	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)C5CCCCC5)cc4CC1=O	CID:44507272	phase I
BRD-K71612465	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507273	phase I
BRD-K52066901	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)C5CC5)cc4CC1=O	CID:44507283	phase I
BRD-K71188711	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507286	phase I
BRD-K74868206	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)Cc3ccc(cc3)C(=O)Nc4ccccc4N)[C@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44507287	phase I
BRD-K67870070	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44507291	phase I
BRD-K95298605	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccccc5)cc4CC1=O	CID:44507299	phase I
BRD-K84450674	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507302	phase I
BRD-K27231781	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NS(=O)(=O)c5ccccc5)cc4CC1=O	CID:44507307	phase I
BRD-K20123385	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4CC1=O	CID:44507309	phase I
BRD-K16995194	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507316	phase I
BRD-K23786503	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5cccc6ccccc56)cc4CC1=O	CID:44507322	phase I
BRD-K58288048	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44507326	phase I
BRD-K35424586	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44507332	phase I
BRD-K86269644	Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc3OCCOc3c2	CID:44507363	phase I
BRD-K88710727	CCOc1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1OCC	CID:44507381	phase I
BRD-K91677732	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44507435	phase I
BRD-K86217343	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507450	phase I
BRD-K04076294	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44507462	phase I
BRD-K05562558	Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(s2)[N+](=O)[O-]	CID:44507495	phase I
BRD-K61105081	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4C1=O)N(C)C	CID:44507712	phase I
BRD-K72505034	C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O	CID:44507722	phase I
BRD-K41668190	Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/C=C/c2ccccc2	CID:44507790	phase I
BRD-K55715339	OCCOc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1	CID:44507806	phase I
BRD-K10649245	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:44507955	phase I
BRD-K53638321	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44507961	phase I
BRD-K53923090	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44507966	phase I
BRD-K51643619	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3c(NC(=O)CCCCCC(=O)Nc4ccccc4N)cccc3C1=O	CID:44507975	phase I
BRD-K82594686	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44507983	phase I
BRD-K03651937	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)C5CCCCC5)cccc4C1=O	CID:44507986	phase I
BRD-K70794677	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)Cc4ccc(cc4)C(=O)Nc5ccccc5N)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44508000	phase I
BRD-K88278225	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc4CC1=O	CID:44508005	phase I
BRD-K08656311	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)C5CCCCC5)cc4CC1=O	CID:44508006	phase I
BRD-K35213218	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44508016	phase I
BRD-K63841267	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)CCC(F)(F)F)cc4CC1=O	CID:44508028	phase I
BRD-K44968548	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44508030	phase I
BRD-K07967886	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NS(=O)(=O)c5cn(C)cn5)cc4CC1=O	CID:44508036	phase I
BRD-A73847809	COc1cccc2cc(oc12)C(=O)C3C(N(C(=O)C3=O)c4nc(C)c(C)s4)c5ccco5	CID:44510770	phase I
BRD-A31801025	CC12CCC3C(CCC4C(=O)C(=O)CCC34C)C2CCC1=O	CID:44511091	phase I
BRD-K04534322	COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(NC(=O)C)c4)c5ccccc53	CID:44511132	phase I
BRD-K08448573	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCC5=O)c6ccccc63	CID:44511133	phase I
BRD-K11181277	OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4csc5ccccc45)cc1	CID:44511151	phase I
BRD-K45842176	COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73	CID:44511205	phase I
BRD-K61175124	COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73	CID:44511206	phase I
BRD-K85580279	OC(=O)c1ccccc1-c1noc(n1)-c1ccccc1F	CID:44517658	phase I
BRD-K44484254	NC(=O)c1ccccc1-c1noc(n1)-c1ccccc1F	CID:44517659	phase I
BRD-A25829966	OC1N2CCCC2=Nc2c(Cl)cc(Cl)cc12	CID:44537690	phase I
BRD-A35141262	OC1N2CCCCC2=Nc2cccc(F)c12	CID:44537691	phase I
BRD-A40560522	OC1N2CCCCCC2=Nc2ccc(Br)cc12	CID:44537693	phase I
BRD-A75106577	OC1N2CCCCCC2=Nc2cccc(F)c12	CID:44537694	phase I
BRD-K25835021	Fc1ccc2nc(SCC(=O)Nc3ccc4CCCc4c3)n(-c3ccccc3)c(=O)c2c1	CID:44537709	phase I
BRD-K38805748	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NS(=O)(=O)c5ccc(C)cc5)cc4CC1=O	CID:44537717	phase I
BRD-K66446284	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44537751	phase I
BRD-K32238524	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44537767	phase I
BRD-K88008216	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:44537781	phase I
BRD-K51302260	Fc1ccc2sn(-c3ccccc3Cl)c(=O)c2c1	CID:44543525	phase I
BRD-K80672993	Nc1cccc(c1)S(=O)(=O)N1CCCN(CC1)S(=O)(=O)c1ccc2OCCOc2c1	CID:44543605	phase I
BRD-K37498076	COc1cc(F)c(c(F)c1)S(=O)(=O)N1CCCN(CC1)S(=O)(=O)c1cccc(N)c1	CID:44543611	phase I
BRD-K15592317	COc1cc2ncnc(-n3nc(nc3N)-c3ccccn3)c2cc1OC	CID:44551660	phase I
BRD-K64979116	Fc1cccc2nc(SCC(=O)Nc3ccc4CCCc4c3)n(-c3ccccc3)c(=O)c12	CID:44552569	phase I
BRD-K61829047	CCOC(=O)\C=C/n1nnc(n1)-c1cccc(Cl)c1	CID:44589607	phase I
BRD-K64606589	CC[C@@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]4CCCCN4C1=O	CID:44593387	phase I
BRD-K92559570	CC(=O)Nc1ccc2sn(-c3ccccc3)c(=O)c2c1	CID:44593869	phase I
BRD-K36153907	FC(F)(F)c1ccc2sn(-c3ccccc3)c(=O)c2c1	CID:44593870	phase I
BRD-K74761218	ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3	CID:44601455	phase I
BRD-K87483782	Clc1ccc(CSc2nnc(-c3ccccn3)n2Cc2ccco2)cc1Cl	CID:44601470	phase I
BRD-K34508425	Cc1ccc(CSc2nnc(-c3ccccn3)n2Cc2cccs2)cc1	CID:44601473	phase I
BRD-K88863622	Clc1ccc(CSc2nnc(-c3ccccn3)n2Cc2cccs2)cc1Cl	CID:44601475	phase I
BRD-K65910366	CCc1ccc(cc1)S(=O)(=O)NCc1ccc(cc1)C(=O)NCCN(C(C)C)Cc1ccccc1	CID:44601476	phase I
BRD-K61717269	Cc1ccc(CNc2nc(nnc2-c2ccccc2)-c2ccccn2)cc1	CID:44602352	phase I
BRD-K81365078	O=C(Cn1sc2ccccc2c1=O)Nc1ccccc1	CID:44602374	phase I
BRD-K39232234	Fc1ccc(NC(=O)Cn2sc3ccccc3c2=O)cc1	CID:44602375	phase I
BRD-K14945759	Brc1ccc(NC(=O)Cn2sc3ccccc3c2=O)cc1	CID:44602376	phase I
BRD-K87446239	O=c1n(sc2cc(ccc12)C#N)-c1ccccc1	CID:44602378	phase I
BRD-K88832793	COc1ccc(cc1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccccc3)n2n1)-c1ccccc1	CID:44602404	phase I
BRD-K82312777	CC(=O)N1CCN(CC1)c1cc(nc2cc(nn12)-c1cccc(Cl)c1)-c1ccccc1	CID:44602405	phase I
BRD-K09138889	O=C(N1CCN(CC1)c1cc(nc2cc(nn12)-c1ccccc1)-c1ccccc1)c1ccoc1	CID:44602406	phase I
BRD-K23531129	Clc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccccc3)n2n1)-c1ccccc1	CID:44602407	phase I
BRD-K73293050	CN1CCN(CC1)c1ccc(Nc2ncc(Cl)c(Oc3cccc(NC(=O)C=C)c3)n2)cc1	CID:44607360	phase I
BRD-K72420232	COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(C)CC1	CID:44607530	phase I
BRD-K73951926	Cc1cccc(C)c1NC(=O)c1ccc(o1)-c1cc(F)ccc1F	CID:44607573	phase I
BRD-K21170640	COc1cccc(OC)c1NC(=O)c1ccc(o1)-c1cc(Cl)ccc1Cl	CID:44607576	phase I
BRD-K99737413	CC(C)c1cccc(C(C)C)c1NC(=O)c1ccc(o1)-c1cc(Cl)ccc1Cl	CID:44607577	phase I
BRD-K09922072	CCc1cccc(CC)c1NC(=O)c1ccc(o1)-c1cc(Cl)ccc1Cl	CID:44607580	phase I
BRD-K75040614	Cc1cscc1-c1ccc(o1)C(=O)Nc1c(C)cccc1C	CID:44607581	phase I
BRD-K05566481	Cc1ccc(cc1)-c1cc2nc(C)cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1	CID:44607584	phase I
BRD-K64822626	Cc1cc(N2CCN(CC2)C(=O)c2ccoc2)n2nc(cc2n1)-c1ccccc1	CID:44607586	phase I
BRD-K43637719	COc1ccc(cc1)-c1cc2nc(C)cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1	CID:44607587	phase I
BRD-K70251741	COc1ccc(cc1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccsc3)n2n1)-c1ccccc1	CID:44607591	phase I
BRD-K29143967	COc1ccc(cc1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)-c1ccccc1	CID:44607592	phase I
BRD-A51666293	O=C1CC(CC2=C1C1(CCCC1)NC(Nc1nc3ccccc3o1)=N2)c1ccccc1	CID:44607600	phase I
BRD-K65404805	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44607850	phase I
BRD-K19985802	Fc1ccc(cc1)S(=O)(=O)C(=C\c1cccn1S(=O)(=O)c1cccc(c1)C#N)\C#N	CID:44607949	phase I
BRD-K29160485	CS(=O)(=O)C(\C#N)=C\c1cccn1S(=O)(=O)c1ccc(cc1)[N+]([O-])=O	CID:44607954	phase I
BRD-K72864428	CS(=O)(=O)C(=C\c1cccn1S(=O)(=O)c1cccc2ccccc12)\C#N	CID:44607958	phase I
BRD-K00256256	[O-][N+](=O)c1cccc(c1)S(=O)(=O)n1cccc1\C=C(/C#N)S(=O)(=O)c1ccc(F)cc1	CID:44607965	phase I
BRD-K64881093	CC(C)(C)S(=O)(=O)C(=C\c1cccn1S(=O)(=O)c1ccccc1)\C#N	CID:44607969	phase I
BRD-K99135512	Fc1ccc(cc1)S(=O)(=O)C(=C\c1cccn1S(=O)(=O)c1ccccc1)\C#N	CID:44607974	phase I
BRD-K86086851	COc1ccc(cc1)-c1cc2nc(C)cc(N3CCN(CC3)C(=O)c3cccnc3)n2n1	CID:44607977	phase I
BRD-K18913711	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4c(cccc4C1=O)N(C)C	CID:44616316	phase I
BRD-K23287115	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44616320	phase I
BRD-K65037509	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44616386	phase I
BRD-K22458275	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44616387	phase I
BRD-K90184854	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44616391	phase I
BRD-K30393343	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44616397	phase I
BRD-K95419055	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44616403	phase I
BRD-K25496062	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)C3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44616413	phase I
BRD-K83601549	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44616428	phase I
BRD-K11889659	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)S(=O)(=O)c3ccccc3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44616431	phase I
BRD-K75969390	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44616453	phase I
BRD-K45222065	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44616467	phase I
BRD-K99439802	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44616498	phase I
BRD-K80786583	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44616501	phase I
BRD-K17401882	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44616505	phase I
BRD-K97973721	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44616514	phase I
BRD-K01528688	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44616530	phase I
BRD-K30726719	CC(C)NC(=O)N(C)C[C@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44616544	phase I
BRD-K86011921	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44616560	phase I
BRD-K84770507	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44616576	phase I
BRD-K39580731	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44616591	phase I
BRD-K28428448	COc1ccc(NC(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)CC4CCCCC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44616599	phase I
BRD-K15328325	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44616619	phase I
BRD-K07060092	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:44616639	phase I
BRD-K06973013	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44616641	phase I
BRD-K05232104	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44616650	phase I
BRD-K02701279	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Nc5ccc6OCOc6c5)cc4CC1=O	CID:44616668	phase I
BRD-K13411622	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(NC(=O)NC(C)C)cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44616686	phase I
BRD-K27173348	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:44616695	phase I
BRD-K15825608	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44616698	phase I
BRD-K13308287	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44616733	phase I
BRD-K60667905	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44616738	phase I
BRD-K28431278	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:44616759	phase I
BRD-K17083260	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44616769	phase I
BRD-K58912123	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44616771	phase I
BRD-K89288521	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44616781	phase I
BRD-K98327170	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44616782	phase I
BRD-K08607084	COc1ccc(NC(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44616788	phase I
BRD-K02964016	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:44616810	phase I
BRD-K08198655	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44616823	phase I
BRD-K26968982	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44616886	phase I
BRD-K10482608	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44616894	phase I
BRD-K93406156	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44616929	phase I
BRD-K69295800	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44616949	phase I
BRD-K68630394	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44616955	phase I
BRD-K95776192	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44616967	phase I
BRD-K44575839	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44616982	phase I
BRD-K45690206	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44616995	phase I
BRD-K13559922	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44617006	phase I
BRD-K36451640	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:44617009	phase I
BRD-K72219469	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44617016	phase I
BRD-K11746559	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44617026	phase I
BRD-K08061170	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:44617034	phase I
BRD-K17492515	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44617069	phase I
BRD-K05150608	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617159	phase I
BRD-K47436535	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)Cc4ccc(Cl)c(Cl)c4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44617171	phase I
BRD-K01615174	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44617175	phase I
BRD-K20624574	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(NC(=O)CCC(F)(F)F)cc4C1=O	CID:44617183	phase I
BRD-K13943990	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44617198	phase I
BRD-K37322457	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44617221	phase I
BRD-K44647644	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:44617225	phase I
BRD-K11366122	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44617229	phase I
BRD-K10946493	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:44617231	phase I
BRD-K85569074	COc1ccc(NC(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)CC4CC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44617236	phase I
BRD-K37149438	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:44617281	phase I
BRD-K16173196	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617289	phase I
BRD-K43014865	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617302	phase I
BRD-K17630163	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44617305	phase I
BRD-K66536842	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617311	phase I
BRD-K13679108	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44617313	phase I
BRD-K16563572	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:44617325	phase I
BRD-K60582191	COc1ccc(NC(=O)N(C)C[C@H]2Oc3ccc(cc3CC(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C)cc1	CID:44617334	phase I
BRD-K04540960	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)C5CCCCC5)cc4CC1=O	CID:44617339	phase I
BRD-K50011261	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44617341	phase I
BRD-K12484748	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44617370	phase I
BRD-K76318793	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44617376	phase I
BRD-K75887136	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44617378	phase I
BRD-K04476933	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:44617408	phase I
BRD-K83431831	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44617409	phase I
BRD-K32605311	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44617432	phase I
BRD-K14593092	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44617441	phase I
BRD-K98832591	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NC(=O)Nc5ccc(F)cc5)cc4CC1=O	CID:44617482	phase I
BRD-K08617930	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44617483	phase I
BRD-K71303366	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44617484	phase I
BRD-K57328348	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44617486	phase I
BRD-K47804338	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)Cc4ccc5OCOc5c4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44617488	phase I
BRD-K95913445	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)NC(C)C)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44617494	phase I
BRD-K27429081	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617502	phase I
BRD-K08251038	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44617508	phase I
BRD-K69406317	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44617510	phase I
BRD-K01427177	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44617549	phase I
BRD-K92431661	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44617555	phase I
BRD-K24722667	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)C4CCCCC4)cc3CC1=O	CID:44617598	phase I
BRD-K44360367	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:44617618	phase I
BRD-K58415436	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:44617646	phase I
BRD-K70397964	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44617670	phase I
BRD-K05469482	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44617693	phase I
BRD-K97671879	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44617719	phase I
BRD-K17954972	COc1cccc(c1)c2cnc3O[C@@H](CN(C)Cc4ccc(F)cc4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44617724	phase I
BRD-K85007671	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:44617726	phase I
BRD-K62291994	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)S(=O)(=O)c3ccc(Cl)cc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44617744	phase I
BRD-K53022123	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44617750	phase I
BRD-K00600835	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44617761	phase I
BRD-K73453061	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44617787	phase I
BRD-K80092909	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44617800	phase I
BRD-K38934024	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44617816	phase I
BRD-K70495648	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617819	phase I
BRD-K02283603	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:44617835	phase I
BRD-K38373457	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44617843	phase I
BRD-K18183699	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44617844	phase I
BRD-K06884091	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44617869	phase I
BRD-K16811158	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:44617870	phase I
BRD-K42454450	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44617880	phase I
BRD-K53437983	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44617904	phase I
BRD-K02025760	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44617931	phase I
BRD-K89034694	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44617953	phase I
BRD-K98936959	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44618011	phase I
BRD-K40724613	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44618016	phase I
BRD-K93459841	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44618017	phase I
BRD-K19166598	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44618018	phase I
BRD-K61373678	COc1ccc(NC(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44618057	phase I
BRD-K54635843	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44618073	phase I
BRD-K89419248	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44618088	phase I
BRD-K99447056	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44618097	phase I
BRD-K11826883	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44618123	phase I
BRD-K22261046	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44618164	phase I
BRD-K86728684	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44618166	phase I
BRD-K73439593	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:44618167	phase I
BRD-K60756411	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44618176	phase I
BRD-K49148689	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44618182	phase I
BRD-K70836798	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44618191	phase I
BRD-K45253154	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44618204	phase I
BRD-K08317416	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44618225	phase I
BRD-K43680293	COc1ccc(NC(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44618254	phase I
BRD-K79326278	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44618270	phase I
BRD-K00362189	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44618274	phase I
BRD-K67868064	COc1ccc(NC(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)Cc4ccc(Cl)c(Cl)c4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44618276	phase I
BRD-K63017287	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)CCC(F)(F)F)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:44618293	phase I
BRD-K97357148	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:44618358	phase I
BRD-K35577141	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44618375	phase I
BRD-K37066706	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44618378	phase I
BRD-K31329249	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44618418	phase I
BRD-K34639619	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44618423	phase I
BRD-K89185880	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44618458	phase I
BRD-K62818989	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4CC1=O)N(C)C	CID:44618470	phase I
BRD-K11624501	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44618473	phase I
BRD-K24319052	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44618474	phase I
BRD-K87426959	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44618507	phase I
BRD-K98731749	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44618522	phase I
BRD-K88748878	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44618542	phase I
BRD-K97961692	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44618620	phase I
BRD-K98044070	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44618633	phase I
BRD-K30934390	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44618659	phase I
BRD-K81496150	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44618662	phase I
BRD-K22450189	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44618671	phase I
BRD-K64615396	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44618702	phase I
BRD-K45835269	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44618747	phase I
BRD-K49669601	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:44618774	phase I
BRD-K68319707	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:44618781	phase I
BRD-K66586010	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:44618790	phase I
BRD-K81646882	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:44618802	phase I
BRD-K44816676	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44618805	phase I
BRD-K00458136	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44618831	phase I
BRD-K23985857	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:44618836	phase I
BRD-K89833083	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44618844	phase I
BRD-K68007270	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44618858	phase I
BRD-K05475237	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:44618860	phase I
BRD-K40160468	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44618900	phase I
BRD-K05353139	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44618908	phase I
BRD-K39211770	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44618932	phase I
BRD-K60760276	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44618954	phase I
BRD-K89194506	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44618963	phase I
BRD-K73459720	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44618970	phase I
BRD-K57900436	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ccc(cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)N(C)C)cc1	CID:44618986	phase I
BRD-K32585359	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:44618988	phase I
BRD-K48195969	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ncc(C#CCC4CCCCC4)cc3C1=O	CID:44619003	phase I
BRD-K47586560	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619021	phase I
BRD-K44036769	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619027	phase I
BRD-K36284700	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:44619031	phase I
BRD-K41593073	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@H](CN(C)Cc4ccc(Cl)c(Cl)c4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44619063	phase I
BRD-K22937431	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44619075	phase I
BRD-K79947405	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44619125	phase I
BRD-K95551268	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619130	phase I
BRD-K77172154	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44619141	phase I
BRD-K67787765	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:44619149	phase I
BRD-K16436767	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)CC4CCCCC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44619176	phase I
BRD-K32593492	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619177	phase I
BRD-K05912972	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44619181	phase I
BRD-K47636083	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44619186	phase I
BRD-K34095629	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3C1=O	CID:44619203	phase I
BRD-K98161915	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:44619237	phase I
BRD-K85642378	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:44619245	phase I
BRD-K28484895	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44619297	phase I
BRD-K68278258	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44619326	phase I
BRD-K74623475	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44619327	phase I
BRD-K00179355	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619373	phase I
BRD-K78525220	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44619374	phase I
BRD-K18891555	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44619395	phase I
BRD-K32389477	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44619439	phase I
BRD-K94633563	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44619469	phase I
BRD-K74121411	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44619499	phase I
BRD-K71935941	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:44619511	phase I
BRD-K58300809	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44619552	phase I
BRD-K71932341	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44619561	phase I
BRD-K25604127	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44619638	phase I
BRD-K48332509	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:44619678	phase I
BRD-K29396015	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44619689	phase I
BRD-K21125707	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:44619742	phase I
BRD-K95976153	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44619763	phase I
BRD-K57204377	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44619765	phase I
BRD-K22280018	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44619818	phase I
BRD-K38454082	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44619827	phase I
BRD-K69672023	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:44619837	phase I
BRD-K53321531	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ccc(NC(=O)Nc5ccc(F)cc5)cc4CC1=O	CID:44619852	phase I
BRD-K53949821	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619904	phase I
BRD-K37459628	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44619911	phase I
BRD-K68911617	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44619926	phase I
BRD-K08461556	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44619937	phase I
BRD-K92884627	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44619940	phase I
BRD-K62083683	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44619943	phase I
BRD-K84536720	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44619957	phase I
BRD-K16360094	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44619967	phase I
BRD-K15284276	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:44619975	phase I
BRD-K96612346	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:44619991	phase I
BRD-K57030368	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)Cc4ccccc4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44620013	phase I
BRD-K92364610	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:44620015	phase I
BRD-K49587132	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44620034	phase I
BRD-K17741643	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44620064	phase I
BRD-K08325197	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44620073	phase I
BRD-K79797751	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44620081	phase I
BRD-K79788021	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44620098	phase I
BRD-K32968870	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)S(=O)(=O)c3ccccc3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:44620106	phase I
BRD-K52047316	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)Cc4ccc5OCOc5c4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:44620117	phase I
BRD-K34981405	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44620120	phase I
BRD-K02589376	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:44620122	phase I
BRD-K22912836	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:44620176	phase I
BRD-K48505466	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44620234	phase I
BRD-K94575695	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44620240	phase I
BRD-K96420933	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44620262	phase I
BRD-K88069074	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44620280	phase I
BRD-K70052069	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:44620299	phase I
BRD-K77939573	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)N(C)C	CID:44620313	phase I
BRD-K53315742	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44620359	phase I
BRD-K36091499	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44620377	phase I
BRD-K61779668	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:44620378	phase I
BRD-K31302860	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:44620440	phase I
BRD-K43327166	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44620448	phase I
BRD-K56584267	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@H](CN(C)S(=O)(=O)c4ccc(Cl)cc4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:44620457	phase I
BRD-K29033329	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44620462	phase I
BRD-K42486494	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:44620495	phase I
BRD-K87449521	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:44620514	phase I
BRD-K40708503	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:44620530	phase I
BRD-K77922066	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44620546	phase I
BRD-K95411194	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44620550	phase I
BRD-K25351202	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44620614	phase I
BRD-K28249211	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44620644	phase I
BRD-K83887149	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:44620657	phase I
BRD-K38725747	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:44620660	phase I
BRD-K92327934	COc1ccc(NC(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44620669	phase I
BRD-K71614913	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:44620686	phase I
BRD-K78944321	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44620704	phase I
BRD-K77750380	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:44620728	phase I
BRD-K03589483	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:44620730	phase I
BRD-K02170312	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:44620732	phase I
BRD-K27742591	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)CCC(F)(F)F)cc3CC1=O	CID:44620743	phase I
BRD-K61556970	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:44620744	phase I
BRD-K43880650	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44620779	phase I
BRD-K97481123	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44620789	phase I
BRD-K74407269	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:44620790	phase I
BRD-K80622828	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44620796	phase I
BRD-K74329753	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:44620812	phase I
BRD-K44559054	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:44620818	phase I
BRD-K76103428	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:44620846	phase I
BRD-K44079161	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:44620847	phase I
BRD-K45156967	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:44620852	phase I
BRD-K19330527	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:44620865	phase I
BRD-K87338781	Cc1ccc(OCCOc2c(Cl)cc(Cl)cc2Cl)c(n1)[N+]([O-])=O	CID:44620882	phase I
BRD-K96072942	[O-][N+](=O)c1ncccc1OCCOc1ccc(Cl)cc1Cl	CID:44620883	phase I
BRD-K71182391	Cc1ccc(OCCCOc2ccc(Cl)cc2Cl)c(n1)[N+]([O-])=O	CID:44620891	phase I
BRD-K14236372	Clc1ccc(OCCOc2ccc(Br)nc2Br)c(Cl)c1	CID:44620892	phase I
BRD-K16618170	Cc1ccc(OCCOc2ccc(Cl)cc2Cl)c(Br)n1	CID:44620895	phase I
BRD-K48969316	CC(C)(C)[C@H](NC(=O)c1ccc(N)c(Cl)c1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(O)=O)C#N	CID:44620939	phase I
BRD-K76846644	CCOC(=O)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)c1ccc(N)c(Cl)c1)C(C)(C)C)C#N	CID:44620944	phase I
BRD-K87547250	CC(=O)Nc1ccc2c(c1)sn(-c1ccccc1)c2=O	CID:44623833	phase I
BRD-K56111351	Cc1ccc(NC(=O)Cn2sc3ccccc3c2=O)cc1	CID:44623834	phase I
BRD-K63326650	Clc1ccc(NC(=O)Cn2sc3ccccc3c2=O)cc1	CID:44623837	phase I
BRD-K19812755	O=c1n(sc2ccc(cc12)C#N)-c1ccccc1	CID:44623838	phase I
BRD-K30606628	Fc1cccc(c1)-c1cc(N2CCN(CC2)C(=O)c2ccoc2)n2nc(cc2n1)-c1cccc(Cl)c1	CID:44623839	phase I
BRD-K61981833	COc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)-c1ccccc1	CID:44623840	phase I
BRD-K96405393	Brc1ccc(cc1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)-c1ccccc1	CID:44623844	phase I
BRD-K70871370	COc1cccc(c1)-c1cc2nc(C)cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1	CID:44623845	phase I
BRD-K78843060	CS(=O)(=O)c1ccc(cc1[N+]([O-])=O)C(=O)OCC(=O)N1CCN(CCC2CCCCC2)CC1	CID:44623849	phase I
BRD-K95352812	CC(C)CN1CCN(CC1)C(=O)COC(=O)c1ccc(c(c1)[N+]([O-])=O)S(C)(=O)=O	CID:44623864	phase I
BRD-K10057859	CS(=O)(=O)c1ccc(cc1[N+]([O-])=O)C(=O)OCC(=O)N1CCOCC1	CID:44623872	phase I
BRD-K86492010	O=C1CCCC2=C1C1(CCCC1)NC(Nc1nc3cc(ccc3o1)-c1ccccc1)=N2	CID:44623881	phase I
BRD-K31600199	Cc1ccc2nc(NC3=NC4=C(C(=O)CCC4)C4(CCCC4)N3)oc2c1	CID:44623882	phase I
BRD-K54470384	Cn1c(NC2=NC3=C(C(=O)CCC3)C3(CCCC3)N2)nc2ccccc12	CID:44623884	phase I
BRD-K26233379	Brc1ccc2oc(NC3=NC4=C(C(=O)CCC4)C4(CCCC4)N3)nc2c1	CID:44623888	phase I
BRD-K51155404	Cc1ccc2oc(NC3=NC4=C(C(=O)CCC4)C4(CCCC4)N3)nc2c1	CID:44623889	phase I
BRD-K13005598	CSCC[C@H](NC=O)C(=O)N[C@@H](CC(O)=O)C(=O)NCC(=O)N[C@@H](CS)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(O)=O	CID:44628955	phase I
BRD-A13346522	CCn1cc(CN2CCCC(C2)C(=O)c3cccc(c3)C(F)(F)F)cn1	CID:44629407	phase I
BRD-K84855052	CC(=O)Nc1c(C#N)c(c(C#N)c(=O)n1c2ccc(C)cc2)c3ccccc3	CID:44629408	phase I
BRD-A02809788	COc1ccc(cc1OC)C(=O)C2CCCN(CCc3ccccc3)C2	CID:44629410	phase I
BRD-K14842454	CC(=O)Nc1ccc(cc1)/C(=N/NC(=O)C2CCCC2)/C	CID:44629411	phase I
BRD-K12621773	Cc1ccc(cc1)c2c(C#N)c(N)n(c3ccccc3C)c(=O)c2C#N	CID:44629412	phase I
BRD-A37656721	COc1ccc(cc1OC)C(=O)C2CCCN(CC3CCCCC3)C2	CID:44629413	phase I
BRD-K02646507	Clc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)-c1cccnc1	CID:44629742	phase I
BRD-K25320246	COc1ccc(cc1)-c1cc2nc(C)c(C)c(N3CCN(CC3)C(=O)c3ccoc3)n2n1	CID:44629744	phase I
BRD-K17023947	COc1cccc(c1)-c1cc(N2CCN(CC2)C(=O)c2ccoc2)n2nc(cc2n1)-c1cccc(Cl)c1	CID:44630538	phase I
BRD-K11015688	Clc1cccc(c1)-c1cc2nc(Cl)cc(N3CCN(CC3)C(=O)c3ccccc3)n2n1	CID:44630539	phase I
BRD-K91937579	Clc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccncc3)n2n1)-c1ccccc1	CID:44630540	phase I
BRD-K92343999	Clc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)-c1ccncc1	CID:44630541	phase I
BRD-K40373196	Clc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)C#C	CID:44631078	phase I
BRD-K08307026	C(Nc1nc(nnc1-c1ccccc1)-c1ccccn1)C1CCCCC1	CID:44631783	phase I
BRD-K74710236	CC(C)(C)CCNc1nc(nnc1-c1ccccc1)-c1ccccn1	CID:44631784	phase I
BRD-A62182663	COc1ccc(cc1)C(=O)CC1(O)C(=O)Nc2c1c(Cl)ccc2Cl	CID:44632017	phase I
BRD-K41845021	Cc1c(n2ccccc2[n+]1CCc1ccccc1)P(=S)(c1ccccc1)c1ccccc1	CID:44634508	phase I
BRD-K51126483	Cc1nc2ccccn2c1C(O)(c1ccccc1)c1ccccc1	CID:44634510	phase I
BRD-K87371039	O=P(c1cnc2ccccn12)(c1ccccc1)c1ccccc1	CID:44634519	phase I
BRD-K21482967	Cc1nc2ccccn2c1P(=O)(c1ccccc1)c1ccccc1	CID:44634521	phase I
BRD-K30781400	Cc1c(n2ccccc2[n+]1C)C(O)(c1ccccc1)c1ccccc1	CID:44634524	phase I
BRD-K78167523	C[n+]1cc(n2ccccc12)C(O)(c1ccccc1)c1ccccc1	CID:44634529	phase I
BRD-K41006959	OC(c1cnc2ccccn12)(c1ccccc1)c1ccccc1	CID:44634533	phase I
BRD-K55557659	Cn1cc(c2ccccc12)P(=S)(c1ccccc1)c1ccccc1	CID:44634539	phase I
BRD-K65774694	Cc1c(c2ccccc2n1C)P(=O)(c1ccccc1)c1ccccc1	CID:44634542	phase I
BRD-K85147876	S=P(c1cnc2ccccn12)(c1ccccc1)c1ccccc1	CID:44634544	phase I
BRD-K11757396	S=P(c1cn(Cc2ccccc2)c2cccc[n+]12)(c1ccccc1)c1ccccc1	CID:44634547	phase I
BRD-K56855930	Cc1nc2ccccn2c1P(=S)(c1ccccc1)c1ccccc1	CID:44634570	phase I
BRD-K37940862	Cc1c(n2ccccc2[n+]1C\C=C\c1ccccc1)P(=S)(c1ccccc1)c1ccccc1	CID:44634573	phase I
BRD-K96134740	CO[C@H]1[C@@H](CC(=O)O[C@H](C)C\C=C/C=C/[C@H](O)[C@H](C)C[C@H](CC=O)[C@@H]1O[C@@H]1O[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC(=O)CC(C)C)[C@@H](O)[C@H](C)O2)[C@@H]([C@H]1O)N(C)C)OC(C)=O	CID:44634697	phase I
BRD-A45140972	CN(C)[C@H]1[C@@H]2[C@@H](O)C3C(C(=O)c4c(O)ccc(Cl)c4C3=C)C(=O)[C@]2(O)C(=O)C(C(=O)N)C1=O	CID:44634699	phase I
BRD-K38061943	Cc1cc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)ccc1Cl	CID:44634865	phase I
BRD-A93942655	CC(OC(=O)c1ccc(c(c1)[N+]([O-])=O)S(C)(=O)=O)C(=O)NC1C2CC3CC(C2)CC1C3	CID:44640136	phase I
BRD-A09719808	CCC(OC(=O)c1ccc(c(c1)[N+]([O-])=O)S(C)(=O)=O)C(=O)NC1C2CC3CC(C2)CC1C3	CID:44640137	phase I
BRD-K07995125	COc1cccc(c1)-c1cc2nc(C)c(C)c(N3CCN(CC3)C(=O)c3ccoc3)n2n1	CID:44640175	phase I
BRD-K15716662	COc1ccccc1-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccco3)n2n1)-c1ccccc1	CID:44640176	phase I
BRD-K50135923	O=C(N1CCN(CC1)c1cc(nc2cc(nn12)-c1ccccc1)-c1ccco1)c1ccoc1	CID:44640177	phase I
BRD-K64409586	COc1ccc(cc1)-c1[nH]nc2nc(cc(c12)C(F)(F)F)N1CCN(CC1)C(=O)c1ccoc1	CID:44640178	phase I
BRD-K73044744	COc1ccc(cc1)-c1cc2nc(C)cc(N3CCN(CC3)C(=O)c3ccco3)n2n1	CID:44640181	phase I
BRD-K51443908	COc1ccccc1-c1cc2nc(cc(N3CCN(CC3)C(=O)c3ccoc3)n2n1)-c1ccccc1	CID:44640183	phase I
BRD-K24538644	COc1ccc(cc1)N1CCN(CCCNC(=O)Cn2c3nccc(C)c3n3cccc3c2=O)CC1	CID:44665680	phase I
BRD-K12437911	COc1cc(CC(=O)C(O)=O)ccc1OCc1ccccc1	CID:44721090	phase I
BRD-K98173387	OC(=O)CCN1C(=S)S\C(=C/c2cccc(OCc3ccc(F)cc3)c2)C1=O	CID:44807133	phase I
BRD-K55890295	CNc1nc(NCc2ccc(NC(=O)c3ccc(F)cc3)cc2)c2ccccc2n1	CID:44818131	phase I
BRD-K83289131	O=C(CCCCCCCn1cc(nn1)-c1cccnc1)Nc1ccccc1-c1ccccc1	CID:44819697	phase I
BRD-K71523760	NCCCNC(=S)NCCCN(Cc1ccc(Cl)cc1)c1ccc(Br)cn1	CID:44820542	phase I
BRD-K82384352	Clc1ccc(CN(CCCNC(=S)NCCCc2c[nH]cn2)c2ccc(Br)cn2)cc1	CID:44820550	phase I
BRD-K33305493	Brc1ccc(nc1)N(CCCNC(=S)NCCCc1c[nH]cn1)Cc1ccccc1	CID:44820554	phase I
BRD-K94296811	CCCCN(CCCNC(=S)NCCCc1c[nH]cn1)c1ccc(Br)cn1	CID:44820562	phase I
BRD-K71029018	CC(=O)NCCCNC(=S)NCCCN(Cc1ccc(Cl)cc1)c1ccc(Br)cn1	CID:44820564	phase I
BRD-K06956503	Clc1ccc(CN(CCCCNC(=S)NCCCc2c[nH]cn2)c2ccc(Br)cn2)cc1	CID:44820570	phase I
BRD-K00925050	OC(=O)c1ccc(cc1)-c1nn2c(nc(cc2=O)N2CCNCC2)s1	CID:44820647	phase I
BRD-K56983253	OC(=O)c1ccc(cc1)-c1cccc(c1)-c1nn2c(nc(cc2=O)N2CCNCC2)s1	CID:44820652	phase I
BRD-K88668992	CCc1nn2c(nc(N3CCNCC3)c(F)c2=O)s1	CID:44820670	phase I
BRD-K19410523	Clc1ccc2c(ccnc2c1)N1CCN(CC1)c1cc(=O)n(C2CCCCC2)c(=O)[nH]1	CID:44825223	phase I
BRD-K05331696	CC(=O)c1cccc(c1)-c1csc2ncnc(Sc3nnnn3C)c12	CID:44825280	phase I
BRD-K75315865	CC(=O)c1ccc(cc1)N1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)C(Cl)(Cl)c2c1	CID:44825304	phase I
BRD-K44893543	Cc1ccc(Nc2ccc(s2)c3ccncc3)c(Br)c1	CID:44826047	phase I
BRD-K37057377	Clc1ccc(cc1)N1CCN(CCCNC(=O)Cn2c3ncccc3n3cccc3c2=O)CC1	CID:44828476	phase I
BRD-K85853911	O=C(Cn1c2ncccc2n2cccc2c1=O)NCCCN1CCN(CC1)c1ccccc1	CID:44828477	phase I
BRD-K40083016	COc1ccc(N2CCN(CCCNC(=O)Cn3c4ncccc4n4cccc4c3=O)CC2)c(OC)c1	CID:44828478	phase I
BRD-K19042873	Oc1ccc(\C=C\c2ccc(\C=C\c3ccc(O)cc3)c(Br)c2)cc1	CID:44828481	phase I
BRD-K78385490	Oc1cccc2cc(Nc3ccccc3)cnc12	CID:44887545	phase I
BRD-K63770300	Oc1cccc2cc(cnc12)-c1ccncc1	CID:44887546	phase I
BRD-K88906571	OC(C1CCN(CCCOc2cccc(c2)C#N)CC1)(c1ccccc1)c1ccccc1	CID:44907115	phase I
BRD-K43992206	OC(C1CCN(CCCOc2ccc(Cl)cc2)CC1)(c1ccccc1)c1ccccc1	CID:44907120	phase I
BRD-K61127831	OC(C1CCN(CCCOc2ccc(F)cc2)CC1)(c1ccccc1)c1ccccc1	CID:44907124	phase I
BRD-K90446130	CCN(Cc1cccs1)c1ncnc2ccc(cc12)-c1ccc2OCOc2c1	CID:44968186	phase I
BRD-K75784474	Fc1c2OCOc2ccc1-c1ccc2ncnc(NCc3cccs3)c2c1	CID:44968206	phase I
BRD-K74980345	Cc1ccc(CNc2ncnc3ccc(cc23)-c2ccoc2C)o1	CID:44968219	phase I
BRD-K17025677	CN(Cc1sccc1C)c1ncnc2ccc(cc12)-c1ccoc1	CID:44968224	phase I
BRD-K92107474	CCOC(=O)c1ccc(o1)-c1ccc2ncnc(N(C)Cc3sccc3C)c2c1	CID:44968227	phase I
BRD-K64835161	Cc1ccc(CNc2ncnc3ccc(cc23)-c2ccc(CO)o2)o1	CID:44968231	phase I
BRD-K21822525	CCOC(=O)c1ccc(o1)-c1ccc2ncnc(NCc3csc(C)n3)c2c1	CID:44968259	phase I
BRD-A66395008	C\C1=C/CC[C@]2(C)OC2[C@H]2OC(=O)C(=C)[C@@H]2CC1	CID:45006067	phase I
BRD-A73909368	CC(C)C1NC(=O)C(NC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C2CCCN2C1=O)C(C)OC(=O)c1ccc(C)c2oc3c(C)c(=O)c(N)c(C(=O)OC(C)C4NC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C5CCCN5C(=O)C(NC4=O)C(C)C)c3nc12	CID:45006140	phase I
BRD-A35912562	CC(=O)[C@H]1CCC2C3CC=C4C[C@H](CC[C@]4(C)C3CC[C@]12C)OC(=O)CCC(O)=O	CID:45006141	phase I
BRD-A25143711	CCCCC(=O)O[C@@]1(CCC2C3CCC4=CC(=O)CC[C@]4(C)C3[C@@H](O)C[C@]12C)C(=O)CO	CID:45006145	phase I
BRD-A27554692	C[C@]12C=CC3=C4CCC(=O)C=C4CCC3C1CC[C@@]2(O)CC=C	CID:45006157	phase I
BRD-A92177080	C[C@H]1CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)COC(C)=O	CID:45006158	phase I
BRD-A49447682	C[C@@H]1CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@H]1C(=O)CO	CID:45006167	phase I
BRD-K81795824	N(c1nc(cs1)-c1ccccc1)c1nc(nnc1-c1ccccc1)-c1ccccn1	CID:45099945	phase I
BRD-K92158425	Clc1ccc2[nH]c(CNc3nc(nc4n(cnc34)-c3ccsc3)N3CCOCC3)nc2c1	CID:45100429	phase I
BRD-K77681376	[O-][N+](=O)c1cccc2[nH]c(CNc3nc(nc4n(cnc34)-c3ccsc3)N3CCOCC3)nc12	CID:45100431	phase I
BRD-K01896723	[O-][N+](=O)c1ccc2[nH]c(CNc3nc(nc4n(cnc34)-c3ccsc3)N3CCOCC3)nc2c1	CID:45100442	phase I
BRD-K10846167	C(Nc1nc(nc2n(cnc12)-c1ccsc1)N1CCOCC1)c1nc2cc3ccccc3cc2[nH]1	CID:45100444	phase I
BRD-K77547509	FC(F)(F)c1cccc(c1)N1CCN(CC1)c1cc(=O)n(C2CCCCC2)c(=O)[nH]1	CID:45100448	phase I
BRD-K79222491	FC(F)(F)c1ccc2[nH]c(CNc3nc(nc4n(cnc34)-c3ccsc3)N3CCOCC3)nc2c1	CID:45100452	phase I
BRD-K02216544	Clc1cccc(N2CCN(CC2)c2cc(=O)n(C3CCCCC3)c(=O)[nH]2)c1Cl	CID:45100455	phase I
BRD-A57457122	Clc1cc(NC(=O)c2ccccn2)ccc1N1C(=O)CC(C1=O)c1ccccc1	CID:45110765	phase I
BRD-A48570745	CCC(C)[C@H]1O[C@]2(CC[C@@H]1C)C[C@@H]1C[C@@H](C\C=C(C)\[C@@H](OC3C[C@H](OC)C(O[C@H]4C[C@H](OC)[C@@H](O)[C@H](C)O4)[C@H](C)O3)[C@@H](C)\C=C\C=C3/CO[C@@H]4[C@H](O)C(C)=C[C@@H](C(=O)O1)[C@]34O)O2	CID:45114068	phase I
BRD-K18453942	CC(C)(C)CCN1CCC[C@@H](C1)NC(=O)COc1ccc(F)c(Cl)c1	CID:45115609	phase I
BRD-A52172093	CC(C)(C)CCN1C[C@H]2C(CNC(=O)c3cc(Cl)cc(Cl)c3)[C@H]2C1	CID:45115620	phase I
BRD-K53780220	C(Nc1nc(nc2n(cnc12)-c1ccsc1)N1CCOCC1)c1nc2ccccc2[nH]1	CID:45115629	phase I
BRD-K41185612	Clc1cc(Cl)cc(c1)S(=O)(=O)N1CCN(CC1)c1nc(nc2ccccc12)-c1cccs1	CID:45136810	phase I
BRD-K49183052	FC(F)(F)S(=O)(=O)c1ccc(CN2CCOCCOCCN(Cc3ccc(cc3)S(=O)(=O)C(F)(F)F)CCOCC2)cc1	CID:45259133	phase I
BRD-K76540910	[O-][N+](=O)c1ccc(CN2CCOCCOCCN(Cc3ccc(cc3Cl)[N+]([O-])=O)CCOCC2)c(Cl)c1	CID:45259135	phase I
BRD-K59795987	Fc1ccc2[nH]c(COCc3nc4cc(F)ccc4[nH]3)nc2c1	CID:45259136	phase I
BRD-K97476371	CN(C)S(=O)(=O)c1ccc2[nH]c(COCc3nc4cc(ccc4[nH]3)S(=O)(=O)N(C)C)nc2c1	CID:45259137	phase I
BRD-K37456065	FC(F)(F)Oc1ccc2N(Cc3ccc(cc3)-c3ccccc3)C(=O)C(=O)c2c1	CID:45281794	phase I
BRD-K66032149	FC(F)(F)Oc1ccc2N(Cc3ccc(cc3)-c3ccsc3)C(=O)C(=O)c2c1	CID:45281797	phase I
BRD-K53732802	FC(F)(F)Oc1ccc2N(Cc3ccc(cc3)-c3ccc(Cl)nc3)C(=O)C(=O)c2c1	CID:45281798	phase I
BRD-K44640865	Fc1ccc(cn1)-c1ccc(CN2C(=O)C(=O)c3cc(OC(F)(F)F)ccc23)cc1	CID:45281801	phase I
BRD-K59460069	COC(=O)c1c(O)ccc2oc3cc(CO)cc(O)c3c(=O)c12	CID:45359153	phase I
BRD-K41415459	CN1CCN(CC1)C(=O)CN[C@@H]1C[C@H]1c1ccc(OCc2ccccc2)cc1	CID:45376076	phase I
BRD-K54687541	CC(C)Cn1c(=O)cc([nH]c1=O)N1CCN(CC1)c1cccc(c1)C(F)(F)F	CID:45382271	phase I
BRD-K06436323	CCn1c(=O)cc([nH]c1=O)N1CCN(CC1)c1cccc(c1)C(F)(F)F	CID:45382284	phase I
BRD-K09716788	CC(C)c1ccc(cc1)C(=O)Nc1cc(Cl)ccc1C(O)=O	CID:45436131	phase I
BRD-K08041211	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:45480087	phase I
BRD-K08640787	FC(F)(F)c1cccc(c1)N1CCN(CC1)c1cc(=O)n(-c2ccccc2)c(=O)[nH]1	CID:45480137	phase I
BRD-A59900482	CC(C)(C)NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C(C)(C)C)c1cccnc1	CID:45489398	phase I
BRD-A68397902	COCC(=O)N(C(C(=O)NC(C)(C)C)c1cccnc1)c1ccc(cc1)C(C)(C)C	CID:45489406	phase I
BRD-A42031983	CC(C)(C)NC(=O)C(N(C(=O)c1cnco1)c1ccc(cc1)C(C)(C)C)c1cccnc1	CID:45489447	phase I
BRD-A89104433	CC(C)(C)NC(=O)C(N(C(=O)c1cccs1)c1ccc(cc1)C(C)(C)C)c1cccnc1	CID:45489449	phase I
BRD-K33459729	Brc1csc(n1)N1CCNCC1	CID:45787501	phase I
BRD-A40431293	CC1(C)C2C=C[C@]3(C)C(CC[C@@]4(C)[C@@H](OC(=O)[C@H]5O[C@@]345)c3ccoc3)[C@@]2(C)C=CC1=O	CID:45934191	phase I
BRD-A54596827	O=C(O[C@H]1CN2CCC1CC2)C1NCc2ccccc2[C@@H]1c1ccccc1	CID:45934210	phase I
BRD-A32440707	CC(=O)[C@H]1CCC2C3CCC4=CC(=O)CC[C@]4(C)C3[C@@H](C[C@]12C)OC(=O)CCC(O)=O	CID:45934211	phase I
BRD-K97516968	Cc1ccc(OCCCN2CCC(CC2)C(O)(c2ccccc2)c2ccccc2)cc1	CID:46172903	phase I
BRD-K36038115	COc1ccc(Oc2c(Cl)cnn(-c3cc(C)cc(C)c3)c2=O)cc1	CID:46172919	phase I
BRD-K34711351	CCc1ccc(Oc2c(Cl)cnn(-c3ccc(C)cc3)c2=O)cc1	CID:46172920	phase I
BRD-K58618158	CCOc1ccc(Oc2c(Cl)cnn(-c3ccc(C)cc3)c2=O)cc1	CID:46172926	phase I
BRD-K45205755	CCc1ccc(cc1)-n1ncc(Cl)c(Oc2ccc(OC)cc2)c1=O	CID:46172935	phase I
BRD-K08325710	CC(=O)N1CCN(CC1)c1cc(nc2cc(nn12)-c1ccccc1)-c1ccco1	CID:46173053	phase I
BRD-K08697762	Nc1ccc(cc1)\C=C\c1cc(O)cc(O)c1	CID:46191176	phase I
BRD-K64800655	CC(C)CC(=O)Nc1n[nH]c2c1CN(C(=O)C1CCN(C)CC1)C2(C)C	CID:46191454	phase I
BRD-K70642949	CNc1nc(cc(n1)-c1ccc2c(N)n[nH]c2c1)N1C[C@H](CC[C@H]1C)C(=O)NC1CCCCC1	CID:46215815	phase I
BRD-K98684188	COC(=O)c1sccc1S(=O)(=O)Nc1ccc(Nc2ccccc2)cc1OC	CID:46233311	phase I
BRD-K06585517	CCCN(CCC)c1nc(N2CCNCC2)c3ccccc3n1	CID:46238405	phase I
BRD-K05114711	CCCN(CCC)c1nc(nc2cc(OC)c(OC)cc12)N3CCCC3	CID:46238422	phase I
BRD-K40480443	COc1cccc(c1)-c1cc2nc(C)c(C)c(N3CCN(Cc4ccco4)CC3)n2n1	CID:46245505	phase I
BRD-A78971512	CC(CCCC(C)(C)O)C1CCC2C1(C)CCC\C2=C/C=C1/CC(O)CCC1=C	CID:46705323	phase I
BRD-A51777634	C1CN(CC1C1CCCCC1)c1nc(nnc1-c1ccccc1)-c1ccccn1	CID:46742339	phase I
BRD-K89093471	Clc1cccc(CNc2nc(nnc2-c2ccccc2)-c2ccccn2)c1	CID:46742340	phase I
BRD-K69097969	CC(C)(C)c1ccc(CNc2nc(nnc2-c2ccccc2)-c2ccccn2)cc1	CID:46742345	phase I
BRD-K44432556	C(Nc1nc(nnc1-c1ccccc1)-c1ccccn1)c1ccc(cc1)-c1ccccc1	CID:46742353	phase I
BRD-K76907295	C(Nc1nc(nnc1-c1ccccc1)-c1ccccn1)c1cccc(c1)-c1ccccc1	CID:46742354	phase I
BRD-A87848830	CCNC(=O)CCC\C=C/CC1C(O)CC(O)[C@@H]1\C=C\C(O)CCc1ccccc1	CID:46780805	phase I
BRD-A01145011	OC[C@H]1O[C@H](C(O)[C@H]1O)n1cccnc1=O	CID:46783268	phase I
BRD-K57353465	C(Nc1nc(nc2ccccc12)N1CCc2ccccc12)c1ccccc1	CID:46829332	phase I
BRD-K21773564	COc1ccc(Oc2c(Cl)cnn(-c3ccc(C(C)C)c(C)c3)c2=O)cc1	CID:46835808	phase I
BRD-A68739437	COc1cc(ccc1Nc1ncc2N(C)C(=O)CC(C)N(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	CID:46843648	phase I
BRD-K50387473	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCC(O)CC1	CID:46843772	phase I
BRD-K01436366	COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	CID:46843906	phase I
BRD-K64857848	COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1	CID:46844147	phase I
BRD-K97522823	COc1ccc(Oc2c(cnn(-c3ccc(C)cc3)c2=O)-c2cccs2)cc1	CID:46846333	phase I
BRD-A29009894	CC(Nc1ncc(Cl)c(Nc2cc(C)[nH]n2)n1)c1ncc(F)cn1	CID:46861588	phase I
BRD-K83010055	COc1cc(NC(=O)c2ccccn2)ccc1NC(=O)c1ccccc1Cl	CID:46869940	phase I
BRD-K39823328	Clc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccccn2)cc1Cl	CID:46869941	phase I
BRD-K84141129	Clc1cc(NC(=O)c2ccccn2)ccc1N1C(=O)CC2(CCCCC2)C1=O	CID:46869951	phase I
BRD-A34208323	CC1(CC(=O)N(C1=O)c1ccc(NC(=O)c2ccccn2)cc1Cl)c1ccccc1	CID:46869952	phase I
BRD-K00366212	COc1cccc2c(NCc3ccccc3)nc(nc12)N1CCOc2ccccc12	CID:46873819	phase I
BRD-K36740062	CCn1cc(c(n1)-c1ccc(NC(=O)N(C)C)cc1)-c1ccnc2[nH]c(cc12)-c1cccc(CN(C)C)c1	CID:46885626	phase I
BRD-K88317944	CC(C)(C)NC(=O)[C@@H](N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1	CID:46897843	phase I
BRD-K59633790	CC(C)(C)NC(=O)[C@H](N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1	CID:46897844	phase I
BRD-K74236984	COc1cc2c(NC3CCN(C)CC3)nc(nc2cc1OCCOCCN(C)C)N1CCCN(C)CC1	CID:46901937	phase I
BRD-K64302725	O[C@H]1C[C@@H](N(Cc2cccs2)C[C@@H]1n1cc(nn1)C1CC1)c1ccc(Cl)cc1	CID:46902718	phase I
BRD-K41916320	CNC[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:46903255	phase I
BRD-K69983865	COc1ccccc1S(=O)(=O)N(C)C[C@H]2Oc3cc(Br)ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO	CID:46903309	phase I
BRD-K90849880	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(Br)ccc3S1(=O)=O	CID:46903337	phase I
BRD-K06450282	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(cc34)N(C)C)[C@H](CO)O2	CID:46903347	phase I
BRD-K32099399	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(Br)ccc3S1(=O)=O	CID:46903353	phase I
BRD-K30180607	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:46903404	phase I
BRD-K25065206	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:46903409	phase I
BRD-K73542906	CCCNC(=O)N(C)C[C@@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:46903414	phase I
BRD-K19396909	COCC(=O)N(C)C[C@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:46903421	phase I
BRD-K49934959	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(C#Cc4cccc(F)c4)ccc3S1(=O)=O	CID:46903423	phase I
BRD-K53185063	C[C@@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:46903425	phase I
BRD-K56375979	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:46903427	phase I
BRD-K87434936	C[C@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:46903432	phase I
BRD-K75997540	COc1ccc(cc1)c2cnc3O[C@@H](CN(C)Cc4ccccc4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:46903448	phase I
BRD-K63807676	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:46903465	phase I
BRD-K86986466	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:46903520	phase I
BRD-K17489199	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:46903526	phase I
BRD-K37226353	COc1cccc(c1)c2ccc3c(O[C@@H](CN(C)C(=O)C4CCOCC4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:46903528	phase I
BRD-K66925231	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:46903542	phase I
BRD-K21494224	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:46903546	phase I
BRD-K03313681	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:46903552	phase I
BRD-K16567490	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:46903556	phase I
BRD-K61050052	CC(C)C#Cc1cnc2O[C@@H](CN(C)Cc3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:46903561	phase I
BRD-K66703091	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:46903562	phase I
BRD-K46849651	CCCC#Cc1cnc2O[C@H](CN(C)C(=O)CCN3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:46903571	phase I
BRD-K20300606	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:46903577	phase I
BRD-K97307478	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:46903580	phase I
BRD-K09167509	CCCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:46903581	phase I
BRD-K70054078	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:46903589	phase I
BRD-K03261284	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:46903678	phase I
BRD-K28882142	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:46903692	phase I
BRD-K73162352	COc1ccccc1S(=O)(=O)N(C)C[C@H]2Oc3cc(Br)ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO	CID:46903710	phase I
BRD-K95500387	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:46903714	phase I
BRD-K12132598	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:46903778	phase I
BRD-K55461955	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)NC3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:46903782	phase I
BRD-K23961390	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:46903784	phase I
BRD-K94979678	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:46903876	phase I
BRD-K76438898	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:46903884	phase I
BRD-K53549851	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2C(=O)O)Oc3ncc(Br)cc3C1=O	CID:46904078	phase I
BRD-K60984759	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3cc(Br)ccc3S1(=O)=O	CID:46904091	phase I
BRD-K76989634	CCCNC(=O)N(C)C[C@H]1Oc2ncc(Br)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:46904117	phase I
BRD-K23166787	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(Br)ccc4S1(=O)=O	CID:46904126	phase I
BRD-K60143275	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(Br)ccc4S1(=O)=O	CID:46904195	phase I
BRD-K91775327	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3cc(Br)ccc3S1(=O)=O	CID:46904202	phase I
BRD-K49031847	CCCNC(=O)N(C)C[C@@H]1Oc2ncc(Br)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:46904239	phase I
BRD-K70838368	COc1ccccc1S(=O)(=O)N(C)C[C@H]2Oc3ncc(Br)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:46904240	phase I
BRD-K46760727	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(Br)cc4C1=O	CID:46904257	phase I
BRD-K89536088	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C(=O)O)Oc3ncc(Br)cc3C1=O	CID:46904260	phase I
BRD-K67742177	O=C(N1CCN(CC1)c1cc(nc2cc(nn12)-c1ccco1)-c1ccco1)c1ccoc1	CID:46905000	phase I
BRD-K18865856	Cc1ccnc(SCc2cc(=O)c(OC(=O)c3ccc(cc3)C#N)co2)n1	CID:46905018	phase I
BRD-K42471691	O=C(Oc1coc(CSc2ncccn2)cc1=O)c1ccc(cc1)C#N	CID:46905029	phase I
BRD-K26304855	Cn1c2ccccc2c(OCCCC(=O)Nc2cc(ccn2)C(F)(F)F)cc1=O	CID:46907611	phase I
BRD-K83670234	Cn1c2ccccc2c(OCCCC(=O)Nc2cc(ccn2)-c2ccncc2)cc1=O	CID:46907618	phase I
BRD-K81814927	Cn1c2ccccc2c(OCCCC(=O)Nc2cc(ccn2)-c2cn[nH]c2)cc1=O	CID:46907621	phase I
BRD-K58853583	Cn1c2ccccc2c(OCCCC(=O)Nc2cc(Br)ccn2)cc1=O	CID:46907631	phase I
BRD-K76363932	CN(C)c1cccc(c1)-c1nccc(n1)N1CCC(CC1)C(N)=O	CID:46907656	phase I
BRD-K61921568	CC(C)Oc1cccc(c1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907658	phase I
BRD-K35514965	COc1cc(OC)cc(c1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907659	phase I
BRD-K94390040	Brc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(=O)N1CCNCC1	CID:46907661	phase I
BRD-K86217247	CN(C)c1cccc(c1)-c1cnc(s1)N1CCC(CC1)C(N)=O	CID:46907664	phase I
BRD-K59754458	CC(C)(C)OC(=O)NC1CCN(CC1)c1nc(cs1)-c1ccc(Br)cc1	CID:46907667	phase I
BRD-K55034844	COc1cc(cc(OC)c1OC)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907669	phase I
BRD-K14914284	CSc1ccc(cc1)-c1cnc(s1)N1CCC(CC1)C(N)=O	CID:46907676	phase I
BRD-K49791723	NC(=O)C1CCN(CC1)c1nc(cs1)-c1ccc(Oc2ccccc2)cc1	CID:46907681	phase I
BRD-K52524742	CC(C)(C)c1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907683	phase I
BRD-K63239300	CC(C)Oc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907689	phase I
BRD-K53461563	Brc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(=O)NCCCc1ccccc1	CID:46907690	phase I
BRD-K76951091	CC(C)COc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907705	phase I
BRD-K17739445	Brc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(=O)NCc1ccccc1	CID:46907707	phase I
BRD-K25784575	NC(=O)C1CCN(CC1)c1ncc(Br)cn1	CID:46907712	phase I
BRD-K85237725	NC(=O)C1CCN(CC1)c1ncc(Br)s1	CID:46907713	phase I
BRD-K74561903	NC(=O)C1CCN(CC1)c1nc(cs1)-c1ccc2OCCCOc2c1	CID:46907714	phase I
BRD-K06555716	CN(C)c1cccc(c1)-c1ccnc(n1)N1CCC(CC1)C(N)=O	CID:46907720	phase I
BRD-K84770158	CN(C)c1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907722	phase I
BRD-K11778076	NC(=O)C1CCN(CC1)c1nc(cs1)-c1ccc(N)cc1	CID:46907727	phase I
BRD-K50907285	NC(=O)C1CCN(CC1)c1nc(cs1)-c1ccc2OCCc2c1	CID:46907734	phase I
BRD-K92981876	Brc1ccc(cc1)-c1csc(n1)N1CCNCC1	CID:46907740	phase I
BRD-K74989018	NC(=O)C1CCN(CC1)c1nc(cs1)-c1ccc(OCc2ccccc2)cc1	CID:46907743	phase I
BRD-K10855750	Brc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C#N	CID:46907752	phase I
BRD-K58935841	CN(C)c1cccc(c1)-c1cnc(nc1)N1CCC(CC1)C(N)=O	CID:46907753	phase I
BRD-K68020183	Brc1ccc(cc1)-c1csc(n1)N1CCC(CC1)c1nn[nH]n1	CID:46907754	phase I
BRD-K17969842	CCOc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:46907757	phase I
BRD-K87426499	COc1ccc(cc1C)S(=O)(=O)N(C)C[C@@H]2Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:46907796	phase I
BRD-K11540476	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc3OCCOc3c2)Oc4c(NC(=O)Nc5cccc6ccccc56)cccc4C1=O	CID:46907798	phase I
BRD-K98896788	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3c(NC(=O)Nc4cccc5ccccc45)cccc3C1=O	CID:46907806	phase I
BRD-K02123250	Cn1cc(cn1)-c1ccc2nnc(n2n1)C(F)(F)c1ccc2ncccc2c1	CID:46911863	phase I
BRD-K65283978	COc1cccc(c1)-c1cc2nc(cc(N3CCN(CC3)C(C)=O)n2n1)-c1ccco1	CID:46912090	phase I
BRD-K41240505	Cc1ccc(cc1)-c1cc2nc(cc(N3CCN(Cc4ccoc4)CC3)n2n1)-c1ccco1	CID:46912091	phase I
BRD-K92793917	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:46912146	phase I
BRD-A17718497	CC1CN(CCN1C(=O)c1ccc(Cl)cc1)c1ccnc2cc(Cl)ccc12	CID:46912148	phase I
BRD-K06206016	Cc1cc2n(C)c3c(cnn(Cc4c(Cl)ccc(C)c4F)c3=O)c2s1	CID:46912192	phase I
BRD-K50218580	Cc1cc2n(C)c3c(cnn(Cc4cc(F)c(F)cc4F)c3=O)c2s1	CID:46912193	phase I
BRD-K28472299	Cc1cc2n(C)c3c(cnn(Cc4cc(F)ccc4F)c3=O)c2s1	CID:46912194	phase I
BRD-K90912239	COc1ccc(cc1)C(=O)Nc1cc(Cl)c(Br)cc1C(O)=O	CID:46916165	phase I
BRD-K65148867	CC(C)(C)c1ccc(cc1)C(=O)Nc1cc(Cl)ccc1-c1nn[nH]n1	CID:46916168	phase I
BRD-K22449070	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)c1nccs1	CID:46916170	phase I
BRD-A81377415	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)C1CCOC1	CID:46916178	phase I
BRD-K99146421	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)C1CCCC1	CID:46916179	phase I
BRD-A83706824	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)C1CCCCO1	CID:46916180	phase I
BRD-A69421747	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)C1CCCOC1	CID:46916182	phase I
BRD-K81214387	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)C1CC1	CID:46916192	phase I
BRD-K02437976	C(Nc1ncnc2ccc(cc12)-c1ccc2OCOc2c1)[C@@H]1CCCO1	CID:46916193	phase I
BRD-K73082558	Cc1ccccc1C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(O)=O)C#N)C(C)(C)C	CID:46916204	phase I
BRD-K66686673	COc1ccc(cc1Cl)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(O)=O)C#N)C(C)(C)C	CID:46916205	phase I
BRD-K15293421	CC(C)(C)[C@H](NC(=O)c1ccc(cc1)C(F)(F)F)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(O)=O)C#N	CID:46916206	phase I
BRD-K18495986	CC(C)(C)[C@H](NC(=O)c1cc(Cl)cc(Cl)c1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(O)=O)C#N	CID:46916207	phase I
BRD-A39599596	Fc1ccc(c(F)c1)-n1ncc2C(CCCc12)NC(=O)Cc1ccccc1	CID:46916306	phase I
BRD-A75558199	Fc1ccc(c(F)c1)-n1ncc2C(CCCc12)NC(=O)c1ccccc1	CID:46916310	phase I
BRD-K56489029	CCOc1ccc(CCNC(=O)c2cc3sccc3n2Cc2ccccc2)cc1OCC	CID:46916320	phase I
BRD-A84445767	Fc1ccc(c(F)c1)-n1ncc2C(CCCc12)NC(=O)c1cccs1	CID:46916321	phase I
BRD-A63949900	Oc1cccc(n1)C(=O)NC1CCCc2c1cnn2-c1ccc(F)cc1F	CID:46916324	phase I
BRD-K95517054	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:46925828	phase I
BRD-K73371640	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:46925839	phase I
BRD-K30836161	FC(F)C(=O)Nc1sc2CNCCc2c1-c1nc2ccccc2s1	CID:46925861	phase I
BRD-K18726304	CC(C)N1CCc2c(C1)sc(NC(=O)CCC#C)c2-c1nc2ccccc2s1	CID:46925865	phase I
BRD-K17754811	FC(F)(F)C(=O)Nc1sc2CNCCc2c1-c1nc2ccccc2s1	CID:46925867	phase I
BRD-K19724398	CC(C)N1CCc2sc(NC(C)=O)c(-c3nc4ccccc4s3)c2CC1	CID:46925870	phase I
BRD-K49477212	CC(=O)Nc1sc2CCNCc2c1-c1nc2ccccc2s1	CID:46925874	phase I
BRD-K00313977	CC(C)N1Cc2sc(NC(C)=O)c(-c3nc4ccccc4s3)c2C1	CID:46925875	phase I
BRD-K09902564	C1Cc2c(CN1)scc2-c1nc2ccccc2s1	CID:46925878	phase I
BRD-K29506255	CC(=O)Nc1sc2COCCc2c1-c1nc2ccccc2s1	CID:46925881	phase I
BRD-K30351863	CC(=O)Nc1sc2CNCc2c1-c1nc2ccccc2s1	CID:46925884	phase I
BRD-K32944375	CC(C)N1CCc2c(C1)sc(NC(C)=O)c2-c1nc(cs1)-c1ccccc1	CID:46925885	phase I
BRD-K18724229	CC(=O)Nc1sc2CNCCCc2c1-c1nc2ccccc2s1	CID:46925886	phase I
BRD-K93623501	CC(=O)Nc1sc2CNCCc2c1-c1cc2ccccc2o1	CID:46925887	phase I
BRD-K84762162	CC(C)N1CCc2c(C1)sc(NC(C)=O)c2-c1nc2ccccc2o1	CID:46925888	phase I
BRD-K03829970	CC(C)N1CCCc2c(C1)sc(NC(C)=O)c2-c1nc2ccccc2s1	CID:46925889	phase I
BRD-K18025010	Cc1ccc(Sc2c([N+]([O-])=O)c(=O)oc3ccccc23)cc1	CID:46926574	phase I
BRD-K32010074	[O-][N+](=O)c1cnc2ccccc2c1Sc1ccccc1	CID:46926575	phase I
BRD-K17823458	CC(C)(C)OC(=O)N[C@H]1CCCCC\C=C/[C@@H]2C[C@@]2(CNS(=O)(=O)C2CC2)NC(=O)[C@@H]2C[C@H](CN2C1=O)OC(=O)N1Cc2cccc(F)c2C1	CID:46931004	phase I
BRD-K17210248	COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](C[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(O)=O	CID:46931007	phase I
BRD-K96147838	CC(C)(C)c1ccc(cc1)C(=O)Nc1cc(Cl)c(Br)cc1C(O)=O	CID:46931017	phase I
BRD-K46681113	OC(c1cn(nn1)C(=O)N1CCC(Cc2ccccc2)CC1)(c1ccccc1)c1ccccc1	CID:46937231	phase I
BRD-A05565054	CCC1CCCCN1C(=O)n1cc(nn1)C(O)(c1ccccc1)c1ccccc1	CID:46937236	phase I
BRD-K89209981	OC(C1CCN(CC1)C(=O)n1cc(nn1)C(O)(c1ccccc1)c1ccccc1)(c1ccccc1)c1ccccc1	CID:46937243	phase I
BRD-K40711313	CC(C)(C)Cc1nnc(NC(=O)COc2ccc(Cl)cc2Cl)o1	CID:46943243	phase I
BRD-K14096083	Fc1ccc(OCC(=O)N[C@H]2CCCN(CC3CC3)C2)cc1Cl	CID:46943258	phase I
BRD-A96749488	COc1cc(O)c(C(CC(=O)N2CCCC(C)C2)c2ccccc2)c(OC)c1	CID:46943317	phase I
BRD-A38793261	COc1cc(O)c([C@@H](CC(=O)N2CC(C)CC(C)C2)c2ccc3OCOc3c2)c(OC)c1	CID:46943339	phase I
BRD-A66846505	COc1cc(O)c(C(CC(=O)N2CC(C)OC(C)C2)c2ccc3OCOc3c2)c(OC)c1	CID:46943351	phase I
BRD-A66604020	COc1cc(O)c(C(CC(=O)N2CCC(C)CC2)c2ccc3OCOc3c2)c(OC)c1	CID:46943400	phase I
BRD-K13318664	CCOc1ccc(CCNC(=O)Cc2ccccc2)cc1OCC	CID:46947844	phase I
BRD-K30434763	CCOc1ccc(CCNC(=O)c2cc3sccc3n2Cc2cccc(C)c2)cc1OCC	CID:46947845	phase I
BRD-K26815099	CCOc1ccc(CCNC(=O)C2CCCCC2)cc1OCC	CID:46947847	phase I
BRD-K82185908	CCOc1ccc(CCNC(=O)c2ccc3[nH]ccc3c2)cc1OCC	CID:46947854	phase I
BRD-K46017542	CCOc1ccc(CCNC(=O)c2ccc(Oc3ccccc3)cc2)cc1OCC	CID:46947855	phase I
BRD-K86273012	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccccc1Cl	CID:46947860	phase I
BRD-K71489689	CC(C)(C)c1ccc(cc1)C(=O)Nc1cc(Cl)c(Cl)cc1C(O)=O	CID:46947875	phase I
BRD-K15440898	CC(=NOC(=O)c1ccc(I)cc1)c1nccs1	CID:46948701	phase I
BRD-A96006241	CC(C)C(NC(=O)C(C)N)C(=O)NC(C)C(=O)Nc1cccc2ccccc12	CID:46948702	phase I
BRD-A61189834	CNC(C)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)Nc1ccc2[nH]ccc2c1	CID:46948703	phase I
BRD-A44862234	CNC(C)C(=O)NC(C(C)C)C(=O)NC(C(C)C)C(=O)Nc1cccc2ccccc12	CID:46948704	phase I
BRD-A94297859	CNC(C)C(=O)NC(C(C)C)C(=O)NC(C)C(=O)Nc1cccc2ccccc12	CID:46948705	phase I
BRD-A02747686	CNC(C)C(=O)NC(C(C)C)C(=O)NC(C)C(=O)NNc1ccccc1	CID:46948706	phase I
BRD-K07790824	CC(=O)Nc1ccc(cc1)C(C)=NNC(=O)C1CCCC1	CID:46948707	phase I
BRD-K18580829	COc1ccc(\C=C\C(=O)NC2=NCCS2)c(OC)c1	CID:47099517	phase I
BRD-K09186807	Fc1ccc(Cn2cccc(C(=O)N[C@@H](COc3ccc4[nH]c(=O)[nH]c4c3)c3ccccc3)c2=O)cc1F	CID:49766501	phase I
BRD-K93060291	Cc1onc(C(=O)N2CCN(CC2)C(c2ccc(F)cc2)c2ccc(F)cc2)c1[N+]([O-])=O	CID:49766518	phase I
BRD-K01877528	Cc1onc(C(=O)N2CCN(CC2)C(c2ccc(Cl)cc2)c2ccc(Cl)cc2)c1[N+]([O-])=O	CID:49766530	phase I
BRD-K50505048	Cc1onc(C(=O)N2CCN(CC2)C(c2ccccc2)c2ccccc2)c1Br	CID:49766538	phase I
BRD-K15166186	COc1ccc(cc1)C(N1CCN(CC1)C(=O)c1noc(C)c1[N+]([O-])=O)c1ccc(OC)cc1	CID:49766549	phase I
BRD-K40955748	CC(C)(C)c1ccc(cc1)C(=O)Nc1cc(Cl)c(F)cc1C(O)=O	CID:49766619	phase I
BRD-K67678077	Fc1ccc2c(c1)nc1sc(Nc3ccc4CCCc4c3)nn1c2=O	CID:49787091	phase I
BRD-K84301121	CC(C)(C)c1ccc(cc1)-c1noc(CCC(=O)NC2CC2)n1	CID:49787124	phase I
BRD-K24686773	Fc1ccc(cc1)C(=O)OCCCCSc1nnc(o1)-c1cccc2ccccc12	CID:49787910	phase I
BRD-K27290412	Fc1ccc(cc1)C(=O)OCc1ccc(CSc2nnc(o2)-c2cccc3ccccc23)cc1	CID:49787911	phase I
BRD-A96791331	O=C1CCCn2cc(COCC3CCCN13)nn2	CID:49818985	phase I
BRD-K57371454	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:49835814	phase I
BRD-K84570482	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:49835817	phase I
BRD-K78812164	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:49835833	phase I
BRD-K71142328	C(c1ncco1)n1nc(-c2ccccc2)c2ccccc12	CID:49835836	phase I
BRD-K90070572	C/C=C/c1cnc2O[C@@H](CN(C)S(=O)(=O)c3ccc(F)cc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:49835840	phase I
BRD-K32112425	COC(=O)Cn1nc(-c2ccccc2)c2cccc(c12)C(F)(F)F	CID:49835842	phase I
BRD-K95688283	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:49835843	phase I
BRD-K11518623	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:49835851	phase I
BRD-K98546361	O=C(Cn1nc(-c2ccccc2)c2ccccc12)Oc1ccccc1	CID:49835857	phase I
BRD-K46062088	On1[n+](c(C#N)c2ccc(cc12)[N+]([O-])=O)-c1ccccc1	CID:49835860	phase I
BRD-K98846091	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:49835862	phase I
BRD-K14324645	COC(=O)Cn1nc(-c2cccc(OC)c2)c2ccccc12	CID:49835877	phase I
BRD-K68594214	OC(=O)CCN1C(=S)S\C(=C/c2ccc(F)cc2F)C1=O	CID:49835913	phase I
BRD-K25536815	COc1ccc(C)cc1-n1c(C)cc(\C=C2\S\C(=N\C)N(C)C2=O)c1C	CID:49835916	phase I
BRD-K17086338	C\N=C1\S\C(=C\c2cc(C)n(c2C)-c2ccc(Cl)cc2F)C(=O)N1C	CID:49835921	phase I
BRD-K12401458	COCC\N=C1/S\C(=C/c2cc(C)n(c2C)-c2ccc(F)cc2F)C(=O)N1C	CID:49835928	phase I
BRD-K26831771	CC\N=C1\S\C(=C\c2cc(C)n(c2C)-c2ccc(Cl)cc2F)C(=O)N1CC	CID:49835932	phase I
BRD-K16940042	C\N=C1\S\C(=C\c2cc(C)n(Cc3ccccc3)c2C)C(=O)N1C	CID:49835933	phase I
BRD-K40175214	CCC(=O)N1CCN(CC1)c1ccc(cc1C(F)(F)F)-n1c2c(ccc1=O)cnc1ccc(cc21)-c1cnc2ccccc2c1	CID:49836027	phase I
BRD-K76079827	O=C(N1CCCC1)n1cc(nn1)-c1ccc(cc1)-c1ccccc1	CID:49837819	phase I
BRD-K47105324	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:49842945	phase I
BRD-K63263229	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)CCCCCC(=O)Nc3ccccc3N)cc2C1=O	CID:49842947	phase I
BRD-K73601942	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:49842952	phase I
BRD-K12189280	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:49842975	phase I
BRD-K98630904	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:49842983	phase I
BRD-K81858524	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:49842987	phase I
BRD-K88722443	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)CC4CCCCC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:49843003	phase I
BRD-K92434623	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:49843012	phase I
BRD-K05563014	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:49843020	phase I
BRD-K86182839	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:49843024	phase I
BRD-K65366129	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:49843054	phase I
BRD-K54517303	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:49843099	phase I
BRD-K60772276	O=C(NC1=NCCS1)\C=C\c1ccc(cc1)-c1ccccc1	CID:49843106	phase I
BRD-K63096635	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:49843125	phase I
BRD-K16257790	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:49843132	phase I
BRD-K07110772	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:49843139	phase I
BRD-K48703351	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:49843144	phase I
BRD-K74127463	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:49843150	phase I
BRD-K99581804	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:49843158	phase I
BRD-K57719270	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:49843205	phase I
BRD-K41042536	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:49843224	phase I
BRD-K12285126	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:49843260	phase I
BRD-K77326001	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:49843262	phase I
BRD-K59201357	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:49843270	phase I
BRD-K35932822	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:49843275	phase I
BRD-K42576592	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:49843290	phase I
BRD-K00185670	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:49843291	phase I
BRD-K49148914	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:49843297	phase I
BRD-K83541009	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:49843306	phase I
BRD-K02290471	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:49843312	phase I
BRD-K27239120	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(cc4C1=O)N(C)C	CID:49843318	phase I
BRD-K16970289	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:49843341	phase I
BRD-K98064019	COc1ccc(NC(=O)Nc2ccc3O[C@@H](CN(C)C(=O)Nc4ccccc4)[C@H](C)CN([C@@H](C)CO)C(=O)Cc3c2)cc1	CID:49843374	phase I
BRD-K49751344	CCCN(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:49843380	phase I
BRD-K01497355	COc1ccc(CN(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:49843384	phase I
BRD-K42303783	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:49843387	phase I
BRD-K35193330	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:49843401	phase I
BRD-K85211514	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:49843416	phase I
BRD-K05647501	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:49843424	phase I
BRD-K38733341	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:49843436	phase I
BRD-K84890987	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)CCCCCC(=O)Nc3ccccc3N)cc2C1=O	CID:49843440	phase I
BRD-K13217265	COc1ccc(NC(=O)N(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:49843441	phase I
BRD-K89000102	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:49843444	phase I
BRD-K48588790	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:49843445	phase I
BRD-K95212245	COc1ccc(COC[C@H](C)N2C[C@@H](C)[C@H](CN(C)S(=O)(=O)c3ccc(F)cc3)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C2=O)cc1	CID:49849909	phase I
BRD-K45399554	C[C@@H](CN(C)C)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:49849912	phase I
BRD-K91442916	C[C@@H](COC(=O)C(C)(C)C)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:49849931	phase I
BRD-K06180729	COCCOC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:49849932	phase I
BRD-K21642343	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:49849996	phase I
BRD-K48478472	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:49850016	phase I
BRD-K23897615	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:49850031	phase I
BRD-K00627859	CN1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO	CID:49850262	phase I
BRD-K05002121	C(Nc1ccnc(n1)N1CCOc2ccccc12)c1ccccc1	CID:49852180	phase I
BRD-K52446745	Clc1ccc(NC(=S)Nc2nnc(s2)-c2ccncc2)cc1Cl	CID:49852226	phase I
BRD-K48844671	Fc1ccc(NC(=O)Nc2nnc(s2)-c2ccncc2)cc1C(F)(F)F	CID:49852229	phase I
BRD-K80962769	CC(C)N1CCc2c(C1)scc2-c1nc2ccccc2s1	CID:49852782	phase I
BRD-K07515761	FC(F)(F)c1cccc(c1)N1CCN(CC1)C(=S)Nc1nccc2ccccc12	CID:49852823	phase I
BRD-K28040935	Fc1ccc(F)c(OCCn2c(CCNC(=O)C3CCCCC3)nc3ccccc23)c1	CID:49852888	phase I
BRD-K76021727	Cc1ccc(OCCn2c(CCNC(=O)C3CCCCCC3)nc3ccccc23)cc1	CID:49852929	phase I
BRD-A31946439	Cc1ccnc(NC(=S)N2CC3CN(CC3C2)c2cccc(c2)C(F)(F)F)c1	CID:49852959	phase I
BRD-K19134488	Cc1cc(C)nc(NC(=S)N2CCN(CC2)c2ccc(Cl)c(Cl)c2)c1	CID:49852967	phase I
BRD-K86846944	CC(C)N1CCc2c(C1)sc(NC(=O)C(F)(F)F)c2-c1nc2ccccc2s1	CID:49853011	phase I
BRD-K21401822	O=C(NCCc1nc2ccccc2n1CCOc1ccc2cccnc2c1)C1CCCCC1	CID:49853159	phase I
BRD-K23165181	Cc1ccnc(NC(=S)N2CCC(CC2)Nc2cccc(c2)C(F)(F)F)c1	CID:49853258	phase I
BRD-K38625260	CC(C)N1CCc2c(C1)sc(NC(=O)C(F)F)c2-c1nc2ccccc2s1	CID:49853292	phase I
BRD-K63308290	Cc1cc(C)nc(NC(=S)N2CCN(CC2)c2ncc(cc2Cl)C(F)(F)F)c1	CID:49853301	phase I
BRD-K08829932	Cc1ccc(OCCn2c(CCNC(=O)c3ccc(F)cc3F)nc3ccccc23)cc1	CID:49853364	phase I
BRD-K12690157	Cc1cc(C)nc(NC(=S)N2CCN(CC2)c2ccc(cn2)C(F)(F)F)c1	CID:49853368	phase I
BRD-K75308783	COc1cc(Nc2nc3ccccc3nc2NS(=O)(=O)c2ccc(NC(=O)c3ccc(C)c(OC)c3)cc2)cc(OC)c1	CID:49867926	phase I
BRD-K16358524	COc1c(ccc2OC(C)(C)C=Cc12)C(=O)\C=C\c1ccccc1	CID:50897562	phase I
BRD-K07521754	COc1ccc2C=CC(C)(C)Oc2c1C(=O)\C=C\c1ccccc1	CID:50897563	phase I
BRD-K99530743	CC1(C)Oc2c(C=C1)ccc(O)c2C(=O)\C=C\c1ccccc1	CID:50897566	phase I
BRD-A38425832	COc1ccc(cc1COc1ccccc1C)C1Nc2ccccc2C(=O)N1Cc1ccco1	CID:50897769	phase I
BRD-K75940587	CCC(=O)Nc1ccc(Cl)cc1C(=O)c1ccc[nH]1	CID:50897777	phase I
BRD-K02381115	C[C@@H](N)C(=O)Nc1ccc(Cl)cc1C(=O)c1ccc[nH]1	CID:50897779	phase I
BRD-A34421300	COc1ccc(cc1COc1c(C)cccc1C)C1Nc2ccccc2C(=O)N1Cc1ccc(C)o1	CID:50897785	phase I
BRD-A21406558	COc1ccc(cc1COc1c(C)cccc1C)C1Nc2ccccc2C(=O)N1Cc1cccs1	CID:50897786	phase I
BRD-K52695588	N[C@H](C(=O)Nc1ccc(Cl)cc1C(=O)c1ccc[nH]1)c1ccccc1	CID:50897790	phase I
BRD-K00637033	NCCC(=O)Nc1ccc(Cl)cc1C(=O)c1ccc[nH]1	CID:50897799	phase I
BRD-A93507363	Cc1cccc(C)c1OCc1cccc(c1)C1Nc2ccccc2C(=O)N1Cc1ccco1	CID:50897801	phase I
BRD-A30612536	COc1ccc(cc1COc1c(C)cc(NC(C)=O)cc1C)C1Nc2ccccc2C(=O)N1Cc1ccco1	CID:50897809	phase I
BRD-A61599461	COc1ccc(cc1COc1c(C)cccc1C)C1Nc2ccccc2C(=O)N1Cc1cccnc1	CID:50897816	phase I
BRD-K90667125	CCOc1ccc(cc1)-c1nc(CSCC(=O)NC2CCC2)c(C)o1	CID:50898021	phase I
BRD-K08447949	CCCCc1ccc(cc1)-c1noc(CCC(=O)NCC)n1	CID:50898027	phase I
BRD-K43149678	CCNC(=O)CCc1nc(no1)-c1ccc(cc1)C(C)C	CID:50898042	phase I
BRD-K98575502	CCOc1ccc(cc1)-c1nc(CSCC(=O)NCC#C)c(C)o1	CID:50898054	phase I
BRD-K69422440	CCCOc1ccc(cc1)-c1nc(CSCC(=O)NC2CC2)c(C)o1	CID:50898056	phase I
BRD-K28215800	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccc(Cl)cc1Cl	CID:50898226	phase I
BRD-K91600270	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccc(cc1)N(C)C	CID:50898228	phase I
BRD-K85937960	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccc2CCCc2c1	CID:50898231	phase I
BRD-K35413818	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccc(F)c(F)c1	CID:50898234	phase I
BRD-K79414420	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccc(OC)c(Cl)c1	CID:50898237	phase I
BRD-K31828306	CCOC(=O)C1CCN(CC1)C(=O)C(C)(C)NC(=O)Nc1ccc(cc1Cl)C(F)(F)F	CID:50898245	phase I
BRD-K31780183	Cc1csc(NC(=O)c2ccc(COc3ccccc3F)o2)n1	CID:50904129	phase I
BRD-K59019422	Cc1csc(NC(=O)c2ccc(COc3cccc(Cl)c3)o2)n1	CID:50904134	phase I
BRD-K09299610	COc1ccc2cc(ccc2c1)-c1cn(nn1)C(=O)N(c1ccccc1)c1ccccc1	CID:50904525	phase I
BRD-K14711204	CC(C)CC(O)(CC(C)C)c1cn(nn1)C(=O)N(c1ccccc1)c1ccccc1	CID:50904528	phase I
BRD-K14749055	OC(c1cn(nn1)C(=O)N1CCc2ccccc2C1)(c1ccccc1)c1ccccc1	CID:50904531	phase I
BRD-K69181860	CCc1ccc(cc1)\C=C\C(=O)NC1=NCCS1	CID:50910523	phase I
BRD-K15206810	COc1cccc2c(NCc3ccccc3)nc(nc12)-n1c(N)nc2cc(Cl)c(Cl)cc12	CID:50918583	phase I
BRD-K20492338	Nc1nc2ccccc2n1-c1nc(NCc2ccccc2)c2ccccc2n1	CID:50918585	phase I
BRD-A93393712	Fc1ccc(cc1)C(=O)C(CN1CCCCC1)c1ccccc1	CID:51003685	phase I
BRD-A83124583	Fc1cccc(c1)C(=O)C(CN1CCOCC1)c1ccccc1	CID:51003694	phase I
BRD-A25088322	CN1CCN(CC(C(=O)c2ccc(F)cc2)c2ccccc2)CC1	CID:51003695	phase I
BRD-A49848186	Fc1ccccc1C(=O)C(CN1CCOCC1)c1ccccc1	CID:51003698	phase I
BRD-K16234721	Cc1csc(NC(=O)c2ccc(COc3ccc(Cl)c(Cl)c3)o2)n1	CID:51003702	phase I
BRD-A50774520	Fc1ccc(cc1)C(=O)C(CN1CCCC1)c1ccccc1	CID:51003716	phase I
BRD-A06929388	CCN(CC)CC(C(=O)c1ccc(F)cc1)c1ccccc1	CID:51003717	phase I
BRD-A59145032	FC(F)(F)c1ccc(cc1)C(=O)C(CN1CCOCC1)c1ccccc1	CID:51003718	phase I
BRD-A80775386	CC(C)C(=O)[C@@]12C(=O)C(CC=C(C)C)C(=O)[C@@](CC=C(C)C)(C[C@H](CC=C(C)C)[C@@]1(C)CCC=C(C)C)C2=O	CID:51348735	phase I
BRD-K68174511	Nc1ccc(cn1)-c1ccc2ncc3ccc(=O)n(-c4cccc(c4)C(F)(F)F)c3c2c1	CID:51358113	phase I
BRD-K15912359	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)N3CCN(C)CC3)OCc4cn(CCCC1=O)nn4	CID:51358831	phase I
BRD-K86638751	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:51358854	phase I
BRD-K11483659	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:51358866	phase I
BRD-K19642661	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:51358867	phase I
BRD-A34037822	Cn1ccc2c(cc3C4CCC(O4)c3c12)-c1ccc(cc1)C(C)(C)C	CID:51360697	phase I
BRD-K81001086	NC(=O)c1cc[n+](CC2=C(N3[C@H](SC2)[C@@H](NC(=O)[C@@H](c2ccccc2)S(O)(=O)=O)C3=O)C(O)=O)cc1	CID:51387307	phase I
BRD-A95074085	CCCC(=O)Nc1ncnc2n(cnc12)[C@H]1O[C@H]2COP(O)(=O)O[C@@H]2[C@@H]1OC(=O)CCC	CID:51397512	phase I
BRD-K01014769	CC(=O)OCC(=O)[C@@]1(O)CC[C@H]2[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]12C	CID:51397657	phase I
BRD-K29731656	C[C@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@H]1CC[C@@H]2C(=O)CO	CID:51414212	phase I
BRD-K99338088	CC(=O)O[C@]1(C(C)=O)C(=C)C[C@@H]2[C@@H]3C=C(C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:51695577	phase I
BRD-K17041687	C[C@H]1C[C@@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(OC(C)=O)C(=O)COC(C)=O	CID:52897293	phase I
BRD-K59067695	CN(c1cccc(Cl)c1)S(=O)(=O)c1ccc2NC(=O)\C(=C\c3[nH]c(C)c(C(=O)N4CCN(C)CC4)c3C)c2c1	CID:52911310	phase I
BRD-K04801023	Cc1ccc(cc1)S(=O)(=O)Nc1nc2ccccc2nc1Nc1cccc2nsnc12	CID:52914932	phase I
BRD-K42918627	COc1nccc(-c2ccc3nccc(-c4ccnnc4)c3c2)c1NS(=O)(=O)c1ccc(F)cc1F	CID:52914946	phase I
BRD-K42728290	CCN1CCN(CC1)c1ccc(Nc2cc(ncn2)N(C)C(=O)Nc2c(Cl)c(OC)cc(OC)c2Cl)cc1	CID:53235510	phase I
BRD-K18964980	Cc1cncc2cccc(c12)S(=O)(=O)N[C@H]1CN[C@H](CO)C1	CID:53245442	phase I
BRD-K03763695	Cc1cncc2cccc(c12)S(=O)(=O)N[C@@H]3CCNC3	CID:53245449	phase I
BRD-K03073752	Cc1cncc2cccc(c12)S(=O)(=O)N3CC[C@H](N)C3	CID:53245456	phase I
BRD-K22828899	CC(=O)NC[C@@H]1C[C@H](CN1)NS(=O)(=O)c1cccc2cncc(C)c12	CID:53245473	phase I
BRD-K05087650	CN1CCN(CC1)C(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccnc1)C(=O)CC1CC1	CID:53299817	phase I
BRD-K14889526	CCS(=O)(=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCCOC	CID:53299819	phase I
BRD-K96411295	CCS(=O)(=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCCOC	CID:53299821	phase I
BRD-K88881681	CCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cncnc1)C(C)=O	CID:53299835	phase I
BRD-K22961642	CCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cncnc1)C(C)=O	CID:53299846	phase I
BRD-K98195492	CCC(=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccccc1OC)C(=O)Nc1nccs1	CID:53299867	phase I
BRD-K98762074	CCN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(\C=C\c4cnc5[nH]ccc5c4OC)c3)cc2C(F)(F)F)CC1	CID:53302361	phase I
BRD-K14177560	CC(=O)O[C@H]1CC[C@@H]2[C@H]3CC[C@@]4(C)[C@H](CC[C@@]4(OC(C)=O)C#C)[C@@H]3CCC2=C1	CID:53315104	phase I
BRD-A56798952	CO[C@H]1\C=C/C=C(C)/C[C@H](C)[C@H](O)[C@H](C)\C=C(C)\C=C(OC)\C(=O)OC1[C@@H](C)[C@@H](O)[C@H](C)[C@@]1(O)C[C@@H](O)[C@H](C)[C@H](O1)C(C)C	CID:53321987	phase I
BRD-A08662020	CNC(C)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)Nc1cccc2ncccc12	CID:53338799	phase I
BRD-K58247702	CCOP(=O)(OCC)c1ccc2-c3ccccc3C(=O)c2c1	CID:53338806	phase I
BRD-K69695287	OP(O)(=O)c1ccc2-c3ccccc3C(=O)c2c1	CID:53338807	phase I
BRD-K43267173	NC(=O)C1CCN(CC1)c1ccnc(Cl)n1	CID:53338826	phase I
BRD-K31887147	CSc1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:53338830	phase I
BRD-K71540055	CN1CCN(CC1)c1ccc(cc1)-c1csc(n1)N1CCC(CC1)C(N)=O	CID:53338836	phase I
BRD-K95985487	COc1ccc(cc1)-n1ncc2cnc(Nc3ccc(N4CCN(C)CC4)c(OC)c3)nc12	CID:53347976	phase I
BRD-K05922103	O=C(Nc1ccccc1-c1nc2ccccc2[nH]c1=O)c1ccccn1	CID:53347979	phase I
BRD-K66645150	Fc1ccc(c(NC(=O)c2cccs2)c1)-c1nc2ccccc2[nH]c1=O	CID:53377419	phase I
BRD-K48188942	CC(C)c1ccc(NC(=O)c2cccs2)c(c1)-c1nc2ccccc2[nH]c1=O	CID:53377448	phase I
BRD-K62804700	COC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2ccccc2F)[C@@H](CO)O1	CID:53382571	phase I
BRD-K42107428	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)NC1CCCCC1	CID:53382623	phase I
BRD-K67733157	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@H]1C	CID:53382626	phase I
BRD-K98814272	CN1CCN(CC1)C(=O)C[C@H]1O[C@H](CO)[C@@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:53382629	phase I
BRD-K76527818	OC[C@H]1O[C@H](CC(=O)NCC2CCCCC2)C=C[C@H]1NC(=O)Nc1cccc(F)c1	CID:53382636	phase I
BRD-K90873269	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@H]1NS(=O)(=O)c1ccccc1	CID:53382638	phase I
BRD-K14413722	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@@H]1NC(=O)c1ccccn1	CID:53382643	phase I
BRD-K68664718	OC[C@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@@H]1NC(=O)c1cnccn1	CID:53382646	phase I
BRD-K30571172	OC[C@H]1O[C@@H](CC(=O)NCC2CC2)C=C[C@H]1NC(=O)c1ccncc1	CID:53382657	phase I
BRD-K14151426	COc1ccc(NC(=O)N[C@H]2CC[C@@H](CC(=O)NC3CCC3)O[C@@H]2CO)cc1	CID:53382659	phase I
BRD-K51339020	OC[C@H]1O[C@H](CC(=O)NCCCN2CCOCC2)C=C[C@@H]1NS(=O)(=O)c1ccccc1F	CID:53382666	phase I
BRD-K57519495	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@H](C)NC[C@@H]1C	CID:53382685	phase I
BRD-K51585944	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:53382697	phase I
BRD-K79367177	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)CN1CCOCC1	CID:53382701	phase I
BRD-K64380616	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H]1C)OC	CID:53382703	phase I
BRD-K51381937	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@H](C)N(CC2CCCCC2)C[C@H]1C	CID:53382706	phase I
BRD-K03301842	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H]1C)OC	CID:53382716	phase I
BRD-K64682090	CCCNC(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@@H]1CO	CID:53382727	phase I
BRD-K46352899	COC(=O)C[C@H]1CC[C@H]2NC[C@@H](O)COC[C@@H]2O1	CID:53382758	phase I
BRD-K39405368	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@@H]2N(Cc2cc(F)ccc2F)C1	CID:53382763	phase I
BRD-K95910173	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:53382764	phase I
BRD-K84853311	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2cccc(F)c2)O1	CID:53382778	phase I
BRD-K12805559	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCCc3ccccc3)CC[C@H]2N(Cc2ccc(Cl)cc2)C1	CID:53382781	phase I
BRD-K23557133	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:53382788	phase I
BRD-K35243934	COC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:53382789	phase I
BRD-K92000256	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@H]2N(Cc2nccs2)C1	CID:53382792	phase I
BRD-A86109770	CC=C1C(=O)CC2C3CCC4=CC(=O)CCC4(C)C3CCC21C	CID:53394010	phase I
BRD-K26573499	CN(C)c1ccc(cc1)\C=C1CCCN=C/1c1cccnc1	CID:53429689	phase I
BRD-K76941385	COc1cc2[C@H]3C[C@@H](O)[C@H](CC(C)C)CN3CCc2cc1O	CID:53487027	phase I
BRD-A96107863	COC(=O)C1C(C(=C(C)N=C1C)C(=O)OCC(C)C)c2ccccc2[N+](=O)[O-]	CID:53729257	phase I
BRD-A20958854	NCCc1ccc(OC2O[C@@H]([C@@H](O)[C@H](O)[C@H]2O)C(O)=O)c(O)c1	CID:53734236	phase I
BRD-A30977374	COC(=O)C1C(C(=C(C)N=C1C)C(=O)OC)c2ccccc2[N+](=O)[O-]	CID:54167661	phase I
BRD-A69927616	COC(=O)C1C(C(=C(C)N=C1C)C(=O)OC(C)C)c2cccc3nonc23	CID:54248788	phase I
BRD-A88774919	CC1C2C(O)C3C(N(C)C)C(=O)C(C(N)=O)C(=O)C3(O)C(=O)C2C(=O)c2c(O)cccc12	CID:54416524	phase I
BRD-K81365479	COCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2S(=O)(=O)c1ccccc1C	CID:54596116	phase I
BRD-K93200353	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)N1CCOCC1)N2S(=O)(=O)c1ccccc1F	CID:54596118	phase I
BRD-K09290524	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2S(=O)(=O)c1cccc(C)c1	CID:54596120	phase I
BRD-K18571495	COCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2S(=O)(=O)c1ccccc1C	CID:54596123	phase I
BRD-K15912020	CS(=O)(=O)N1[C@@H]2Cn3c(cccc3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCc1ccccc1	CID:54596125	phase I
BRD-K91892860	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2S(=O)(=O)c1cccc(C)c1	CID:54596130	phase I
BRD-K58466974	CC(=O)NC[C@H]1C[C@H](CN1)N(C(C)=O)S(=O)(=O)c1cccc2cncc(C)c12	CID:54596134	phase I
BRD-K14096157	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)N1CCOCC1)N2S(=O)(=O)c1ccccc1F	CID:54596141	phase I
BRD-K04643052	CS(=O)(=O)N1[C@H]2Cn3c(cccc3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCc1ccccc1	CID:54596142	phase I
BRD-K35669573	Cc1cncc2cccc(c12)S(=O)(=O)N[C@H]3CCNC3	CID:54596143	phase I
BRD-K78639526	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)C4CCCCC4)cc3CC1=O	CID:54613797	phase I
BRD-K28317853	COc1ccc(NC(=O)Nc2ccc3O[C@H](CN(C)CC4CCCCC4)[C@@H](C)CN([C@H](C)CO)C(=O)Cc3c2)cc1	CID:54613802	phase I
BRD-K60067222	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(cc4C1=O)N(C)C	CID:54613883	phase I
BRD-K95409124	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)Cc3ccc4OCOc4c3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:54613903	phase I
BRD-K06146388	CC(C)NC(=O)N(C)C[C@@H]1Oc2ccc(NC(=O)Cc3cn(C)c4ccccc34)cc2CC(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54613904	phase I
BRD-K29639729	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCN4CCOCC4)cc3C1=O	CID:54613905	phase I
BRD-K31251993	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:54613906	phase I
BRD-K83718139	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:54613907	phase I
BRD-K24736231	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:54613908	phase I
BRD-K53227073	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2CC1=O	CID:54613909	phase I
BRD-K77221801	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:54613910	phase I
BRD-K66966735	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Cn4cnnn4)cc3C1=O	CID:54613911	phase I
BRD-K40365006	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCN(C)C)cc3CC1=O	CID:54613912	phase I
BRD-K56984065	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCN(C)C)cc3CC1=O	CID:54613913	phase I
BRD-K06663126	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54613914	phase I
BRD-K01348631	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)Nc3cccc4ccccc34)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54613915	phase I
BRD-K99487580	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:54613916	phase I
BRD-K83385358	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:54613917	phase I
BRD-K24798550	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4CC1=O	CID:54613918	phase I
BRD-K04380254	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4C1=O	CID:54613919	phase I
BRD-K02987635	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54613920	phase I
BRD-K97939101	COc1ccc(CN(C)C[C@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54613921	phase I
BRD-K43605845	COc1ccc(CN(C)C[C@@H]2Oc3ccc(NC(=O)NC4CCCCC4)cc3CC(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54613922	phase I
BRD-K73199200	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4ccc(NC(=O)CCCN(C)C)cc4C1=O	CID:54613923	phase I
BRD-K84290569	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:54613924	phase I
BRD-K98194167	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:54613925	phase I
BRD-K03289154	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ccc(NC(=O)Nc3cccc4ccccc34)cc2CC1=O	CID:54613926	phase I
BRD-K91738333	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54613927	phase I
BRD-K59482768	CNC[C@H]1Oc2ccc(NC(=O)Nc3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54613928	phase I
BRD-K77545824	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)CC3CC3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:54613929	phase I
BRD-K89298751	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)CC3CC3)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:54613930	phase I
BRD-K95416928	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)CC3CC3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:54613931	phase I
BRD-K79758054	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NS(=O)(=O)C)cc3CC1=O	CID:54613932	phase I
BRD-K04328580	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc3ccccc23)Oc4ccc(NS(=O)(=O)C)cc4CC1=O	CID:54613933	phase I
BRD-K86910216	CC(C)NC(=O)Nc1ccc2O[C@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)Cc2c1	CID:54613934	phase I
BRD-K04993985	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:54613935	phase I
BRD-K65093687	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ccc(NC(=O)Cc5cn(C)c6ccccc56)cc4C1=O	CID:54613965	phase I
BRD-K40461288	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3CC1=O	CID:54614162	phase I
BRD-K18876264	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4ccccc4)cc3CC1=O	CID:54614166	phase I
BRD-K88290000	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)c4ccncc4)cc3CC1=O	CID:54614174	phase I
BRD-K70804088	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3CC1=O	CID:54614176	phase I
BRD-K20625691	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)C4CC4)cc3CC1=O	CID:54614204	phase I
BRD-K88529044	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3ccc(NC(=O)NC4CCCCC4)cc3CC1=O	CID:54614219	phase I
BRD-K59887251	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3CC1=O	CID:54614223	phase I
BRD-K25214457	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccccc4)cc3CC1=O	CID:54614231	phase I
BRD-K38803221	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)NC4CCCCC4)cc3CC1=O	CID:54614240	phase I
BRD-K55137639	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3CC1=O	CID:54614241	phase I
BRD-K66793411	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:54614256	phase I
BRD-K44421266	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:54614262	phase I
BRD-K09596790	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Cc4cn(C)c5ccccc45)cc3CC1=O	CID:54614268	phase I
BRD-K15634164	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3CC1=O	CID:54614320	phase I
BRD-K87367419	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3CC1=O	CID:54614335	phase I
BRD-K47419679	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3CC1=O	CID:54614400	phase I
BRD-K88817140	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)NC5CCCCC5)cc4CC1=O	CID:54614404	phase I
BRD-K86606617	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)C4CCCCC4)cc3CC1=O	CID:54614411	phase I
BRD-K02519835	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:54614427	phase I
BRD-K43226598	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ccc(NC(=O)CCCCCC(=O)Nc5ccccc5N)cc4CC1=O	CID:54614463	phase I
BRD-K53293903	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc3CC1=O	CID:54614484	phase I
BRD-K74020160	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54614525	phase I
BRD-K18832733	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3CC1=O	CID:54614526	phase I
BRD-K09423613	CC(C)NC(=O)Nc1ccc2O[C@@H](CN(C)C(=O)Nc3ccc4OCOc4c3)[C@H](C)CN([C@@H](C)CO)C(=O)Cc2c1	CID:54614567	phase I
BRD-K57678861	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4c(NC(=O)Nc5ccccc5)cccc4C1=O	CID:54614568	phase I
BRD-K75051049	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)Oc4ccc(NS(=O)(=O)c5ccccc5)cc4CC1=O	CID:54614602	phase I
BRD-K00431438	CNC[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614640	phase I
BRD-K00867929	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614641	phase I
BRD-K01678149	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)NC(C)C)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54614646	phase I
BRD-K03391109	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54614655	phase I
BRD-K10716948	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54614681	phase I
BRD-K17103381	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54614702	phase I
BRD-K17698750	CNC[C@@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc(F)cc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54614707	phase I
BRD-K26817071	CCCN(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)C)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614768	phase I
BRD-K29081238	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3cn(C)cn3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54614783	phase I
BRD-K91833864	CNC[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614938	phase I
BRD-K42035280	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54614978	phase I
BRD-K68325161	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54614979	phase I
BRD-K17288883	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54614980	phase I
BRD-K73121863	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614981	phase I
BRD-K28918096	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54614982	phase I
BRD-K10008415	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614983	phase I
BRD-K04592856	CC(C)NC(=O)N(C)C[C@@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614984	phase I
BRD-K36466190	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54614985	phase I
BRD-K70496443	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54614986	phase I
BRD-K14363876	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54614987	phase I
BRD-K47295867	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54614988	phase I
BRD-K20949245	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54614989	phase I
BRD-K53220080	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54614990	phase I
BRD-K79131144	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54614991	phase I
BRD-K79260832	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54614992	phase I
BRD-K03245321	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54614993	phase I
BRD-K15950605	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54614994	phase I
BRD-K07039703	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54614995	phase I
BRD-K61991236	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54614996	phase I
BRD-K01329157	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54614997	phase I
BRD-K01739339	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54614998	phase I
BRD-K20139170	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54614999	phase I
BRD-K79112806	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615000	phase I
BRD-K38700430	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54615001	phase I
BRD-K80138901	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54615002	phase I
BRD-K90748376	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54615003	phase I
BRD-K14078057	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615004	phase I
BRD-K51388814	CCCN(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54615005	phase I
BRD-K73517272	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615006	phase I
BRD-K52220918	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)C(=O)CCC(F)(F)F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54615008	phase I
BRD-K62431786	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54615009	phase I
BRD-K76859558	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H](C)CCCCO[C@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54615010	phase I
BRD-K41889859	CCCN(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54615011	phase I
BRD-K69598982	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54615012	phase I
BRD-K03050720	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC(C)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615013	phase I
BRD-K96385755	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54615014	phase I
BRD-K16050964	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54615015	phase I
BRD-K52856667	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54615016	phase I
BRD-K42006110	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615017	phase I
BRD-K93971021	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615018	phase I
BRD-K66361302	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@@H](CN(C)C(=O)NC(C)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615019	phase I
BRD-K64951577	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615020	phase I
BRD-K44421914	CC(C)NC(=O)N(C)C[C@H]1OCCCC[C@H](C)Oc2ccc(NC(=O)C3CCCCC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54615021	phase I
BRD-K32885145	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615022	phase I
BRD-K93158953	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615023	phase I
BRD-K31697605	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615024	phase I
BRD-K41871066	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615025	phase I
BRD-K28083085	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615026	phase I
BRD-K19818442	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615027	phase I
BRD-K14433433	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54615028	phase I
BRD-K42841961	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54615029	phase I
BRD-K02515288	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54615030	phase I
BRD-K46629170	COc1ccc(CN(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54615031	phase I
BRD-K75035820	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)OCCCC[C@H](C)Oc2ccc(NC(=O)c3ccncc3)cc2C1=O	CID:54615032	phase I
BRD-K92740670	CC(C)NC(=O)Nc1ccc2O[C@H](C)CCCCO[C@@H](CN(C)C(=O)NC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615033	phase I
BRD-K37631226	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615034	phase I
BRD-K55185663	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615035	phase I
BRD-K06064877	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615036	phase I
BRD-K50058777	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615037	phase I
BRD-K94809766	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615038	phase I
BRD-K30126976	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615039	phase I
BRD-K12744202	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615040	phase I
BRD-K96309168	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615041	phase I
BRD-K35090513	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615042	phase I
BRD-K47396627	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615043	phase I
BRD-K00188019	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615044	phase I
BRD-K22951866	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(cc3C1=O)N(C)C	CID:54615045	phase I
BRD-K13346599	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54615046	phase I
BRD-K73434976	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54615047	phase I
BRD-K36206486	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54615048	phase I
BRD-K67484450	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54615049	phase I
BRD-K15179096	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)C)cc3C1=O	CID:54615050	phase I
BRD-K46610687	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615051	phase I
BRD-K96903074	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54615052	phase I
BRD-K31485493	CC(C)NC(=O)Nc1ccc2O[C@@H](C)CCCCO[C@H](CN(C)CC3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54615053	phase I
BRD-K78544941	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54615054	phase I
BRD-K00819343	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54615055	phase I
BRD-K09019812	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54615056	phase I
BRD-K53790075	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54615057	phase I
BRD-K94501123	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615058	phase I
BRD-K54730162	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615059	phase I
BRD-K56646986	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615060	phase I
BRD-K25870200	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615061	phase I
BRD-K19549666	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615062	phase I
BRD-K29256470	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615063	phase I
BRD-K15790516	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615064	phase I
BRD-K91016007	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:54615065	phase I
BRD-K08014780	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:54615066	phase I
BRD-K31998493	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:54615067	phase I
BRD-K38313084	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:54615068	phase I
BRD-K70595737	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:54615069	phase I
BRD-K72913953	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615070	phase I
BRD-K36596997	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615071	phase I
BRD-K12345237	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615072	phase I
BRD-K54010839	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615073	phase I
BRD-K37340147	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615074	phase I
BRD-K47636932	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@H](CN(C)CC4CC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54615075	phase I
BRD-K16464815	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@H](CN(C)CC4CC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54615076	phase I
BRD-K43253317	COc1ccc(NC(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)CC4CC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54615077	phase I
BRD-K80058284	COc1ccc(NC(=O)Nc2ccc3O[C@@H](C)CCCCO[C@H](CN(C)CC4CC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54615078	phase I
BRD-K76850979	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)CC4CC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54615079	phase I
BRD-K43453714	COc1ccc(NC(=O)Nc2ccc3O[C@H](C)CCCCO[C@@H](CN(C)CC4CC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54615080	phase I
BRD-K29451642	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:54615081	phase I
BRD-K43838150	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:54615082	phase I
BRD-K79489641	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:54615083	phase I
BRD-K88522059	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54615084	phase I
BRD-K91390083	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54615085	phase I
BRD-K47081163	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54615086	phase I
BRD-K20531360	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:54615087	phase I
BRD-K66812281	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:54615088	phase I
BRD-K28743085	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615089	phase I
BRD-K31822300	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615090	phase I
BRD-K56899980	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615091	phase I
BRD-K02917242	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615092	phase I
BRD-K05211263	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4c(C)noc4C)cc3C1=O	CID:54615093	phase I
BRD-K05351800	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:54615094	phase I
BRD-K09054764	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:54615095	phase I
BRD-K52675185	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:54615096	phase I
BRD-K44465671	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:54615097	phase I
BRD-K33979365	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:54615098	phase I
BRD-K73388776	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615099	phase I
BRD-K02418197	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615100	phase I
BRD-K77741497	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615101	phase I
BRD-K31175437	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615102	phase I
BRD-K41069217	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615103	phase I
BRD-K34798063	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615104	phase I
BRD-K63880531	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615105	phase I
BRD-K24776959	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:54615106	phase I
BRD-K30309936	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:54615107	phase I
BRD-K31380618	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:54615108	phase I
BRD-K15050703	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:54615109	phase I
BRD-K54263226	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:54615110	phase I
BRD-K31999759	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4c(C)noc4C)cc3C1=O	CID:54615111	phase I
BRD-K46448313	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54615112	phase I
BRD-K30633722	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54615113	phase I
BRD-K38459107	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54615114	phase I
BRD-K64272762	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54615115	phase I
BRD-K55699053	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54615116	phase I
BRD-K01981286	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54615117	phase I
BRD-K70590207	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54615118	phase I
BRD-K01404579	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54615119	phase I
BRD-K46047563	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54615120	phase I
BRD-K09031632	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54615121	phase I
BRD-K75781834	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54615122	phase I
BRD-K32444480	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCCCC[C@H](C)Oc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54615123	phase I
BRD-K63230271	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:54615594	phase I
BRD-K56664261	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc3ccccc23)OCCCC[C@H](C)Oc4ccc(NS(=O)(=O)c5cccs5)cc4C1=O	CID:54615606	phase I
BRD-K94725447	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:54615628	phase I
BRD-K22663811	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:54615631	phase I
BRD-K44562105	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54615634	phase I
BRD-K43286821	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54615637	phase I
BRD-K20616644	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:54615639	phase I
BRD-K49797414	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:54615640	phase I
BRD-K59562667	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:54615655	phase I
BRD-K90608600	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:54615662	phase I
BRD-K13468108	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)NC4CCCCC4)cc3C1=O	CID:54615666	phase I
BRD-K05718365	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C1=O	CID:54615681	phase I
BRD-K81665681	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:54615696	phase I
BRD-K53228569	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:54615699	phase I
BRD-K42478751	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:54615702	phase I
BRD-K07531476	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54615718	phase I
BRD-K72808738	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:54615827	phase I
BRD-K70559158	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cn(C)cn4)cc3C1=O	CID:54615828	phase I
BRD-K65494396	COc1ccc(NC(=O)N(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54615933	phase I
BRD-K07734969	COc1ccc(NC(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54615934	phase I
BRD-K40606280	COc1ccc(NC(=O)N(C)C[C@@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54615937	phase I
BRD-K34544769	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:54615949	phase I
BRD-K11672081	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCCCC[C@@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:54615950	phase I
BRD-K56243496	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(NC(=O)C5CCCCC5)cc4C1=O	CID:54615952	phase I
BRD-K90734182	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54615956	phase I
BRD-K76758536	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54615958	phase I
BRD-K37226311	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C1=O	CID:54615967	phase I
BRD-K93219845	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccncc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54615969	phase I
BRD-K80598371	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54615984	phase I
BRD-K70337365	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:54616023	phase I
BRD-K42400758	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:54616024	phase I
BRD-K75949681	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:54616027	phase I
BRD-K79407655	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@@H](C)Oc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2C1=O	CID:54616049	phase I
BRD-K91735860	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)C4CCCCC4)cc3C1=O	CID:54616054	phase I
BRD-K98196975	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:54616112	phase I
BRD-K26391060	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:54616115	phase I
BRD-K64643280	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4cccs4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54616134	phase I
BRD-K01093405	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54616180	phase I
BRD-K93340102	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)c4ccccc4)cc3C1=O	CID:54616268	phase I
BRD-K64693729	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54616296	phase I
BRD-K91250867	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54616297	phase I
BRD-K78484446	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCCCC[C@H](C)Oc4ccc(NS(=O)(=O)c5c(C)noc5C)cc4C1=O	CID:54616384	phase I
BRD-K85305147	COc1ccc(NC(=O)Nc2ccc3O[C@@H](C)CCCCO[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54616417	phase I
BRD-K20382089	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:54616535	phase I
BRD-K41328253	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54616675	phase I
BRD-K14781269	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:54616742	phase I
BRD-K97466946	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C1=O	CID:54616967	phase I
BRD-K83007718	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:54616971	phase I
BRD-K66261897	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCC(F)(F)F)cc3C1=O	CID:54616981	phase I
BRD-K07577534	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54616988	phase I
BRD-K51522005	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54617019	phase I
BRD-K06432527	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54617020	phase I
BRD-K54756845	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54617021	phase I
BRD-K97863769	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54617022	phase I
BRD-K61612515	COc1ccc(CN(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54617031	phase I
BRD-K10879245	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54617032	phase I
BRD-K90619727	COc1ccc(CN(C)C[C@H]2OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54617035	phase I
BRD-K95195947	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCCN(C)C)OCCCC[C@H](C)Oc2ccc(NC(=O)Nc3ccc(F)cc3)cc2C1=O	CID:54617058	phase I
BRD-K98427832	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54617209	phase I
BRD-K21110399	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)CCCN(C)C)cc3C1=O	CID:54617262	phase I
BRD-K48454318	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54617267	phase I
BRD-K29143341	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4cccc5ccccc45)cc3C1=O	CID:54617365	phase I
BRD-K02677403	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C1=O	CID:54617432	phase I
BRD-K35210537	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccccc4)cc3C1=O	CID:54617719	phase I
BRD-K72539944	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Cc4ccccc4)cc3C1=O	CID:54617742	phase I
BRD-K41390249	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc5OCOc5c4)cc3C1=O	CID:54617759	phase I
BRD-K35247118	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:54617777	phase I
BRD-K52955163	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:54617778	phase I
BRD-K01763173	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:54617779	phase I
BRD-K37765157	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C1=O	CID:54617781	phase I
BRD-K32974773	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C1=O	CID:54617783	phase I
BRD-K36192494	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Cl)c(Cl)c2)OCCCC[C@@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C1=O	CID:54617784	phase I
BRD-K70489510	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C1=O	CID:54617932	phase I
BRD-K61102114	COc1ccc(NC(=O)N(C)C[C@H]2OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54618067	phase I
BRD-K83457129	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)OCCCC[C@H](C)Oc3ccc(NS(=O)(=O)c4ccccc4)cc3C1=O	CID:54618085	phase I
BRD-K88934376	CCCNC(=O)N(C)C[C@@H]1Oc2ncc(Br)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618098	phase I
BRD-K12913157	C/C=C/c1cnc2O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618099	phase I
BRD-K96839003	COc1ccc(cc1)c2cnc3O[C@H](CN(C)C(=O)C4CCCCC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618100	phase I
BRD-K94303022	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618101	phase I
BRD-K55434198	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618102	phase I
BRD-K39332692	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618103	phase I
BRD-K51234905	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618104	phase I
BRD-K14396276	COCC#Cc1cnc2O[C@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618105	phase I
BRD-K69503483	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618106	phase I
BRD-K60656884	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618107	phase I
BRD-K28077119	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618108	phase I
BRD-K26245595	COCC#Cc1cnc2O[C@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618109	phase I
BRD-K20806007	COc1ccccc1C#Cc2ccc3c(O[C@H](CN(C)Cc4cccnc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618110	phase I
BRD-K48816779	C/C=C/c1cnc2O[C@@H](CN(C)Cc3cccc(c3)C(=O)O)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618111	phase I
BRD-K25290948	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618112	phase I
BRD-K18854347	CCCC#Cc1cnc2O[C@@H](CN(C)C(=O)CCN3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618113	phase I
BRD-K26421164	COc1cccc(c1)c2ccc3c(O[C@H](CN(C)C(=O)C4CCOCC4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618114	phase I
BRD-K08288431	COc1ccc(cc1)c2cnc3O[C@H](CN(C)C(=O)C4CCCCC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618115	phase I
BRD-K09779552	COc1ccccc1c2ccc3c(O[C@@H](CN(C)C(=O)c4cccnc4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618116	phase I
BRD-K63345683	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618117	phase I
BRD-K43634429	C/C=C/c1ccc2c(O[C@H](CN(C)S(=O)(=O)c3ccc(F)cc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618120	phase I
BRD-K35810638	CC(C)CC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3cnccn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618121	phase I
BRD-K07464613	CCCNC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3cncnc3	CID:54618122	phase I
BRD-K47123716	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618123	phase I
BRD-K56051237	COCC#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618124	phase I
BRD-K78978845	CCCC#Cc1cnc2O[C@H](CN(C)C(=O)CCN3CCCCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618125	phase I
BRD-K20875709	CC(C)CC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3cnccn3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618126	phase I
BRD-K06042430	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618127	phase I
BRD-K28397270	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618128	phase I
BRD-K15502712	C/C=C/c1cnc2O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618129	phase I
BRD-K22325899	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618130	phase I
BRD-K73871495	CCCC#Cc1cnc2O[C@@H](CN(C)C(=O)CCN3CCCCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618131	phase I
BRD-K10301293	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618132	phase I
BRD-K35689168	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618133	phase I
BRD-K68690449	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618134	phase I
BRD-K87990527	C/C=C/c1cnc2O[C@@H](CN(C)Cc3cccc(c3)C(=O)O)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618135	phase I
BRD-K38996795	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618136	phase I
BRD-K20347745	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618137	phase I
BRD-K68546494	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618138	phase I
BRD-K41350512	COc1ccccc1c2ccc3c(O[C@@H](CN(C)C(=O)c4cccnc4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618139	phase I
BRD-K92967681	COc1ccccc1C#Cc2ccc3c(O[C@@H](CN(C)Cc4cccnc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618140	phase I
BRD-K36156445	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618141	phase I
BRD-K41743657	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618142	phase I
BRD-K61861910	COCC#Cc1cnc2O[C@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618143	phase I
BRD-K66573697	CCCC#Cc1ccc2c(O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618144	phase I
BRD-K40109091	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618145	phase I
BRD-K27841704	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618146	phase I
BRD-K21152785	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618147	phase I
BRD-K76892938	CC(C)CC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3cnccn3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618148	phase I
BRD-K29799191	C/C=C/c1cnc2O[C@H](CN(C)Cc3cccc(c3)C(=O)O)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618149	phase I
BRD-K04278887	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618150	phase I
BRD-K95488294	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618151	phase I
BRD-K93494062	COc1cccc(c1)c2ccc3c(O[C@@H](CN(C)C(=O)C4CCOCC4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618152	phase I
BRD-K30477337	COc1cccc(c1)c2ccc3c(O[C@H](CN(C)C(=O)C4CCOCC4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618153	phase I
BRD-K63948704	C/C=C/c1ccc2c(O[C@H](CN(C)S(=O)(=O)c3ccc(F)cc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618154	phase I
BRD-K54935014	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618155	phase I
BRD-K83082136	COc1ccccc1c2ccc3c(O[C@@H](CN(C)C(=O)c4cccnc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618156	phase I
BRD-K78218619	COCC#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618157	phase I
BRD-K65196043	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618158	phase I
BRD-K78961368	CCCC#Cc1ccc2c(O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618159	phase I
BRD-K76960042	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618160	phase I
BRD-K18724553	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618161	phase I
BRD-K23713813	C/C=C/c1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccc(F)cc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618162	phase I
BRD-K17339982	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618163	phase I
BRD-K13999467	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618164	phase I
BRD-K96198015	CC(C)CC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3cnccn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618165	phase I
BRD-K92655621	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618166	phase I
BRD-K93368389	C/C=C/c1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccc(F)cc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618167	phase I
BRD-K98611274	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618168	phase I
BRD-K34576879	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618169	phase I
BRD-K51502980	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618170	phase I
BRD-K77069371	C/C=C/c1cnc2O[C@H](CN(C)Cc3cccc(c3)C(=O)O)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618171	phase I
BRD-K67407970	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618172	phase I
BRD-K59524902	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618173	phase I
BRD-K92889073	CCCNC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3cncnc3	CID:54618174	phase I
BRD-K06486491	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54618175	phase I
BRD-K25344230	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:54618176	phase I
BRD-K84271926	CCCNC(=O)N(C)C[C@H]1Oc2ncc(Br)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618177	phase I
BRD-K84260700	CCCNC(=O)N(C)C[C@H]1Oc2ncc(Br)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618178	phase I
BRD-K47203692	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618179	phase I
BRD-K44387261	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618180	phase I
BRD-K44422244	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618181	phase I
BRD-K51202492	COCC#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618182	phase I
BRD-K72913973	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618183	phase I
BRD-K61412007	CCCC#Cc1ccc2c(O[C@@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618184	phase I
BRD-K89137409	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618185	phase I
BRD-K66803141	COc1ccccc1c2ccc3c(O[C@H](CN(C)C(=O)c4cccnc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618186	phase I
BRD-K36276950	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618187	phase I
BRD-K67240417	COc1cccc(c1)c2ccc3c(O[C@@H](CN(C)C(=O)C4CCOCC4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618188	phase I
BRD-K35615823	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:54618189	phase I
BRD-K71216533	COc1cccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:54618190	phase I
BRD-K70055050	COCC#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618191	phase I
BRD-K67727634	C/C=C/c1cnc2O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618192	phase I
BRD-K09206831	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618193	phase I
BRD-K47031124	CCCC#Cc1cnc2O[C@H](CN(C)C(=O)CCN3CCCCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618194	phase I
BRD-K15684061	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618195	phase I
BRD-K40814141	COc1ccc(cc1)c2cnc3O[C@@H](CN(C)C(=O)C4CCCCC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618196	phase I
BRD-K69054398	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618197	phase I
BRD-K73643601	C/C=C/c1cnc2O[C@H](CN(C)Cc3cccc(c3)C(=O)O)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618198	phase I
BRD-K41970046	COc1ccc(cc1)c2cnc3O[C@@H](CN(C)C(=O)C4CCCCC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618199	phase I
BRD-K79145797	C/C=C/c1cnc2O[C@H](CN(C)Cc3cccc(c3)C(=O)O)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618200	phase I
BRD-K14990409	C/C=C/c1cnc2O[C@@H](CN(C)Cc3cccc(c3)C(=O)O)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618201	phase I
BRD-K62599086	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618202	phase I
BRD-K60820896	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618203	phase I
BRD-K22098045	COc1ccccc1S(=O)(=O)N(C)C[C@H]2Oc3ncc(Br)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54618204	phase I
BRD-K60527064	COc1ccccc1C#Cc2ccc3c(O[C@@H](CN(C)Cc4cccnc4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618205	phase I
BRD-K65461993	CNC[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccc(C#N)cc3	CID:54618206	phase I
BRD-K34787855	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618207	phase I
BRD-K66110520	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54618208	phase I
BRD-K29350630	CCCNC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3cncnc3	CID:54618209	phase I
BRD-K82957261	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618210	phase I
BRD-K86872145	COc1ccccc1C#Cc2ccc3c(O[C@@H](CN(C)Cc4cccnc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618211	phase I
BRD-K77423370	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54618212	phase I
BRD-K50965411	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618213	phase I
BRD-K74145465	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54618214	phase I
BRD-K73282213	COCC#Cc1cnc2O[C@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618215	phase I
BRD-K69827766	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618216	phase I
BRD-K08942755	C/C=C/c1cnc2O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618217	phase I
BRD-K83712984	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618218	phase I
BRD-K59539129	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618219	phase I
BRD-K10287595	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618220	phase I
BRD-K63757709	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618221	phase I
BRD-K01573538	COc1ccccc1c2cnc3O[C@H](CN(C)CC4CCOCC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618222	phase I
BRD-K01463627	COc1ccccc1C#Cc2ccc3c(O[C@H](CN(C)Cc4cccnc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618223	phase I
BRD-K11930946	CCCNC(=O)N(C)C[C@@H]1Oc2ncc(Br)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618224	phase I
BRD-K29438074	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:54618225	phase I
BRD-K75460409	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618226	phase I
BRD-K16136812	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618227	phase I
BRD-K27709404	COc1ccccc1c2cnc3O[C@@H](CN(C)CC4CCOCC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618228	phase I
BRD-K37722208	CCCC#Cc1ccc2c(O[C@@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618229	phase I
BRD-K76973159	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618230	phase I
BRD-K92208021	COCC#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618231	phase I
BRD-K64930281	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618232	phase I
BRD-K78223464	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618233	phase I
BRD-K48918933	CC(C)CC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3cnccn3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618234	phase I
BRD-K57461880	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618235	phase I
BRD-K99171789	COCC#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618236	phase I
BRD-K05570331	C/C=C/c1cnc2O[C@@H](CN(C)Cc3cccc(c3)C(=O)O)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618237	phase I
BRD-K53798768	COCC#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618238	phase I
BRD-K45787391	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54618239	phase I
BRD-K25476619	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618240	phase I
BRD-K14602451	COc1ccccc1c2ccc3c(O[C@H](CN(C)C(=O)c4cccnc4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618241	phase I
BRD-K06900263	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618242	phase I
BRD-K33768761	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618243	phase I
BRD-K54595160	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618244	phase I
BRD-K47272214	COCC#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618245	phase I
BRD-K20582542	CCCC#Cc1ccc2c(O[C@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618246	phase I
BRD-K29908513	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618247	phase I
BRD-K75636715	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618248	phase I
BRD-K37813153	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618249	phase I
BRD-K37403152	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618250	phase I
BRD-K94465870	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618251	phase I
BRD-K56592974	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618252	phase I
BRD-K80442083	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618253	phase I
BRD-K05653239	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618254	phase I
BRD-K60741970	COCC#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618255	phase I
BRD-K57758244	COc1cccc(c1)c2ccc3c(O[C@@H](CN(C)C(=O)C4CCOCC4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618256	phase I
BRD-K53350977	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618257	phase I
BRD-K66149578	CCCNC(=O)N(C)C[C@@H]1Oc2ncc(Br)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618258	phase I
BRD-K19724753	C/C=C/c1cnc2O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618259	phase I
BRD-K53477720	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54618260	phase I
BRD-K52062350	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618261	phase I
BRD-K79932545	CCCNC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3cncnc3	CID:54618262	phase I
BRD-K41790019	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618263	phase I
BRD-K93011670	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618264	phase I
BRD-K13653700	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618265	phase I
BRD-K62047982	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618266	phase I
BRD-K80000073	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618267	phase I
BRD-K64233461	CC(C)C#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618268	phase I
BRD-K54278059	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618269	phase I
BRD-K39068840	COc1ccccc1c2ccc3c(O[C@@H](CN(C)C(=O)c4cccnc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618270	phase I
BRD-K24975719	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618271	phase I
BRD-K01556781	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618272	phase I
BRD-K23992348	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618273	phase I
BRD-K17618128	CCCC#Cc1ccc2c(O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618274	phase I
BRD-K63870957	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618275	phase I
BRD-K45613561	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618276	phase I
BRD-K85158753	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618277	phase I
BRD-K99514625	CC(C)CC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3cnccn3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618278	phase I
BRD-K86816409	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618279	phase I
BRD-K09076022	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618280	phase I
BRD-K17965071	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618281	phase I
BRD-K27728416	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618282	phase I
BRD-K08110534	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618283	phase I
BRD-K08828851	C/C=C/c1cnc2O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618284	phase I
BRD-K77221985	COc1ccccc1c2cnc3O[C@@H](CN(C)CC4CCOCC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618285	phase I
BRD-K22485649	COc1ccc(cc1)c2cnc3O[C@@H](CN(C)C(=O)C4CCCCC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618286	phase I
BRD-K17583574	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618287	phase I
BRD-K12163240	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618288	phase I
BRD-K98216700	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618289	phase I
BRD-K30573524	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618290	phase I
BRD-K19414061	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618291	phase I
BRD-K12092185	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618292	phase I
BRD-K34666250	COc1ccccc1C#Cc2ccc3c(O[C@H](CN(C)Cc4cccnc4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618293	phase I
BRD-K38263412	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54618294	phase I
BRD-K35174435	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618295	phase I
BRD-K72318460	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618296	phase I
BRD-K19122760	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54618297	phase I
BRD-K34937870	CCCNC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3cncnc3	CID:54618298	phase I
BRD-K06806702	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618299	phase I
BRD-K77703574	COc1cccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54618300	phase I
BRD-K87260976	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618301	phase I
BRD-K07481069	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618302	phase I
BRD-K79861274	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618303	phase I
BRD-K57230817	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618304	phase I
BRD-K14844214	CC(C)CC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3cnccn3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618305	phase I
BRD-K19472114	CC(C)C#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618306	phase I
BRD-K56634255	COc1ccccc1C#Cc2ccc3c(O[C@H](CN(C)Cc4cccnc4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618307	phase I
BRD-K13365737	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618308	phase I
BRD-K60997369	CC(C)CC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3cnccn3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618309	phase I
BRD-K68246656	COc1ccccc1c2ccc3c(O[C@H](CN(C)C(=O)c4cccnc4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618310	phase I
BRD-K39562569	COc1ccccc1c2ccc3c(O[C@H](CN(C)C(=O)c4cccnc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618311	phase I
BRD-K63484613	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3ncccc3C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54618312	phase I
BRD-K97709323	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618313	phase I
BRD-K40052948	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618314	phase I
BRD-K12230293	COc1ccccc1c2cnc3O[C@H](CN(C)CC4CCOCC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618315	phase I
BRD-K57169040	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618316	phase I
BRD-K78120854	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618317	phase I
BRD-K98833727	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618318	phase I
BRD-K27656392	CCCNC(=O)N(C)C[C@H]1Oc2ncc(Br)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618319	phase I
BRD-K55681368	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618320	phase I
BRD-K05130619	COc1ccc(cc1)c2cnc3O[C@H](CN(C)C(=O)C4CCCCC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618321	phase I
BRD-K12633506	CC(C)NC(=O)N(C)C[C@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618322	phase I
BRD-K26652457	COc1cccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:54618323	phase I
BRD-K64217340	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618324	phase I
BRD-K99432717	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618325	phase I
BRD-K55300135	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618326	phase I
BRD-K80747759	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618327	phase I
BRD-K47716199	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618328	phase I
BRD-K25056189	CCCC#Cc1ccc2c(O[C@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618329	phase I
BRD-K43782664	COc1ccccc1C#Cc2ccc3c(O[C@@H](CN(C)Cc4cccnc4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618330	phase I
BRD-K99805333	CC(C)C#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618331	phase I
BRD-K67771738	CCCNC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3cncnc3	CID:54618332	phase I
BRD-K49309964	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618333	phase I
BRD-K67862892	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618334	phase I
BRD-K71004332	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618335	phase I
BRD-K38665228	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618336	phase I
BRD-K62881454	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618337	phase I
BRD-K53121826	CC(C)C#Cc1ccc2c(O[C@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618338	phase I
BRD-K57756744	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618339	phase I
BRD-K77264230	CCCC#Cc1ccc2c(O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618340	phase I
BRD-K29974036	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618341	phase I
BRD-K03958946	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618342	phase I
BRD-K33348232	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618343	phase I
BRD-K78380744	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618344	phase I
BRD-K47991733	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618345	phase I
BRD-K26957826	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618346	phase I
BRD-K87721831	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618347	phase I
BRD-K92627732	COc1ccc(cc1)c2cnc3O[C@H](CN(C)C(=O)C4CCCCC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618348	phase I
BRD-K55415928	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4cncnc4	CID:54618349	phase I
BRD-K35712980	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54618350	phase I
BRD-K05686172	COc1cccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:54618351	phase I
BRD-K12589632	COCC#Cc1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccc(OC)cc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618352	phase I
BRD-K59155687	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618353	phase I
BRD-K22065094	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618354	phase I
BRD-K90827020	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618355	phase I
BRD-K94789179	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618356	phase I
BRD-K97217923	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)C5=CCCCC5	CID:54618357	phase I
BRD-K65313110	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54618358	phase I
BRD-K27224038	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618359	phase I
BRD-K03591925	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618360	phase I
BRD-K23801936	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618361	phase I
BRD-K45699165	COc1cccc(c1)c2ccc3c(O[C@H](CN(C)C(=O)C4CCOCC4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618362	phase I
BRD-K78118043	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618363	phase I
BRD-K58079191	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618364	phase I
BRD-K25533536	COc1ccccc1c2cnc3O[C@@H](CN(C)CC4CCOCC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618365	phase I
BRD-K45628229	COc1ccccc1c2cnc3O[C@H](CN(C)CC4CCOCC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618366	phase I
BRD-K48775846	COc1ccccc1c2cnc3O[C@@H](CN(C)CC4CCOCC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618367	phase I
BRD-K69096174	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618368	phase I
BRD-K21000135	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618369	phase I
BRD-K01651394	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618370	phase I
BRD-K32648402	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618371	phase I
BRD-K14161261	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54618372	phase I
BRD-K57017252	CCCC#Cc1cnc2O[C@H](CN(C)C(=O)CCN3CCCCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618373	phase I
BRD-K52660225	CC(C)NC(=O)N(C)C[C@@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618374	phase I
BRD-K46622484	COc1ccccc1c2cnc3O[C@H](CN(C)CC4CCOCC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618375	phase I
BRD-K50108835	CCCNC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3cncnc3	CID:54618376	phase I
BRD-K00463020	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618377	phase I
BRD-K87126403	CCCNC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3cncnc3	CID:54618378	phase I
BRD-K92841908	COCC#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618379	phase I
BRD-K42241928	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54618380	phase I
BRD-K19554975	C/C=C/c1cnc2O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618381	phase I
BRD-K33960497	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3cc(C#CC(C)(C)O)ccc3S1(=O)=O	CID:54618382	phase I
BRD-K09749233	COCC#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3cc(F)ccc3F)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618383	phase I
BRD-K24638771	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618384	phase I
BRD-K04798077	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2cccnc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54618385	phase I
BRD-K78232231	COc1cccc(c1)c2ccc3c(O[C@H](CN(C)C(=O)C4CCOCC4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618386	phase I
BRD-K55522699	C/C=C/c1cnc2O[C@@H](CN(C)S(=O)(=O)c3cn(C)cn3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618387	phase I
BRD-K66599765	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CC4(O)CCCC4)ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54618388	phase I
BRD-K89995901	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54618389	phase I
BRD-K60865324	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618390	phase I
BRD-K54261877	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:54618393	phase I
BRD-K91491104	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618394	phase I
BRD-K44245916	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618395	phase I
BRD-K86762131	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618396	phase I
BRD-K33518436	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618397	phase I
BRD-K52797126	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618398	phase I
BRD-K02756145	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ncc(C#CCc4ccccc4)cc3C1=O	CID:54618399	phase I
BRD-K33593585	C/C=C/c1cnc2O[C@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618400	phase I
BRD-K30357474	CC(C)NC(=O)N(C)C[C@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618401	phase I
BRD-K58775116	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618402	phase I
BRD-K20877213	COc1cccc(NC(=O)N(C)C[C@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54618403	phase I
BRD-K40321450	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618404	phase I
BRD-K90912017	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618405	phase I
BRD-K01162658	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54618406	phase I
BRD-K42357106	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618407	phase I
BRD-K00241248	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ncc(C#CCc4ccccc4)cc3C1=O	CID:54618408	phase I
BRD-K27824357	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618409	phase I
BRD-K02072940	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ncc(C#CCc4ccccc4)cc3C1=O	CID:54618410	phase I
BRD-K41235383	CC(C)CC#Cc1cnc2O[C@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618411	phase I
BRD-K64979177	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618412	phase I
BRD-K88306141	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618415	phase I
BRD-K05111274	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618416	phase I
BRD-K72766058	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618417	phase I
BRD-K90146121	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618418	phase I
BRD-K91898214	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618419	phase I
BRD-K27428408	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618420	phase I
BRD-K54381125	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618421	phase I
BRD-K88597074	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618422	phase I
BRD-K73360774	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618423	phase I
BRD-K35152204	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618424	phase I
BRD-K77304272	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)C4=CCCCC4	CID:54618425	phase I
BRD-K87062384	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618426	phase I
BRD-K62442112	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618427	phase I
BRD-K78764313	CC(C)NC(=O)N(C)C[C@@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618428	phase I
BRD-K83241810	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618429	phase I
BRD-K39245533	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3	CID:54618430	phase I
BRD-K39227212	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618431	phase I
BRD-K97492549	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618432	phase I
BRD-K40837535	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618433	phase I
BRD-K03995514	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618434	phase I
BRD-K93549834	CCCC#Cc1ccc2c(O[C@H](CN(C)C(=O)Nc3ccccc3F)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618435	phase I
BRD-K51390937	COCC(=O)N(C)C[C@@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618436	phase I
BRD-K86420846	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618437	phase I
BRD-K60056908	COCC(=O)N(C)C[C@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618438	phase I
BRD-K59475561	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618439	phase I
BRD-K35854261	CC(C)NC(=O)N(C)C[C@@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618440	phase I
BRD-K18493795	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)C4=CCCCC4	CID:54618441	phase I
BRD-K37090607	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618442	phase I
BRD-K61965677	CCCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)Nc3ccccc3F)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618443	phase I
BRD-K26309991	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:54618444	phase I
BRD-K20119687	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618445	phase I
BRD-K62780697	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618446	phase I
BRD-K29824954	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(C#CCC4CCCC4)ccc3S1(=O)=O	CID:54618447	phase I
BRD-K07581216	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618448	phase I
BRD-K79275879	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618449	phase I
BRD-K41340267	CCCN(C)C[C@@H]1Oc2cc(C#Cc3cccc(OC)c3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618450	phase I
BRD-K80649837	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618451	phase I
BRD-K84447176	CCCN(C)C[C@@H]1Oc2cc(C#Cc3cccc(OC)c3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618452	phase I
BRD-K29890753	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618453	phase I
BRD-K53601225	COCC(=O)N(C)C[C@@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618454	phase I
BRD-K92191596	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618455	phase I
BRD-K51512723	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618456	phase I
BRD-K28394201	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618457	phase I
BRD-K32796290	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618458	phase I
BRD-K87811893	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618459	phase I
BRD-K43714340	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618460	phase I
BRD-K68311329	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618461	phase I
BRD-K30234379	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618462	phase I
BRD-K23506413	COCC(=O)N(C)C[C@@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618463	phase I
BRD-K62051893	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618464	phase I
BRD-K14327282	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618465	phase I
BRD-K51803154	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618466	phase I
BRD-K26449125	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618467	phase I
BRD-K87217296	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ncc(C#CCc4ccccc4)cc3C1=O	CID:54618468	phase I
BRD-K60963631	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618469	phase I
BRD-K98803880	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618470	phase I
BRD-K74962003	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618471	phase I
BRD-K27451531	CC(C)NC(=O)N(C)C[C@@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618472	phase I
BRD-K33148516	CCCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)Nc3ccccc3F)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618473	phase I
BRD-K48733306	COCC(=O)N(C)C[C@@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618474	phase I
BRD-K86524553	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618475	phase I
BRD-K06884108	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Cc3cccnc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618476	phase I
BRD-K19147816	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618477	phase I
BRD-K45941745	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618478	phase I
BRD-K49723079	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618479	phase I
BRD-K33603918	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54618480	phase I
BRD-K47788371	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618481	phase I
BRD-K65409714	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618482	phase I
BRD-K52032805	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3cccc(F)c3	CID:54618483	phase I
BRD-K20019319	COCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccccc3F	CID:54618484	phase I
BRD-K84909597	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618485	phase I
BRD-K67321912	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618486	phase I
BRD-K69697800	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618487	phase I
BRD-K47499097	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618488	phase I
BRD-K77987559	CCCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)Nc3ccccc3F)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618489	phase I
BRD-K22576413	C/C=C/c1cnc2O[C@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618490	phase I
BRD-K31786211	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618491	phase I
BRD-K61070477	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618492	phase I
BRD-K30857143	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618493	phase I
BRD-K40630529	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618494	phase I
BRD-K77924862	COc1ccc(C#Cc2ccc3c(O[C@H](CN(C)C(=O)CN4CCOCC4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2)cc1	CID:54618495	phase I
BRD-K37815632	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618496	phase I
BRD-K99192901	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618497	phase I
BRD-K62602051	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)O)Oc3ncc(C#CCc4ccccc4)cc3C1=O	CID:54618498	phase I
BRD-K60339813	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)C4=CCCCC4	CID:54618499	phase I
BRD-K66204187	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618500	phase I
BRD-K92639644	COc1ccc(C#Cc2ccc3c(O[C@H](CN(C)C(=O)CN4CCOCC4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2)cc1	CID:54618501	phase I
BRD-K55282910	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)c3ccccc3	CID:54618502	phase I
BRD-K23304679	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618503	phase I
BRD-K69805180	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618504	phase I
BRD-K42509645	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Cc3cccnc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618505	phase I
BRD-K67936348	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618506	phase I
BRD-K54419202	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618507	phase I
BRD-K57690336	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618508	phase I
BRD-K02882069	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Cc3cccnc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618509	phase I
BRD-K19593188	COc1ccc(C#Cc2ccc3c(O[C@@H](CN(C)C(=O)CN4CCOCC4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2)cc1	CID:54618510	phase I
BRD-K00278564	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618511	phase I
BRD-K53985154	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618512	phase I
BRD-K33238309	CC(C)CC#Cc1cnc2O[C@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618513	phase I
BRD-K87087278	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618514	phase I
BRD-K46718584	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618515	phase I
BRD-K32051704	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618516	phase I
BRD-K22673215	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618517	phase I
BRD-K93545352	COc1ccc(C#Cc2ccc3c(O[C@@H](CN(C)C(=O)CN4CCOCC4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2)cc1	CID:54618518	phase I
BRD-K40959498	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618519	phase I
BRD-K57082361	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618520	phase I
BRD-K76547245	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618521	phase I
BRD-K90445273	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618522	phase I
BRD-K43017765	CC(C)CC#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccc(F)c3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618523	phase I
BRD-K05041276	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618524	phase I
BRD-K11054980	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618525	phase I
BRD-K67209190	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618526	phase I
BRD-K01023753	COCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3F	CID:54618527	phase I
BRD-K99691991	COCC(=O)N(C)C[C@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618528	phase I
BRD-K10182851	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618529	phase I
BRD-K71839385	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618530	phase I
BRD-K81080300	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618531	phase I
BRD-K25125608	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618532	phase I
BRD-K72623425	COCC(=O)N(C)C[C@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618533	phase I
BRD-K25441114	COCC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccccc3F	CID:54618534	phase I
BRD-K12091863	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618535	phase I
BRD-K46663433	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618536	phase I
BRD-K41974651	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618537	phase I
BRD-K44407752	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)c3ccccc3	CID:54618538	phase I
BRD-K72980834	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618539	phase I
BRD-K38051696	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618540	phase I
BRD-K64217932	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618541	phase I
BRD-K22385434	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccccc3	CID:54618542	phase I
BRD-K54789622	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618543	phase I
BRD-K31439714	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Cc3cccnc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618544	phase I
BRD-K20103689	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618545	phase I
BRD-K21987633	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618546	phase I
BRD-K57133453	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618547	phase I
BRD-K22801678	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54618548	phase I
BRD-K61208213	CC(C)NC(=O)N(C)C[C@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618549	phase I
BRD-K82367827	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54618550	phase I
BRD-K04618303	COc1cccc(NC(=O)N(C)C[C@@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:54618551	phase I
BRD-K20806847	CC(C)CC#Cc1cnc2O[C@H](CN(C)C(=O)c3cccc(F)c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618552	phase I
BRD-K10385416	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618553	phase I
BRD-K31955163	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618554	phase I
BRD-K32271530	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618555	phase I
BRD-K72515004	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)C4=CCCCC4	CID:54618556	phase I
BRD-K24161447	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618557	phase I
BRD-K77644960	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618558	phase I
BRD-K30723822	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618559	phase I
BRD-K12815005	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618560	phase I
BRD-K22945779	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618561	phase I
BRD-K69672299	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#Cc4ccccc4F)cc3C1=O	CID:54618562	phase I
BRD-K68876477	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618563	phase I
BRD-K02655584	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618564	phase I
BRD-K79064458	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618565	phase I
BRD-K53978628	CCCC#Cc1ccc2c(O[C@H](CN(C)C(=O)Nc3ccccc3F)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618566	phase I
BRD-K09244864	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5cncnc5	CID:54618567	phase I
BRD-K37168393	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618568	phase I
BRD-K04007716	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618569	phase I
BRD-K91573667	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)C4=CCCCC4	CID:54618570	phase I
BRD-K78908189	COc1ccc(C#Cc2ccc3c(O[C@@H](CN(C)C(=O)CN4CCOCC4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2)cc1	CID:54618571	phase I
BRD-K31036503	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618572	phase I
BRD-K38589316	COc1ccc(C#Cc2ccc3c(O[C@@H](CN(C)C(=O)CN4CCOCC4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2)cc1	CID:54618573	phase I
BRD-K13719685	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618574	phase I
BRD-K11792293	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618575	phase I
BRD-K30079954	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618576	phase I
BRD-K42279779	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618577	phase I
BRD-K53255530	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618578	phase I
BRD-K11400546	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618579	phase I
BRD-K97615779	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Cc3cccnc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618580	phase I
BRD-K53756103	CC(C)NC(=O)N(C)C[C@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618581	phase I
BRD-K35234011	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618582	phase I
BRD-K57579659	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618583	phase I
BRD-K92372623	COCC(=O)N(C)C[C@@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618584	phase I
BRD-K50639228	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618585	phase I
BRD-K55343182	C[C@@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618586	phase I
BRD-K50801330	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618587	phase I
BRD-K11976754	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618588	phase I
BRD-K53700261	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54618589	phase I
BRD-K84113859	C[C@H](O)C#Cc1cnc2O[C@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618590	phase I
BRD-K77422873	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618591	phase I
BRD-K89801405	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618592	phase I
BRD-K64552378	CC(C)NC(=O)N(C)C[C@@H]1Oc2ncc(C#CC3CC3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618593	phase I
BRD-K14203250	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618594	phase I
BRD-K07208716	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618595	phase I
BRD-K44446302	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54618596	phase I
BRD-K93165404	C/C=C/c1cnc2O[C@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618597	phase I
BRD-K62462045	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4C	CID:54618598	phase I
BRD-K40567080	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618599	phase I
BRD-K46658587	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618600	phase I
BRD-K29255825	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618601	phase I
BRD-K25583560	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618602	phase I
BRD-K69516264	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618603	phase I
BRD-K01619611	CCCC#Cc1ccc2c(O[C@H](CN(C)C(=O)Nc3ccccc3F)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618604	phase I
BRD-K12834930	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618605	phase I
BRD-K45258986	CCCN(C)C[C@H]1Oc2cc(C#Cc3cccc(OC)c3)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618606	phase I
BRD-K27539003	C[C@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618607	phase I
BRD-K94882528	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)C4=CCCCC4	CID:54618608	phase I
BRD-K29290722	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618609	phase I
BRD-K62114978	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618610	phase I
BRD-K30516885	CC(C)CC#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618611	phase I
BRD-K16210823	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618612	phase I
BRD-K36394966	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618613	phase I
BRD-K01355066	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54618614	phase I
BRD-K52654243	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618615	phase I
BRD-K49345388	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618616	phase I
BRD-K86752593	COCC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3F	CID:54618617	phase I
BRD-K68233995	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCC5	CID:54618618	phase I
BRD-K88606952	COCC(=O)N(C)C[C@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618619	phase I
BRD-K80694691	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3	CID:54618620	phase I
BRD-K36702054	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618621	phase I
BRD-K77282409	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618622	phase I
BRD-K78976513	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618623	phase I
BRD-K38774907	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(/C=C/c4ccccc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54618624	phase I
BRD-K37231045	COc1ccc(C#Cc2ccc3c(O[C@H](CN(C)C(=O)CN4CCOCC4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2)cc1	CID:54618625	phase I
BRD-K20009726	COCC(=O)N(C)C[C@@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618626	phase I
BRD-K79367755	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618627	phase I
BRD-K06295532	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618628	phase I
BRD-K26759399	CCCC#Cc1ccc2c(O[C@H](CN(C)C(=O)Nc3ccccc3F)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618629	phase I
BRD-K58404149	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Cc3cccnc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618630	phase I
BRD-K20093888	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618631	phase I
BRD-K81121951	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618632	phase I
BRD-K29060081	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Cc3cccnc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618633	phase I
BRD-K42899395	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618634	phase I
BRD-K64558129	COCC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3ccccc3F	CID:54618635	phase I
BRD-K12108140	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618636	phase I
BRD-K78380066	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2C(=O)O)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54618637	phase I
BRD-K43436404	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618638	phase I
BRD-K36801622	COCC(=O)N(C)C[C@H]1Oc2cc(C#Cc3cccnc3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618639	phase I
BRD-K92748025	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618640	phase I
BRD-K56945633	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618641	phase I
BRD-K69194443	COc1ccc(C#Cc2ccc3c(O[C@H](CN(C)C(=O)CN4CCOCC4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2)cc1	CID:54618642	phase I
BRD-K27918075	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)Oc2ncc(cc2C1=O)c3ccc(C)cc3	CID:54618643	phase I
BRD-K59551872	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618644	phase I
BRD-K11548496	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618645	phase I
BRD-K34055449	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618646	phase I
BRD-K00083176	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618647	phase I
BRD-K46450665	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Cc3cccnc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618648	phase I
BRD-K49125116	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618649	phase I
BRD-K01847595	COCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3F	CID:54618650	phase I
BRD-K63539924	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618651	phase I
BRD-K31096204	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618652	phase I
BRD-K26214776	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3	CID:54618653	phase I
BRD-K12942263	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)c4cccc(c4)C(=O)N(C)C)cc1	CID:54618654	phase I
BRD-K37058154	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618655	phase I
BRD-K36333904	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54618656	phase I
BRD-K43966462	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)C4=CCCCC4	CID:54618657	phase I
BRD-K71819159	COCC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3F	CID:54618658	phase I
BRD-K01604266	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3cccc(F)c3	CID:54618659	phase I
BRD-K60245465	CCCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)Nc3ccccc3F)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618660	phase I
BRD-K51791261	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618661	phase I
BRD-K48228567	CC(C)CC#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618662	phase I
BRD-K15619703	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618663	phase I
BRD-K81859633	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54618664	phase I
BRD-K48582996	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618665	phase I
BRD-K88786138	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618666	phase I
BRD-K95438730	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4ncc(cc4C1=O)c5cncnc5	CID:54618667	phase I
BRD-K30377659	COc1cccc(NC(=O)N(C)C[C@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:54618668	phase I
BRD-K08844227	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5cncnc5	CID:54618669	phase I
BRD-K27543325	COc1cccc(NC(=O)N(C)C[C@H]2Oc3ncc(C#Cc4ccncc4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:54618670	phase I
BRD-K87791256	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618671	phase I
BRD-K14131832	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)Oc2cc(C#Cc3ccccn3)ccc2S1(=O)=O	CID:54618672	phase I
BRD-K75418563	CCCN(C)C[C@H]1Oc2cc(C#Cc3cccc(OC)c3)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618673	phase I
BRD-K62283710	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3cccc(F)c3	CID:54618674	phase I
BRD-K54560380	C/C=C/c1cnc2O[C@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618675	phase I
BRD-K78657294	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3	CID:54618676	phase I
BRD-K48527688	COc1ccccc1C#Cc2cnc3O[C@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618677	phase I
BRD-K83435763	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)Oc3ncc(cc3C1=O)c4ccc(cc4)C(=O)N(C)C	CID:54618678	phase I
BRD-K59174091	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54618679	phase I
BRD-K28065812	C[C@@H](O)C#Cc1cnc2O[C@@H](CN(C)C(=O)Cc3ccncc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618680	phase I
BRD-K59730983	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618681	phase I
BRD-K53792011	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618682	phase I
BRD-K33575007	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4cc(ccc4S1(=O)=O)c5ccccc5	CID:54618683	phase I
BRD-K97959949	CC(C)CC#Cc1cnc2O[C@H](CN(C)C(=O)c3cccc(F)c3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618684	phase I
BRD-K86023266	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618685	phase I
BRD-K88914803	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CC(C)(C)O)cc3C1=O	CID:54618686	phase I
BRD-K67365258	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)S(=O)(=O)c4cn(C)cn4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54618687	phase I
BRD-K33894111	COCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3ccccc3F	CID:54618688	phase I
BRD-K57009782	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54618689	phase I
BRD-K69349639	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54618690	phase I
BRD-K57537921	COc1ccccc1C#Cc2cnc3O[C@@H](CN(C)C(=O)c4ccc5OCOc5c4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54618691	phase I
BRD-K83631404	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618692	phase I
BRD-K45515828	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618695	phase I
BRD-K28467343	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618696	phase I
BRD-K27807043	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618697	phase I
BRD-K84838433	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618698	phase I
BRD-K80003719	CC(C)C#Cc1cnc2O[C@H](CN(C)Cc3cncnc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618699	phase I
BRD-K13464529	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)C(=O)CC4CC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54618700	phase I
BRD-K14409255	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618701	phase I
BRD-K50696746	CNC[C@H]1Oc2ncc(C#Cc3cccc(OC)c3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618702	phase I
BRD-K97951470	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618703	phase I
BRD-K83344091	COc1ccc(C#Cc2cnc3O[C@H](CN(C)C(=O)CC4CC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54618704	phase I
BRD-K43690686	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54618705	phase I
BRD-K13166308	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618706	phase I
BRD-K98238711	COc1ccccc1NC(=O)N(C)C[C@@H]2Oc3ncc(C#CC(C)C)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54618707	phase I
BRD-K57016057	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)C3=CCCCC3	CID:54618708	phase I
BRD-K03050455	COCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618709	phase I
BRD-K86250672	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618710	phase I
BRD-K12642652	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618711	phase I
BRD-K65997856	CNC[C@@H]1Oc2ncc(/C=C/c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618712	phase I
BRD-K02014458	COc1ccc(C#Cc2cnc3O[C@H](CN(C)C(=O)CC4CC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54618713	phase I
BRD-K69429207	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618714	phase I
BRD-K31559406	CCCNC(=O)N(C)C[C@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618717	phase I
BRD-K80531070	COc1ccccc1c2ccc3c(O[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618718	phase I
BRD-K07489121	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618719	phase I
BRD-K03458571	COc1ccccc1c2ccc3c(O[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618720	phase I
BRD-K60343011	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618721	phase I
BRD-K44194212	COCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccccc3F)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618722	phase I
BRD-K17619044	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618723	phase I
BRD-K03251393	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618724	phase I
BRD-K63406313	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618725	phase I
BRD-K70744040	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618726	phase I
BRD-K70018966	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618727	phase I
BRD-K39841630	C[C@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618728	phase I
BRD-K95400509	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618729	phase I
BRD-K51848823	CC(C)C#Cc1cnc2O[C@H](CN(C)C(=O)c3cccnc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618730	phase I
BRD-K78832647	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618731	phase I
BRD-K23240038	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618732	phase I
BRD-K02559684	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618733	phase I
BRD-K46489288	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618734	phase I
BRD-K57272712	C[C@@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618735	phase I
BRD-K17193648	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618736	phase I
BRD-K55452151	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618737	phase I
BRD-K75393430	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618738	phase I
BRD-K35111787	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618739	phase I
BRD-K22721982	CC(C)C#Cc1cnc2O[C@H](CN(C)Cc3cncnc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618740	phase I
BRD-K97648508	CCCNC(=O)N(C)C[C@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618741	phase I
BRD-K16480639	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618742	phase I
BRD-K77424821	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618743	phase I
BRD-K87286000	COCC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccccc3F)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618744	phase I
BRD-K83369119	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618745	phase I
BRD-K43440986	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618746	phase I
BRD-K79345052	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618747	phase I
BRD-K94292824	CCCNC(=O)N(C)C[C@@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618748	phase I
BRD-K62214276	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618749	phase I
BRD-K88223257	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618750	phase I
BRD-K48097043	CCCC#Cc1cnc2O[C@@H](CN(C)Cc3ccccc3F)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618751	phase I
BRD-K84358317	CC(C)C#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618752	phase I
BRD-K04605510	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)C(=O)CC4CC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54618753	phase I
BRD-K53914976	CCCNC(=O)N(C)C[C@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618754	phase I
BRD-K36935776	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618755	phase I
BRD-K10432434	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618756	phase I
BRD-K82881395	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618757	phase I
BRD-K12796341	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618758	phase I
BRD-K50126643	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618759	phase I
BRD-K68670732	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618760	phase I
BRD-K44978017	COCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618761	phase I
BRD-K84797651	C[C@@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618762	phase I
BRD-K33808757	CC(C)C#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618763	phase I
BRD-K77954087	C[C@@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618764	phase I
BRD-K34096870	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618765	phase I
BRD-K19678433	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618766	phase I
BRD-K40904431	CNC[C@@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618767	phase I
BRD-K93958918	CNC[C@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618768	phase I
BRD-K65999663	CNC[C@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618769	phase I
BRD-K83831887	C[C@@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618770	phase I
BRD-K63431240	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618771	phase I
BRD-K95190454	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618772	phase I
BRD-K13848456	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618773	phase I
BRD-K38688128	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618774	phase I
BRD-K14408783	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CN2CCOCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618775	phase I
BRD-K10493820	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618776	phase I
BRD-K17868036	CCCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618777	phase I
BRD-K56961909	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618778	phase I
BRD-K42864285	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618779	phase I
BRD-K48656305	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618780	phase I
BRD-K91684468	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)C3CCOCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618781	phase I
BRD-K19189563	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618782	phase I
BRD-K50360395	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618783	phase I
BRD-K21084378	COc1ccccc1c2ccc3c(O[C@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618784	phase I
BRD-K59099936	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54618785	phase I
BRD-K76450606	COc1ccccc1c2ccc3c(O[C@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618786	phase I
BRD-K27558213	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618787	phase I
BRD-K02201521	COCC(=O)N(C)C[C@@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618788	phase I
BRD-K60056824	CCCC#Cc1cnc2O[C@@H](CN(C)Cc3ccccc3F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618789	phase I
BRD-K95664364	CC(C)C#Cc1cnc2O[C@H](CN(C)Cc3cncnc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618790	phase I
BRD-K02985669	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618791	phase I
BRD-K76227258	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618792	phase I
BRD-K12016928	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54618793	phase I
BRD-K64882872	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618794	phase I
BRD-K33514849	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618795	phase I
BRD-K23011225	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618796	phase I
BRD-K48840041	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618797	phase I
BRD-K89326053	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618798	phase I
BRD-K82903423	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618799	phase I
BRD-K26006030	COCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618800	phase I
BRD-K88033714	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618801	phase I
BRD-K57902493	CC(C)C#Cc1cnc2O[C@@H](CN(C)Cc3cncnc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618802	phase I
BRD-K05625127	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Nc3cccc(F)c3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618803	phase I
BRD-K29458822	COCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618804	phase I
BRD-K27735716	CC(C)C#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618805	phase I
BRD-K92635027	CCCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618806	phase I
BRD-K30738885	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618807	phase I
BRD-K25119693	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618808	phase I
BRD-K61535492	CC(C)C#Cc1cnc2O[C@H](CN(C)Cc3cncnc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618809	phase I
BRD-K44436874	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618810	phase I
BRD-K15849229	CC(C)C#Cc1cnc2O[C@H](CN(C)C(=O)c3cccnc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618811	phase I
BRD-K37929770	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54618812	phase I
BRD-K34102596	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618813	phase I
BRD-K85301720	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618814	phase I
BRD-K80866161	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618815	phase I
BRD-K12263461	CNC[C@@H]1Oc2ncc(C#Cc3cccc(OC)c3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618816	phase I
BRD-K98970645	C[C@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618817	phase I
BRD-K90734139	CNC[C@H]1Oc2ncc(C#Cc3cccc(OC)c3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618818	phase I
BRD-K74843557	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54618819	phase I
BRD-K84522516	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618820	phase I
BRD-K63947305	C/C=C/c1cnc2O[C@H](CN(C)C(=O)C3CCOCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618821	phase I
BRD-K53861829	CCCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618822	phase I
BRD-K21980308	C/C=C/c1cnc2O[C@H](CN(C)C(=O)C3CCOCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618823	phase I
BRD-K69892607	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618824	phase I
BRD-K30316035	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)C(=O)CC4CC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54618825	phase I
BRD-K91757634	COCC(=O)N(C)C[C@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618826	phase I
BRD-K14212121	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)Oc3ncc(cc3C1=O)c4cccnc4	CID:54618827	phase I
BRD-K71329594	C[C@@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618828	phase I
BRD-K54676281	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54618829	phase I
BRD-K88849270	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618830	phase I
BRD-K74885091	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618831	phase I
BRD-K18229142	COCC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccccc3F)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618832	phase I
BRD-K47728674	COCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618833	phase I
BRD-K47647527	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618834	phase I
BRD-K87387784	COCC(=O)N(C)C[C@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618835	phase I
BRD-K14850613	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54618836	phase I
BRD-K35231228	CC(C)C#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccnc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618837	phase I
BRD-K99732047	C[C@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618838	phase I
BRD-K76321890	COc1ccccc1c2ccc3c(O[C@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618839	phase I
BRD-K94766884	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618840	phase I
BRD-K44589075	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54618841	phase I
BRD-K43419088	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Nc3cccc(F)c3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618842	phase I
BRD-K07426711	COCC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccccc3F)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618843	phase I
BRD-K66211423	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618844	phase I
BRD-K66698705	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618845	phase I
BRD-K86693846	CCCC#Cc1cnc2O[C@H](CN(C)Cc3ccccc3F)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618846	phase I
BRD-K24124456	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618847	phase I
BRD-K52373514	CCCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618848	phase I
BRD-K04260462	CNC[C@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618849	phase I
BRD-K06449093	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618850	phase I
BRD-K44752001	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618851	phase I
BRD-K64831080	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618852	phase I
BRD-K54543443	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618853	phase I
BRD-K54347561	COCC#Cc1ccc2c(O[C@H](CN(C)Cc3ccccn3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618854	phase I
BRD-K54857308	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618855	phase I
BRD-K05463922	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618856	phase I
BRD-K45850369	CCCNC(=O)N(C)C[C@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618857	phase I
BRD-K65611481	COCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccccc3F)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618858	phase I
BRD-K76996839	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618859	phase I
BRD-K87276639	COCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccccc3F)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618860	phase I
BRD-K02341409	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618861	phase I
BRD-K55482336	CCCC#Cc1cnc2O[C@H](CN(C)Cc3ccccc3F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618862	phase I
BRD-K73911580	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618863	phase I
BRD-K18710049	C[C@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618864	phase I
BRD-K48954843	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618865	phase I
BRD-K13898895	CC(C)C#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618866	phase I
BRD-K28922292	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618867	phase I
BRD-K40487298	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CN2CCOCC2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618868	phase I
BRD-K79240958	CCCC#Cc1cnc2O[C@H](CN(C)Cc3ccccc3F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618869	phase I
BRD-K47277477	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Nc3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618870	phase I
BRD-K04261044	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54618871	phase I
BRD-K64147637	COCC#Cc1ccc2c(O[C@H](CN(C)Cc3ccccn3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618872	phase I
BRD-K18754288	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54618873	phase I
BRD-K78556523	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Nc3cccc(F)c3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618874	phase I
BRD-K94267488	CCCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618875	phase I
BRD-K51757031	C[C@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618876	phase I
BRD-K73928524	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618877	phase I
BRD-K67891857	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618878	phase I
BRD-K37959950	C/C=C/c1cnc2O[C@H](CN(C)C(=O)C3CCOCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618879	phase I
BRD-K63448182	COc1ccccc1c2ccc3c(O[C@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54618880	phase I
BRD-K51031805	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618881	phase I
BRD-K69142462	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618882	phase I
BRD-K41761879	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618883	phase I
BRD-K92741883	COCC(=O)N(C)C[C@@H]1Oc2ncc(C#CC(C)(C)O)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618884	phase I
BRD-K07852185	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618885	phase I
BRD-K86482074	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)C3CCOCC3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618886	phase I
BRD-K56274797	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618887	phase I
BRD-K81464255	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618888	phase I
BRD-K36045097	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618889	phase I
BRD-K91019833	COc1ccccc1NC(=O)N(C)C[C@@H]2Oc3ncc(C#CC(C)C)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54618890	phase I
BRD-K38814572	COc1ccccc1c2ccc3c(O[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618891	phase I
BRD-K94346523	COc1ccc(cc1)S(=O)(=O)N(C)C[C@@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54618892	phase I
BRD-K45794109	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618893	phase I
BRD-K07315344	CCCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618894	phase I
BRD-K89074352	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618895	phase I
BRD-K90108396	CC(C)C#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccnc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618896	phase I
BRD-K05363386	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@@H](C)CO)C3=CCCCC3	CID:54618897	phase I
BRD-K15513663	CCCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)c3cccc(OC)c3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618898	phase I
BRD-K36801517	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618899	phase I
BRD-K51169491	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618900	phase I
BRD-K27503016	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618901	phase I
BRD-K23378122	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618902	phase I
BRD-K56562216	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618903	phase I
BRD-K93569047	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618904	phase I
BRD-K00133896	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618905	phase I
BRD-K68216590	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618906	phase I
BRD-K81291261	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618907	phase I
BRD-K10771753	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618908	phase I
BRD-K55504273	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618909	phase I
BRD-K06361641	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618910	phase I
BRD-K49258369	COc1ccccc1c2ccc3c(O[C@@H](CN(C)S(=O)(=O)c4ccc(F)cc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54618911	phase I
BRD-K92014291	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618912	phase I
BRD-K32816753	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618913	phase I
BRD-K99808647	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618914	phase I
BRD-K55657259	COCC#Cc1ccc2c(O[C@H](CN(C)Cc3ccccn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618915	phase I
BRD-K72999223	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618916	phase I
BRD-K31825071	COCC#Cc1ccc2c(O[C@H](CN(C)Cc3ccccn3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618917	phase I
BRD-K65598823	CC(C)C#Cc1cnc2O[C@H](CN(C)C(=O)c3cccnc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618918	phase I
BRD-K28714324	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618919	phase I
BRD-K31310964	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618920	phase I
BRD-K01060955	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Nc3cccc(F)c3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618921	phase I
BRD-K05295391	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cnccn2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54618922	phase I
BRD-K02806746	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Nc3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618923	phase I
BRD-K18071543	COc1ccccc1NC(=O)N(C)C[C@H]2Oc3ncc(C#CC(C)C)cc3C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54618924	phase I
BRD-K60732356	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618925	phase I
BRD-K18532833	COc1ccccc1NC(=O)N(C)C[C@@H]2Oc3ncc(C#CC(C)C)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54618926	phase I
BRD-K77805051	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618927	phase I
BRD-K49739160	CNC[C@@H]1Oc2ncc(C#Cc3cccc(OC)c3)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618928	phase I
BRD-K52465094	CNC[C@@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618929	phase I
BRD-K60069548	CNC[C@@H]1Oc2ncc(/C=C/c3ccccc3)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618930	phase I
BRD-K11231529	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CCC(C)C)ccc3S(=O)(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54618931	phase I
BRD-K23491633	CC(C)C#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccnc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618932	phase I
BRD-K94534355	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(C#Cc4ccncc4)ccc3S1(=O)=O	CID:54618933	phase I
BRD-K51004501	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618934	phase I
BRD-K66457675	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618935	phase I
BRD-K95096346	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618936	phase I
BRD-K15761174	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618937	phase I
BRD-K17157581	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618938	phase I
BRD-K57218871	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)C3CCOCC3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618939	phase I
BRD-K50282595	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)Oc4cc(C#Cc5ccncc5)ccc4S1(=O)=O	CID:54618940	phase I
BRD-K54049773	CC(C)C#Cc1cnc2O[C@@H](CN(C)Cc3cncnc3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618941	phase I
BRD-K21509488	C[C@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618942	phase I
BRD-K47371343	CCCC#Cc1cnc2O[C@@H](CN(C)Cc3ccccc3F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618943	phase I
BRD-K30174465	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)C3CCOCC3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618944	phase I
BRD-K95852551	CC(C)C#Cc1cnc2O[C@@H](CN(C)Cc3cncnc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618945	phase I
BRD-K42359528	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618946	phase I
BRD-K66975912	COc1ccc(C#Cc2cnc3O[C@H](CN(C)C(=O)CC4CC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54618947	phase I
BRD-K76893224	C/C=C/c1cnc2O[C@H](CN(C)C(=O)C3CCOCC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618948	phase I
BRD-K01204681	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54618949	phase I
BRD-K27957164	COCC#Cc1ccc2c(O[C@@H](CN(C)Cc3ccccn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618950	phase I
BRD-K30478013	CC(C)C#Cc1cnc2O[C@H](CN(C)C(=O)c3cccnc3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618951	phase I
BRD-K04284624	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618952	phase I
BRD-K94974633	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccccn4)cc3C1=O	CID:54618953	phase I
BRD-K14518066	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Nc3cccc(F)c3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618954	phase I
BRD-K54735832	CNC[C@@H]1Oc2ncc(/C=C/c3ccccc3)cc2C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54618955	phase I
BRD-K94597513	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618956	phase I
BRD-K35380368	COc1ccccc1NC(=O)N(C)C[C@H]2Oc3ncc(C#CC(C)C)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54618957	phase I
BRD-K29946624	CC(C)C#Cc1cnc2O[C@@H](CN(C)C(=O)c3cccnc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618958	phase I
BRD-K57179401	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618959	phase I
BRD-K64894352	COCC#Cc1ccc2c(O[C@@H](CN(C)Cc3ccccn3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618960	phase I
BRD-K91353140	CNC[C@@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618961	phase I
BRD-K46123637	C[C@@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618962	phase I
BRD-K16948767	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618963	phase I
BRD-K76582515	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54618964	phase I
BRD-K19418666	CCCNC(=O)N(C)C[C@@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54618965	phase I
BRD-K71964750	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618966	phase I
BRD-K45803728	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3ncc(C#CC4(O)CCCC4)cc3C1=O	CID:54618967	phase I
BRD-K67944552	C[C@H](O)C#Cc1ccc2c(O[C@@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618968	phase I
BRD-K61391179	COc1ccc(cc1)S(=O)(=O)N(C)C[C@H]2Oc3ncc(C#CC4(O)CCCC4)cc3C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54618969	phase I
BRD-K65529687	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54618970	phase I
BRD-K29107762	COc1ccccc1NC(=O)N(C)C[C@H]2Oc3ncc(C#CC(C)C)cc3C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54618971	phase I
BRD-K47020544	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cccnc2)Oc3cc(C#CC4(O)CCCC4)ccc3S1(=O)=O	CID:54618972	phase I
BRD-K85064040	COCC#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccccc3F)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618973	phase I
BRD-K65708449	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618974	phase I
BRD-K13118417	CNC[C@H]1Oc2cc(C#CC3(O)CCCC3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54618975	phase I
BRD-K52476750	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618976	phase I
BRD-K47810177	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Nc3cccc(F)c3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54618977	phase I
BRD-K07081072	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)C3=CCCCC3	CID:54618978	phase I
BRD-K12342216	COCC#Cc1ccc2c(O[C@H](CN(C)C(=O)c3ccccc3F)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618979	phase I
BRD-K05357743	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54618980	phase I
BRD-K00799745	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54618981	phase I
BRD-K42581894	C[C@@H](O)C#Cc1ccc2c(O[C@H](CN(C)Cc3ccc(cc3)c4ccccc4)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618982	phase I
BRD-K24750847	COCC#Cc1cnc2O[C@@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618983	phase I
BRD-K93494624	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)c4ccccc4F	CID:54618984	phase I
BRD-K44070326	CCCC#Cc1cnc2O[C@@H](CN(C)Cc3ccccc3F)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618985	phase I
BRD-K67291850	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618986	phase I
BRD-K76132378	COCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)C)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618987	phase I
BRD-K28833951	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54618988	phase I
BRD-K19755908	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)C(=O)CC4CC4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54618989	phase I
BRD-K10108893	COCC#Cc1ccc2c(O[C@@H](CN(C)Cc3ccccn3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618990	phase I
BRD-K42092012	COCC#Cc1cnc2O[C@H](CN(C)S(=O)(=O)C)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54618991	phase I
BRD-K38588505	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C)Oc2cc(C#Cc3ccc(F)cc3)ccc2S1(=O)=O	CID:54618992	phase I
BRD-K60638204	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54618993	phase I
BRD-K12438144	CC(C)C#Cc1ccc2c(O[C@@H](CN(C)C(=O)c3ccncc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54618994	phase I
BRD-K51252203	CC(C)C#Cc1cnc2O[C@@H](CN(C)Cc3cncnc3)[C@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54618995	phase I
BRD-K87886529	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)c4ccc(cc4)C(=O)N(C)C	CID:54618996	phase I
BRD-K03683936	COc1ccc(C#Cc2cnc3O[C@H](CN(C)C(=O)CC4CC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54618997	phase I
BRD-K84405221	CCCNC(=O)N(C)C[C@@H]1Oc2cc(C#CC(C)(C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54618998	phase I
BRD-K35095050	C/C=C/c1ccc2c(O[C@@H](CN(C)CC3CCOCC3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54619008	phase I
BRD-K57079327	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54619012	phase I
BRD-K55218950	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54619016	phase I
BRD-K52435112	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54619019	phase I
BRD-K73080020	COc1ccccc1S(=O)(=O)N(C)C[C@H]2Oc3cc(C#CCC4CCCC4)ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54619020	phase I
BRD-K02654447	CNC[C@H]1Oc2cc(/C=C/C)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54619028	phase I
BRD-K63157607	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54619030	phase I
BRD-K94034047	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54619034	phase I
BRD-K33218708	CNC[C@@H]1Oc2cc(C#Cc3ccccc3F)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54619037	phase I
BRD-K85413794	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3F	CID:54619048	phase I
BRD-K84023371	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3F	CID:54619055	phase I
BRD-K02375958	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54619056	phase I
BRD-K16717061	CCCC#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54619060	phase I
BRD-K20578716	CCCC#Cc1cnc2O[C@@H](CN(C)C(=O)Nc3cccc(F)c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54619062	phase I
BRD-K47906330	CCCC#Cc1cnc2O[C@H](CN(C)C(=O)Nc3cccc(F)c3)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54619065	phase I
BRD-K95435237	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54619066	phase I
BRD-K52908798	CNC[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3cccc(c3)C(=O)N(C)C	CID:54619080	phase I
BRD-K22458526	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54619105	phase I
BRD-K22420960	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccn2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54619119	phase I
BRD-K94005961	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54619129	phase I
BRD-K92666980	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54619138	phase I
BRD-K05278519	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54619148	phase I
BRD-K16479870	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54619161	phase I
BRD-K03056434	CNC[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)C3=CCCC3	CID:54619193	phase I
BRD-K64618192	C/C=C/c1ccc2c(O[C@H](CN(C)CC3CCOCC3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54619218	phase I
BRD-K83941994	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54619252	phase I
BRD-K63199400	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54619258	phase I
BRD-K71448503	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54619269	phase I
BRD-K86265745	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54619271	phase I
BRD-K99259037	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(C#CC4CCCC4)ccc3S1(=O)=O	CID:54619273	phase I
BRD-K21407905	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)C3=CCCCC3	CID:54619353	phase I
BRD-K91568452	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCOCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54619367	phase I
BRD-K97335870	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54619402	phase I
BRD-K08318631	CCCN(C)C[C@@H]1Oc2cc(C#CCC3CCCC3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54619426	phase I
BRD-K00177096	CCCN(C)C[C@H]1Oc2cc(C#CCC3CCCC3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54619430	phase I
BRD-K02537686	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)C3=CCCCC3	CID:54619435	phase I
BRD-K59549646	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)C3=CCCCC3	CID:54619457	phase I
BRD-K72055444	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54619462	phase I
BRD-K79080366	CCCN(C)C[C@@H]1Oc2ncc(C#Cc3ccccc3OC)cc2C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54619464	phase I
BRD-K76970388	CNC[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3ccccc3F	CID:54619466	phase I
BRD-K01048404	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54619475	phase I
BRD-K89390280	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54619477	phase I
BRD-K30935394	CNC[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3F	CID:54619491	phase I
BRD-K47077178	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccc(OC)cc3	CID:54619492	phase I
BRD-K18545493	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)C3=CCCCC3	CID:54619494	phase I
BRD-K45700898	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccc(OC)cc3	CID:54619503	phase I
BRD-K83155387	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54619510	phase I
BRD-K81732150	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54619535	phase I
BRD-K81654062	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54619536	phase I
BRD-K50351738	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)C3=CCCCC3	CID:54619572	phase I
BRD-K98621344	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)C3=CCCCC3	CID:54619574	phase I
BRD-K08614872	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54619640	phase I
BRD-K01251033	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54619651	phase I
BRD-K81373254	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54619652	phase I
BRD-K46211110	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54619703	phase I
BRD-K19601332	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(C)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54619738	phase I
BRD-K92043077	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccccc3C	CID:54619902	phase I
BRD-K09964242	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccc(C#N)cc3	CID:54619906	phase I
BRD-K27732957	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54619971	phase I
BRD-K85347477	COc1cccc(c1)c2cnc3O[C@H](CN(C)CC4CCCC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54619975	phase I
BRD-K00248354	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)C3CCCCC3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54619990	phase I
BRD-K66288362	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54619996	phase I
BRD-K47724214	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccc(C#N)cc3	CID:54620005	phase I
BRD-K68315360	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54620037	phase I
BRD-K35443780	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54620040	phase I
BRD-K29097491	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3cc(C#Cc4cccnc4)ccc3S1(=O)=O	CID:54620047	phase I
BRD-K88925856	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3cc(C#Cc4cccnc4)ccc3S1(=O)=O	CID:54620051	phase I
BRD-K07922534	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3ccc(C#N)cc3	CID:54620066	phase I
BRD-K59261651	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54620067	phase I
BRD-K69936404	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCOCC2)Oc3cc(C#Cc4ccccc4F)ccc3S1(=O)=O	CID:54620069	phase I
BRD-K66581298	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54620121	phase I
BRD-K71982936	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54620131	phase I
BRD-K29211776	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54620145	phase I
BRD-K95593113	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#Cc4cccnc4)cc3C1=O	CID:54620164	phase I
BRD-K98790311	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54620190	phase I
BRD-K27961885	C/C=C/c1ccc2c(O[C@H](CN(C)Cc3cccc(F)c3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54620198	phase I
BRD-K53986871	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620215	phase I
BRD-K14000735	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620217	phase I
BRD-K80212510	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620218	phase I
BRD-K59159285	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620221	phase I
BRD-K99830292	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620222	phase I
BRD-K00144236	CCCN(C)C[C@@H]1Oc2cc(C#Cc3ccncc3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54620273	phase I
BRD-K34314104	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3ncc(/C=C/c4ccccc4)cc3C1=O	CID:54620330	phase I
BRD-K39420925	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620413	phase I
BRD-K17897186	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620414	phase I
BRD-K05745188	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620415	phase I
BRD-K16376056	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620416	phase I
BRD-K25895238	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620418	phase I
BRD-K32069250	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620419	phase I
BRD-K92370559	COc1ccc(C#Cc2cnc3O[C@H](CN(C)CC4CCCC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54620486	phase I
BRD-K48619543	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)CC4CCCC4)[C@@H](C)CN([C@H](C)CO)C(=O)c3c2)cc1	CID:54620487	phase I
BRD-K65243627	COc1ccc(C#Cc2cnc3O[C@H](CN(C)CC4CCCC4)[C@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:54620488	phase I
BRD-K14383710	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4cccc(F)c4)cc3C1=O	CID:54620506	phase I
BRD-K78777980	C/C=C/c1ccc2c(O[C@H](CN(C)Cc3ccccc3F)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54620917	phase I
BRD-K32297746	C/C=C/c1ccc2c(O[C@H](CN(C)Cc3ccccc3F)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54620918	phase I
BRD-K47517065	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620981	phase I
BRD-K20347026	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620982	phase I
BRD-K73434853	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620983	phase I
BRD-K17705111	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620984	phase I
BRD-K18004653	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620986	phase I
BRD-K42731451	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620987	phase I
BRD-K17155259	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54620988	phase I
BRD-K57182060	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621024	phase I
BRD-K24752075	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621025	phase I
BRD-K56384721	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621026	phase I
BRD-K74647590	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621027	phase I
BRD-K23844489	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621028	phase I
BRD-K99311962	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621029	phase I
BRD-K19668893	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54621030	phase I
BRD-K19033697	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54621064	phase I
BRD-K05051664	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)c4ccncc4	CID:54621065	phase I
BRD-K45056194	CNC[C@@H]1Oc2cc(C#C[C@@H](C)O)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54621135	phase I
BRD-K30611309	CNC[C@@H]1Oc2cc(C#C[C@H](C)O)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54621137	phase I
BRD-K67925802	CCCN(C)C[C@H]1Oc2cc(C#Cc3ccccc3F)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54621292	phase I
BRD-K30315899	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Cc3ccccn3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54621317	phase I
BRD-K76710817	CNC[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)c3ccccc3OC	CID:54621324	phase I
BRD-K32035967	CNC[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3OC	CID:54621325	phase I
BRD-K61050695	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccccc3OC	CID:54621466	phase I
BRD-K30040610	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54621587	phase I
BRD-K99333268	CNC[C@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54621646	phase I
BRD-K64257929	CNC[C@@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54621647	phase I
BRD-K12385780	CNC[C@@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54621648	phase I
BRD-K35432283	CNC[C@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54621649	phase I
BRD-K44363090	CNC[C@@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54621650	phase I
BRD-K53223020	CNC[C@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54621651	phase I
BRD-K41732846	CNC[C@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO	CID:54621652	phase I
BRD-K07768565	CNC[C@@H]1Oc2cc(C#CCN(C)C)ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54621653	phase I
BRD-K57884454	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54621691	phase I
BRD-K74042299	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54621859	phase I
BRD-K89354557	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54621966	phase I
BRD-K04457555	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54622047	phase I
BRD-K48755012	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(cc3C1=O)c4cccc(C#N)c4	CID:54622048	phase I
BRD-K19838409	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccc(C)cc3	CID:54622572	phase I
BRD-K73230533	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54622611	phase I
BRD-K89637993	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ncc(C#CCN(C)C)cc4C1=O	CID:54622909	phase I
BRD-K82440152	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)c3ccccc3)Oc4ncc(C#CCN(C)C)cc4C1=O	CID:54622912	phase I
BRD-K91094904	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C)Oc2cc(ccc2S1(=O)=O)C3=CCCC3	CID:54622989	phase I
BRD-K54837534	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54623073	phase I
BRD-K30058879	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54623074	phase I
BRD-K19033174	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54624299	phase I
BRD-K35462725	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)c3cccc(F)c3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54624302	phase I
BRD-K34836852	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54624303	phase I
BRD-K34136030	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)c3cccc(F)c3)[C@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54624304	phase I
BRD-K45386827	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(ccc2S1(=O)=O)c3ccc(F)cc3	CID:54624404	phase I
BRD-K82263627	C/C=C/c1ccc2c(O[C@H](CN(C)C)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54624431	phase I
BRD-K34545919	C/C=C/c1ccc2c(O[C@H](CN(C)C)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54624434	phase I
BRD-K64160028	COc1cccc(c1)c2cnc3O[C@@H](CN(C)Cc4ccc(F)cc4)[C@H](C)CN([C@H](C)CO)C(=O)c3c2	CID:54624441	phase I
BRD-K29794647	COc1cccc(c1)c2cnc3O[C@H](CN(C)Cc4ccc(F)cc4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2	CID:54624442	phase I
BRD-K53642448	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CN(C)C)Oc2ncc(C#Cc3ccncc3)cc2C1=O	CID:54624472	phase I
BRD-K03840522	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CN(C)C)Oc2ncc(C#Cc3ccncc3)cc2C1=O	CID:54624473	phase I
BRD-K51934037	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccccc4	CID:54624541	phase I
BRD-K15234288	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3cc(ccc3S1(=O)=O)c4ccccc4	CID:54624543	phase I
BRD-K44161636	C/C=C/c1ccc2c(O[C@@H](CN(C)S(=O)(=O)c3ccccc3)[C@@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54624606	phase I
BRD-K99839793	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@H](C)CO)c3cccnc3	CID:54624614	phase I
BRD-K84244541	CCCN(C)C[C@@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3cccnc3	CID:54624615	phase I
BRD-K74554256	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3cccnc3	CID:54624616	phase I
BRD-K45695360	CCCN(C)C[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3cccnc3	CID:54624619	phase I
BRD-K88844437	CCCN(C)C[C@H]1Oc2ncc(C#Cc3ccc(OC)cc3)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54624752	phase I
BRD-K09110452	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CN2CCOCC2)Oc3ncc(cc3C1=O)c4ccncc4	CID:54624763	phase I
BRD-K15863674	CCCN(C)C[C@H]1Oc2ncc(C#CCN(C)C)cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54624798	phase I
BRD-K81930842	CCCN(C)C[C@H]1Oc2ncc(C#CCN(C)C)cc2C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54624799	phase I
BRD-K75904236	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54624827	phase I
BRD-K09553491	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54624828	phase I
BRD-K38841486	CCCN(C)C[C@H]1Oc2cc(C#Cc3ccccc3)ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54624850	phase I
BRD-K74547048	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54624984	phase I
BRD-K25485361	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54624985	phase I
BRD-K43049540	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54624986	phase I
BRD-K33637182	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54624989	phase I
BRD-K71855503	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54624990	phase I
BRD-K55341496	CCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)C3=CCCC3	CID:54625138	phase I
BRD-K02990757	CCC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)C3=CCCC3	CID:54625139	phase I
BRD-K00663064	CCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)C3=CCCC3	CID:54625140	phase I
BRD-K95951626	CCC(=O)N(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)C3=CCCC3	CID:54625142	phase I
BRD-K44368508	CCC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@@H](C)CO)C3=CCCC3	CID:54625143	phase I
BRD-K27009196	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625159	phase I
BRD-K33061098	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625160	phase I
BRD-K01228394	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625161	phase I
BRD-K44640039	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625162	phase I
BRD-K12878711	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)c3ccc(F)cc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54625177	phase I
BRD-K64180195	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625239	phase I
BRD-K39101193	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625242	phase I
BRD-K91731568	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625243	phase I
BRD-K15126665	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625244	phase I
BRD-K04104496	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625245	phase I
BRD-K90149465	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625293	phase I
BRD-K86832444	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625294	phase I
BRD-K88962898	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)Oc4cc(C#CCN(C)C)ccc4S1(=O)=O	CID:54625295	phase I
BRD-K36633782	CNC[C@H]1Oc2ncc(cc2C(=O)N(C[C@H]1C)[C@H](C)CO)c3ccc(C)cc3	CID:54625379	phase I
BRD-K09996575	CNC[C@@H]1Oc2ncc(cc2C(=O)N(C[C@@H]1C)[C@@H](C)CO)c3ccc(C)cc3	CID:54625380	phase I
BRD-K84951011	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(ccc2S1(=O)=O)c3cccc(C#N)c3	CID:54625394	phase I
BRD-K39144410	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(ccc2S1(=O)=O)c3cccc(C#N)c3	CID:54625397	phase I
BRD-K43550773	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625451	phase I
BRD-K87500884	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625452	phase I
BRD-K38615358	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625454	phase I
BRD-K22577612	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625455	phase I
BRD-K12017137	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625456	phase I
BRD-K86537726	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625457	phase I
BRD-K39561907	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54625458	phase I
BRD-K97641878	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625468	phase I
BRD-K30150248	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625469	phase I
BRD-K79103937	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625470	phase I
BRD-K24348220	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625471	phase I
BRD-K71585907	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54625472	phase I
BRD-K54302962	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54625500	phase I
BRD-K78518750	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54625501	phase I
BRD-K77760488	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(F)cc4	CID:54625502	phase I
BRD-K60783789	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3ccc(F)cc3	CID:54625517	phase I
BRD-K49098390	COc1cccc(C#Cc2ccc3c(O[C@@H](CN(C)C)[C@H](C)CN([C@@H](C)CO)S3(=O)=O)c2)c1	CID:54625522	phase I
BRD-K02549628	COc1cccc(C#Cc2ccc3c(O[C@@H](CN(C)C)[C@H](C)CN([C@H](C)CO)S3(=O)=O)c2)c1	CID:54625523	phase I
BRD-K89161054	C/C=C/c1ccc2c(O[C@H](CN(C)C(=O)c3ccncc3)[C@@H](C)CN([C@H](C)CO)S2(=O)=O)c1	CID:54625567	phase I
BRD-K15559773	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54625611	phase I
BRD-K13226037	C/C=C/c1cnc2O[C@@H](CN(C)Cc3ccc(F)cc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54625621	phase I
BRD-K86335338	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54625679	phase I
BRD-K03188480	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54625680	phase I
BRD-K30342454	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54625687	phase I
BRD-K47992037	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54625688	phase I
BRD-K28013436	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54625689	phase I
BRD-K01575212	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54625692	phase I
BRD-K07642375	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(/C=C/c4ccccc4)ccc3S1(=O)=O	CID:54625694	phase I
BRD-K15525241	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54625696	phase I
BRD-K23384658	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54625698	phase I
BRD-K70492429	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54625700	phase I
BRD-K86948282	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54625701	phase I
BRD-K05678583	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(C#CC4CC4)ccc3S1(=O)=O	CID:54625702	phase I
BRD-K84724939	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)Oc3ncc(cc3C1=O)c4ccc(C)cc4	CID:54625716	phase I
BRD-K07820537	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625719	phase I
BRD-K07275374	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625720	phase I
BRD-K75557837	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625721	phase I
BRD-K65809558	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625722	phase I
BRD-K07438289	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625723	phase I
BRD-K37203945	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625724	phase I
BRD-K09597785	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625725	phase I
BRD-K71328603	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54625726	phase I
BRD-K96194602	CCCC#Cc1ccc2c(O[C@@H](CN(C)Cc3ccncc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54625750	phase I
BRD-K92646316	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ncc(C#CCN(C)C)cc4C1=O	CID:54625780	phase I
BRD-K33350866	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)Oc4ncc(C#CCN(C)C)cc4C1=O	CID:54625783	phase I
BRD-K26778237	COc1ccccc1C#Cc2ccc3c(O[C@@H](CN(C)Cc4ccccc4)[C@@H](C)CN([C@H](C)CO)S3(=O)=O)c2	CID:54625812	phase I
BRD-K74200139	COc1ccccc1C#Cc2ccc3c(O[C@@H](CN(C)Cc4ccccc4)[C@@H](C)CN([C@@H](C)CO)S3(=O)=O)c2	CID:54625815	phase I
BRD-K26553253	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54626030	phase I
BRD-K56116682	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54626033	phase I
BRD-K99495107	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54626141	phase I
BRD-K43848904	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54626142	phase I
BRD-K79481905	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54626143	phase I
BRD-K76294510	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54626145	phase I
BRD-K49733809	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626155	phase I
BRD-K36278687	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626157	phase I
BRD-K83874987	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626158	phase I
BRD-K46791751	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626159	phase I
BRD-K42584632	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626160	phase I
BRD-K28135985	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626161	phase I
BRD-K19159562	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54626195	phase I
BRD-K34206995	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54626196	phase I
BRD-K48679006	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54626197	phase I
BRD-K82117061	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54626200	phase I
BRD-K71493061	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54626201	phase I
BRD-K74757268	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54626406	phase I
BRD-K15638296	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54626407	phase I
BRD-K68541237	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54626408	phase I
BRD-K75856618	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4ccc(C#N)cc4	CID:54626409	phase I
BRD-K56842656	CCCN(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@@H]1C)[C@H](C)CO)c3cccc(C#N)c3	CID:54626418	phase I
BRD-K83498497	CCCN(C)C[C@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@@H](C)CO)c3cccc(C#N)c3	CID:54626419	phase I
BRD-K79982586	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626526	phase I
BRD-K43905345	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cc(F)ccc2F)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:54626527	phase I
BRD-K17180926	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54626572	phase I
BRD-K19431609	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54626573	phase I
BRD-K02043218	C/C=C/c1ccc2c(O[C@@H](CN(C)C(=O)Nc3ccc(F)cc3)[C@H](C)CN([C@@H](C)CO)S2(=O)=O)c1	CID:54626596	phase I
BRD-K31992949	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(C#CCN(C)C)ccc2S1(=O)=O	CID:54626632	phase I
BRD-K85908443	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccccc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54626847	phase I
BRD-K99994453	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54626992	phase I
BRD-K82469231	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54626993	phase I
BRD-K22983069	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54626997	phase I
BRD-K48031880	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54626998	phase I
BRD-K92659561	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5ccncc5	CID:54627208	phase I
BRD-K37743233	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5ccncc5	CID:54627209	phase I
BRD-K71894218	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5ccncc5	CID:54627210	phase I
BRD-K04309313	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5ccncc5	CID:54627211	phase I
BRD-K28036193	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4cc(ccc4S1(=O)=O)c5ccncc5	CID:54627213	phase I
BRD-K78496556	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54627254	phase I
BRD-K05225561	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)Oc3cc(ccc3S1(=O)=O)c4cccc(C#N)c4	CID:54627261	phase I
BRD-K51970157	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54627270	phase I
BRD-K02256002	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCOCC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54627271	phase I
BRD-K94293016	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCOCC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54627272	phase I
BRD-K32132728	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54627273	phase I
BRD-K73365449	C/C=C/c1cnc2O[C@H](CN(C)S(=O)(=O)c3ccccc3)[C@@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:54627288	phase I
BRD-K05322955	COc1ccc(NC(=O)N(C)C[C@H]2Oc3cc(C#CCN(C)C)ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:54627368	phase I
BRD-K44660322	COc1ccc(NC(=O)N(C)C[C@@H]2Oc3cc(C#CCN(C)C)ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54627369	phase I
BRD-K14721343	C/C=C/c1cnc2O[C@@H](CN(C)C(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](C)CN([C@H](C)CO)C(=O)c2c1	CID:54627377	phase I
BRD-K39030761	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54627464	phase I
BRD-K05615182	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCOCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54627465	phase I
BRD-K17144088	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCOCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54627467	phase I
BRD-K40576182	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)c4cccnc4	CID:54628019	phase I
BRD-K43623238	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628092	phase I
BRD-K31749518	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628093	phase I
BRD-K08781018	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:54628647	phase I
BRD-K12973880	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628724	phase I
BRD-K72430479	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628725	phase I
BRD-K77235585	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628726	phase I
BRD-K37237818	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628727	phase I
BRD-K07033348	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628728	phase I
BRD-K40324831	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628729	phase I
BRD-K37516186	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54628794	phase I
BRD-K56928281	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54628797	phase I
BRD-K66351990	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)Oc2cc(ccc2S1(=O)=O)C3=CCCCC3	CID:54628893	phase I
BRD-K40034229	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2cc(ccc2S1(=O)=O)C3=CCCCC3	CID:54628894	phase I
BRD-K71032892	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C)Oc2cc(ccc2S1(=O)=O)C3=CCCCC3	CID:54628895	phase I
BRD-K28583191	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628987	phase I
BRD-K05205967	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628988	phase I
BRD-K45937240	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628989	phase I
BRD-K27775808	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54628990	phase I
BRD-K56250581	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54629011	phase I
BRD-K48723823	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629090	phase I
BRD-K72147201	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629095	phase I
BRD-K54577741	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629096	phase I
BRD-K93410934	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629097	phase I
BRD-K18377730	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629126	phase I
BRD-K20098898	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629128	phase I
BRD-K72234025	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629129	phase I
BRD-K29702325	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629162	phase I
BRD-K77899084	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54629195	phase I
BRD-K88756517	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54629196	phase I
BRD-K12844656	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54629197	phase I
BRD-K17627540	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54629198	phase I
BRD-K59680547	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54629199	phase I
BRD-K66617214	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629227	phase I
BRD-K79437066	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629230	phase I
BRD-K86888704	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CC2CC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54629231	phase I
BRD-K11620284	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54629279	phase I
BRD-K90077012	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54629280	phase I
BRD-K57134435	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54629281	phase I
BRD-K55187504	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cncnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54629285	phase I
BRD-K37315860	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cncnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54629286	phase I
BRD-K55385841	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)c4ccccc4F	CID:54630363	phase I
BRD-K41377239	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630616	phase I
BRD-K19607523	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630617	phase I
BRD-K71059148	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630618	phase I
BRD-K48680503	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630619	phase I
BRD-K26370510	CCCNC(=O)N(C)C[C@@H]1Oc2cc(ccc2S(=O)(=O)N(C[C@H]1C)[C@H](C)CO)C3=CCCCC3	CID:54630622	phase I
BRD-K08179047	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630661	phase I
BRD-K22435870	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630662	phase I
BRD-K94312010	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630663	phase I
BRD-K62854197	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630665	phase I
BRD-K46599299	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630666	phase I
BRD-K93156709	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630667	phase I
BRD-K29407738	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630674	phase I
BRD-K68672034	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630683	phase I
BRD-K39379715	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630684	phase I
BRD-K00409424	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630686	phase I
BRD-K54986816	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630687	phase I
BRD-K18863894	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630688	phase I
BRD-K38044934	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630689	phase I
BRD-K98560805	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccn2)Oc3cc(ccc3S1(=O)=O)C4=CCCCC4	CID:54630690	phase I
BRD-K96398395	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@H](C)CO)C4=CCCC4	CID:54630715	phase I
BRD-K85119394	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@H]2C)[C@@H](C)CO)C4=CCCC4	CID:54630716	phase I
BRD-K15478534	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2Oc3cc(ccc3S(=O)(=O)N(C[C@@H]2C)[C@@H](C)CO)C4=CCCC4	CID:54630721	phase I
BRD-K29253960	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54630745	phase I
BRD-K92498491	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54630746	phase I
BRD-K60693111	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54630748	phase I
BRD-K40927841	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccccc2F)Oc3ncc(cc3C1=O)C4=CCCCC4	CID:54630750	phase I
BRD-K69482343	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630769	phase I
BRD-K80767319	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630770	phase I
BRD-K25304254	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630791	phase I
BRD-K95521279	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630792	phase I
BRD-K46936109	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630794	phase I
BRD-K24002047	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccncc2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54630795	phase I
BRD-K82392710	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(cc3C1=O)C4=CCCC4	CID:54630816	phase I
BRD-K33165698	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc3OCOc3c2)Oc4ncc(cc4C1=O)C5=CCCCC5	CID:54630847	phase I
BRD-K90108753	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(cc3C1=O)c4ccc(C)cc4	CID:54631009	phase I
BRD-K14499901	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(cc3C1=O)c4ccc(C)cc4	CID:54631010	phase I
BRD-K22610673	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54631021	phase I
BRD-K21017376	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccc(F)cc4	CID:54631025	phase I
BRD-K16503119	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3cc(ccc3S1(=O)=O)C4=CCCC4	CID:54631042	phase I
BRD-K44624970	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54631053	phase I
BRD-K82340687	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54631054	phase I
BRD-K65741216	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54631055	phase I
BRD-K75388977	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(C#Cc4ccncc4)cc3C1=O	CID:54631056	phase I
BRD-K25876174	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54631091	phase I
BRD-K14121002	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCC2)Oc3ncc(cc3C1=O)c4ccc(C#N)cc4	CID:54631092	phase I
BRD-K07298554	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccc(C)cc4	CID:54631154	phase I
BRD-K71006572	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54631158	phase I
BRD-K77051246	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CCCCC2)Oc3ncc(C#CC4CCCCC4)cc3C1=O	CID:54631159	phase I
BRD-K95815724	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCCC2)Oc3ncc(cc3C1=O)c4ccccc4C	CID:54631205	phase I
BRD-K70068608	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54631219	phase I
BRD-K19870323	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54631220	phase I
BRD-K97787842	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54631221	phase I
BRD-K08428488	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54631222	phase I
BRD-K27431449	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54631223	phase I
BRD-K84559549	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc3cc(ccc3S1(=O)=O)c4ccc(C)cc4	CID:54631225	phase I
BRD-K01176062	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(cc2)C(F)(F)F)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:54631235	phase I
BRD-K68690198	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(Oc3ccccc3)cc2)Oc4c(NC(=O)NC5CCCCC5)cccc4C1=O	CID:54631247	phase I
BRD-K54061956	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(cc2)C(=O)Nc3ccccc3N)OCc4cn(CCCC1=O)nn4	CID:54631254	phase I
BRD-K09080977	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2cc(F)ccc2F)C[C@H]1C	CID:54631279	phase I
BRD-K63938446	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@H]1C)OC	CID:54631280	phase I
BRD-K98321674	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631281	phase I
BRD-K20729616	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)Cc1ccccn1	CID:54631282	phase I
BRD-K27467349	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)cc2OC[C@H](C)NC[C@H]1C	CID:54631283	phase I
BRD-K27811024	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631284	phase I
BRD-K00061590	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(Cc2ccc(OC)cc2)C[C@@H]1C	CID:54631285	phase I
BRD-K24486079	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631286	phase I
BRD-K89896024	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631287	phase I
BRD-K67187917	CCCNC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H]1C)OC	CID:54631288	phase I
BRD-K91694818	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631289	phase I
BRD-K37517867	CCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631290	phase I
BRD-K39475284	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631291	phase I
BRD-K06240911	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631292	phase I
BRD-K34692511	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc(cc3)C(F)(F)F)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631293	phase I
BRD-K12610781	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631294	phase I
BRD-K08540981	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631295	phase I
BRD-K66975725	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631296	phase I
BRD-K01977318	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3Cl)cc2OC[C@H](C)NC[C@H]1C	CID:54631297	phase I
BRD-K89165671	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@H](C)N(C[C@H]1C)S(C)(=O)=O	CID:54631298	phase I
BRD-K62237490	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)C1CCOCC1	CID:54631299	phase I
BRD-K46419847	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@H](C)NC[C@H]1C	CID:54631300	phase I
BRD-K46959535	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54631301	phase I
BRD-K01335229	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631302	phase I
BRD-K98622504	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccc(F)c3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631303	phase I
BRD-K98783629	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54631304	phase I
BRD-K79330967	CCCC(=O)Nc1ccc2OC[C@H](C)N(CC3CCCC3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631305	phase I
BRD-K17554230	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H](C)NC[C@H]1C	CID:54631306	phase I
BRD-K51849024	CCCNC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631307	phase I
BRD-K16339566	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631308	phase I
BRD-K95549765	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@H](C)N(C)C[C@H]1C	CID:54631309	phase I
BRD-K73146135	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631310	phase I
BRD-K17333907	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631311	phase I
BRD-K53987979	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631312	phase I
BRD-K22210284	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631313	phase I
BRD-K87258520	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631314	phase I
BRD-K07250107	CCCC(=O)Nc1ccc2OC[C@@H](C)N(CC3CCCC3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631315	phase I
BRD-K70633610	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@H](C)N(C)C[C@H]1C	CID:54631316	phase I
BRD-K07817703	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631317	phase I
BRD-K87109962	CCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631318	phase I
BRD-K16714380	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1cccnc1	CID:54631319	phase I
BRD-K76224440	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631320	phase I
BRD-K43971874	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631321	phase I
BRD-K89133991	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631322	phase I
BRD-K00498462	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)C1CCOCC1	CID:54631323	phase I
BRD-K01284917	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1ccc(F)cc1	CID:54631324	phase I
BRD-K57641516	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@H](C)NC[C@H]1C	CID:54631325	phase I
BRD-K56124197	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631326	phase I
BRD-K00927991	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631327	phase I
BRD-K15178090	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631328	phase I
BRD-K78699095	CCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631329	phase I
BRD-K92028820	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631330	phase I
BRD-K68887696	CCCC(=O)Nc1ccc2OC[C@H](C)N(CC3CCCC3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631331	phase I
BRD-K71904020	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54631332	phase I
BRD-K67628477	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc(cc3)C(F)(F)F)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631333	phase I
BRD-K46359800	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@H](C)NC[C@H]1C	CID:54631334	phase I
BRD-K76258424	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631335	phase I
BRD-K48270072	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631336	phase I
BRD-K30953566	CCCNC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631337	phase I
BRD-K44011183	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631338	phase I
BRD-K63903580	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54631339	phase I
BRD-K17506650	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCCCC3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54631340	phase I
BRD-K35944454	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631341	phase I
BRD-K28370158	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631342	phase I
BRD-K12012973	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631343	phase I
BRD-K66046471	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631344	phase I
BRD-K21627123	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631345	phase I
BRD-K66944475	CCCC(=O)Nc1ccc2OC[C@@H](C)N(CC3CCCC3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631346	phase I
BRD-K28752165	CCCNC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631347	phase I
BRD-K20555183	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccn3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1ccccc1Cl	CID:54631348	phase I
BRD-K30706668	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631349	phase I
BRD-K81810761	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631350	phase I
BRD-K66687431	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1cccnc1	CID:54631351	phase I
BRD-K24781739	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)CN(C)C)ccc2OC[C@@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631352	phase I
BRD-K58472651	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631353	phase I
BRD-K42011191	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631354	phase I
BRD-K90897407	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)CN(C)C)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccncc1	CID:54631355	phase I
BRD-K47119747	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631356	phase I
BRD-K81721884	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccc(F)c3)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631357	phase I
BRD-K95814669	COCC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3cccc(F)c3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631358	phase I
BRD-K79516068	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2cc(F)ccc2F)C[C@@H]1C	CID:54631359	phase I
BRD-K85721574	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631360	phase I
BRD-K41421455	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3Cl)cc2OC[C@H](C)NC[C@@H]1C	CID:54631361	phase I
BRD-K32629755	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631362	phase I
BRD-K22743786	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631363	phase I
BRD-K05531636	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631364	phase I
BRD-K20032520	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631365	phase I
BRD-K02943940	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)C1CCOCC1	CID:54631366	phase I
BRD-K48479537	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631367	phase I
BRD-K37608670	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631368	phase I
BRD-K84921800	CCCNC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631369	phase I
BRD-K24758440	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631370	phase I
BRD-K48553449	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631371	phase I
BRD-K06250012	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631372	phase I
BRD-K38740852	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54631373	phase I
BRD-K88269272	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(CC2CCOCC2)C[C@@H]1C	CID:54631374	phase I
BRD-K75717096	CCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccno3)cc2OC[C@H]1C)OC	CID:54631375	phase I
BRD-K87524836	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631376	phase I
BRD-K01006500	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54631377	phase I
BRD-K32324469	COCC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3cccc(F)c3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631378	phase I
BRD-K51217456	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1cccnc1	CID:54631379	phase I
BRD-K02356765	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54631380	phase I
BRD-K23060864	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(CC2CCOCC2)C[C@@H]1C	CID:54631381	phase I
BRD-K27998900	CCCNC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H]1C)OC	CID:54631382	phase I
BRD-K44207800	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(CC2CCOCC2)C[C@H]1C	CID:54631383	phase I
BRD-K80550858	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@H]1C)OC	CID:54631384	phase I
BRD-K92978187	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)Cc1ccccn1	CID:54631385	phase I
BRD-K34786682	CCCNC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H]1C)OC	CID:54631386	phase I
BRD-K86335374	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631387	phase I
BRD-K66714409	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631388	phase I
BRD-K14209633	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631389	phase I
BRD-K33909932	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631390	phase I
BRD-K26461874	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631391	phase I
BRD-K99949435	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccc(F)cc1	CID:54631392	phase I
BRD-K20877010	CCCNC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631393	phase I
BRD-K19357327	CCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631394	phase I
BRD-K03804563	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)Cc1ccccn1	CID:54631395	phase I
BRD-K74591286	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc(cc3)C(F)(F)F)ccc2OC[C@H](C)NC[C@H]1C	CID:54631396	phase I
BRD-K59323544	CCCNC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631397	phase I
BRD-K64955433	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631398	phase I
BRD-K40063896	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631399	phase I
BRD-K80866887	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631400	phase I
BRD-K00526921	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631401	phase I
BRD-K75596743	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631402	phase I
BRD-K89679058	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@H]1C)OC	CID:54631403	phase I
BRD-K51725102	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@H]1C)OC	CID:54631404	phase I
BRD-K89416483	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631405	phase I
BRD-K19949652	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)C1CCOCC1	CID:54631406	phase I
BRD-K37639981	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccc(F)cc1	CID:54631407	phase I
BRD-K99469929	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631408	phase I
BRD-K79512815	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631409	phase I
BRD-K61164584	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631410	phase I
BRD-K91292927	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(CC2CCOCC2)C[C@@H]1C	CID:54631411	phase I
BRD-K00566471	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(CC2CCOCC2)C[C@H]1C	CID:54631412	phase I
BRD-K44119437	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631413	phase I
BRD-K62753164	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631414	phase I
BRD-K74162965	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631415	phase I
BRD-K30228236	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631416	phase I
BRD-K32809121	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631417	phase I
BRD-K77700305	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631418	phase I
BRD-K63415335	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631419	phase I
BRD-K16955082	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631420	phase I
BRD-K71073890	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccc(F)c3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631421	phase I
BRD-K90173466	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631422	phase I
BRD-K59909245	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631423	phase I
BRD-K84078621	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631424	phase I
BRD-K54029516	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54631425	phase I
BRD-K00196194	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54631426	phase I
BRD-K16925239	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@@H](C)N(Cc2cccc(c2)C(F)(F)F)C[C@H]1C	CID:54631427	phase I
BRD-K00575615	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631428	phase I
BRD-K59336577	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)Cc1ccccn1	CID:54631429	phase I
BRD-K83896715	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2OC[C@@H](C)N(Cc2ccccn2)C[C@H]1C	CID:54631430	phase I
BRD-K54456094	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631431	phase I
BRD-K89432015	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631432	phase I
BRD-K79881395	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)c1ccc(Cl)cc1	CID:54631433	phase I
BRD-K68836298	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc(cc3)C(F)(F)F)ccc2OC[C@H](C)NC[C@H]1C	CID:54631434	phase I
BRD-K55232867	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631435	phase I
BRD-K62676049	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1cccnc1	CID:54631436	phase I
BRD-K06897051	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2cc(F)ccc2F)C[C@@H]1C	CID:54631437	phase I
BRD-K45591070	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631438	phase I
BRD-K29996103	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631439	phase I
BRD-K02576169	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(Cc2ccc(OC)cc2)C[C@H]1C	CID:54631440	phase I
BRD-K82053812	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631441	phase I
BRD-K46792957	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631442	phase I
BRD-K82062446	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631443	phase I
BRD-K52628302	CCCNC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H]1C)OC	CID:54631444	phase I
BRD-K92975271	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631445	phase I
BRD-K09640010	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)C1CCOCC1	CID:54631446	phase I
BRD-K77793090	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(OC)c3)cc2OC[C@@H]1C)OC	CID:54631447	phase I
BRD-K80603893	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631448	phase I
BRD-K44562621	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3nc4ccccc4s3)ccc2OC[C@@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631449	phase I
BRD-K53155533	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@@H](C)N(C[C@@H]1C)S(C)(=O)=O	CID:54631450	phase I
BRD-K05581223	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631451	phase I
BRD-K17806071	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)Cc1cccnc1	CID:54631452	phase I
BRD-K96871778	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631453	phase I
BRD-K19019278	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631454	phase I
BRD-K41700431	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631455	phase I
BRD-K86522396	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cccc(OC)c3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)C1CCCCC1	CID:54631458	phase I
BRD-K93109423	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc(Oc4ccccc4)cc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631459	phase I
BRD-K37225168	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1cccnc1	CID:54631460	phase I
BRD-K40410846	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3OC)cc2OC[C@@H](C)N(Cc2ccccc2C(O)=O)C[C@H]1C	CID:54631461	phase I
BRD-K58731341	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1ccccc1F	CID:54631462	phase I
BRD-K35965314	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cc(on3)-c3ccccc3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631463	phase I
BRD-K85891179	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)CN2CCOCC2)c1	CID:54631464	phase I
BRD-K19340473	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631465	phase I
BRD-K12089955	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631466	phase I
BRD-K48662018	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@H](C)NC[C@H]1C	CID:54631467	phase I
BRD-K32602441	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631468	phase I
BRD-K83694683	CCCNC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631469	phase I
BRD-K52564648	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54631470	phase I
BRD-K22583762	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631471	phase I
BRD-K98626176	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3Cl)cc2OC[C@H](C)NC[C@H]1C	CID:54631472	phase I
BRD-K09411281	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631473	phase I
BRD-K58499277	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@H](C)N(C[C@H]1C)S(C)(=O)=O	CID:54631474	phase I
BRD-K17134074	CCCC(=O)Nc1ccc2OC[C@@H](C)N(CC3CCCC3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631475	phase I
BRD-K91969329	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)cc2OC[C@H](C)NC[C@H]1C	CID:54631476	phase I
BRD-K15695045	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(CC2CCOCC2)C[C@H]1C	CID:54631477	phase I
BRD-K65127260	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)NC[C@H]1C	CID:54631480	phase I
BRD-K27424042	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3nc4ccccc4s3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631481	phase I
BRD-K31392657	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccc(F)cc1	CID:54631482	phase I
BRD-K57375725	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631483	phase I
BRD-K17157530	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54631484	phase I
BRD-K74378303	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631485	phase I
BRD-K31163805	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)C1CCOCC1	CID:54631486	phase I
BRD-K47501069	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631487	phase I
BRD-K35727710	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)C1CCOCC1	CID:54631488	phase I
BRD-K98194519	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631489	phase I
BRD-K03276924	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(Cc2ccc(OC)cc2)C[C@@H]1C	CID:54631490	phase I
BRD-K24821098	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631491	phase I
BRD-K87410008	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc(cc3)C(F)(F)F)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631492	phase I
BRD-K39435863	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccc(F)cc1	CID:54631493	phase I
BRD-K90947365	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631494	phase I
BRD-K60826706	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54631495	phase I
BRD-K54003568	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cc(C)on3)cc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)c1ccc(F)cc1	CID:54631496	phase I
BRD-K33368990	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631497	phase I
BRD-K74345748	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631498	phase I
BRD-K26507936	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631499	phase I
BRD-K13324372	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccc(F)c3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631500	phase I
BRD-K80472474	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(CC2CCOCC2)C[C@@H]1C	CID:54631501	phase I
BRD-K79793338	CCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631502	phase I
BRD-K28021369	CCCNC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631503	phase I
BRD-K36424250	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54631504	phase I
BRD-K18097652	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)C1CCOCC1	CID:54631505	phase I
BRD-K96077293	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(Cc2ccc(OC)cc2)C[C@H]1C	CID:54631506	phase I
BRD-K84516003	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631507	phase I
BRD-K82599388	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631508	phase I
BRD-K36144252	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)NC[C@H]1C	CID:54631509	phase I
BRD-K88074877	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631510	phase I
BRD-K58733842	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631511	phase I
BRD-K27788917	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631512	phase I
BRD-K40676967	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cccnc3)cc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631513	phase I
BRD-K09453969	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631514	phase I
BRD-K89304341	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631515	phase I
BRD-K02653676	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H](C)NC[C@H]1C	CID:54631516	phase I
BRD-K28871766	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631517	phase I
BRD-K94669078	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3c(C)noc3C)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631518	phase I
BRD-K69573138	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631519	phase I
BRD-K31846842	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1ccccc1OC	CID:54631520	phase I
BRD-K12019169	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@@H]1C)OC	CID:54631521	phase I
BRD-K58743986	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3C)ccc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)c1ccccc1	CID:54631522	phase I
BRD-K42831041	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631523	phase I
BRD-K55381473	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3Cl)ccc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)CC(F)(F)F	CID:54631524	phase I
BRD-K28831272	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(CC2CCOCC2)C[C@H]1C	CID:54631525	phase I
BRD-K80890401	CCCNC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H]1C)OC	CID:54631526	phase I
BRD-K20107219	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631527	phase I
BRD-K24927839	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631528	phase I
BRD-K47994485	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(OC)cc3)ccc2OC[C@@H](C)N(Cc2cc(F)ccc2F)C[C@H]1C	CID:54631529	phase I
BRD-K98997045	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2cc(F)ccc2F)C[C@H]1C	CID:54631530	phase I
BRD-K00816633	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631531	phase I
BRD-K83121797	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)CC(F)(F)F	CID:54631532	phase I
BRD-K39878860	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54631533	phase I
BRD-K09366813	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631534	phase I
BRD-K86107831	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@@H]1C)OC	CID:54631535	phase I
BRD-K72241566	CCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631536	phase I
BRD-K73474555	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1ccc(F)cc1	CID:54631537	phase I
BRD-K96745884	CCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)CC	CID:54631538	phase I
BRD-K50755896	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54631539	phase I
BRD-K08570368	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3Cl)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631540	phase I
BRD-K00549770	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631541	phase I
BRD-K21305994	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631542	phase I
BRD-K80932888	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631543	phase I
BRD-K91665395	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631544	phase I
BRD-K70459579	CO[C@@H]1CN(C)C(=O)c2ccc(N)cc2OC[C@@H](C)NC[C@H]1C	CID:54631545	phase I
BRD-K70751797	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631546	phase I
BRD-K51592421	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631547	phase I
BRD-K53394241	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631548	phase I
BRD-K97727749	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631549	phase I
BRD-K62214646	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc4OCOc4c3)cc2OC[C@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631550	phase I
BRD-K10774870	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631551	phase I
BRD-K15172981	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54631552	phase I
BRD-K83756286	CCCNC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1F	CID:54631553	phase I
BRD-K82869179	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC3CCCCC3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631554	phase I
BRD-K22356946	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631555	phase I
BRD-K52812196	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc(cc3)C(F)(F)F)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631556	phase I
BRD-K88022263	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631557	phase I
BRD-K68903590	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)Cc1cccnc1	CID:54631558	phase I
BRD-K87851508	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@@H]1C)OC	CID:54631559	phase I
BRD-K71857815	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631560	phase I
BRD-K26319806	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54631561	phase I
BRD-K66533845	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631562	phase I
BRD-K40840224	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2cc(F)ccc2F)C[C@H]1C	CID:54631563	phase I
BRD-K44980533	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631564	phase I
BRD-K56004278	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cnccn3)ccc2OC[C@@H]1C)OC	CID:54631565	phase I
BRD-K69589246	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631566	phase I
BRD-K32992890	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54631567	phase I
BRD-K48327915	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(C[C@H]1C)C(=O)Cc1ccccn1	CID:54631568	phase I
BRD-K03779476	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54631569	phase I
BRD-K64778483	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)Cc1ccccn1	CID:54631570	phase I
BRD-K91721610	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54631571	phase I
BRD-K03438483	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631572	phase I
BRD-K24562909	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccc2OCOc2c1	CID:54631573	phase I
BRD-K14958998	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)N(Cc2nccs2)C[C@H]1C	CID:54631574	phase I
BRD-K46980879	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631575	phase I
BRD-K25198488	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631576	phase I
BRD-K85672685	CCCC(=O)Nc1ccc2OC[C@H](C)N(CC3CCCC3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631577	phase I
BRD-K66755238	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631578	phase I
BRD-K20763958	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631579	phase I
BRD-K95786246	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631580	phase I
BRD-K52124071	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3Cl)cc2OC[C@@H](C)NC[C@H]1C	CID:54631581	phase I
BRD-K38889985	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631582	phase I
BRD-K13759728	CCCNC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H]1C)OC	CID:54631583	phase I
BRD-K58590337	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2cc(F)ccc2F)C[C@H]1C	CID:54631584	phase I
BRD-K88352433	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631585	phase I
BRD-K25481209	CCCC(=O)Nc1ccc2OC[C@H](C)N(CC3CCCC3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631586	phase I
BRD-K27161788	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631587	phase I
BRD-K32654925	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc(F)cc3)ccc2OC[C@@H](C)N(Cc2cocn2)C[C@@H]1C	CID:54631588	phase I
BRD-K14123146	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631589	phase I
BRD-K94206926	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3c(C)noc3C)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631590	phase I
BRD-K34766381	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccc(C)cc3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54631591	phase I
BRD-K39379309	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631592	phase I
BRD-K74711277	CCCNC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H]1C)OC	CID:54631593	phase I
BRD-K57792211	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cn(C)cn3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54631594	phase I
BRD-K33504592	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccc(F)cc1	CID:54631595	phase I
BRD-K85667213	CCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccncc3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631596	phase I
BRD-K56219224	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@@H]1C)OC	CID:54631597	phase I
BRD-K14496573	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631598	phase I
BRD-K69837023	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H]1C)OC	CID:54631599	phase I
BRD-K17122162	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H]1C)OC	CID:54631600	phase I
BRD-K59536184	CCCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631601	phase I
BRD-K39056847	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631602	phase I
BRD-K95246884	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631603	phase I
BRD-K37760698	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631604	phase I
BRD-K49473389	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631605	phase I
BRD-K95371508	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccccc1	CID:54631606	phase I
BRD-K81606899	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631607	phase I
BRD-K00262440	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631608	phase I
BRD-K49014970	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@H](C)NC[C@H]1C	CID:54631609	phase I
BRD-K69021148	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@@H]1C	CID:54631610	phase I
BRD-K53290343	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631611	phase I
BRD-K52838656	CCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@H]1C)OC	CID:54631612	phase I
BRD-K11158154	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631613	phase I
BRD-K53980138	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(Cc2ccccc2OC)C[C@@H]1C	CID:54631614	phase I
BRD-K38304019	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631615	phase I
BRD-K10081616	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccc1F	CID:54631616	phase I
BRD-K32209551	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54631617	phase I
BRD-K39659850	CCCC(=O)Nc1ccc2c(OC[C@@H](C)NC[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631618	phase I
BRD-K65342196	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54631619	phase I
BRD-K62185604	CCCC(=O)Nc1ccc2c(OC[C@@H](C)NC[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631620	phase I
BRD-K69310574	CCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccncc3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631621	phase I
BRD-K92818291	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54631622	phase I
BRD-K28777623	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631623	phase I
BRD-K61268714	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccccc1F	CID:54631624	phase I
BRD-K07197565	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccnc3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631625	phase I
BRD-K88959773	CCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@H]1C)OC	CID:54631626	phase I
BRD-K12882397	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631627	phase I
BRD-K59757264	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccc1F	CID:54631628	phase I
BRD-K64630692	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631629	phase I
BRD-K61998593	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccc1	CID:54631630	phase I
BRD-K69420053	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631631	phase I
BRD-K39352275	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631632	phase I
BRD-K37838939	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(cc3)-c3ccccc3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631633	phase I
BRD-K51328581	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631634	phase I
BRD-K33689388	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@@H]1C)OC	CID:54631635	phase I
BRD-K25525438	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccccc1	CID:54631636	phase I
BRD-K45174347	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@@H]1C)OC	CID:54631637	phase I
BRD-K97986353	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@H]1C)OC	CID:54631638	phase I
BRD-K87175237	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)C1CCC1	CID:54631639	phase I
BRD-K36951400	CCCNC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@H]1C)OC	CID:54631640	phase I
BRD-K03891150	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@@H]1C)OC	CID:54631641	phase I
BRD-K60237462	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccnc3)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631642	phase I
BRD-K02675466	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631643	phase I
BRD-K28862419	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(cc3)-c3ccccc3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631644	phase I
BRD-K39036510	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54631645	phase I
BRD-K38320477	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)NC[C@H]1C	CID:54631646	phase I
BRD-K50819157	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(Cc2ccccc2OC)C[C@H]1C	CID:54631647	phase I
BRD-K32380790	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631648	phase I
BRD-K69414416	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631649	phase I
BRD-K07275921	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631650	phase I
BRD-K33635485	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(CC3CC3)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631651	phase I
BRD-K87687716	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@H](C)NC[C@H]1C	CID:54631652	phase I
BRD-K08210330	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccno3)ccc2OC[C@H](C)N(C[C@H]1C)S(C)(=O)=O	CID:54631653	phase I
BRD-K46396728	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)C2CCOCC2)c1	CID:54631654	phase I
BRD-K84651951	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)C3CCCCC3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631655	phase I
BRD-K38561684	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631656	phase I
BRD-K54145771	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631657	phase I
BRD-K86741607	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631658	phase I
BRD-K36018407	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@H]1C)OC	CID:54631659	phase I
BRD-K03180599	CCCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631660	phase I
BRD-K33961995	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631661	phase I
BRD-K21179706	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631662	phase I
BRD-K76472157	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccnc3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631663	phase I
BRD-K88671928	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631664	phase I
BRD-K63458711	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631665	phase I
BRD-K20754058	CCCC(=O)Nc1ccc2OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631666	phase I
BRD-K94889220	COCC(=O)Nc1ccc2c(OC[C@H](C)N(CC3CC3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631667	phase I
BRD-K08521815	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631668	phase I
BRD-K03142004	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CN1CCOCC1	CID:54631669	phase I
BRD-K77966217	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(Cc2cccnc2)C[C@H]1C	CID:54631670	phase I
BRD-K38557047	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631671	phase I
BRD-K97359152	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631672	phase I
BRD-K92573321	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)C1CCC1	CID:54631673	phase I
BRD-K59550348	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631674	phase I
BRD-K39158620	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(CCC(F)(F)F)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631675	phase I
BRD-K01547088	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631676	phase I
BRD-K86888602	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631677	phase I
BRD-K62748060	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(Cc2ccccc2OC)C[C@@H]1C	CID:54631678	phase I
BRD-K39703302	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631679	phase I
BRD-K60778274	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)C2CCOCC2)c1	CID:54631680	phase I
BRD-K61404768	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631681	phase I
BRD-K95489112	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccccc1F	CID:54631682	phase I
BRD-K50008654	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(CCC(F)(F)F)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631683	phase I
BRD-K11156132	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631686	phase I
BRD-K73555595	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631687	phase I
BRD-K68236123	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC3CCCCC3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631688	phase I
BRD-K49215584	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@H](C)NC[C@H]1C	CID:54631689	phase I
BRD-K94116832	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54631690	phase I
BRD-K70260471	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3cccnc3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631691	phase I
BRD-K88404561	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3ccc(F)cc3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631692	phase I
BRD-K98950492	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccccc1	CID:54631693	phase I
BRD-K68921379	COCC(=O)Nc1ccc2c(OC[C@H](C)N(CC3CC3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631694	phase I
BRD-K67322403	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631695	phase I
BRD-K73141149	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@H]1C)OC	CID:54631696	phase I
BRD-K11194815	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631697	phase I
BRD-K72993421	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@H]1C)OC	CID:54631698	phase I
BRD-K74817145	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54631699	phase I
BRD-K60286124	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631700	phase I
BRD-K18350116	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@H]1C)OC	CID:54631701	phase I
BRD-K87643614	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@H](C)N(Cc2ccccc2F)C[C@@H]1C	CID:54631702	phase I
BRD-K20741178	CCCNC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@@H]1C)OC	CID:54631703	phase I
BRD-K01624114	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H]1C)OC	CID:54631704	phase I
BRD-K51052187	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54631705	phase I
BRD-K31716313	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(Cc2ccccc2OC)C[C@H]1C	CID:54631708	phase I
BRD-K33324635	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631709	phase I
BRD-K02541615	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@@H]1C)OC	CID:54631710	phase I
BRD-K97657359	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631711	phase I
BRD-K91922990	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631712	phase I
BRD-K14378954	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@@H]1C)OC	CID:54631713	phase I
BRD-K06651637	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631714	phase I
BRD-K09700964	CCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@@H]1C)OC	CID:54631715	phase I
BRD-K07237640	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H]1C)OC	CID:54631716	phase I
BRD-K58300499	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)C2CCOCC2)c1	CID:54631717	phase I
BRD-K94198920	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@H]1C)OC	CID:54631718	phase I
BRD-K75985729	CCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@H]1C)OC	CID:54631719	phase I
BRD-K25249292	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccccc1F	CID:54631720	phase I
BRD-K21968411	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cc(C)on3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)C1CCC1	CID:54631721	phase I
BRD-K79157597	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631722	phase I
BRD-K24196267	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631723	phase I
BRD-K33258193	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@@H]1C	CID:54631724	phase I
BRD-K18406496	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3ccc(F)cc3)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631725	phase I
BRD-K69293497	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)C1CCC1	CID:54631726	phase I
BRD-K73898073	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(Cc2ccccc2OC)C[C@H]1C	CID:54631727	phase I
BRD-K87854506	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631728	phase I
BRD-K41641829	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631729	phase I
BRD-K43571148	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)C2CCOCC2)c1	CID:54631730	phase I
BRD-K41539628	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC3CCCCC3)cc2OC[C@@H](C)N(CC2CCOCC2)C[C@H]1C	CID:54631731	phase I
BRD-K49430514	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631732	phase I
BRD-K11458523	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)CN1CCOCC1	CID:54631733	phase I
BRD-K73504196	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631734	phase I
BRD-K06475386	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631735	phase I
BRD-K60149889	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cccc(OC)c3)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631736	phase I
BRD-K59291587	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631737	phase I
BRD-K16506419	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631738	phase I
BRD-K92942746	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631739	phase I
BRD-K51147721	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)CN1CCOCC1	CID:54631740	phase I
BRD-K29635534	CCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccncc3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631741	phase I
BRD-K75381775	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631742	phase I
BRD-K84702181	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631743	phase I
BRD-K03046744	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(Cc2cccnc2)C[C@H]1C	CID:54631744	phase I
BRD-K49956785	CCCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3nccs3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631745	phase I
BRD-K39906469	CCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccncc3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631746	phase I
BRD-K32665240	CCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccncc3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631747	phase I
BRD-K67786373	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631748	phase I
BRD-K70318404	CCCC(=O)Nc1ccc2c(OC[C@H](C)NC[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631749	phase I
BRD-K82803470	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631750	phase I
BRD-K38467418	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631751	phase I
BRD-K28256231	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54631752	phase I
BRD-K29324759	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@H]1C)OC	CID:54631753	phase I
BRD-K16752930	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631754	phase I
BRD-K99104612	CCC(=O)Nc1ccc2c(OC[C@H](C)N(CCc3ccccc3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631755	phase I
BRD-K68955961	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(Cc2cccnc2)C[C@@H]1C	CID:54631756	phase I
BRD-K35414268	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)NC[C@H]1C	CID:54631757	phase I
BRD-K15687395	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@@H]1C)OC	CID:54631758	phase I
BRD-K88762178	CCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccncc3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631759	phase I
BRD-K69962604	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)C1CCC1	CID:54631760	phase I
BRD-K30836174	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)CN1CCOCC1	CID:54631761	phase I
BRD-K19223413	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@@H]1C)OC	CID:54631762	phase I
BRD-K61164776	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H](C)NC[C@H]1C	CID:54631763	phase I
BRD-K34758135	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631764	phase I
BRD-K24779930	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccccc1	CID:54631765	phase I
BRD-K02401733	CCCC(=O)Nc1ccc2c(OC[C@@H](C)NC[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631766	phase I
BRD-K66960754	CCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@H]1C)OC	CID:54631767	phase I
BRD-K90960272	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(Cc2cccnc2)C[C@@H]1C	CID:54631768	phase I
BRD-K79719155	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3ccc(F)cc3)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631769	phase I
BRD-K01373529	CCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccncc3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631770	phase I
BRD-K43615608	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631771	phase I
BRD-K38547930	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@H]1C)OC	CID:54631772	phase I
BRD-K43717413	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H](C)NC[C@@H]1C	CID:54631773	phase I
BRD-K19657374	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631774	phase I
BRD-K93744771	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631775	phase I
BRD-K91674938	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631776	phase I
BRD-K50608366	CCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@@H]1C)OC	CID:54631777	phase I
BRD-K74506609	CCCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccc3C(O)=O)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631778	phase I
BRD-K97766167	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631779	phase I
BRD-K43744546	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccc1	CID:54631780	phase I
BRD-K67839548	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(CCC(F)(F)F)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631781	phase I
BRD-K23674983	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631782	phase I
BRD-K63484733	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(CCC(F)(F)F)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631783	phase I
BRD-K26857129	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54631784	phase I
BRD-K18383512	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(CC3CC3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631785	phase I
BRD-K28377322	CCCNC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@@H]1C)OC	CID:54631786	phase I
BRD-K49354529	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCOCC3)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1ccccc1	CID:54631787	phase I
BRD-K94579454	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631788	phase I
BRD-K15639930	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631789	phase I
BRD-K05156496	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631790	phase I
BRD-K18153171	CCCNC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@H]1C)OC	CID:54631791	phase I
BRD-K05214965	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631792	phase I
BRD-K18817373	CCCNC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@@H]1C)OC	CID:54631793	phase I
BRD-K04566325	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631794	phase I
BRD-K22451143	CCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2OC[C@@H]1C)OC	CID:54631795	phase I
BRD-K05398363	CCCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3nccs3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631796	phase I
BRD-K96611378	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H](C)NC[C@H]1C	CID:54631797	phase I
BRD-K13418716	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(CC3CC3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631798	phase I
BRD-K86719628	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H]1C)OC	CID:54631799	phase I
BRD-K50805111	CCC(=O)Nc1ccc2c(OC[C@@H](C)N(CCc3ccccc3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631800	phase I
BRD-K81974123	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@@H]1C)OC	CID:54631801	phase I
BRD-K66147676	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631802	phase I
BRD-K73969578	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@H]1C)OC	CID:54631803	phase I
BRD-K51538472	COCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631804	phase I
BRD-K76527508	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@H]1C)OC	CID:54631805	phase I
BRD-K20757362	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3cccnc3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631806	phase I
BRD-K09260588	CCC(=O)Nc1ccc2c(OC[C@@H](C)N(CCc3ccccc3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631807	phase I
BRD-K83251511	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(Cc3cccnc3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631808	phase I
BRD-K53923842	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631809	phase I
BRD-K58196326	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631810	phase I
BRD-K49166646	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(cc3)-c3ccccc3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631811	phase I
BRD-K02003138	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631812	phase I
BRD-K76293253	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631813	phase I
BRD-K93247546	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@@H]1C)OC	CID:54631814	phase I
BRD-K48603187	CCC(=O)Nc1ccc2c(OC[C@H](C)N(CCc3ccccc3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631815	phase I
BRD-K75486920	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(Cc2cccnc2)C[C@H]1C	CID:54631816	phase I
BRD-K60413918	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631817	phase I
BRD-K41042783	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@H]1C)OC	CID:54631818	phase I
BRD-K41957723	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(CCC(F)(F)F)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631819	phase I
BRD-K37779687	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@@H]1C	CID:54631820	phase I
BRD-K94223259	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631821	phase I
BRD-K80843514	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631822	phase I
BRD-K79027750	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H](C)NC[C@H]1C	CID:54631823	phase I
BRD-K11901011	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1cnccn1	CID:54631824	phase I
BRD-K95722922	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631825	phase I
BRD-K04772033	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H]1C)OC	CID:54631826	phase I
BRD-K10864752	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(Cc2ccccc2OC)C[C@@H]1C	CID:54631827	phase I
BRD-K99515159	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)C2CCOCC2)c1	CID:54631828	phase I
BRD-K81403739	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631829	phase I
BRD-K35039537	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccno3)ccc2OC[C@H](C)N(C[C@@H]1C)S(C)(=O)=O	CID:54631830	phase I
BRD-K07918661	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631831	phase I
BRD-K31207674	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54631832	phase I
BRD-K87269491	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(Cc2cncnc2)C[C@H]1C	CID:54631833	phase I
BRD-K41023039	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631834	phase I
BRD-K71520313	CCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccncc3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631835	phase I
BRD-K68057497	CCCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631836	phase I
BRD-K85058337	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)CN1CCOCC1	CID:54631837	phase I
BRD-K06723172	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631838	phase I
BRD-K67660075	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@H]1C)OC	CID:54631839	phase I
BRD-K42397226	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccn3)cc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54631840	phase I
BRD-K82772827	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631841	phase I
BRD-K54543575	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccc4OCOc4c3)ccc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631842	phase I
BRD-K98793371	CCCC(=O)Nc1ccc2OC[C@H](C)N(Cc3nccs3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631843	phase I
BRD-K55432508	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631844	phase I
BRD-K57616212	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H]1C)OC	CID:54631845	phase I
BRD-K87300242	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631846	phase I
BRD-K28489983	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@H]1C)OC	CID:54631847	phase I
BRD-K24269428	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631848	phase I
BRD-K95515654	CCCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631849	phase I
BRD-K25196723	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)C1CCC1	CID:54631850	phase I
BRD-K53101279	CCCC(=O)Nc1ccc2c(OC[C@H](C)NC[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631851	phase I
BRD-K66850406	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccno3)ccc2OC[C@@H](C)N(C[C@H]1C)S(C)(=O)=O	CID:54631852	phase I
BRD-K34982474	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)C1CCC1	CID:54631853	phase I
BRD-K20091307	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccno3)ccc2OC[C@@H](C)N(C[C@H]1C)S(C)(=O)=O	CID:54631854	phase I
BRD-K25097708	CCCC(=O)Nc1ccc2OC[C@H](C)N(Cc3nccs3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631855	phase I
BRD-K24685884	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccccc1F	CID:54631856	phase I
BRD-K56990873	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3ccc(F)cc3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631857	phase I
BRD-K84003657	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccno3)ccc2OC[C@@H](C)N(C[C@@H]1C)S(C)(=O)=O	CID:54631858	phase I
BRD-K82644788	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(CC3CC3)C[C@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631859	phase I
BRD-K88809956	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@H](C)NC[C@@H]1C	CID:54631860	phase I
BRD-K67718916	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631861	phase I
BRD-K52097822	CCCC(=O)Nc1ccc2OC[C@H](C)N(Cc3nccs3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631862	phase I
BRD-K08080638	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@H](C)NC[C@H]1C	CID:54631863	phase I
BRD-K30860517	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631864	phase I
BRD-K60050469	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631865	phase I
BRD-K87445129	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3cccc(OC)c3)ccc2OC[C@@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54631866	phase I
BRD-K49579550	CCCC(=O)Nc1ccc2OC[C@H](C)N(Cc3nccs3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631867	phase I
BRD-K94390294	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631868	phase I
BRD-K64478751	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631869	phase I
BRD-K34327142	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)C1CCC1	CID:54631870	phase I
BRD-K87972129	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631871	phase I
BRD-K22944564	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@H](C)NC[C@H]1C	CID:54631872	phase I
BRD-K55819735	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@H](C)NC[C@H]1C	CID:54631873	phase I
BRD-K78954318	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631874	phase I
BRD-K26555669	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631875	phase I
BRD-K57204946	CCCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631876	phase I
BRD-K69487032	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc2OC[C@@H]1C)OC	CID:54631877	phase I
BRD-K69441986	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccc(cc3)-c3ccccc3)cc2OC[C@H](C)NC[C@H]1C	CID:54631878	phase I
BRD-K32636206	CCCNC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3cccnc3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631879	phase I
BRD-K17891672	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(Cc2cccnc2)C[C@H]1C	CID:54631880	phase I
BRD-K67641117	CCCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631881	phase I
BRD-K64939621	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCC3)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631882	phase I
BRD-K80630466	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@H]1C)OC	CID:54631883	phase I
BRD-K78226445	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631884	phase I
BRD-K54972173	CCCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3nccs3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631885	phase I
BRD-K20089037	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54631886	phase I
BRD-K57060993	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(Cc2cccnc2)C[C@@H]1C	CID:54631887	phase I
BRD-K18310625	CCCNC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@H]1C)OC	CID:54631888	phase I
BRD-K41952303	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H]1C)OC	CID:54631889	phase I
BRD-K24390300	COCC(=O)Nc1ccc2c(OC[C@H](C)N(CC3CC3)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54631890	phase I
BRD-K90601358	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@@H](C)N(Cc2cocn2)C[C@H]1C	CID:54631891	phase I
BRD-K43013792	COCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccc1	CID:54631892	phase I
BRD-K27858373	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccc(OC)cc3)cc2OC[C@@H]1C)OC	CID:54631893	phase I
BRD-K27571934	CCCC(=O)Nc1ccc2OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC)C(=O)c1ccccn1	CID:54631894	phase I
BRD-K86715531	CCCNC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)C2CCOCC2)c1	CID:54631895	phase I
BRD-K79118917	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631896	phase I
BRD-K02817669	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3F)cc2OC[C@H]1C)OC	CID:54631897	phase I
BRD-K69367836	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54631898	phase I
BRD-K50981189	CO[C@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(Cc2ccccc2OC)C[C@@H]1C	CID:54631899	phase I
BRD-K43503317	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@H]1C)OC	CID:54631900	phase I
BRD-K59377703	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(Cc2cccnc2)C[C@@H]1C	CID:54631901	phase I
BRD-K13714335	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)C1CCC1	CID:54631902	phase I
BRD-K13498994	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CN1CCOCC1	CID:54631903	phase I
BRD-K44737208	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Cc3ccccc3)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1ccccc1F	CID:54631904	phase I
BRD-K08971733	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3OC)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631905	phase I
BRD-K48860322	CCC(=O)Nc1ccc2c(OC[C@@H](C)N(CCc3ccccc3)C[C@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631906	phase I
BRD-K82710433	CCC(=O)Nc1ccc2c(OC[C@H](C)N(CCc3ccccc3)C[C@@H](C)[C@H](CN(C)C2=O)OC)c1	CID:54631907	phase I
BRD-K28431554	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)CN(C)C)c1	CID:54631908	phase I
BRD-K82447793	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccccc3OC)cc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54631909	phase I
BRD-K89697867	CCCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3nccs3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631910	phase I
BRD-K72872827	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3OC)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631911	phase I
BRD-K79106177	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631912	phase I
BRD-K69880993	CO[C@@H]1CN(C)C(=O)c2cc(NC(C)=O)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1cnccn1	CID:54631913	phase I
BRD-K22246751	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3ccccc3F)ccc2OC[C@@H]1C)OC	CID:54631914	phase I
BRD-K73324958	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1c(C)noc1C	CID:54631917	phase I
BRD-K74260403	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54631918	phase I
BRD-K31067719	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631919	phase I
BRD-K30803694	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631920	phase I
BRD-K52544910	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@@H](C)N(Cc2ccccn2)C[C@@H]1C	CID:54631921	phase I
BRD-K02061388	CCCNC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@@H]1C)OC	CID:54631922	phase I
BRD-K91188527	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)Cc1cccnc1	CID:54631923	phase I
BRD-K49810938	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54631924	phase I
BRD-K88085458	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3F)cc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631925	phase I
BRD-K99626027	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3cc(F)ccc3F)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631926	phase I
BRD-K93450738	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54631927	phase I
BRD-K72316999	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631928	phase I
BRD-K52880714	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)c2cccnc2)c1	CID:54631929	phase I
BRD-K61220066	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3cc(F)ccc3F)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631930	phase I
BRD-K83397037	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@H](C)NC[C@H]1C	CID:54631931	phase I
BRD-K31248348	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631932	phase I
BRD-K43048602	CCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@@H]1C)OC	CID:54631933	phase I
BRD-K16172779	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCCCC3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631934	phase I
BRD-K72360839	CCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)c2ccc(F)cc2)c1	CID:54631935	phase I
BRD-K59472190	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54631936	phase I
BRD-K59974052	CO[C@H]1CN(C)C(=O)c2ccc(cc2OC[C@H](C)NC[C@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54631939	phase I
BRD-K08006444	CCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@@H]1C)OC	CID:54631940	phase I
BRD-K27817945	CCCNC(=O)Nc1ccc2OC[C@@H](C)NC[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631941	phase I
BRD-K27292311	CO[C@@H]1CN(C)C(=O)c2ccc(cc2OC[C@@H](C)NC[C@@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54631942	phase I
BRD-K38092925	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(Cc2ccccc2)C[C@@H]1C	CID:54631943	phase I
BRD-K81140509	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3F)cc2OC[C@H](C)NC[C@H]1C	CID:54631944	phase I
BRD-K34385682	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(Cc2ccccc2)C[C@H]1C	CID:54631945	phase I
BRD-K42613785	CCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@H]1C)OC	CID:54631946	phase I
BRD-K48052985	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54631947	phase I
BRD-K95896215	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)Nc1c(C)noc1C	CID:54631948	phase I
BRD-K72232421	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54631949	phase I
BRD-K82176569	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H](C)N(Cc2cccnc2)C[C@H]1C	CID:54631950	phase I
BRD-K85588347	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54631951	phase I
BRD-K50673380	CCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)c2ccc(F)cc2)c1	CID:54631952	phase I
BRD-K18384660	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccno3)cc2OC[C@H](C)NC[C@@H]1C	CID:54631953	phase I
BRD-K83826057	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54631954	phase I
BRD-K65517548	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C)C[C@H]1C	CID:54631955	phase I
BRD-K28658046	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631956	phase I
BRD-K45115014	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H]1C)OC	CID:54631957	phase I
BRD-K98582396	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631958	phase I
BRD-K10762274	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631959	phase I
BRD-K68629330	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631960	phase I
BRD-K18321170	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54631961	phase I
BRD-K48545097	CCCNC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@H]1C)OC	CID:54631962	phase I
BRD-K02928994	CCCNC(=O)Nc1ccc2OC[C@H](C)NC[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631963	phase I
BRD-K22959724	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@@H]1C)OC	CID:54631964	phase I
BRD-K50408407	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3F)cc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631965	phase I
BRD-K87840555	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631966	phase I
BRD-K80412673	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54631967	phase I
BRD-K60602279	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54631968	phase I
BRD-K89284683	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(Cc2ccccc2)C[C@H]1C	CID:54631969	phase I
BRD-K70012251	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631970	phase I
BRD-K55637344	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631971	phase I
BRD-K19042305	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccn1	CID:54631972	phase I
BRD-K38681012	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54631973	phase I
BRD-K77719922	CO[C@H]1CN(C)C(=O)c2ccc(cc2OC[C@@H](C)NC[C@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54631974	phase I
BRD-K89479751	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54631975	phase I
BRD-K65900075	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@H](C)N(Cc2ccccn2)C[C@H]1C	CID:54631976	phase I
BRD-K55197905	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(Cc2ccccc2F)C[C@@H]1C	CID:54631977	phase I
BRD-K53914164	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3cc(F)ccc3F)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54631978	phase I
BRD-K49623506	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H]1C)OC	CID:54631979	phase I
BRD-K80503839	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@H]1C)OC	CID:54631980	phase I
BRD-K97116995	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631981	phase I
BRD-K36651002	CCCN1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@@H]1C)OC	CID:54631982	phase I
BRD-K87967185	CCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)c2ccc(F)cc2)c1	CID:54631983	phase I
BRD-K63841469	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)NC[C@H]1C	CID:54631984	phase I
BRD-K83426111	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54631985	phase I
BRD-K21747841	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54631986	phase I
BRD-K94385358	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H]1C)OC	CID:54631987	phase I
BRD-K32916048	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCCCC3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54631988	phase I
BRD-K78074929	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@H]1C	CID:54631989	phase I
BRD-K28810861	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54631990	phase I
BRD-K61596998	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54631991	phase I
BRD-K26929400	CCCNC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@H]1C)OC	CID:54631992	phase I
BRD-K82824976	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54631993	phase I
BRD-K86149851	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54631994	phase I
BRD-K29266727	CCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@@H]1C)OC	CID:54631995	phase I
BRD-K87408386	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54631996	phase I
BRD-K70860307	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54631997	phase I
BRD-K00346458	COCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54631998	phase I
BRD-K56603522	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54631999	phase I
BRD-K04443175	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)Nc1c(C)noc1C	CID:54632000	phase I
BRD-K48114548	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54632001	phase I
BRD-K91857575	CCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@@H]1C)OC	CID:54632002	phase I
BRD-K87976657	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54632003	phase I
BRD-K78970311	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54632004	phase I
BRD-K35089608	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54632005	phase I
BRD-K04251331	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccno3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54632006	phase I
BRD-K68320080	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54632007	phase I
BRD-K14460076	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54632008	phase I
BRD-K44097254	CCCNC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@@H]1C)OC	CID:54632009	phase I
BRD-K71205264	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632010	phase I
BRD-K12988428	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3F)cc2OC[C@H](C)NC[C@@H]1C	CID:54632011	phase I
BRD-K40724605	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54632012	phase I
BRD-K72795491	CCCC(=O)Nc1ccc2c(OC[C@H](C)NC[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54632013	phase I
BRD-K73290601	CCCNC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@H]1C)OC	CID:54632014	phase I
BRD-K40628295	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54632015	phase I
BRD-K84103449	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H]1C)OC	CID:54632016	phase I
BRD-K27411066	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@@H]1C	CID:54632017	phase I
BRD-K59746807	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54632018	phase I
BRD-K82462147	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54632019	phase I
BRD-K09303054	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@H](C)N(Cc2cccnc2)C[C@@H]1C	CID:54632020	phase I
BRD-K80059960	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632021	phase I
BRD-K63403474	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54632022	phase I
BRD-K31900068	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H]1C)OC	CID:54632023	phase I
BRD-K15719180	CCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@H]1C)OC	CID:54632024	phase I
BRD-K47724900	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2ccccc2F)C[C@@H]1C	CID:54632025	phase I
BRD-K71781760	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccccn1	CID:54632026	phase I
BRD-K89222788	CCCNC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@H]1C)OC	CID:54632027	phase I
BRD-K43188042	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54632028	phase I
BRD-K44579616	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54632029	phase I
BRD-K08720480	CCCNC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@@H]1C)OC	CID:54632030	phase I
BRD-K62199122	CO[C@H]1CN(C)C(=O)c2ccc(cc2OC[C@@H](C)NC[C@@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54632031	phase I
BRD-K64440942	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54632032	phase I
BRD-K93105623	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632033	phase I
BRD-K70068422	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54632034	phase I
BRD-K28646532	CCCNC(=O)Nc1ccc2OC[C@@H](C)NC[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632035	phase I
BRD-K85259624	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H]1C)OC	CID:54632036	phase I
BRD-K52353085	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54632037	phase I
BRD-K64428314	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54632038	phase I
BRD-K01626010	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@H](C)NC[C@H]1C	CID:54632039	phase I
BRD-K61586432	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C)C[C@@H]1C	CID:54632040	phase I
BRD-K71841447	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54632041	phase I
BRD-K46653995	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@H](C)NC[C@@H]1C	CID:54632042	phase I
BRD-K39662808	CCCNC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)CCC)ccc2OC[C@@H]1C)OC	CID:54632043	phase I
BRD-K07809895	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccno3)cc2OC[C@H](C)NC[C@H]1C	CID:54632044	phase I
BRD-K13633691	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C)C[C@H]1C	CID:54632045	phase I
BRD-K26298689	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)CC1CC1	CID:54632046	phase I
BRD-K75199888	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)Cc1cccnc1	CID:54632047	phase I
BRD-K07937631	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccno3)cc2OC[C@@H](C)NC[C@H]1C	CID:54632048	phase I
BRD-K17491544	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)Cc1cccnc1	CID:54632049	phase I
BRD-K62314156	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54632050	phase I
BRD-K71604153	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)NC[C@H]1C	CID:54632051	phase I
BRD-K93672121	CCCNC(=O)Nc1ccc2OC[C@H](C)NC[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632052	phase I
BRD-K67215210	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@H](C)NC[C@H]1C	CID:54632053	phase I
BRD-K73427206	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@@H](C)NC[C@H]1C	CID:54632054	phase I
BRD-K89998644	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54632055	phase I
BRD-K99880843	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(Cc2nccs2)C[C@H]1C	CID:54632056	phase I
BRD-K10838258	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54632057	phase I
BRD-K36296949	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)c2cccnc2)c1	CID:54632058	phase I
BRD-K98468968	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54632059	phase I
BRD-K40603797	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@H](C)N(C)C[C@H]1C	CID:54632060	phase I
BRD-K99567057	CCCN1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@@H]1C)OC	CID:54632061	phase I
BRD-K60272067	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54632062	phase I
BRD-K76257863	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@H](C)N(CC2CCCCC2)C[C@H]1C	CID:54632063	phase I
BRD-K82279920	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54632064	phase I
BRD-K37714126	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccn1	CID:54632065	phase I
BRD-K66401835	COCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54632066	phase I
BRD-K75867134	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54632067	phase I
BRD-K63651474	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)Cc1cccnc1	CID:54632068	phase I
BRD-K59314947	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632069	phase I
BRD-K98135954	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3ccno3)cc2OC[C@H](C)NC[C@@H]1C	CID:54632070	phase I
BRD-K68552135	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H]1C)OC	CID:54632071	phase I
BRD-K72051249	CO[C@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@H](C)N(C)C[C@@H]1C	CID:54632072	phase I
BRD-K99978152	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@H](C)NC[C@H]1C	CID:54632073	phase I
BRD-K07424227	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@H](C)N(Cc2ccccn2)C[C@@H]1C	CID:54632074	phase I
BRD-K47514459	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3cc(F)ccc3F)C[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632075	phase I
BRD-K38493271	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@@H](C)N(Cc2ccccn2)C[C@@H]1C	CID:54632076	phase I
BRD-K12896711	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@H](C)N(C)C[C@H]1C	CID:54632077	phase I
BRD-K65750227	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@H]1C	CID:54632078	phase I
BRD-K16942988	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(Cc2ccccc2)C[C@@H]1C	CID:54632079	phase I
BRD-K59904884	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632080	phase I
BRD-K10429990	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)Cc1cccnc1	CID:54632081	phase I
BRD-K59000636	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54632082	phase I
BRD-K43732469	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632083	phase I
BRD-K29004135	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632084	phase I
BRD-K13835847	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54632085	phase I
BRD-K28336972	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54632086	phase I
BRD-K73671483	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)c2cccnc2)c1	CID:54632087	phase I
BRD-K10701306	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3cc(F)ccc3F)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54632088	phase I
BRD-K91720591	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H]1C)OC	CID:54632089	phase I
BRD-K94766424	CCCNC(=O)Nc1ccc2OC[C@@H](C)NC[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54632090	phase I
BRD-K97749477	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H](C)N(CCc2ccccc2)C[C@H]1C	CID:54632091	phase I
BRD-K38311495	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632092	phase I
BRD-K61968247	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632093	phase I
BRD-K31613395	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54632094	phase I
BRD-K48415574	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2ccncc2)C[C@H]1C	CID:54632095	phase I
BRD-K10054282	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)Nc1c(C)noc1C	CID:54632096	phase I
BRD-K84210283	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCCCC3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632097	phase I
BRD-K15028327	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)CC(F)(F)F)cc2OC[C@H](C)N(C[C@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54632098	phase I
BRD-K24496965	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)Nc1c(C)noc1C	CID:54632099	phase I
BRD-K13591554	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2ccncc2)C[C@H]1C	CID:54632100	phase I
BRD-K21600166	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@H](C)N(Cc2nccs2)C[C@H]1C	CID:54632101	phase I
BRD-K76571344	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54632102	phase I
BRD-K93986444	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54632103	phase I
BRD-K68118564	CCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)c2ccc(F)cc2)c1	CID:54632104	phase I
BRD-K84432438	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54632105	phase I
BRD-K36054906	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)N(C[C@@H]1C)C(C)=O	CID:54632106	phase I
BRD-K13707774	CCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)c2ccc(F)cc2)c1	CID:54632107	phase I
BRD-K96345282	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@@H](C)N(C)C[C@H]1C	CID:54632108	phase I
BRD-K68441823	COCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54632109	phase I
BRD-K16158586	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3F)cc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632110	phase I
BRD-K29924325	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H]1C)OC	CID:54632111	phase I
BRD-K77402297	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632112	phase I
BRD-K58879212	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3cc(F)ccc3F)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632113	phase I
BRD-K62060607	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54632114	phase I
BRD-K52076988	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3F)cc2OC[C@@H](C)NC[C@H]1C	CID:54632115	phase I
BRD-K50984462	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632116	phase I
BRD-K40260510	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)c2cccnc2)c1	CID:54632117	phase I
BRD-K55730324	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632118	phase I
BRD-K37219781	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)NC[C@@H]1C	CID:54632119	phase I
BRD-K73307873	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3F)cc2OC[C@H](C)NC[C@H]1C	CID:54632120	phase I
BRD-K01405464	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)c1ccccn1	CID:54632121	phase I
BRD-K26663582	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2ccncc2)C[C@@H]1C	CID:54632122	phase I
BRD-K78913846	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54632123	phase I
BRD-K30750630	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@H](C)N(C)C[C@H]1C	CID:54632124	phase I
BRD-K46261417	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(Cc2nccs2)C[C@H]1C	CID:54632125	phase I
BRD-K62601469	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(Cc2ccccc2)C[C@@H]1C	CID:54632126	phase I
BRD-K47078472	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54632127	phase I
BRD-K05261220	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@H](C)NC[C@H]1C	CID:54632128	phase I
BRD-K54602409	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54632129	phase I
BRD-K86078446	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54632130	phase I
BRD-K89833114	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H](C)N(CCc2ccccc2)C[C@@H]1C	CID:54632131	phase I
BRD-K05432839	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54632132	phase I
BRD-K48528697	CO[C@@H]1CN(C)C(=O)c2ccc(cc2OC[C@H](C)NC[C@@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54632133	phase I
BRD-K63047641	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccccn1	CID:54632134	phase I
BRD-K05951707	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3ccccc3F)cc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54632135	phase I
BRD-K90610504	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)c1ccccn1	CID:54632136	phase I
BRD-K33530763	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54632137	phase I
BRD-K27803932	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54632138	phase I
BRD-K86631750	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54632139	phase I
BRD-K36908385	CCCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)c2cccnc2)c1	CID:54632140	phase I
BRD-K81545342	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632141	phase I
BRD-K89920769	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1c(C)noc1C	CID:54632142	phase I
BRD-K18345986	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3F)cc2OC[C@@H](C)NC[C@@H]1C	CID:54632143	phase I
BRD-K14263251	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@H](C)[C@@H](CN(C)C2=O)OC)C(=O)c2cccnc2)c1	CID:54632144	phase I
BRD-K08183383	CO[C@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3F)cc2OC[C@@H](C)NC[C@H]1C	CID:54632145	phase I
BRD-K68776823	CO[C@@H]1CN(C)C(=O)c2cc(NS(C)(=O)=O)ccc2OC[C@@H](C)N(C)C[C@H]1C	CID:54632146	phase I
BRD-K63921140	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@H]1C	CID:54632147	phase I
BRD-K05543852	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)NC[C@H]1C	CID:54632148	phase I
BRD-K71505729	CO[C@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(Cc2nccs2)C[C@@H]1C	CID:54632149	phase I
BRD-K06326887	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cc(F)ccc3F)ccc2OC[C@@H](C)NC[C@H]1C	CID:54632150	phase I
BRD-K13648511	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(Cc2ccccc2)C[C@@H]1C	CID:54632151	phase I
BRD-K46273627	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54632152	phase I
BRD-K39738296	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54632153	phase I
BRD-K98062520	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(Cc2ccccc2)C[C@H]1C	CID:54632154	phase I
BRD-K95814727	CO[C@@H]1CN(C)C(=O)c2ccc(cc2OC[C@@H](C)NC[C@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54632155	phase I
BRD-K40060962	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2ccncc2)C[C@H]1C	CID:54632156	phase I
BRD-K71550516	CCC(=O)Nc1ccc2OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC)C(=O)Nc1ccccc1F	CID:54632157	phase I
BRD-K49114771	COCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@H]1C)OC	CID:54632158	phase I
BRD-K49158673	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cccc(F)c3)cc2OC[C@@H](C)NC[C@H]1C	CID:54632159	phase I
BRD-K14558018	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3cccc(F)c3)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)Cc1cccnc1	CID:54632160	phase I
BRD-K74852367	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H]1C)OC	CID:54632161	phase I
BRD-K41703587	CO[C@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@H](C)N(Cc2ccccc2F)C[C@H]1C	CID:54632162	phase I
BRD-K96406750	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@@H](C)N(C)C[C@@H]1C	CID:54632163	phase I
BRD-K76510844	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@@H](C)N(CCC(F)(F)F)C[C@@H]1C	CID:54632164	phase I
BRD-K36415399	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(=O)Nc1c(C)noc1C	CID:54632165	phase I
BRD-K82825326	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H]1C)OC	CID:54632166	phase I
BRD-K72463020	COCC(=O)Nc1ccc2OC[C@H](C)N(Cc3cc(F)ccc3F)C[C@@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632167	phase I
BRD-K99950451	CCCNC(=O)Nc1ccc2OC[C@H](C)NC[C@H](C)[C@@H](CN(C)C(=O)c2c1)OC	CID:54632168	phase I
BRD-K36512157	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)CC(F)(F)F)cc2OC[C@@H](C)N(C[C@@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54632169	phase I
BRD-K64070950	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632170	phase I
BRD-K19455915	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)CC(F)(F)F)cc2OC[C@@H](C)N(C[C@@H]1C)S(=O)(=O)c1cn(C)cn1	CID:54632171	phase I
BRD-K37928755	CCCC(=O)Nc1ccc2c(OC[C@@H](C)N(Cc3ccccc3OC)C[C@@H](C)[C@@H](CN(C)C2=O)OC)c1	CID:54632172	phase I
BRD-K04371396	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54632173	phase I
BRD-K68687385	CCCN1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@H]1C)OC	CID:54632174	phase I
BRD-K96989541	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)NC(C)C)cc2OC[C@H](C)N(Cc2ccccn2)C[C@H]1C	CID:54632175	phase I
BRD-K90898708	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632176	phase I
BRD-K51179640	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@@H](C)N(Cc2ccccc2)C[C@H]1C	CID:54632177	phase I
BRD-K73478880	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCCCC3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632178	phase I
BRD-K51040159	CCS(=O)(=O)Nc1ccc2OC[C@@H](C)N(Cc3ccccn3)C[C@@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54632179	phase I
BRD-K24257383	CO[C@@H]1CN(C)C(=O)c2ccc(NC(C)=O)cc2OC[C@@H](C)N(Cc2ccc(cc2)-c2ccccn2)C[C@H]1C	CID:54632180	phase I
BRD-K53349319	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(CC2CC2)C[C@@H]1C	CID:54632181	phase I
BRD-K76403391	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632182	phase I
BRD-K21094215	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCOCC3)ccc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54632183	phase I
BRD-K43218507	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)NC[C@H]1C	CID:54632184	phase I
BRD-K77726270	CCS(=O)(=O)Nc1ccc2OC[C@H](C)N(Cc3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54632185	phase I
BRD-K37777176	COCC(=O)Nc1ccc2OC[C@@H](C)N(Cc3cc(F)ccc3F)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54632186	phase I
BRD-K60706752	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@H](C)N(CC2CC2)C[C@H]1C	CID:54632187	phase I
BRD-K97821886	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2ccncc2)C[C@@H]1C	CID:54632188	phase I
BRD-K17429946	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3cc(F)ccc3F)cc2OC[C@@H](C)N(C)C[C@H]1C	CID:54632189	phase I
BRD-K77629773	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)Nc1c(C)noc1C	CID:54632190	phase I
BRD-K10734177	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54632191	phase I
BRD-K72072435	CO[C@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@@H](C)N(C[C@H]1C)C(=O)NC(C)C	CID:54632192	phase I
BRD-K01317665	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54632193	phase I
BRD-K46005840	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@@H](C)N(C)C[C@H]1C	CID:54632194	phase I
BRD-K42393177	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)C3CC3)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54632195	phase I
BRD-K39805076	CCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@H]1C)OC	CID:54632196	phase I
BRD-K31112909	CCC(=O)Nc1ccc2c(OC[C@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)c2ccc(F)cc2)c1	CID:54632197	phase I
BRD-K03079643	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)c3ccccc3F)ccc2OC[C@@H](C)N(C[C@H]1C)S(C)(=O)=O	CID:54632198	phase I
BRD-K24506271	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54632199	phase I
BRD-K61756858	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H](C)N(C[C@H]1C)S(=O)(=O)c1cccc(C)c1	CID:54632200	phase I
BRD-K92209998	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3ccc(cc3)-c3ccccc3)ccc2OC[C@H]1C)OC	CID:54632201	phase I
BRD-K29532955	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)N(C[C@H]1C)C(C)=O	CID:54632202	phase I
BRD-K99136192	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@@H](C)NC[C@H]1C	CID:54632203	phase I
BRD-K04627808	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632204	phase I
BRD-K08159565	CO[C@@H]1CN(C)C(=O)c2ccc(NS(C)(=O)=O)cc2OC[C@@H](C)N(Cc2nccs2)C[C@H]1C	CID:54632205	phase I
BRD-K88352009	COCC(=O)N1C[C@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)Nc3cccc(F)c3)ccc2OC[C@H]1C)OC	CID:54632206	phase I
BRD-K64497523	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)c3ccc4OCOc4c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632207	phase I
BRD-K92096002	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)c3ccccc3F)ccc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54632208	phase I
BRD-K74294292	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2ccncc2)C[C@@H]1C	CID:54632209	phase I
BRD-K40240180	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)c3ccccc3C)cc2OC[C@H](C)N(C)C[C@@H]1C	CID:54632210	phase I
BRD-K09641927	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@@H]1C)OC	CID:54632211	phase I
BRD-K37457040	CCCN1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(NS(=O)(=O)c3cn(C)cn3)cc2OC[C@H]1C)OC	CID:54632212	phase I
BRD-K31682048	CO[C@@H]1CN(C)C(=O)c2ccc(cc2OC[C@H](C)NC[C@H]1C)NS(=O)(=O)c1cccc(Cl)c1	CID:54632213	phase I
BRD-K77888550	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54632214	phase I
BRD-K93369639	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)Cc3ccccc3)ccc2OC[C@H](C)NC[C@@H]1C	CID:54632215	phase I
BRD-K64023191	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCC3)cc2OC[C@@H](C)N(CC2CCCCC2)C[C@@H]1C	CID:54632216	phase I
BRD-K63366453	COCC(=O)N1C[C@@H](C)[C@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H]1C)OC	CID:54632217	phase I
BRD-K61344432	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@H](C)N(Cc2ccncc2)C[C@@H]1C	CID:54632218	phase I
BRD-K05275169	CCC(=O)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(NC(=O)c3ccccc3)cc2OC[C@H]1C)OC	CID:54632219	phase I
BRD-K03888308	CO[C@@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(OC)c3)ccc2OC[C@@H](C)N(CC2CC2)C[C@@H]1C	CID:54632220	phase I
BRD-K21285939	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@H](C)N(C[C@H]1C)C(C)=O	CID:54632221	phase I
BRD-K56150975	COCC(=O)Nc1ccc2c(OC[C@@H](C)N(C[C@@H](C)[C@@H](CN(C)C2=O)OC)C(=O)NC(C)C)c1	CID:54632222	phase I
BRD-K14255719	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cnccn3)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)Nc1ccccc1OC	CID:54632223	phase I
BRD-K39701065	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Cc3ccccc3)ccc2OC[C@@H](C)N(C[C@@H]1C)C(C)=O	CID:54632224	phase I
BRD-K54074847	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)C3CCCC3)cc2OC[C@@H](C)N(C[C@@H]1C)C(=O)CC1CC1	CID:54632225	phase I
BRD-K71877850	CO[C@@H]1CN(C)C(=O)c2cc(NS(=O)(=O)CC(F)(F)F)ccc2OC[C@H](C)N(C[C@@H]1C)C(=O)NC(C)C	CID:54632226	phase I
BRD-K43057855	COCC(=O)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2cc(NC(=O)c3cc(C)on3)ccc2OC[C@H]1C)OC	CID:54632227	phase I
BRD-K57140889	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)Nc3cccc(Cl)c3)ccc2OC[C@@H](C)NC[C@@H]1C	CID:54632228	phase I
BRD-K79992300	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)C3CC3)cc2OC[C@@H](C)N(Cc2ccncc2)C[C@H]1C	CID:54632229	phase I
BRD-K72464155	CO[C@H]1CN(C)C(=O)c2ccc(NC(=O)Nc3c(C)noc3C)cc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54632230	phase I
BRD-K14187559	CO[C@@H]1CN(C)C(=O)c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OC[C@@H](C)N(C[C@H]1C)C(=O)c1ccc2OCOc2c1	CID:54632474	phase I
BRD-K51626376	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)C3CCCCC3)ccc2OC[C@H](C)N(C[C@H]1C)C(=O)c1ccccc1	CID:54632493	phase I
BRD-K28080909	CO[C@@H]1CN(C)C(=O)c2ccc(NC(=O)c3cccc(OC)c3)cc2OC[C@@H](C)N(CC2CC2)C[C@H]1C	CID:54633555	phase I
BRD-K98645985	CO[C@H]1CN(C)C(=O)c2cc(NC(=O)NC(C)C)ccc2OC[C@H](C)N(Cc2ccc(cc2)-c2ccccn2)C[C@@H]1C	CID:54633693	phase I
BRD-K21001652	CCCC(=O)Nc1ccc2OC[C@H](C)N(Cc3ccc(cc3)-c3ccccn3)C[C@H](C)[C@H](CN(C)C(=O)c2c1)OC	CID:54636786	phase I
BRD-K39629581	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO)c4ccccc4	CID:54637640	phase I
BRD-K84749975	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO)c4ccccc4	CID:54637641	phase I
BRD-K83311395	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO)c4ccccc4	CID:54637642	phase I
BRD-K84691165	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO)c4ccccc4	CID:54637643	phase I
BRD-K04570341	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO)c4ccccc4	CID:54637644	phase I
BRD-K37847786	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO)c4ccccc4	CID:54637645	phase I
BRD-K84104483	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO)c4ccccc4	CID:54637646	phase I
BRD-K70433089	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637647	phase I
BRD-K17139610	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637648	phase I
BRD-K34922409	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637649	phase I
BRD-K91379182	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637650	phase I
BRD-K71204485	COc1ccccc1CN(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54637651	phase I
BRD-K90630790	COc1cccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54637652	phase I
BRD-K24167577	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54637653	phase I
BRD-K05519665	COc1cccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:54637654	phase I
BRD-K63832750	COc1cccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:54637655	phase I
BRD-K84596673	CC(C)COC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54637656	phase I
BRD-K28076694	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637657	phase I
BRD-K56962853	CC(C)COC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54637658	phase I
BRD-K62590938	CC(C)COC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54637659	phase I
BRD-K99224100	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637660	phase I
BRD-K88318034	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637661	phase I
BRD-K80211979	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637662	phase I
BRD-K54457715	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637663	phase I
BRD-K21852581	CO[C@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637664	phase I
BRD-K02475229	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637665	phase I
BRD-K32326107	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637666	phase I
BRD-K93738295	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637667	phase I
BRD-K39635970	CO[C@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637668	phase I
BRD-K06892639	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637669	phase I
BRD-K51643793	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637670	phase I
BRD-K56890651	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637671	phase I
BRD-K06725649	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:54637672	phase I
BRD-K55129824	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637673	phase I
BRD-K11468634	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637674	phase I
BRD-K40997335	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637675	phase I
BRD-K50347701	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637676	phase I
BRD-K19589763	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637677	phase I
BRD-K96804382	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637678	phase I
BRD-K42969667	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637679	phase I
BRD-K55943540	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637680	phase I
BRD-K91572503	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637681	phase I
BRD-K63494246	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637682	phase I
BRD-K51556413	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637683	phase I
BRD-K66442181	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637684	phase I
BRD-K18883945	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637685	phase I
BRD-K64169482	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637686	phase I
BRD-K48877010	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637687	phase I
BRD-K63424643	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637688	phase I
BRD-K00064877	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637689	phase I
BRD-K92441219	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637690	phase I
BRD-K50761336	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637691	phase I
BRD-K99191181	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637692	phase I
BRD-K00765103	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4ccccc4C1=O	CID:54637693	phase I
BRD-K11577165	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4ccccc4C1=O	CID:54637694	phase I
BRD-K97277752	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4ccccc4C1=O	CID:54637695	phase I
BRD-K67766243	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637696	phase I
BRD-K78822642	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637697	phase I
BRD-K01727336	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637698	phase I
BRD-K09526594	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637699	phase I
BRD-K96257627	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637700	phase I
BRD-K38517635	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637701	phase I
BRD-K45231555	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637702	phase I
BRD-K53285126	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637703	phase I
BRD-K10279767	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637704	phase I
BRD-K58719691	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637705	phase I
BRD-K34433706	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637706	phase I
BRD-K57552506	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637707	phase I
BRD-K89551576	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637708	phase I
BRD-K99638701	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637709	phase I
BRD-K42610174	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637710	phase I
BRD-K26626929	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637711	phase I
BRD-K72303429	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637712	phase I
BRD-K11022579	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4ccccc4C1=O	CID:54637713	phase I
BRD-K21317335	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4ccccc4C1=O	CID:54637714	phase I
BRD-K77791851	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4ccccc4C1=O	CID:54637715	phase I
BRD-K55293774	COc1ccc(CNC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54637716	phase I
BRD-K29987902	COc1ccc(CNC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54637717	phase I
BRD-K62975098	COc1ccc(CNC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54637718	phase I
BRD-K27872553	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637719	phase I
BRD-K45998529	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637720	phase I
BRD-K78542975	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637721	phase I
BRD-K24855614	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637722	phase I
BRD-K85332209	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637723	phase I
BRD-K85536714	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637724	phase I
BRD-K31975688	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637725	phase I
BRD-K40276799	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637726	phase I
BRD-K29381365	COc1ccccc1NC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54637727	phase I
BRD-K43556160	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54637728	phase I
BRD-K54618558	COc1ccccc1NC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54637729	phase I
BRD-K33116513	COc1ccccc1NC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54637730	phase I
BRD-K98005081	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:54637731	phase I
BRD-K33054146	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:54637732	phase I
BRD-K64701969	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:54637733	phase I
BRD-K53621751	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:54637734	phase I
BRD-K02653582	COc1ccc(CNC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45)cc1	CID:54637735	phase I
BRD-K27525788	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637738	phase I
BRD-K32559936	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637739	phase I
BRD-K57638192	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:54637740	phase I
BRD-K58925245	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:54637741	phase I
BRD-K01691627	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:54637742	phase I
BRD-K23731136	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:54637743	phase I
BRD-K34799054	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:54637744	phase I
BRD-K62561943	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:54637745	phase I
BRD-K80391949	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637746	phase I
BRD-K73942053	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637747	phase I
BRD-K47131467	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637748	phase I
BRD-K79652816	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637749	phase I
BRD-K49567165	COc1ccc(OC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54637752	phase I
BRD-K20255967	COc1ccc(OC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO)cc1	CID:54637753	phase I
BRD-K61963347	COc1ccc(OC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:54637754	phase I
BRD-K09424864	COc1ccc(OC(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:54637755	phase I
BRD-K31494307	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637756	phase I
BRD-K77608736	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637757	phase I
BRD-K60841303	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637758	phase I
BRD-K26425257	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637759	phase I
BRD-K66559265	CNC[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637760	phase I
BRD-K11171096	CNC[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54637761	phase I
BRD-K16741885	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637762	phase I
BRD-K56322026	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637763	phase I
BRD-K65752719	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637764	phase I
BRD-K75403700	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637765	phase I
BRD-K82909508	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:54637766	phase I
BRD-K02112931	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:54637767	phase I
BRD-K78300612	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:54637768	phase I
BRD-K50325283	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:54637769	phase I
BRD-K37398676	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637770	phase I
BRD-K10893406	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637771	phase I
BRD-K71532462	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637772	phase I
BRD-K00434250	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637773	phase I
BRD-K39696539	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637774	phase I
BRD-K93459801	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637775	phase I
BRD-K70377370	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637776	phase I
BRD-K15973523	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637777	phase I
BRD-K27718415	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637778	phase I
BRD-K99219003	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637779	phase I
BRD-K85957472	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637780	phase I
BRD-K89597637	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637781	phase I
BRD-K23871470	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637782	phase I
BRD-K66877406	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:54637783	phase I
BRD-K23373611	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637784	phase I
BRD-K26427778	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637785	phase I
BRD-K07613753	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637786	phase I
BRD-K22778679	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637787	phase I
BRD-K15389391	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637788	phase I
BRD-K63946052	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637789	phase I
BRD-K61190439	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637790	phase I
BRD-K81799166	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637791	phase I
BRD-K11556486	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637792	phase I
BRD-K11296387	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc3OCCCOc23)OCc4ccccc4-c5ccccc5C1=O	CID:54637793	phase I
BRD-K45713168	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4ccccc4-c5ccccc5C1=O	CID:54637794	phase I
BRD-K80342168	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc3OCCCOc23)OCc4ccccc4-c5ccccc5C1=O	CID:54637795	phase I
BRD-K95284932	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:54637796	phase I
BRD-K26545050	COc1ccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:54637797	phase I
BRD-K08105592	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:54637798	phase I
BRD-K99048249	COc1ccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:54637799	phase I
BRD-K08706435	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54637800	phase I
BRD-K95196306	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54637801	phase I
BRD-K88384060	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54637802	phase I
BRD-K09796735	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54637803	phase I
BRD-K91244634	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54637804	phase I
BRD-K63201679	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637805	phase I
BRD-K03706963	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637806	phase I
BRD-K56712828	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637807	phase I
BRD-K13060097	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637808	phase I
BRD-K24282403	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637809	phase I
BRD-K27452198	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637810	phase I
BRD-K99349510	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637811	phase I
BRD-K22324798	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637812	phase I
BRD-K29385065	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637813	phase I
BRD-K65968856	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637814	phase I
BRD-K94224651	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637815	phase I
BRD-K50342369	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637816	phase I
BRD-K38963656	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637817	phase I
BRD-K89502948	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:54637818	phase I
BRD-K90074540	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637819	phase I
BRD-K66771647	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637820	phase I
BRD-K84306552	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637821	phase I
BRD-K34347561	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637822	phase I
BRD-K46533463	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:54637823	phase I
BRD-K61873274	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:54637824	phase I
BRD-K76749891	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:54637825	phase I
BRD-K18244645	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:54637826	phase I
BRD-K81332205	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:54637827	phase I
BRD-K72095065	CCCN(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54637828	phase I
BRD-K08963966	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637829	phase I
BRD-K87748653	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637830	phase I
BRD-K40455893	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637831	phase I
BRD-K45892018	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:54637832	phase I
BRD-K44511222	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:54637833	phase I
BRD-K80094052	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:54637834	phase I
BRD-K92604082	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:54637835	phase I
BRD-K31487013	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:54637836	phase I
BRD-K37357048	COc1ccc(CNC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45)cc1	CID:54637839	phase I
BRD-K25385069	COc1ccc(CNC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45)cc1	CID:54637840	phase I
BRD-K63140065	COc1ccc(CNC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45)cc1	CID:54637841	phase I
BRD-K38663221	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637842	phase I
BRD-K23985677	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637843	phase I
BRD-K84475927	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637844	phase I
BRD-K91849632	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637845	phase I
BRD-K78122632	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:54637846	phase I
BRD-K21683946	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54637847	phase I
BRD-K33454337	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO	CID:54637848	phase I
BRD-K05690403	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:54637849	phase I
BRD-K51662742	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO	CID:54637850	phase I
BRD-K87311987	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637851	phase I
BRD-K85197047	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637854	phase I
BRD-K49111930	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637855	phase I
BRD-K39597586	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637856	phase I
BRD-K25420921	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:54637857	phase I
BRD-K06421369	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637858	phase I
BRD-K67374281	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637859	phase I
BRD-K56757089	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637860	phase I
BRD-K17903303	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637861	phase I
BRD-K36553386	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637862	phase I
BRD-K21209030	COc1cccc(CN(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@H](C)CO)c1	CID:54637863	phase I
BRD-K13587575	COc1cccc(CN(C)C[C@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:54637864	phase I
BRD-K38304289	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637865	phase I
BRD-K47612243	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637866	phase I
BRD-K72204100	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637867	phase I
BRD-K49921033	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:54637868	phase I
BRD-K53528245	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637869	phase I
BRD-K42902917	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637870	phase I
BRD-K32833573	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637871	phase I
BRD-K77381468	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54637872	phase I
BRD-K20251969	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637873	phase I
BRD-K79967274	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637874	phase I
BRD-K99985506	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637875	phase I
BRD-K81945689	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637876	phase I
BRD-K44021875	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637877	phase I
BRD-K65300017	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637878	phase I
BRD-K70202431	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637879	phase I
BRD-K15895141	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637880	phase I
BRD-K90028787	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637881	phase I
BRD-K55897144	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637882	phase I
BRD-K17263374	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637883	phase I
BRD-K23455135	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637884	phase I
BRD-K83147038	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@H](C)CO)n(C)c4ccccc34	CID:54637885	phase I
BRD-K04153348	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@H](C)CO)n(C)c4ccccc34	CID:54637886	phase I
BRD-K08750028	CC(C)COC(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@@H](C)CO)n(C)c4ccccc34	CID:54637887	phase I
BRD-K49860242	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@@H](C)CO)n(C)c4ccccc34	CID:54637888	phase I
BRD-K32532498	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637889	phase I
BRD-K12827775	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637890	phase I
BRD-K34412442	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637891	phase I
BRD-K31284555	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637892	phase I
BRD-K61819258	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:54637893	phase I
BRD-K07253943	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:54637894	phase I
BRD-K10682047	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:54637895	phase I
BRD-K80410762	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:54637896	phase I
BRD-K96538394	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637897	phase I
BRD-K71944426	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637898	phase I
BRD-K83266926	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637899	phase I
BRD-K59709493	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)CC2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637900	phase I
BRD-K71040278	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:54637901	phase I
BRD-K83547636	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:54637902	phase I
BRD-K43604368	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:54637903	phase I
BRD-K96688934	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:54637904	phase I
BRD-K28018597	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:54637905	phase I
BRD-K51712294	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637906	phase I
BRD-K46522835	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637907	phase I
BRD-K59453266	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637908	phase I
BRD-K62008506	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637909	phase I
BRD-K16399103	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637910	phase I
BRD-K35886478	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637911	phase I
BRD-K79027739	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637912	phase I
BRD-K37316418	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637913	phase I
BRD-K71195237	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637914	phase I
BRD-K15224350	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637915	phase I
BRD-K33303625	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637916	phase I
BRD-K39248781	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637917	phase I
BRD-K16256442	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637918	phase I
BRD-K94032641	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637919	phase I
BRD-K75308057	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637920	phase I
BRD-K47006988	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637921	phase I
BRD-K30347205	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637922	phase I
BRD-K34320757	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637923	phase I
BRD-K60019754	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637924	phase I
BRD-K75733071	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637925	phase I
BRD-K04669648	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637926	phase I
BRD-K65222708	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637927	phase I
BRD-K85359245	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637928	phase I
BRD-K71357056	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637929	phase I
BRD-K18304318	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637930	phase I
BRD-K85169571	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637931	phase I
BRD-K39063656	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637932	phase I
BRD-K85124606	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637933	phase I
BRD-K00478394	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637934	phase I
BRD-K72529818	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637935	phase I
BRD-K48575680	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637936	phase I
BRD-K08970510	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637937	phase I
BRD-K50404714	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637938	phase I
BRD-K50309272	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637939	phase I
BRD-K91133575	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54637940	phase I
BRD-K27951502	CC(C)OC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637941	phase I
BRD-K40507170	CC(C)OC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54637942	phase I
BRD-K51019170	CC(C)OC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637943	phase I
BRD-K40123785	CC(C)OC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54637944	phase I
BRD-K39768328	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637945	phase I
BRD-K18296113	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637946	phase I
BRD-K39412479	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637947	phase I
BRD-K30785989	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637948	phase I
BRD-K06401240	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637949	phase I
BRD-K21959862	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(O)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54637950	phase I
BRD-K02306470	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637951	phase I
BRD-K55880295	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637952	phase I
BRD-K93011030	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637953	phase I
BRD-K14228330	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637954	phase I
BRD-K05032830	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637955	phase I
BRD-K11112971	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637956	phase I
BRD-K17402942	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637957	phase I
BRD-K31933349	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637958	phase I
BRD-K58360282	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637959	phase I
BRD-K39006362	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637960	phase I
BRD-K35928056	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637961	phase I
BRD-K18306851	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637962	phase I
BRD-K54391669	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637963	phase I
BRD-K55667009	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637964	phase I
BRD-K85742570	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637965	phase I
BRD-K29035246	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637966	phase I
BRD-K57216724	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637967	phase I
BRD-K83335786	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637968	phase I
BRD-K51143622	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637969	phase I
BRD-K63631822	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637970	phase I
BRD-K58098983	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637971	phase I
BRD-K85258684	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637972	phase I
BRD-K18822535	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637973	phase I
BRD-K50195301	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637974	phase I
BRD-K05500678	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637975	phase I
BRD-K19054197	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637976	phase I
BRD-K26576471	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637977	phase I
BRD-K82083906	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:54637978	phase I
BRD-K69318356	CC(C)[C@H](C)NC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637979	phase I
BRD-K35189425	CC(C)[C@@H](C)NC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637980	phase I
BRD-K71710045	CC(C)[C@H](C)NC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54637981	phase I
BRD-K11031937	CC(C)[C@@H](C)NC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:54637982	phase I
BRD-K93657737	CC(C)[C@@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637983	phase I
BRD-K61929092	CC(C)[C@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@H](C)CO	CID:54637984	phase I
BRD-K35404971	CC(C)[C@@H](C)NC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:54637985	phase I
BRD-K21364577	CC(C)[C@H](C)NC(=O)N(C)C[C@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:54637986	phase I
BRD-K38865695	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637987	phase I
BRD-K41996639	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637988	phase I
BRD-K47036878	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:54637989	phase I
BRD-K27647724	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@H](C)CO)n(C)c5ccccc45)c1	CID:54637990	phase I
BRD-K11787592	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45)c1	CID:54637991	phase I
BRD-K22518694	COc1cccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c1	CID:54637992	phase I
BRD-K36314330	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c1	CID:54637993	phase I
BRD-K61113746	CNC[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@H](C)CO)n(C)c4ccccc34	CID:54637994	phase I
BRD-K61796480	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637995	phase I
BRD-K94161851	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637996	phase I
BRD-K83468907	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637997	phase I
BRD-K19275171	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54637998	phase I
BRD-K73824371	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54637999	phase I
BRD-K11517399	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54638000	phase I
BRD-K62951188	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54638001	phase I
BRD-K92730269	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:54638002	phase I
BRD-K64075070	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638003	phase I
BRD-K17910135	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638004	phase I
BRD-K51776699	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638005	phase I
BRD-K56883821	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638006	phase I
BRD-K32827537	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638007	phase I
BRD-K73658839	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54638008	phase I
BRD-K29427427	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54638009	phase I
BRD-K40141271	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54638010	phase I
BRD-K97448504	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:54638011	phase I
BRD-K00930335	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54638012	phase I
BRD-K16110862	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54638013	phase I
BRD-K79986209	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54638014	phase I
BRD-K42968051	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:54638015	phase I
BRD-K59324394	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54638016	phase I
BRD-K45571747	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54638017	phase I
BRD-K63591202	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54638018	phase I
BRD-K64127467	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:54638019	phase I
BRD-K18327813	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638020	phase I
BRD-K51574318	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638021	phase I
BRD-K05498469	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638022	phase I
BRD-K67123444	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54638023	phase I
BRD-K82621995	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54638024	phase I
BRD-K50665432	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54638025	phase I
BRD-K25473383	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)Cc2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:54638026	phase I
BRD-K35885715	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638027	phase I
BRD-K83033340	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638028	phase I
BRD-K56950264	C[C@@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638029	phase I
BRD-K13515789	C[C@H](CO)N1C[C@@H](C)[C@@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:54638030	phase I
BRD-K03013810	OC[C@H]1O[C@@H](CC(=O)Nc2ccccc2)CC[C@H]1NC(=O)C1CC1	CID:54638216	phase I
BRD-K91787616	OC[C@@H]1O[C@H](CC(=O)Nc2ccccc2)CC[C@@H]1NC(=O)C1CC1	CID:54638217	phase I
BRD-K16752617	OC[C@H]1O[C@H](CC(=O)Nc2ccccc2)CC[C@@H]1NC(=O)C1CC1	CID:54638218	phase I
BRD-K57166447	OC[C@@H]1O[C@@H](CC(=O)Nc2ccccc2)CC[C@H]1NC(=O)C1CC1	CID:54638219	phase I
BRD-K68870366	OC[C@H]1O[C@@H](CC(=O)Nc2ccccc2)CC[C@@H]1NC(=O)C1CC1	CID:54638220	phase I
BRD-K33891131	OC[C@@H]1O[C@H](CC(=O)Nc2ccccc2)CC[C@H]1NC(=O)C1CC1	CID:54638221	phase I
BRD-K17554130	COc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)NCCc2ccncc2)O[C@@H]1CO	CID:54638222	phase I
BRD-K99055802	COc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)NCCc2ccncc2)O[C@H]1CO	CID:54638223	phase I
BRD-K65395273	COc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)NCCc2ccncc2)O[C@@H]1CO	CID:54638224	phase I
BRD-K67780021	COc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)NCCc2ccncc2)O[C@H]1CO	CID:54638225	phase I
BRD-K75703168	COc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)NCCc2ccncc2)O[C@@H]1CO	CID:54638226	phase I
BRD-K16257721	COc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)NCCc2ccncc2)O[C@H]1CO	CID:54638227	phase I
BRD-K79997126	COc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)NCCc2ccncc2)O[C@@H]1CO	CID:54638228	phase I
BRD-K56904840	COc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)NCCc2ccncc2)O[C@H]1CO	CID:54638229	phase I
BRD-K41423295	N[C@@H]1CC[C@@H](CCn2cc(nn2)C2(O)CCCC2)O[C@H]1CO	CID:54638230	phase I
BRD-K25427024	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)C=C[C@H]1NC(=O)NC1CCCCC1	CID:54638231	phase I
BRD-K43420611	OC[C@@H]1O[C@@H](CC(=O)N2CCOCC2)C=C[C@@H]1NC(=O)NC1CCCCC1	CID:54638232	phase I
BRD-K86524002	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)C=C[C@H]1NC(=O)NC1CCCCC1	CID:54638233	phase I
BRD-K07727895	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)C=C[C@@H]1NC(=O)NC1CCCCC1	CID:54638234	phase I
BRD-K25646871	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)C=C[C@@H]1NC(=O)NC1CCCCC1	CID:54638235	phase I
BRD-K50223932	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)C=C[C@H]1NC(=O)NC1CCCCC1	CID:54638238	phase I
BRD-K04632406	OC[C@H]1O[C@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638239	phase I
BRD-K79184162	OC[C@@H]1O[C@@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638240	phase I
BRD-K46707636	OC[C@H]1O[C@@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638241	phase I
BRD-K27442643	OC[C@@H]1O[C@@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638242	phase I
BRD-K77070775	OC[C@H]1O[C@@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638243	phase I
BRD-K76366810	OC[C@@H]1O[C@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638244	phase I
BRD-K24658364	OC[C@H]1O[C@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638245	phase I
BRD-K89114227	OC[C@@H]1O[C@H](CCNC(=O)c2ccc3OCOc3c2)CC[C@H]1NS(=O)(=O)c1ccc(Cl)cc1	CID:54638246	phase I
BRD-K85055995	COC(=O)C[C@@H]1O[C@@H](CO)[C@@H](N)C=C1	CID:54638247	phase I
BRD-K64344970	COC(=O)C[C@H]1O[C@@H](CO)[C@H](N)C=C1	CID:54638248	phase I
BRD-K56189188	CC(C)NC(=O)NCC[C@@H]1CC[C@@H](NC(=O)CCN2CCCCC2)[C@@H](CO)O1	CID:54638249	phase I
BRD-K73873786	CC(C)NC(=O)NCC[C@H]1CC[C@H](NC(=O)CCN2CCCCC2)[C@H](CO)O1	CID:54638250	phase I
BRD-K71779338	CC(C)NC(=O)NCC[C@H]1CC[C@@H](NC(=O)CCN2CCCCC2)[C@@H](CO)O1	CID:54638251	phase I
BRD-K09929530	CC(C)NC(=O)NCC[C@H]1CC[C@@H](NC(=O)CCN2CCCCC2)[C@H](CO)O1	CID:54638252	phase I
BRD-K47214596	CC(C)NC(=O)NCC[C@H]1CC[C@H](NC(=O)CCN2CCCCC2)[C@@H](CO)O1	CID:54638253	phase I
BRD-K19303070	CC(C)NC(=O)NCC[C@@H]1CC[C@H](NC(=O)CCN2CCCCC2)[C@H](CO)O1	CID:54638254	phase I
BRD-K36870972	CC(C)NC(=O)NCC[C@@H]1CC[C@H](NC(=O)CCN2CCCCC2)[C@@H](CO)O1	CID:54638255	phase I
BRD-K39728090	CC(C)NC(=O)NCC[C@@H]1CC[C@@H](NC(=O)CCN2CCCCC2)[C@H](CO)O1	CID:54638256	phase I
BRD-K31812348	OC[C@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638257	phase I
BRD-K03257659	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638258	phase I
BRD-K72299443	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638259	phase I
BRD-K46796516	OC[C@@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638260	phase I
BRD-K44635753	OC[C@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638261	phase I
BRD-K48571121	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638262	phase I
BRD-K92061784	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638263	phase I
BRD-K86853253	OC[C@@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C=C[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638264	phase I
BRD-K42450605	COc1ccccc1-c1cn(CC[C@@H]2CC[C@@H](NC(=O)c3cnccn3)[C@@H](CO)O2)nn1	CID:54638265	phase I
BRD-K34798777	COc1ccccc1-c1cn(CC[C@H]2CC[C@H](NC(=O)c3cnccn3)[C@H](CO)O2)nn1	CID:54638266	phase I
BRD-K39911043	COc1ccccc1-c1cn(CC[C@@H]2CC[C@H](NC(=O)c3cnccn3)[C@@H](CO)O2)nn1	CID:54638267	phase I
BRD-K50883617	COc1ccccc1-c1cn(CC[C@H]2CC[C@@H](NC(=O)c3cnccn3)[C@H](CO)O2)nn1	CID:54638268	phase I
BRD-K79302166	COc1ccccc1-c1cn(CC[C@H]2CC[C@@H](NC(=O)c3cnccn3)[C@@H](CO)O2)nn1	CID:54638269	phase I
BRD-K09632545	COc1ccccc1-c1cn(CC[C@@H]2CC[C@H](NC(=O)c3cnccn3)[C@H](CO)O2)nn1	CID:54638270	phase I
BRD-K41613119	COc1ccccc1-c1cn(CC[C@H]2CC[C@H](NC(=O)c3cnccn3)[C@@H](CO)O2)nn1	CID:54638271	phase I
BRD-K99775849	COc1ccccc1-c1cn(CC[C@@H]2CC[C@@H](NC(=O)c3cnccn3)[C@H](CO)O2)nn1	CID:54638272	phase I
BRD-K38542964	Cn1cnc(c1)S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)NCC2CCCCC2)O[C@@H]1CO	CID:54638273	phase I
BRD-K40608370	Cn1cnc(c1)S(=O)(=O)N[C@H]1CC[C@H](CC(=O)NCC2CCCCC2)O[C@H]1CO	CID:54638274	phase I
BRD-K94765019	Cn1cnc(c1)S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)NCC2CCCCC2)O[C@@H]1CO	CID:54638275	phase I
BRD-K68340318	Cn1cnc(c1)S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)NCC2CCCCC2)O[C@H]1CO	CID:54638276	phase I
BRD-K31671785	Cn1cnc(c1)S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)NCC2CCCCC2)O[C@H]1CO	CID:54638277	phase I
BRD-K52369815	Cn1cnc(c1)S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)NCC2CCCCC2)O[C@@H]1CO	CID:54638278	phase I
BRD-K01316590	Cn1cnc(c1)S(=O)(=O)N[C@H]1CC[C@H](CC(=O)NCC2CCCCC2)O[C@@H]1CO	CID:54638279	phase I
BRD-K55806039	Cn1cnc(c1)S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)NCC2CCCCC2)O[C@H]1CO	CID:54638280	phase I
BRD-K32323656	C[C@@H](NC(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638281	phase I
BRD-K04533640	C[C@H](NC(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638282	phase I
BRD-K76644587	C[C@@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638283	phase I
BRD-K48753787	C[C@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638284	phase I
BRD-K07807999	C[C@H](NC(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638285	phase I
BRD-K00801770	C[C@@H](NC(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638286	phase I
BRD-K87755452	C[C@@H](NC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638287	phase I
BRD-K41173255	C[C@H](NC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638288	phase I
BRD-K47173028	C[C@H](NC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638289	phase I
BRD-K65735929	C[C@@H](NC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638290	phase I
BRD-K26173688	C[C@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638291	phase I
BRD-K85593835	C[C@@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638292	phase I
BRD-K78343029	C[C@H](NC(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638293	phase I
BRD-K83388394	C[C@@H](NC(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638294	phase I
BRD-K03676054	C[C@H](NC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638295	phase I
BRD-K26327304	C[C@@H](NC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Cc2ccccn2)C=C1)c1ccccc1	CID:54638296	phase I
BRD-K69498175	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H](NC(=O)Nc2c(C)noc2C)[C@@H](CO)O1	CID:54638297	phase I
BRD-K38933129	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H](NC(=O)Nc2c(C)noc2C)[C@H](CO)O1	CID:54638298	phase I
BRD-K42679345	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H](NC(=O)Nc2c(C)noc2C)[C@@H](CO)O1	CID:54638299	phase I
BRD-K78229216	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H](NC(=O)Nc2c(C)noc2C)[C@H](CO)O1	CID:54638300	phase I
BRD-K01241136	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H](NC(=O)Nc2c(C)noc2C)[C@@H](CO)O1	CID:54638301	phase I
BRD-K42361507	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H](NC(=O)Nc2c(C)noc2C)[C@H](CO)O1	CID:54638302	phase I
BRD-K68370959	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H](NC(=O)Nc2c(C)noc2C)[C@@H](CO)O1	CID:54638303	phase I
BRD-K75353513	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H](NC(=O)Nc2c(C)noc2C)[C@H](CO)O1	CID:54638304	phase I
BRD-K55013500	OC[C@H]1O[C@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@H]1NC(=O)Cc1cccnc1	CID:54638305	phase I
BRD-K67716641	OC[C@@H]1O[C@@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54638306	phase I
BRD-K22694382	OC[C@H]1O[C@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54638307	phase I
BRD-K08403039	OC[C@@H]1O[C@@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@H]1NC(=O)Cc1cccnc1	CID:54638308	phase I
BRD-K29312193	OC[C@H]1O[C@@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@H]1NC(=O)Cc1cccnc1	CID:54638309	phase I
BRD-K63618292	OC[C@@H]1O[C@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54638310	phase I
BRD-K48102470	OC[C@H]1O[C@@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54638311	phase I
BRD-K77970970	OC[C@@H]1O[C@H](CCNS(=O)(=O)c2ccccc2Cl)CC[C@H]1NC(=O)Cc1cccnc1	CID:54638312	phase I
BRD-K73044562	COc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@@H]1CO	CID:54638313	phase I
BRD-K97748079	COc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@H]1CO	CID:54638314	phase I
BRD-K21528100	COc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@@H]1CO	CID:54638315	phase I
BRD-K00314651	COc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@H]1CO	CID:54638316	phase I
BRD-K69886508	COc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@@H]1CO	CID:54638317	phase I
BRD-K43151809	COc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@H]1CO	CID:54638318	phase I
BRD-K65437607	COc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@@H]1CO	CID:54638319	phase I
BRD-K89715659	COc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)O[C@H]1CO	CID:54638320	phase I
BRD-K89609393	COc1ccc(NC(=O)N[C@@H]2CC[C@H](CCNC(=O)Nc3cc(F)ccc3F)O[C@H]2CO)cc1	CID:54638321	phase I
BRD-K01070670	COc1ccc(NC(=O)N[C@@H]2CC[C@H](CCNC(=O)Nc3cc(F)ccc3F)O[C@@H]2CO)cc1	CID:54638322	phase I
BRD-K06650679	COc1ccc(NC(=O)N[C@H]2CC[C@@H](CCNC(=O)Nc3cc(F)ccc3F)O[C@H]2CO)cc1	CID:54638323	phase I
BRD-K52178187	COc1ccc(NC(=O)N[C@H]2CC[C@H](CCNC(=O)Nc3cc(F)ccc3F)O[C@@H]2CO)cc1	CID:54638324	phase I
BRD-K08240821	COc1ccc(NC(=O)N[C@H]2CC[C@@H](CCNC(=O)Nc3cc(F)ccc3F)O[C@@H]2CO)cc1	CID:54638325	phase I
BRD-K34549246	OC[C@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638326	phase I
BRD-K34019494	OC[C@@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638327	phase I
BRD-K81288057	OC[C@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638328	phase I
BRD-K80514140	OC[C@@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638329	phase I
BRD-K94690761	OC[C@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638330	phase I
BRD-K55331619	OC[C@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638331	phase I
BRD-K02409808	OC[C@@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638332	phase I
BRD-K44205194	OC[C@@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638333	phase I
BRD-K31385226	OC[C@@H]1O[C@@H](CC(=O)NCCc2cscn2)C=C[C@@H]1NC(=O)C1CCOCC1	CID:54638334	phase I
BRD-K74550836	OC[C@H]1O[C@H](CC(=O)NCCc2cscn2)C=C[C@@H]1NC(=O)C1CCOCC1	CID:54638335	phase I
BRD-K49781215	OC[C@H]1O[C@H](CCn2cc(nn2)C2CCCCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638336	phase I
BRD-K21549522	OC[C@@H]1O[C@@H](CCn2cc(nn2)C2CCCCC2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638337	phase I
BRD-K70983703	OC[C@@H]1O[C@@H](CCn2cc(nn2)C2CCCCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638338	phase I
BRD-K53619921	OC[C@H]1O[C@@H](CCn2cc(nn2)C2CCCCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638339	phase I
BRD-K18999740	OC[C@@H]1O[C@H](CCn2cc(nn2)C2CCCCC2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638340	phase I
BRD-K38498572	OC[C@H]1O[C@H](CCn2cc(nn2)C2CCCCC2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638341	phase I
BRD-K08369728	OC[C@H]1O[C@@H](CCn2cc(nn2)C2CCCCC2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638342	phase I
BRD-K37848804	OC[C@@H]1O[C@H](CCn2cc(nn2)C2CCCCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638343	phase I
BRD-K43374517	OC[C@H]1O[C@H](CC(=O)NCCCN2CCOCC2)CC[C@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638344	phase I
BRD-K98099906	OC[C@@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)CC[C@@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638345	phase I
BRD-K61541040	OC[C@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)CC[C@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638346	phase I
BRD-K72461570	OC[C@@H]1O[C@H](CC(=O)NCCCN2CCOCC2)CC[C@@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638347	phase I
BRD-K99533437	OC[C@H]1O[C@H](CC(=O)NCCCN2CCOCC2)CC[C@@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638348	phase I
BRD-K71032175	OC[C@@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)CC[C@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638349	phase I
BRD-K80723382	OC[C@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)CC[C@@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638350	phase I
BRD-K71302181	OC[C@@H]1O[C@H](CC(=O)NCCCN2CCOCC2)CC[C@H]1NC(=O)Nc1ccc2OCOc2c1	CID:54638351	phase I
BRD-K67399667	Cn1cnc(c1)S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@@H]1CO	CID:54638352	phase I
BRD-K47881779	Cn1cnc(c1)S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@H]1CO	CID:54638353	phase I
BRD-K40225343	Cn1cnc(c1)S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@H]1CO	CID:54638354	phase I
BRD-K68007071	Cn1cnc(c1)S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@@H]1CO	CID:54638355	phase I
BRD-K97489107	Cn1cnc(c1)S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@H]1CO	CID:54638356	phase I
BRD-K30855709	Cn1cnc(c1)S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@@H]1CO	CID:54638357	phase I
BRD-K10951564	Cn1cnc(c1)S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)O[C@H]1CO	CID:54638358	phase I
BRD-K91269653	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C=C[C@H]1NC(=O)c1cccnc1	CID:54638359	phase I
BRD-K60151092	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C=C[C@@H]1NC(=O)c1cccnc1	CID:54638360	phase I
BRD-K19251038	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C=C[C@H]1NC(=O)c1cccnc1	CID:54638361	phase I
BRD-K36618611	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C=C[C@@H]1NC(=O)c1cccnc1	CID:54638362	phase I
BRD-K23586462	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C=C[C@@H]1NC(=O)c1cccnc1	CID:54638363	phase I
BRD-K65608865	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C=C[C@H]1NC(=O)c1cccnc1	CID:54638364	phase I
BRD-K04009734	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C=C[C@@H]1NC(=O)c1cccnc1	CID:54638365	phase I
BRD-K62724755	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C=C[C@H]1NC(=O)c1cccnc1	CID:54638366	phase I
BRD-K06158553	OC[C@H]1O[C@H](CC(=O)NCc2ccncn2)CC[C@H]1NC(=O)c1ccc(F)cc1	CID:54638367	phase I
BRD-K88617254	OC[C@@H]1O[C@@H](CC(=O)NCc2ccncn2)CC[C@@H]1NC(=O)c1ccc(F)cc1	CID:54638368	phase I
BRD-K95982530	OC[C@H]1O[C@@H](CC(=O)NCc2ccncn2)CC[C@H]1NC(=O)c1ccc(F)cc1	CID:54638369	phase I
BRD-K85088178	OC[C@@H]1O[C@H](CC(=O)NCc2ccncn2)CC[C@@H]1NC(=O)c1ccc(F)cc1	CID:54638370	phase I
BRD-K41139858	OC[C@H]1O[C@H](CC(=O)NCc2ccncn2)CC[C@@H]1NC(=O)c1ccc(F)cc1	CID:54638371	phase I
BRD-K49290616	OC[C@@H]1O[C@@H](CC(=O)NCc2ccncn2)CC[C@H]1NC(=O)c1ccc(F)cc1	CID:54638372	phase I
BRD-K76223260	OC[C@H]1O[C@@H](CC(=O)NCc2ccncn2)CC[C@@H]1NC(=O)c1ccc(F)cc1	CID:54638373	phase I
BRD-K86618560	OC[C@@H]1O[C@H](CC(=O)NCc2ccncn2)CC[C@H]1NC(=O)c1ccc(F)cc1	CID:54638374	phase I
BRD-K49172498	COc1cccc(NC(=O)N[C@@H]2C=C[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2CO)c1	CID:54638375	phase I
BRD-K90338784	COc1cccc(NC(=O)N[C@H]2C=C[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2CO)c1	CID:54638376	phase I
BRD-K95360473	COc1cccc(NC(=O)N[C@H]2C=C[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2CO)c1	CID:54638377	phase I
BRD-K29776425	COc1cccc(NC(=O)N[C@H]2C=C[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2CO)c1	CID:54638378	phase I
BRD-K22428007	COc1cccc(NC(=O)N[C@@H]2C=C[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2CO)c1	CID:54638379	phase I
BRD-K44996602	COc1cccc(NC(=O)N[C@H]2C=C[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2CO)c1	CID:54638380	phase I
BRD-K83095440	COc1cccc(NC(=O)N[C@@H]2C=C[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2CO)c1	CID:54638381	phase I
BRD-K33750632	COCCNC(=O)C[C@@H]1CC[C@@H](NC(=O)NC2CCCCC2)[C@@H](CO)O1	CID:54638382	phase I
BRD-K84907327	COCCNC(=O)C[C@H]1CC[C@H](NC(=O)NC2CCCCC2)[C@H](CO)O1	CID:54638383	phase I
BRD-K74964997	COCCNC(=O)C[C@H]1CC[C@@H](NC(=O)NC2CCCCC2)[C@@H](CO)O1	CID:54638384	phase I
BRD-K87878143	COCCNC(=O)C[C@@H]1CC[C@H](NC(=O)NC2CCCCC2)[C@H](CO)O1	CID:54638385	phase I
BRD-K57841225	COCCNC(=O)C[C@@H]1CC[C@H](NC(=O)NC2CCCCC2)[C@@H](CO)O1	CID:54638386	phase I
BRD-K15171837	COCCNC(=O)C[C@H]1CC[C@@H](NC(=O)NC2CCCCC2)[C@H](CO)O1	CID:54638387	phase I
BRD-K71156053	COCCNC(=O)C[C@H]1CC[C@H](NC(=O)NC2CCCCC2)[C@@H](CO)O1	CID:54638388	phase I
BRD-K61338389	COCCNC(=O)C[C@@H]1CC[C@@H](NC(=O)NC2CCCCC2)[C@H](CO)O1	CID:54638389	phase I
BRD-K76688996	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@@H](CCNC(=O)C2CCOCC2)O[C@@H]1CO	CID:54638390	phase I
BRD-K39430900	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@H](CCNC(=O)C2CCOCC2)O[C@H]1CO	CID:54638391	phase I
BRD-K32233845	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@@H](CCNC(=O)C2CCOCC2)O[C@@H]1CO	CID:54638392	phase I
BRD-K79944151	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@H](CCNC(=O)C2CCOCC2)O[C@H]1CO	CID:54638393	phase I
BRD-K37303684	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@H](CCNC(=O)C2CCOCC2)O[C@@H]1CO	CID:54638394	phase I
BRD-K12826563	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@@H](CCNC(=O)C2CCOCC2)O[C@H]1CO	CID:54638395	phase I
BRD-K61219693	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@H](CCNC(=O)C2CCOCC2)O[C@@H]1CO	CID:54638396	phase I
BRD-K74594501	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@@H](CCNC(=O)C2CCOCC2)O[C@H]1CO	CID:54638397	phase I
BRD-K26003427	CN(C)C(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638398	phase I
BRD-K79410674	CN(C)C(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638399	phase I
BRD-K21463062	CN(C)C(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638400	phase I
BRD-K04831789	CN(C)C(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638401	phase I
BRD-K09852122	CN(C)C(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638402	phase I
BRD-K61083743	CN(C)C(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638403	phase I
BRD-K59022317	CN(C)C(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638404	phase I
BRD-K56665985	CN(C)C(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)c2ccc(F)cc2)C=C1	CID:54638405	phase I
BRD-K98062568	COc1ccccc1NC(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@@H]1CO	CID:54638406	phase I
BRD-K26924060	COc1ccccc1NC(=O)N[C@H]1CC[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@H]1CO	CID:54638407	phase I
BRD-K91194423	COc1ccccc1NC(=O)N[C@@H]1CC[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@@H]1CO	CID:54638408	phase I
BRD-K50808811	COc1ccccc1NC(=O)N[C@H]1CC[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@H]1CO	CID:54638409	phase I
BRD-K57055053	COc1ccccc1NC(=O)N[C@H]1CC[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@@H]1CO	CID:54638410	phase I
BRD-K97001739	COc1ccccc1NC(=O)N[C@@H]1CC[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@H]1CO	CID:54638411	phase I
BRD-K42743267	COc1ccccc1NC(=O)N[C@H]1CC[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@@H]1CO	CID:54638412	phase I
BRD-K35060817	COc1ccccc1NC(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)O[C@H]1CO	CID:54638413	phase I
BRD-K54247306	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C=C[C@H]1NC(=O)CC1CC1	CID:54638414	phase I
BRD-K54964414	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C=C[C@@H]1NC(=O)CC1CC1	CID:54638415	phase I
BRD-K55767126	OC[C@H]1O[C@H](CC(=O)NCC(F)(F)F)C=C[C@@H]1NC(=O)CC1CC1	CID:54638416	phase I
BRD-K37655007	OC[C@@H]1O[C@@H](CC(=O)NCC(F)(F)F)C=C[C@H]1NC(=O)CC1CC1	CID:54638417	phase I
BRD-K46714753	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C=C[C@@H]1NC(=O)CC1CC1	CID:54638418	phase I
BRD-K27720649	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C=C[C@H]1NC(=O)CC1CC1	CID:54638419	phase I
BRD-K53943507	CCS(=O)(=O)NCC[C@H]1CC[C@@H](NC(=O)C2CCCCC2)[C@H](CO)O1	CID:54638420	phase I
BRD-K89994146	CCS(=O)(=O)NCC[C@H]1CC[C@H](NC(=O)C2CCCCC2)[C@@H](CO)O1	CID:54638421	phase I
BRD-K19696710	CCS(=O)(=O)NCC[C@@H]1CC[C@@H](NC(=O)C2CCCCC2)[C@H](CO)O1	CID:54638422	phase I
BRD-K47691029	CN(C)CCCNC(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638423	phase I
BRD-K66640841	CN(C)CCCNC(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638424	phase I
BRD-K35470597	CN(C)CCCNC(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638425	phase I
BRD-K94726713	CN(C)CCCNC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638426	phase I
BRD-K43601041	CN(C)CCCNC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638427	phase I
BRD-K44867089	CN(C)CCCNC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638428	phase I
BRD-K47366586	CN(C)CCCNC(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638429	phase I
BRD-K53359544	CN(C)CCCNC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Nc2c(C)noc2C)C=C1	CID:54638430	phase I
BRD-K63376220	COc1ccccc1CNC(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)CN(C)C)C=C1	CID:54638431	phase I
BRD-K63671514	COc1ccccc1CNC(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)CN(C)C)C=C1	CID:54638432	phase I
BRD-K23688566	COc1ccccc1CNC(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)CN(C)C)C=C1	CID:54638433	phase I
BRD-K33668351	COc1ccccc1CNC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)CN(C)C)C=C1	CID:54638434	phase I
BRD-K72347310	COc1ccccc1CNC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)CN(C)C)C=C1	CID:54638435	phase I
BRD-K60703313	COc1ccccc1CNC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)CN(C)C)C=C1	CID:54638436	phase I
BRD-K71531260	COc1ccccc1CNC(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)CN(C)C)C=C1	CID:54638437	phase I
BRD-K12888055	COc1ccccc1CNC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)CN(C)C)C=C1	CID:54638438	phase I
BRD-K88391199	NCC[C@@H]1CC[C@@H](NC(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638439	phase I
BRD-K54431311	NCC[C@H]1CC[C@H](NC(=O)c2ccccc2F)[C@H](CO)O1	CID:54638440	phase I
BRD-K60809157	NCC[C@H]1CC[C@@H](NC(=O)c2ccccc2F)[C@H](CO)O1	CID:54638441	phase I
BRD-K13428252	NCC[C@H]1CC[C@H](NC(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638442	phase I
BRD-K72915790	NCC[C@H]1CC[C@@H](NC(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638443	phase I
BRD-K80726792	NCC[C@@H]1CC[C@H](NC(=O)c2ccccc2F)[C@H](CO)O1	CID:54638444	phase I
BRD-K18683499	NCC[C@@H]1CC[C@H](NC(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638445	phase I
BRD-K37752193	NCC[C@@H]1CC[C@@H](NC(=O)c2ccccc2F)[C@H](CO)O1	CID:54638446	phase I
BRD-K63798874	OC[C@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@H]1NC(=O)c1cnccn1	CID:54638447	phase I
BRD-K11062991	OC[C@@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@@H]1NC(=O)c1cnccn1	CID:54638448	phase I
BRD-K45711268	OC[C@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@H]1NC(=O)c1cnccn1	CID:54638449	phase I
BRD-K96269157	OC[C@@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@@H]1NC(=O)c1cnccn1	CID:54638450	phase I
BRD-K13860832	OC[C@@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@H]1NC(=O)c1cnccn1	CID:54638451	phase I
BRD-K14471942	OC[C@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@@H]1NC(=O)c1cnccn1	CID:54638452	phase I
BRD-K80171496	OC[C@@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)C=C[C@H]1NC(=O)c1cnccn1	CID:54638453	phase I
BRD-K20310932	OC[C@H]1O[C@H](CC(=O)NCCCN2CCOCC2)C=C[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638454	phase I
BRD-K76454674	OC[C@@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)C=C[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638455	phase I
BRD-K91924645	OC[C@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)C=C[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638456	phase I
BRD-K30620974	OC[C@@H]1O[C@H](CC(=O)NCCCN2CCOCC2)C=C[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638457	phase I
BRD-K23794511	OC[C@@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)C=C[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638458	phase I
BRD-K89699317	OC[C@H]1O[C@@H](CC(=O)NCCCN2CCOCC2)C=C[C@@H]1NS(=O)(=O)c1ccccc1F	CID:54638459	phase I
BRD-K60471354	OC[C@@H]1O[C@H](CC(=O)NCCCN2CCOCC2)C=C[C@H]1NS(=O)(=O)c1ccccc1F	CID:54638460	phase I
BRD-K80408402	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)CC[C@H]1NC(=O)c1ccccn1	CID:54638461	phase I
BRD-K49417484	OC[C@@H]1O[C@@H](CC(=O)N2CCOCC2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638462	phase I
BRD-K02117849	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)CC[C@H]1NC(=O)c1ccccn1	CID:54638463	phase I
BRD-K14159335	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638464	phase I
BRD-K64864583	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638465	phase I
BRD-K34431359	OC[C@@H]1O[C@@H](CC(=O)N2CCOCC2)CC[C@H]1NC(=O)c1ccccn1	CID:54638466	phase I
BRD-K99115033	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638467	phase I
BRD-K82071478	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)CC[C@H]1NC(=O)c1ccccn1	CID:54638468	phase I
BRD-K73876582	COCc1cn(CC[C@@H]2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](CO)O2)nn1	CID:54638469	phase I
BRD-K60857329	COCc1cn(CC[C@H]2CC[C@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@H](CO)O2)nn1	CID:54638470	phase I
BRD-K48724570	COCc1cn(CC[C@H]2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](CO)O2)nn1	CID:54638471	phase I
BRD-K85194284	COCc1cn(CC[C@H]2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@H](CO)O2)nn1	CID:54638472	phase I
BRD-K92758184	COCc1cn(CC[C@@H]2CC[C@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@H](CO)O2)nn1	CID:54638473	phase I
BRD-K37552925	COCc1cn(CC[C@@H]2CC[C@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](CO)O2)nn1	CID:54638474	phase I
BRD-K27198844	COCc1cn(CC[C@H]2CC[C@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@@H](CO)O2)nn1	CID:54638475	phase I
BRD-K39799535	COCc1cn(CC[C@@H]2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)[C@H](CO)O2)nn1	CID:54638476	phase I
BRD-K92593565	C[C@H](NC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638477	phase I
BRD-K91730835	C[C@H](NC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638478	phase I
BRD-K26840329	C[C@@H](NC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638479	phase I
BRD-K67319066	C[C@@H](NC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638480	phase I
BRD-K77162730	C[C@@H](NC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638481	phase I
BRD-K78528600	C[C@H](NC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638482	phase I
BRD-K47686295	C[C@@H](NC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638483	phase I
BRD-K40506152	C[C@H](NC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638484	phase I
BRD-K78849449	C[C@H](NC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638485	phase I
BRD-K71752918	C[C@@H](NC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638486	phase I
BRD-K19677752	C[C@H](NC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638487	phase I
BRD-K43216840	C[C@@H](NC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638488	phase I
BRD-K38011931	C[C@@H](NC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638489	phase I
BRD-K09454555	C[C@H](NC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2cccc(F)c2)[C@@H](CO)O1)c1ccccc1	CID:54638490	phase I
BRD-K94688728	C[C@@H](NC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638491	phase I
BRD-K14736141	C[C@H](NC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2cccc(F)c2)[C@H](CO)O1)c1ccccc1	CID:54638492	phase I
BRD-K93240833	OC[C@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638493	phase I
BRD-K52954098	OC[C@@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638494	phase I
BRD-K84143894	OC[C@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638495	phase I
BRD-K77831863	OC[C@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638496	phase I
BRD-K24820558	OC[C@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638497	phase I
BRD-K63922933	OC[C@@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638498	phase I
BRD-K69672581	OC[C@@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638499	phase I
BRD-K72443777	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638500	phase I
BRD-K50218765	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638501	phase I
BRD-K01711704	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638502	phase I
BRD-K50611992	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638503	phase I
BRD-K82986138	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638504	phase I
BRD-K93330237	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638505	phase I
BRD-K84468307	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638506	phase I
BRD-K39255658	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638507	phase I
BRD-K26038019	CC(C)NC(=O)N[C@@H]1C=C[C@@H](CC(=O)NC2Cc3ccccc3C2)O[C@@H]1CO	CID:54638508	phase I
BRD-K89386994	CC(C)NC(=O)N[C@H]1C=C[C@H](CC(=O)NC2Cc3ccccc3C2)O[C@H]1CO	CID:54638509	phase I
BRD-K90061989	CC(C)NC(=O)N[C@@H]1C=C[C@H](CC(=O)NC2Cc3ccccc3C2)O[C@@H]1CO	CID:54638510	phase I
BRD-K73804157	CC(C)NC(=O)N[C@H]1C=C[C@@H](CC(=O)NC2Cc3ccccc3C2)O[C@H]1CO	CID:54638511	phase I
BRD-K84718005	CC(C)NC(=O)N[C@H]1C=C[C@@H](CC(=O)NC2Cc3ccccc3C2)O[C@@H]1CO	CID:54638512	phase I
BRD-K76876037	CC(C)NC(=O)N[C@@H]1C=C[C@H](CC(=O)NC2Cc3ccccc3C2)O[C@H]1CO	CID:54638513	phase I
BRD-K51620275	CC(C)NC(=O)N[C@H]1C=C[C@H](CC(=O)NC2Cc3ccccc3C2)O[C@@H]1CO	CID:54638514	phase I
BRD-K92134560	CC(C)NC(=O)N[C@@H]1C=C[C@@H](CC(=O)NC2Cc3ccccc3C2)O[C@H]1CO	CID:54638515	phase I
BRD-K62814224	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2ccc(C)cc2)[C@@H](CO)O1	CID:54638516	phase I
BRD-K19770227	CN(C)CCCNC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)[C@H](CO)O1	CID:54638517	phase I
BRD-K85208848	CN(C)CCCNC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2ccc(C)cc2)[C@@H](CO)O1	CID:54638518	phase I
BRD-K10014225	CN(C)CCCNC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)[C@H](CO)O1	CID:54638519	phase I
BRD-K92958239	CN(C)CCCNC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)[C@@H](CO)O1	CID:54638520	phase I
BRD-K91508497	CN(C)CCCNC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2ccc(C)cc2)[C@H](CO)O1	CID:54638521	phase I
BRD-K33038714	CN(C)CCCNC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)[C@@H](CO)O1	CID:54638522	phase I
BRD-K99567611	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2ccc(C)cc2)[C@H](CO)O1	CID:54638523	phase I
BRD-K90089455	OC[C@H]1O[C@H](CCNC(=O)Cc2ccccn2)CC[C@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638524	phase I
BRD-K92493271	OC[C@@H]1O[C@@H](CCNC(=O)Cc2ccccn2)CC[C@@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638525	phase I
BRD-K40383467	OC[C@H]1O[C@H](CCNC(=O)Cc2ccccn2)CC[C@@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638526	phase I
BRD-K22451824	OC[C@@H]1O[C@@H](CCNC(=O)Cc2ccccn2)CC[C@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638527	phase I
BRD-K76688397	OC[C@H]1O[C@@H](CCNC(=O)Cc2ccccn2)CC[C@@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638528	phase I
BRD-K63811860	OC[C@H]1O[C@@H](CCNC(=O)Cc2ccccn2)CC[C@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638529	phase I
BRD-K34404012	OC[C@@H]1O[C@H](CCNC(=O)Cc2ccccn2)CC[C@@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638530	phase I
BRD-K24199200	OC[C@@H]1O[C@H](CCNC(=O)Cc2ccccn2)CC[C@H]1NC(=O)Nc1ccc(Cl)cc1	CID:54638531	phase I
BRD-K15013036	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C=C[C@@H]1NC(=O)C1CC1	CID:54638534	phase I
BRD-K44338067	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C=C[C@@H]1NC(=O)C1CC1	CID:54638535	phase I
BRD-K47587697	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C=C[C@H]1NC(=O)C1CC1	CID:54638536	phase I
BRD-K86938339	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C=C[C@@H]1NC(=O)C1CC1	CID:54638537	phase I
BRD-K85025453	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C=C[C@H]1NC(=O)C1CC1	CID:54638538	phase I
BRD-K80232076	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@H]1NC(=O)c1ccccn1	CID:54638539	phase I
BRD-K98909007	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@@H]1NC(=O)c1ccccn1	CID:54638540	phase I
BRD-K82814298	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@H]1NC(=O)c1ccccn1	CID:54638541	phase I
BRD-K61782241	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@@H]1NC(=O)c1ccccn1	CID:54638542	phase I
BRD-K49595590	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@@H]1NC(=O)c1ccccn1	CID:54638543	phase I
BRD-K17181267	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@H]1NC(=O)c1ccccn1	CID:54638544	phase I
BRD-K45496021	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)C=C[C@H]1NC(=O)c1ccccn1	CID:54638545	phase I
BRD-K32519217	OC[C@H]1O[C@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@H]1NC(=O)Nc1cccc(F)c1	CID:54638546	phase I
BRD-K24217589	OC[C@@H]1O[C@@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638547	phase I
BRD-K79382100	OC[C@@H]1O[C@@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@H]1NC(=O)Nc1cccc(F)c1	CID:54638548	phase I
BRD-K80019738	OC[C@H]1O[C@@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@H]1NC(=O)Nc1cccc(F)c1	CID:54638549	phase I
BRD-K29711801	OC[C@@H]1O[C@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638550	phase I
BRD-K23564937	OC[C@H]1O[C@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638551	phase I
BRD-K90915722	OC[C@H]1O[C@@H](CCNS(=O)(=O)c2cccc(Cl)c2)CC[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638552	phase I
BRD-K94172147	OC[C@@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638555	phase I
BRD-K93510852	OC[C@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638556	phase I
BRD-K36026160	OC[C@@H]1O[C@H](CC(=O)NCc2cccc(F)c2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638557	phase I
BRD-K95578893	OC[C@H]1O[C@H](CC(=O)NCc2cccc(F)c2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638558	phase I
BRD-K81954574	OC[C@@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638559	phase I
BRD-K67694126	OC[C@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638560	phase I
BRD-K39530782	OC[C@@H]1O[C@H](CC(=O)NCc2cccc(F)c2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638561	phase I
BRD-K03245480	CCCNC(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@@H]1CO	CID:54638562	phase I
BRD-K73639776	CCCNC(=O)N[C@H]1CC[C@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@H]1CO	CID:54638563	phase I
BRD-K61428915	CCCNC(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@H]1CO	CID:54638564	phase I
BRD-K93007240	CCCNC(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@@H]1CO	CID:54638565	phase I
BRD-K02241254	CCCNC(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@H]1CO	CID:54638566	phase I
BRD-K00474848	CCCNC(=O)N[C@H]1CC[C@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@@H]1CO	CID:54638567	phase I
BRD-K64549867	CCCNC(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)-c2cccc(F)c2)O[C@H]1CO	CID:54638568	phase I
BRD-K35660899	CCS(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54638569	phase I
BRD-K33537450	CCS(=O)(=O)N[C@H]1CC[C@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54638570	phase I
BRD-K31784555	COc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@@H](CCN)O[C@@H]1CO	CID:54638571	phase I
BRD-K77314783	COc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@H](CCN)O[C@H]1CO	CID:54638572	phase I
BRD-K77931347	COc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@H](CCN)O[C@@H]1CO	CID:54638573	phase I
BRD-K13529284	COc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@H](CCN)O[C@H]1CO	CID:54638574	phase I
BRD-K43467947	COc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@H](CCN)O[C@@H]1CO	CID:54638575	phase I
BRD-K60462241	COc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@@H](CCN)O[C@H]1CO	CID:54638576	phase I
BRD-K13626437	COc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@@H](CCN)O[C@@H]1CO	CID:54638577	phase I
BRD-K90947049	COc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@@H](CCN)O[C@H]1CO	CID:54638578	phase I
BRD-K37556205	OC[C@H]1O[C@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@H]1NC(=O)C1CCOCC1	CID:54638579	phase I
BRD-K42419992	OC[C@@H]1O[C@@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@@H]1NC(=O)C1CCOCC1	CID:54638580	phase I
BRD-K10562742	OC[C@H]1O[C@@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@H]1NC(=O)C1CCOCC1	CID:54638581	phase I
BRD-K39635618	OC[C@@H]1O[C@@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@H]1NC(=O)C1CCOCC1	CID:54638582	phase I
BRD-K10578850	OC[C@@H]1O[C@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@@H]1NC(=O)C1CCOCC1	CID:54638583	phase I
BRD-K73860091	OC[C@H]1O[C@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@@H]1NC(=O)C1CCOCC1	CID:54638584	phase I
BRD-K27767004	OC[C@H]1O[C@@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@@H]1NC(=O)C1CCOCC1	CID:54638585	phase I
BRD-K04515815	OC[C@@H]1O[C@H](CCNC(=O)c2cc(Cl)cc(Cl)c2)CC[C@H]1NC(=O)C1CCOCC1	CID:54638586	phase I
BRD-K53263381	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C=C[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638587	phase I
BRD-K00575273	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C=C[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638588	phase I
BRD-K22433696	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C=C[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638589	phase I
BRD-K61255273	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C=C[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638590	phase I
BRD-K39151337	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C=C[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638591	phase I
BRD-K85471465	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C=C[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638592	phase I
BRD-K80457386	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C=C[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638593	phase I
BRD-K43518940	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C=C[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638594	phase I
BRD-K70630513	Cc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@@H](CCNC(=O)c2cnccn2)O[C@@H]1CO	CID:54638595	phase I
BRD-K33130522	Cc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@H](CCNC(=O)c2cnccn2)O[C@H]1CO	CID:54638596	phase I
BRD-K68409203	Cc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@H](CCNC(=O)c2cnccn2)O[C@@H]1CO	CID:54638597	phase I
BRD-K36747900	Cc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@H](CCNC(=O)c2cnccn2)O[C@H]1CO	CID:54638598	phase I
BRD-K53740625	Cc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@@H](CCNC(=O)c2cnccn2)O[C@H]1CO	CID:54638599	phase I
BRD-K14295062	Cc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@@H](CCNC(=O)c2cnccn2)O[C@@H]1CO	CID:54638600	phase I
BRD-K57497528	Cc1cccc(c1)S(=O)(=O)N[C@H]1CC[C@H](CCNC(=O)c2cnccn2)O[C@@H]1CO	CID:54638601	phase I
BRD-K80821495	Cc1cccc(c1)S(=O)(=O)N[C@@H]1CC[C@@H](CCNC(=O)c2cnccn2)O[C@H]1CO	CID:54638602	phase I
BRD-K41675418	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)-c2cccnc2)O[C@@H]1CO	CID:54638603	phase I
BRD-K44586044	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CCn2cc(nn2)-c2cccnc2)O[C@H]1CO	CID:54638604	phase I
BRD-K96207987	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)-c2cccnc2)O[C@@H]1CO	CID:54638605	phase I
BRD-K37710486	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)-c2cccnc2)O[C@H]1CO	CID:54638606	phase I
BRD-K02240493	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)-c2cccnc2)O[C@H]1CO	CID:54638607	phase I
BRD-K61531144	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)-c2cccnc2)O[C@@H]1CO	CID:54638608	phase I
BRD-K84195984	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CCn2cc(nn2)-c2cccnc2)O[C@@H]1CO	CID:54638609	phase I
BRD-K70874643	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)-c2cccnc2)O[C@H]1CO	CID:54638610	phase I
BRD-K58962381	OC[C@H]1O[C@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@H]1NC(=O)c1cccnc1	CID:54638611	phase I
BRD-K48515753	OC[C@@H]1O[C@@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@@H]1NC(=O)c1cccnc1	CID:54638612	phase I
BRD-K55065943	OC[C@@H]1O[C@@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@H]1NC(=O)c1cccnc1	CID:54638613	phase I
BRD-K82041810	OC[C@H]1O[C@@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@@H]1NC(=O)c1cccnc1	CID:54638614	phase I
BRD-K49702326	OC[C@H]1O[C@@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@H]1NC(=O)c1cccnc1	CID:54638615	phase I
BRD-K47569804	OC[C@@H]1O[C@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@@H]1NC(=O)c1cccnc1	CID:54638616	phase I
BRD-K22070096	OC[C@H]1O[C@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@@H]1NC(=O)c1cccnc1	CID:54638617	phase I
BRD-K04643065	OC[C@@H]1O[C@H](CCNC(=O)Nc2ccc(cc2)C(F)(F)F)CC[C@H]1NC(=O)c1cccnc1	CID:54638618	phase I
BRD-K22643403	CN1CCN(CC1)C(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638619	phase I
BRD-K98607641	CN1CCN(CC1)C(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638620	phase I
BRD-K59247792	CN1CCN(CC1)C(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638621	phase I
BRD-K45355730	CN1CCN(CC1)C(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638622	phase I
BRD-K22719646	CN1CCN(CC1)C(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638623	phase I
BRD-K55597137	CN1CCN(CC1)C(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638624	phase I
BRD-K25096430	CN1CCN(CC1)C(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638625	phase I
BRD-K71921803	CN1CCN(CC1)C(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccccc2F)C=C1	CID:54638626	phase I
BRD-K61636401	COC(=O)C[C@H]1CC[C@@H](N)[C@@H](CO)O1	CID:54638627	phase I
BRD-K99809487	COC(=O)C[C@H]1CC[C@@H](N)[C@H](CO)O1	CID:54638628	phase I
BRD-K97741410	COC(=O)C[C@H]1CC[C@H](N)[C@@H](CO)O1	CID:54638629	phase I
BRD-K22291343	CC(C)c1cn(CC[C@@H]2CC[C@@H](NC(=O)C3CC3)[C@@H](CO)O2)nn1	CID:54638630	phase I
BRD-K35199432	CC(C)c1cn(CC[C@H]2CC[C@H](NC(=O)C3CC3)[C@H](CO)O2)nn1	CID:54638631	phase I
BRD-K01572707	CC(C)c1cn(CC[C@@H]2CC[C@H](NC(=O)C3CC3)[C@@H](CO)O2)nn1	CID:54638632	phase I
BRD-K46709181	CC(C)c1cn(CC[C@H]2CC[C@@H](NC(=O)C3CC3)[C@H](CO)O2)nn1	CID:54638633	phase I
BRD-K62372763	CC(C)c1cn(CC[C@H]2CC[C@@H](NC(=O)C3CC3)[C@@H](CO)O2)nn1	CID:54638634	phase I
BRD-K13513398	CC(C)c1cn(CC[C@@H]2CC[C@H](NC(=O)C3CC3)[C@H](CO)O2)nn1	CID:54638635	phase I
BRD-K74513776	CC(C)c1cn(CC[C@H]2CC[C@H](NC(=O)C3CC3)[C@@H](CO)O2)nn1	CID:54638636	phase I
BRD-K31561199	CC(C)c1cn(CC[C@@H]2CC[C@@H](NC(=O)C3CC3)[C@H](CO)O2)nn1	CID:54638637	phase I
BRD-K11868205	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@H]1NS(=O)(=O)c1ccccc1	CID:54638638	phase I
BRD-K63531989	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@@H]1NS(=O)(=O)c1ccccc1	CID:54638639	phase I
BRD-K59404663	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@@H]1NS(=O)(=O)c1ccccc1	CID:54638640	phase I
BRD-K23191900	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@@H]1NS(=O)(=O)c1ccccc1	CID:54638641	phase I
BRD-K02897131	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@H]1NS(=O)(=O)c1ccccc1	CID:54638642	phase I
BRD-K37344040	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@@H]1NS(=O)(=O)c1ccccc1	CID:54638643	phase I
BRD-K33368320	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)C=C[C@H]1NS(=O)(=O)c1ccccc1	CID:54638644	phase I
BRD-K30361687	COc1cccc(NC(=O)N[C@@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@@H]2CO)c1	CID:54638645	phase I
BRD-K07493900	COc1cccc(NC(=O)N[C@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@H]2CO)c1	CID:54638646	phase I
BRD-K11401851	COc1cccc(NC(=O)N[C@@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@@H]2CO)c1	CID:54638647	phase I
BRD-K88973556	COc1cccc(NC(=O)N[C@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@H]2CO)c1	CID:54638648	phase I
BRD-K75467206	COc1cccc(NC(=O)N[C@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@@H]2CO)c1	CID:54638649	phase I
BRD-K70868165	COc1cccc(NC(=O)N[C@@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@H]2CO)c1	CID:54638650	phase I
BRD-K52887203	COc1cccc(NC(=O)N[C@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@@H]2CO)c1	CID:54638651	phase I
BRD-K61202234	COc1cccc(NC(=O)N[C@@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@H]2CO)c1	CID:54638652	phase I
BRD-K24890551	COc1cccc(CNC(=O)C[C@H]2O[C@H](CO)[C@H](NC(=O)C3CCC3)C=C2)c1	CID:54638653	phase I
BRD-K99944604	COc1cccc(CNC(=O)C[C@@H]2O[C@@H](CO)[C@@H](NC(=O)C3CCC3)C=C2)c1	CID:54638654	phase I
BRD-K82003968	COc1cccc(CNC(=O)C[C@@H]2O[C@H](CO)[C@H](NC(=O)C3CCC3)C=C2)c1	CID:54638655	phase I
BRD-K75111717	COc1cccc(CNC(=O)C[C@H]2O[C@@H](CO)[C@@H](NC(=O)C3CCC3)C=C2)c1	CID:54638656	phase I
BRD-K92219497	COc1cccc(CNC(=O)C[C@H]2O[C@H](CO)[C@@H](NC(=O)C3CCC3)C=C2)c1	CID:54638657	phase I
BRD-K39241486	COc1cccc(CNC(=O)C[C@@H]2O[C@@H](CO)[C@H](NC(=O)C3CCC3)C=C2)c1	CID:54638658	phase I
BRD-K69280720	COc1cccc(CNC(=O)C[C@@H]2O[C@H](CO)[C@@H](NC(=O)C3CCC3)C=C2)c1	CID:54638659	phase I
BRD-K77835518	COc1cccc(CNC(=O)C[C@H]2O[C@@H](CO)[C@H](NC(=O)C3CCC3)C=C2)c1	CID:54638660	phase I
BRD-K22097595	OC[C@@H]1O[C@@H](CC(=O)NCC2CCCCC2)C=C[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638661	phase I
BRD-K73336648	OC[C@H]1O[C@@H](CC(=O)NCC2CCCCC2)C=C[C@H]1NC(=O)Nc1cccc(F)c1	CID:54638662	phase I
BRD-K95352879	OC[C@@H]1O[C@H](CC(=O)NCC2CCCCC2)C=C[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638663	phase I
BRD-K35944577	OC[C@H]1O[C@H](CC(=O)NCC2CCCCC2)C=C[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638664	phase I
BRD-K40591230	OC[C@@H]1O[C@@H](CC(=O)NCC2CCCCC2)C=C[C@H]1NC(=O)Nc1cccc(F)c1	CID:54638665	phase I
BRD-K31418530	OC[C@H]1O[C@@H](CC(=O)NCC2CCCCC2)C=C[C@@H]1NC(=O)Nc1cccc(F)c1	CID:54638666	phase I
BRD-K44806584	OC[C@@H]1O[C@H](CC(=O)NCC2CCCCC2)C=C[C@H]1NC(=O)Nc1cccc(F)c1	CID:54638667	phase I
BRD-K78584123	OC[C@H]1O[C@H](CCNC(=O)Cc2ccncc2)CC[C@H]1NC(=O)C1CCC1	CID:54638668	phase I
BRD-K30377297	OC[C@@H]1O[C@@H](CCNC(=O)Cc2ccncc2)CC[C@@H]1NC(=O)C1CCC1	CID:54638669	phase I
BRD-K42182933	OC[C@H]1O[C@H](CCNC(=O)Cc2ccncc2)CC[C@@H]1NC(=O)C1CCC1	CID:54638670	phase I
BRD-K13706246	OC[C@@H]1O[C@@H](CCNC(=O)Cc2ccncc2)CC[C@H]1NC(=O)C1CCC1	CID:54638671	phase I
BRD-K05391634	OC[C@H]1O[C@@H](CCNC(=O)Cc2ccncc2)CC[C@@H]1NC(=O)C1CCC1	CID:54638672	phase I
BRD-K74192638	OC[C@H]1O[C@@H](CCNC(=O)Cc2ccncc2)CC[C@H]1NC(=O)C1CCC1	CID:54638673	phase I
BRD-K07748118	OC[C@@H]1O[C@H](CCNC(=O)Cc2ccncc2)CC[C@@H]1NC(=O)C1CCC1	CID:54638674	phase I
BRD-K66149656	OC[C@@H]1O[C@H](CCNC(=O)Cc2ccncc2)CC[C@H]1NC(=O)C1CCC1	CID:54638675	phase I
BRD-K46206861	CCCNC(=O)N[C@@H]1C=C[C@@H](CC(=O)NCCc2ccccc2)O[C@@H]1CO	CID:54638676	phase I
BRD-K74370838	CCCNC(=O)N[C@H]1C=C[C@H](CC(=O)NCCc2ccccc2)O[C@H]1CO	CID:54638677	phase I
BRD-K03876750	CCCNC(=O)N[C@@H]1C=C[C@H](CC(=O)NCCc2ccccc2)O[C@@H]1CO	CID:54638678	phase I
BRD-K35957449	CCCNC(=O)N[C@H]1C=C[C@@H](CC(=O)NCCc2ccccc2)O[C@H]1CO	CID:54638679	phase I
BRD-K22886798	CCCNC(=O)N[C@H]1C=C[C@@H](CC(=O)NCCc2ccccc2)O[C@@H]1CO	CID:54638680	phase I
BRD-K33012050	CCCNC(=O)N[C@@H]1C=C[C@H](CC(=O)NCCc2ccccc2)O[C@H]1CO	CID:54638681	phase I
BRD-K04680237	CCCNC(=O)N[C@H]1C=C[C@H](CC(=O)NCCc2ccccc2)O[C@@H]1CO	CID:54638682	phase I
BRD-K34407245	CCCNC(=O)N[C@@H]1C=C[C@@H](CC(=O)NCCc2ccccc2)O[C@H]1CO	CID:54638683	phase I
BRD-K62985789	CCS(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2ccccn2)O[C@@H]1CO	CID:54638684	phase I
BRD-K56581148	CCS(=O)(=O)N[C@H]1CC[C@@H](CC(=O)NCc2ccccn2)O[C@H]1CO	CID:54638685	phase I
BRD-K21478308	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638686	phase I
BRD-K19487261	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638687	phase I
BRD-K00150267	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638688	phase I
BRD-K68644714	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638689	phase I
BRD-K65378566	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638690	phase I
BRD-K94300226	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638691	phase I
BRD-K27927067	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638692	phase I
BRD-K51050762	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638693	phase I
BRD-K92986600	Cc1noc(C)c1NC(=O)NCC[C@@H]1CC[C@@H](NC(=O)c2ccc(F)cc2)[C@@H](CO)O1	CID:54638694	phase I
BRD-K72424685	Cc1noc(C)c1NC(=O)NCC[C@H]1CC[C@H](NC(=O)c2ccc(F)cc2)[C@H](CO)O1	CID:54638695	phase I
BRD-K28585560	Cc1noc(C)c1NC(=O)NCC[C@H]1CC[C@@H](NC(=O)c2ccc(F)cc2)[C@@H](CO)O1	CID:54638696	phase I
BRD-K69197680	Cc1noc(C)c1NC(=O)NCC[C@H]1CC[C@@H](NC(=O)c2ccc(F)cc2)[C@H](CO)O1	CID:54638697	phase I
BRD-K00382464	Cc1noc(C)c1NC(=O)NCC[C@H]1CC[C@H](NC(=O)c2ccc(F)cc2)[C@@H](CO)O1	CID:54638698	phase I
BRD-K21630495	Cc1noc(C)c1NC(=O)NCC[C@@H]1CC[C@H](NC(=O)c2ccc(F)cc2)[C@H](CO)O1	CID:54638699	phase I
BRD-K02847640	Cc1noc(C)c1NC(=O)NCC[C@@H]1CC[C@H](NC(=O)c2ccc(F)cc2)[C@@H](CO)O1	CID:54638700	phase I
BRD-K98980304	Cc1noc(C)c1NC(=O)NCC[C@@H]1CC[C@@H](NC(=O)c2ccc(F)cc2)[C@H](CO)O1	CID:54638701	phase I
BRD-K17655522	OC[C@H]1O[C@H](CC(=O)Nc2nccs2)C=C[C@H]1NC(=O)c1cccc(F)c1	CID:54638702	phase I
BRD-K84321619	OC[C@@H]1O[C@@H](CC(=O)Nc2nccs2)C=C[C@@H]1NC(=O)c1cccc(F)c1	CID:54638703	phase I
BRD-K66185487	OC[C@H]1O[C@@H](CC(=O)Nc2nccs2)C=C[C@H]1NC(=O)c1cccc(F)c1	CID:54638704	phase I
BRD-K19213530	OC[C@@H]1O[C@H](CC(=O)Nc2nccs2)C=C[C@@H]1NC(=O)c1cccc(F)c1	CID:54638705	phase I
BRD-K25037118	OC[C@H]1O[C@H](CC(=O)Nc2nccs2)C=C[C@@H]1NC(=O)c1cccc(F)c1	CID:54638706	phase I
BRD-K79277758	OC[C@@H]1O[C@@H](CC(=O)Nc2nccs2)C=C[C@H]1NC(=O)c1cccc(F)c1	CID:54638707	phase I
BRD-K52149447	OC[C@H]1O[C@@H](CC(=O)Nc2nccs2)C=C[C@@H]1NC(=O)c1cccc(F)c1	CID:54638708	phase I
BRD-K89299922	OC[C@@H]1O[C@H](CC(=O)Nc2nccs2)C=C[C@H]1NC(=O)c1cccc(F)c1	CID:54638709	phase I
BRD-K35786295	CCC(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2ccccc2F)O[C@@H]1CO	CID:54638710	phase I
BRD-K22664171	CCC(=O)N[C@H]1CC[C@H](CC(=O)NCc2ccccc2F)O[C@H]1CO	CID:54638711	phase I
BRD-K46561506	CCC(=O)N[C@@H]1CC[C@H](CC(=O)NCc2ccccc2F)O[C@@H]1CO	CID:54638712	phase I
BRD-K75894982	CCC(=O)N[C@H]1CC[C@@H](CC(=O)NCc2ccccc2F)O[C@H]1CO	CID:54638713	phase I
BRD-K32049912	CCC(=O)N[C@H]1CC[C@@H](CC(=O)NCc2ccccc2F)O[C@@H]1CO	CID:54638714	phase I
BRD-K87669574	CCC(=O)N[C@@H]1CC[C@H](CC(=O)NCc2ccccc2F)O[C@H]1CO	CID:54638715	phase I
BRD-K79145303	CCC(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2ccccc2F)O[C@H]1CO	CID:54638716	phase I
BRD-K16974571	COc1ccc(cc1)-c1cn(CC[C@@H]2CC[C@@H](NC(=O)CCN3CCCCC3)[C@@H](CO)O2)nn1	CID:54638717	phase I
BRD-K69722708	COc1ccc(cc1)-c1cn(CC[C@H]2CC[C@H](NC(=O)CCN3CCCCC3)[C@H](CO)O2)nn1	CID:54638718	phase I
BRD-K18589989	COc1ccc(cc1)-c1cn(CC[C@H]2CC[C@@H](NC(=O)CCN3CCCCC3)[C@H](CO)O2)nn1	CID:54638719	phase I
BRD-K36149190	COc1ccc(cc1)-c1cn(CC[C@H]2CC[C@@H](NC(=O)CCN3CCCCC3)[C@@H](CO)O2)nn1	CID:54638720	phase I
BRD-K85802361	COc1ccc(cc1)-c1cn(CC[C@@H]2CC[C@H](NC(=O)CCN3CCCCC3)[C@H](CO)O2)nn1	CID:54638721	phase I
BRD-K00946569	COc1ccc(cc1)-c1cn(CC[C@@H]2CC[C@H](NC(=O)CCN3CCCCC3)[C@@H](CO)O2)nn1	CID:54638722	phase I
BRD-K15750053	COc1ccc(cc1)-c1cn(CC[C@H]2CC[C@H](NC(=O)CCN3CCCCC3)[C@@H](CO)O2)nn1	CID:54638723	phase I
BRD-K64704452	COc1ccc(cc1)-c1cn(CC[C@@H]2CC[C@@H](NC(=O)CCN3CCCCC3)[C@H](CO)O2)nn1	CID:54638724	phase I
BRD-K88385750	CN(C)C(=O)C[C@@H]1CC[C@@H](NC(=O)C2CCOCC2)[C@@H](CO)O1	CID:54638725	phase I
BRD-K08005469	CN(C)C(=O)C[C@H]1CC[C@H](NC(=O)C2CCOCC2)[C@H](CO)O1	CID:54638726	phase I
BRD-K22275321	CN(C)C(=O)C[C@H]1CC[C@@H](NC(=O)C2CCOCC2)[C@@H](CO)O1	CID:54638727	phase I
BRD-K23958338	CN(C)C(=O)C[C@@H]1CC[C@H](NC(=O)C2CCOCC2)[C@H](CO)O1	CID:54638728	phase I
BRD-K43714262	CN(C)C(=O)C[C@@H]1CC[C@H](NC(=O)C2CCOCC2)[C@@H](CO)O1	CID:54638729	phase I
BRD-K14952621	CN(C)C(=O)C[C@H]1CC[C@@H](NC(=O)C2CCOCC2)[C@H](CO)O1	CID:54638730	phase I
BRD-K89321975	CN(C)C(=O)C[C@H]1CC[C@H](NC(=O)C2CCOCC2)[C@@H](CO)O1	CID:54638731	phase I
BRD-K91498722	CN(C)C(=O)C[C@@H]1CC[C@@H](NC(=O)C2CCOCC2)[C@H](CO)O1	CID:54638732	phase I
BRD-K67663786	OC[C@H]1O[C@H](CC(O)=O)C=C[C@H]1NC(=O)c1ccccc1F	CID:54638733	phase I
BRD-K85644737	OC[C@@H]1O[C@@H](CC(O)=O)C=C[C@@H]1NC(=O)c1ccccc1F	CID:54638734	phase I
BRD-K80101280	OC[C@@H]1O[C@H](CC(O)=O)C=C[C@@H]1NC(=O)c1ccccc1F	CID:54638735	phase I
BRD-K75996234	OC[C@H]1O[C@H](CC(O)=O)C=C[C@@H]1NC(=O)c1ccccc1F	CID:54638736	phase I
BRD-K03088187	OC[C@@H]1O[C@@H](CC(O)=O)C=C[C@H]1NC(=O)c1ccccc1F	CID:54638737	phase I
BRD-K74042281	OC[C@H]1O[C@@H](CC(O)=O)C=C[C@@H]1NC(=O)c1ccccc1F	CID:54638738	phase I
BRD-K13012607	OC[C@@H]1O[C@H](CC(O)=O)C=C[C@H]1NC(=O)c1ccccc1F	CID:54638739	phase I
BRD-K67359324	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638740	phase I
BRD-K42478399	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638741	phase I
BRD-K85079232	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638742	phase I
BRD-K62773636	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638743	phase I
BRD-K85699864	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638744	phase I
BRD-K02041150	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638745	phase I
BRD-K78227082	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638746	phase I
BRD-K82462389	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)cc(F)c2)CC[C@H]1NC(=O)Nc1ccc(cc1)C(F)(F)F	CID:54638747	phase I
BRD-K20163346	OC[C@H]1O[C@H](CCNC(=O)CCN2CCCCC2)CC[C@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638748	phase I
BRD-K10657952	OC[C@H]1O[C@@H](CCNC(=O)CCN2CCCCC2)CC[C@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638749	phase I
BRD-K50115811	OC[C@@H]1O[C@@H](CCNC(=O)CCN2CCCCC2)CC[C@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638750	phase I
BRD-K81559336	OC[C@@H]1O[C@H](CCNC(=O)CCN2CCCCC2)CC[C@@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638751	phase I
BRD-K47018052	OC[C@H]1O[C@H](CCNC(=O)CCN2CCCCC2)CC[C@@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638752	phase I
BRD-K84935712	OC[C@H]1O[C@@H](CCNC(=O)CCN2CCCCC2)CC[C@@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638753	phase I
BRD-K08040026	OC[C@@H]1O[C@H](CCNC(=O)CCN2CCCCC2)CC[C@H]1NS(=O)(=O)c1cccc(Cl)c1	CID:54638754	phase I
BRD-K39929061	COC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638755	phase I
BRD-K83322422	COC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2ccccc2F)[C@H](CO)O1	CID:54638756	phase I
BRD-K16195900	COC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638757	phase I
BRD-K22447604	COC(=O)C[C@@H]1CC[C@H](NS(=O)(=O)c2ccccc2F)[C@H](CO)O1	CID:54638758	phase I
BRD-K58610656	COC(=O)C[C@H]1CC[C@@H](NS(=O)(=O)c2ccccc2F)[C@H](CO)O1	CID:54638759	phase I
BRD-K09032125	COC(=O)C[C@H]1CC[C@H](NS(=O)(=O)c2ccccc2F)[C@@H](CO)O1	CID:54638760	phase I
BRD-K49093373	COC(=O)C[C@@H]1CC[C@@H](NS(=O)(=O)c2ccccc2F)[C@H](CO)O1	CID:54638761	phase I
BRD-K53507509	CC(C)NC(=O)NCC[C@@H]1CC[C@@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@@H](CO)O1	CID:54638762	phase I
BRD-K85528826	CC(C)NC(=O)NCC[C@H]1CC[C@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@H](CO)O1	CID:54638763	phase I
BRD-K12970833	CC(C)NC(=O)NCC[C@H]1CC[C@@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@H](CO)O1	CID:54638764	phase I
BRD-K52904986	CC(C)NC(=O)NCC[C@H]1CC[C@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@@H](CO)O1	CID:54638765	phase I
BRD-K27299383	CC(C)NC(=O)NCC[C@H]1CC[C@@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@@H](CO)O1	CID:54638766	phase I
BRD-K90208654	CC(C)NC(=O)NCC[C@@H]1CC[C@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@H](CO)O1	CID:54638767	phase I
BRD-K66184091	CC(C)NC(=O)NCC[C@@H]1CC[C@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@@H](CO)O1	CID:54638768	phase I
BRD-K67661368	CC(C)NC(=O)NCC[C@@H]1CC[C@@H](NS(=O)(=O)c2ccc(Oc3ccccc3)cc2)[C@H](CO)O1	CID:54638769	phase I
BRD-K49907578	COC(=O)C[C@H]1O[C@H](CO)[C@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638770	phase I
BRD-K56945204	COC(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638771	phase I
BRD-K13779607	COC(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638772	phase I
BRD-K77273736	COC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638773	phase I
BRD-K36513323	COC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638774	phase I
BRD-K39132590	COC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638775	phase I
BRD-K07382790	COC(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638776	phase I
BRD-K28358982	COC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C=C1	CID:54638777	phase I
BRD-K76688030	OC[C@H]1O[C@@H](C=C[C@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638778	phase I
BRD-K21033948	OC[C@@H]1O[C@H](C=C[C@@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638779	phase I
BRD-K08920503	OC[C@H]1O[C@H](C=C[C@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638780	phase I
BRD-K44229115	OC[C@@H]1O[C@@H](C=C[C@@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638781	phase I
BRD-K49276305	OC[C@H]1O[C@@H](C=C[C@@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638782	phase I
BRD-K73400194	OC[C@@H]1O[C@H](C=C[C@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638783	phase I
BRD-K83072410	OC[C@H]1O[C@H](C=C[C@@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638784	phase I
BRD-K38188442	OC[C@@H]1O[C@@H](C=C[C@H]1NC(=O)Cc1cccnc1)CC(=O)Nc1ccccc1	CID:54638785	phase I
BRD-K93140279	OC[C@H]1O[C@H](CC(=O)N2CCCCC2)C=C[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638786	phase I
BRD-K41571462	OC[C@@H]1O[C@@H](CC(=O)N2CCCCC2)C=C[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638787	phase I
BRD-K92810472	OC[C@H]1O[C@@H](CC(=O)N2CCCCC2)C=C[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638788	phase I
BRD-K05726929	OC[C@@H]1O[C@H](CC(=O)N2CCCCC2)C=C[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638789	phase I
BRD-K11081110	OC[C@H]1O[C@H](CC(=O)N2CCCCC2)C=C[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638790	phase I
BRD-K96160456	OC[C@@H]1O[C@@H](CC(=O)N2CCCCC2)C=C[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638791	phase I
BRD-K95244186	OC[C@H]1O[C@@H](CC(=O)N2CCCCC2)C=C[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638792	phase I
BRD-K78467731	OC[C@@H]1O[C@H](CC(=O)N2CCCCC2)C=C[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638793	phase I
BRD-K24339152	Cc1ccc(cc1)S(=O)(=O)NCC[C@@H]1CC[C@@H](NC(=O)CC2CC2)[C@@H](CO)O1	CID:54638794	phase I
BRD-K00695053	Cc1ccc(cc1)S(=O)(=O)NCC[C@H]1CC[C@H](NC(=O)CC2CC2)[C@H](CO)O1	CID:54638795	phase I
BRD-K58072864	Cc1ccc(cc1)S(=O)(=O)NCC[C@H]1CC[C@@H](NC(=O)CC2CC2)[C@@H](CO)O1	CID:54638796	phase I
BRD-K15142057	Cc1ccc(cc1)S(=O)(=O)NCC[C@H]1CC[C@@H](NC(=O)CC2CC2)[C@H](CO)O1	CID:54638797	phase I
BRD-K19729667	Cc1ccc(cc1)S(=O)(=O)NCC[C@H]1CC[C@H](NC(=O)CC2CC2)[C@@H](CO)O1	CID:54638798	phase I
BRD-K31931379	Cc1ccc(cc1)S(=O)(=O)NCC[C@@H]1CC[C@H](NC(=O)CC2CC2)[C@H](CO)O1	CID:54638799	phase I
BRD-K94177318	Cc1ccc(cc1)S(=O)(=O)NCC[C@@H]1CC[C@H](NC(=O)CC2CC2)[C@@H](CO)O1	CID:54638800	phase I
BRD-K68201904	Cc1ccc(cc1)S(=O)(=O)NCC[C@@H]1CC[C@@H](NC(=O)CC2CC2)[C@H](CO)O1	CID:54638801	phase I
BRD-K33761091	CN(C)Cc1cn(CC[C@@H]2CC[C@@H](NC(=O)Cc3cccnc3)[C@@H](CO)O2)nn1	CID:54638802	phase I
BRD-K89255395	CN(C)Cc1cn(CC[C@H]2CC[C@H](NC(=O)Cc3cccnc3)[C@H](CO)O2)nn1	CID:54638803	phase I
BRD-K62220055	CN(C)Cc1cn(CC[C@@H]2CC[C@H](NC(=O)Cc3cccnc3)[C@@H](CO)O2)nn1	CID:54638804	phase I
BRD-K50608891	CN(C)Cc1cn(CC[C@H]2CC[C@@H](NC(=O)Cc3cccnc3)[C@H](CO)O2)nn1	CID:54638805	phase I
BRD-K46096244	CN(C)Cc1cn(CC[C@H]2CC[C@H](NC(=O)Cc3cccnc3)[C@@H](CO)O2)nn1	CID:54638806	phase I
BRD-K18844601	CN(C)Cc1cn(CC[C@H]2CC[C@@H](NC(=O)Cc3cccnc3)[C@@H](CO)O2)nn1	CID:54638807	phase I
BRD-K45682001	CN(C)Cc1cn(CC[C@@H]2CC[C@H](NC(=O)Cc3cccnc3)[C@H](CO)O2)nn1	CID:54638808	phase I
BRD-K82118651	CN(C)Cc1cn(CC[C@@H]2CC[C@@H](NC(=O)Cc3cccnc3)[C@H](CO)O2)nn1	CID:54638809	phase I
BRD-K48703433	COCC(=O)N[C@@H]1C=C[C@H](O[C@@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638810	phase I
BRD-K32350897	COCC(=O)N[C@H]1C=C[C@@H](O[C@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638811	phase I
BRD-K09130601	COCC(=O)N[C@@H]1C=C[C@@H](O[C@@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638812	phase I
BRD-K62465706	COCC(=O)N[C@H]1C=C[C@H](O[C@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638813	phase I
BRD-K18234030	COCC(=O)N[C@H]1C=C[C@H](O[C@@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638814	phase I
BRD-K47368357	COCC(=O)N[C@@H]1C=C[C@@H](O[C@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638815	phase I
BRD-K24213763	COCC(=O)N[C@H]1C=C[C@@H](O[C@@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638816	phase I
BRD-K74390607	COCC(=O)N[C@@H]1C=C[C@H](O[C@H]1CO)CC(=O)NCc1ccc(Cl)cc1	CID:54638817	phase I
BRD-K78830924	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@H]1NC(=O)CC1CC1	CID:54638818	phase I
BRD-K82488679	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@@H]1NC(=O)CC1CC1	CID:54638819	phase I
BRD-K15892609	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@H]1NC(=O)CC1CC1	CID:54638820	phase I
BRD-K87361616	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@@H]1NC(=O)CC1CC1	CID:54638821	phase I
BRD-K48211564	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@@H]1NC(=O)CC1CC1	CID:54638822	phase I
BRD-K82096551	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@H]1NC(=O)CC1CC1	CID:54638823	phase I
BRD-K14768863	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@@H]1NC(=O)CC1CC1	CID:54638824	phase I
BRD-K76574148	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)CC[C@H]1NC(=O)CC1CC1	CID:54638825	phase I
BRD-K60474343	COc1ccccc1S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54638826	phase I
BRD-K40064462	COc1ccccc1S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54638827	phase I
BRD-K21855096	COc1ccccc1S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54638828	phase I
BRD-K86857638	COc1ccccc1S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54638829	phase I
BRD-K31545458	COc1ccccc1S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54638830	phase I
BRD-K28968484	COc1ccccc1S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54638831	phase I
BRD-K36708799	COc1ccccc1S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54638832	phase I
BRD-K07563916	COc1ccccc1S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54638833	phase I
BRD-K31028119	OC[C@H]1O[C@H](CC(=O)Nc2nccs2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54638834	phase I
BRD-K15178935	OC[C@@H]1O[C@@H](CC(=O)Nc2nccs2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54638835	phase I
BRD-K57277442	OC[C@H]1O[C@H](CC(=O)Nc2nccs2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54638836	phase I
BRD-K89029303	OC[C@@H]1O[C@@H](CC(=O)Nc2nccs2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54638837	phase I
BRD-K11266478	OC[C@H]1O[C@@H](CC(=O)Nc2nccs2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54638838	phase I
BRD-K23584424	OC[C@@H]1O[C@H](CC(=O)Nc2nccs2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54638839	phase I
BRD-K61025685	OC[C@H]1O[C@H](CCn2cc(nn2)-c2ccccc2F)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638840	phase I
BRD-K55341911	OC[C@@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2F)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638841	phase I
BRD-K93525097	OC[C@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2F)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638842	phase I
BRD-K80213755	OC[C@@H]1O[C@H](CCn2cc(nn2)-c2ccccc2F)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54638843	phase I
BRD-K18567420	OC[C@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2F)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638844	phase I
BRD-K19915020	OC[C@@H]1O[C@H](CCn2cc(nn2)-c2ccccc2F)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54638845	phase I
BRD-K51810646	OC[C@H]1O[C@H](CCNC(=O)C2CCCCC2)CC[C@H]1NC(=O)Nc1ccccc1F	CID:54638846	phase I
BRD-K18480277	OC[C@H]1O[C@@H](CCNC(=O)C2CCCCC2)CC[C@H]1NC(=O)Nc1ccccc1F	CID:54638849	phase I
BRD-K19426893	OC[C@@H]1O[C@H](CCNC(=O)C2CCCCC2)CC[C@@H]1NC(=O)Nc1ccccc1F	CID:54638850	phase I
BRD-K09397553	OC[C@H]1O[C@H](CCNC(=O)C2CCCCC2)CC[C@@H]1NC(=O)Nc1ccccc1F	CID:54638851	phase I
BRD-K87517219	OC[C@H]1O[C@@H](CCNC(=O)C2CCCCC2)CC[C@@H]1NC(=O)Nc1ccccc1F	CID:54638852	phase I
BRD-K76166520	OC[C@@H]1O[C@H](CCNC(=O)C2CCCCC2)CC[C@H]1NC(=O)Nc1ccccc1F	CID:54638853	phase I
BRD-K75095704	COc1cccc(c1)-c1cn(CC[C@@H]2CC[C@@H](NS(=O)(=O)Cc3ccccc3)[C@@H](CO)O2)nn1	CID:54638854	phase I
BRD-K21643869	COc1cccc(c1)-c1cn(CC[C@H]2CC[C@H](NS(=O)(=O)Cc3ccccc3)[C@H](CO)O2)nn1	CID:54638855	phase I
BRD-K26862028	COc1cccc(c1)-c1cn(CC[C@H]2CC[C@@H](NS(=O)(=O)Cc3ccccc3)[C@@H](CO)O2)nn1	CID:54638856	phase I
BRD-K88652561	COc1cccc(c1)-c1cn(CC[C@@H]2CC[C@H](NS(=O)(=O)Cc3ccccc3)[C@H](CO)O2)nn1	CID:54638857	phase I
BRD-K73701301	COc1cccc(c1)-c1cn(CC[C@H]2CC[C@H](NS(=O)(=O)Cc3ccccc3)[C@@H](CO)O2)nn1	CID:54638858	phase I
BRD-K08972808	COc1cccc(c1)-c1cn(CC[C@@H]2CC[C@@H](NS(=O)(=O)Cc3ccccc3)[C@H](CO)O2)nn1	CID:54638859	phase I
BRD-K41597316	COc1ccccc1NC(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)C2(O)CCCC2)O[C@@H]1CO	CID:54638860	phase I
BRD-K63285694	COc1ccccc1NC(=O)N[C@H]1CC[C@H](CCn2cc(nn2)C2(O)CCCC2)O[C@H]1CO	CID:54638861	phase I
BRD-K27483344	COc1ccccc1NC(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)C2(O)CCCC2)O[C@H]1CO	CID:54638862	phase I
BRD-K29371459	COc1ccccc1NC(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)C2(O)CCCC2)O[C@@H]1CO	CID:54638863	phase I
BRD-K52473019	COc1ccccc1NC(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)C2(O)CCCC2)O[C@H]1CO	CID:54638864	phase I
BRD-K38037265	COc1ccccc1NC(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)C2(O)CCCC2)O[C@@H]1CO	CID:54638865	phase I
BRD-K21536131	COc1ccccc1NC(=O)N[C@H]1CC[C@H](CCn2cc(nn2)C2(O)CCCC2)O[C@@H]1CO	CID:54638866	phase I
BRD-K76462626	COc1ccccc1NC(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)C2(O)CCCC2)O[C@H]1CO	CID:54638867	phase I
BRD-K09623383	OC[C@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638868	phase I
BRD-K84024786	OC[C@@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638871	phase I
BRD-K13275849	OC[C@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638872	phase I
BRD-K13299591	OC[C@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638873	phase I
BRD-K74511610	OC[C@@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@@H]1NC(=O)CN1CCOCC1	CID:54638874	phase I
BRD-K12718908	OC[C@@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@H]1NC(=O)CN1CCOCC1	CID:54638875	phase I
BRD-K58539957	OC[C@H]1O[C@H](CC(=O)NCC2CC2)C=C[C@H]1NC(=O)c1ccncc1	CID:54638876	phase I
BRD-K67673602	OC[C@@H]1O[C@@H](CC(=O)NCC2CC2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54638877	phase I
BRD-K37684537	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54638878	phase I
BRD-K22215387	OC[C@H]1O[C@H](CC(=O)NCC2CC2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54638879	phase I
BRD-K84715825	OC[C@@H]1O[C@@H](CC(=O)NCC2CC2)C=C[C@H]1NC(=O)c1ccncc1	CID:54638880	phase I
BRD-K64120525	OC[C@H]1O[C@@H](CC(=O)NCC2CC2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54638881	phase I
BRD-K66378473	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)C=C[C@H]1NC(=O)c1ccncc1	CID:54638882	phase I
BRD-K22109269	Cc1ccccc1S(=O)(=O)NCC[C@@H]1CC[C@@H](NS(=O)(=O)c2ccccc2C)[C@@H](CO)O1	CID:54638883	phase I
BRD-K13304927	Cc1ccccc1S(=O)(=O)NCC[C@H]1CC[C@H](NS(=O)(=O)c2ccccc2C)[C@H](CO)O1	CID:54638884	phase I
BRD-K62917551	Cc1ccccc1S(=O)(=O)NCC[C@@H]1CC[C@H](NS(=O)(=O)c2ccccc2C)[C@@H](CO)O1	CID:54638885	phase I
BRD-K73340768	Cc1ccccc1S(=O)(=O)NCC[C@H]1CC[C@@H](NS(=O)(=O)c2ccccc2C)[C@H](CO)O1	CID:54638886	phase I
BRD-K25688236	Cc1ccccc1S(=O)(=O)NCC[C@H]1CC[C@@H](NS(=O)(=O)c2ccccc2C)[C@@H](CO)O1	CID:54638887	phase I
BRD-K24084946	Cc1ccccc1S(=O)(=O)NCC[C@@H]1CC[C@H](NS(=O)(=O)c2ccccc2C)[C@H](CO)O1	CID:54638888	phase I
BRD-K41927787	Cc1ccccc1S(=O)(=O)NCC[C@H]1CC[C@H](NS(=O)(=O)c2ccccc2C)[C@@H](CO)O1	CID:54638889	phase I
BRD-K88114920	Cc1ccccc1S(=O)(=O)NCC[C@@H]1CC[C@@H](NS(=O)(=O)c2ccccc2C)[C@H](CO)O1	CID:54638890	phase I
BRD-K63813530	C[C@@H](NC(=O)C[C@H]1CC[C@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638891	phase I
BRD-K95041551	C[C@H](NC(=O)C[C@H]1CC[C@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638892	phase I
BRD-K93763482	C[C@H](NC(=O)C[C@@H]1CC[C@@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638893	phase I
BRD-K77660367	C[C@@H](NC(=O)C[C@@H]1CC[C@@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638894	phase I
BRD-K77182083	C[C@@H](NC(=O)C[C@H]1CC[C@@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638895	phase I
BRD-K25234731	C[C@H](NC(=O)C[C@H]1CC[C@@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638896	phase I
BRD-K66910993	C[C@@H](NC(=O)C[C@@H]1CC[C@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638897	phase I
BRD-K78419283	C[C@H](NC(=O)C[C@@H]1CC[C@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638898	phase I
BRD-K89062214	C[C@H](NC(=O)C[C@@H]1CC[C@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638899	phase I
BRD-K97440159	C[C@@H](NC(=O)C[C@@H]1CC[C@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638900	phase I
BRD-K77221189	C[C@H](NC(=O)C[C@H]1CC[C@@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638901	phase I
BRD-K62213032	C[C@@H](NC(=O)C[C@H]1CC[C@@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638902	phase I
BRD-K59183712	C[C@@H](NC(=O)C[C@H]1CC[C@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638903	phase I
BRD-K21472896	C[C@H](NC(=O)C[C@H]1CC[C@H](NC(=O)c2cccnc2)[C@@H](CO)O1)c1ccccc1	CID:54638904	phase I
BRD-K71552149	C[C@@H](NC(=O)C[C@@H]1CC[C@@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638905	phase I
BRD-K88104720	C[C@H](NC(=O)C[C@@H]1CC[C@@H](NC(=O)c2cccnc2)[C@H](CO)O1)c1ccccc1	CID:54638906	phase I
BRD-K54199214	OC[C@H]1O[C@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@H]1NC(=O)c1ccccn1	CID:54638907	phase I
BRD-K82062373	OC[C@@H]1O[C@@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638908	phase I
BRD-K92951265	OC[C@H]1O[C@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638909	phase I
BRD-K40478655	OC[C@@H]1O[C@@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@H]1NC(=O)c1ccccn1	CID:54638910	phase I
BRD-K02545368	OC[C@H]1O[C@@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638911	phase I
BRD-K26399147	OC[C@H]1O[C@@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@H]1NC(=O)c1ccccn1	CID:54638912	phase I
BRD-K09845511	OC[C@@H]1O[C@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@@H]1NC(=O)c1ccccn1	CID:54638913	phase I
BRD-K19752742	OC[C@@H]1O[C@H](CCNS(=O)(=O)c2ccc(Cl)cc2)CC[C@H]1NC(=O)c1ccccn1	CID:54638914	phase I
BRD-K29567467	OC[C@H]1O[C@H](CCn2cc(nn2)C2CC2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638915	phase I
BRD-K54202584	OC[C@@H]1O[C@@H](CCn2cc(nn2)C2CC2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638916	phase I
BRD-K31705167	OC[C@@H]1O[C@@H](CCn2cc(nn2)C2CC2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638917	phase I
BRD-K32972218	OC[C@H]1O[C@@H](CCn2cc(nn2)C2CC2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638918	phase I
BRD-K23872111	OC[C@H]1O[C@@H](CCn2cc(nn2)C2CC2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638919	phase I
BRD-K06380464	OC[C@@H]1O[C@H](CCn2cc(nn2)C2CC2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638920	phase I
BRD-K23301583	OC[C@H]1O[C@H](CCn2cc(nn2)C2CC2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638921	phase I
BRD-K35035541	OC[C@@H]1O[C@H](CCn2cc(nn2)C2CC2)CC[C@H]1NC(=O)Nc1cc(F)ccc1F	CID:54638922	phase I
BRD-K60092199	CC(C)NC(=O)N[C@@H]1CC[C@@H](CCN)O[C@@H]1CO	CID:54638923	phase I
BRD-K92036763	CC(C)NC(=O)N[C@H]1CC[C@H](CCN)O[C@H]1CO	CID:54638924	phase I
BRD-K56298028	CC(C)NC(=O)N[C@@H]1CC[C@H](CCN)O[C@H]1CO	CID:54638925	phase I
BRD-K09804899	CC(C)NC(=O)N[C@H]1CC[C@H](CCN)O[C@@H]1CO	CID:54638926	phase I
BRD-K42256568	CC(C)NC(=O)N[C@@H]1CC[C@H](CCN)O[C@@H]1CO	CID:54638927	phase I
BRD-K64497770	CC(C)NC(=O)N[C@H]1CC[C@@H](CCN)O[C@H]1CO	CID:54638928	phase I
BRD-K23876588	CC(C)NC(=O)N[C@@H]1CC[C@@H](CCN)O[C@H]1CO	CID:54638929	phase I
BRD-K00262667	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638930	phase I
BRD-K07456098	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638931	phase I
BRD-K44801029	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638932	phase I
BRD-K10134498	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638933	phase I
BRD-K36232819	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638934	phase I
BRD-K30377815	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638935	phase I
BRD-K70447364	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638936	phase I
BRD-K19325173	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)c(Cl)c2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54638937	phase I
BRD-K93713304	OC[C@H]1O[C@H](CC(=O)NC2CCC2)C=C[C@H]1NC(=O)C1CC1	CID:54638938	phase I
BRD-K00544996	OC[C@@H]1O[C@@H](CC(=O)NC2CCC2)C=C[C@@H]1NC(=O)C1CC1	CID:54638939	phase I
BRD-K88328468	OC[C@H]1O[C@@H](CC(=O)NC2CCC2)C=C[C@H]1NC(=O)C1CC1	CID:54638940	phase I
BRD-K52971351	OC[C@@H]1O[C@H](CC(=O)NC2CCC2)C=C[C@@H]1NC(=O)C1CC1	CID:54638941	phase I
BRD-K80893668	OC[C@H]1O[C@H](CC(=O)NC2CCC2)C=C[C@@H]1NC(=O)C1CC1	CID:54638942	phase I
BRD-K27699706	OC[C@@H]1O[C@@H](CC(=O)NC2CCC2)C=C[C@H]1NC(=O)C1CC1	CID:54638943	phase I
BRD-K00175211	OC[C@H]1O[C@@H](CC(=O)NC2CCC2)C=C[C@@H]1NC(=O)C1CC1	CID:54638944	phase I
BRD-K94711641	OC[C@@H]1O[C@H](CC(=O)NC2CCC2)C=C[C@H]1NC(=O)C1CC1	CID:54638945	phase I
BRD-K70766049	OC[C@H]1O[C@H](CCn2cc(nn2)-c2ccccc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638946	phase I
BRD-K83400219	OC[C@@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638947	phase I
BRD-K85806228	OC[C@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638948	phase I
BRD-K85664836	OC[C@@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638949	phase I
BRD-K77564294	OC[C@@H]1O[C@H](CCn2cc(nn2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638950	phase I
BRD-K74140407	OC[C@H]1O[C@H](CCn2cc(nn2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638951	phase I
BRD-K45358679	OC[C@H]1O[C@@H](CCn2cc(nn2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638952	phase I
BRD-K54627309	OC[C@@H]1O[C@H](CCn2cc(nn2)-c2ccccc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638953	phase I
BRD-K41440211	C[C@@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638954	phase I
BRD-K60188503	C[C@@H](NC(=O)C[C@@H]1O[C@H](CO)[C@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638955	phase I
BRD-K15477190	C[C@H](NC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638956	phase I
BRD-K77918164	C[C@@H](NC(=O)C[C@H]1O[C@@H](CO)[C@@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638957	phase I
BRD-K52938793	C[C@H](NC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638958	phase I
BRD-K89112856	C[C@@H](NC(=O)C[C@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638959	phase I
BRD-K82991167	C[C@@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638960	phase I
BRD-K73573525	C[C@H](NC(=O)C[C@@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638961	phase I
BRD-K75938736	C[C@@H](NC(=O)C[C@@H]1O[C@H](CO)[C@@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638962	phase I
BRD-K07678162	C[C@H](NC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638963	phase I
BRD-K20220643	C[C@@H](NC(=O)C[C@H]1O[C@@H](CO)[C@H](NC(=O)Nc2ccc3OCOc3c2)C=C1)c1ccccc1	CID:54638964	phase I
BRD-K81189877	OC[C@H]1O[C@H](CCNC(=O)c2ccc(F)cc2)CC[C@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638965	phase I
BRD-K70237789	OC[C@@H]1O[C@@H](CCNC(=O)c2ccc(F)cc2)CC[C@@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638966	phase I
BRD-K31099173	OC[C@@H]1O[C@@H](CCNC(=O)c2ccc(F)cc2)CC[C@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638967	phase I
BRD-K06155953	OC[C@H]1O[C@@H](CCNC(=O)c2ccc(F)cc2)CC[C@@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638968	phase I
BRD-K47995524	OC[C@H]1O[C@@H](CCNC(=O)c2ccc(F)cc2)CC[C@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638969	phase I
BRD-K20307883	OC[C@@H]1O[C@H](CCNC(=O)c2ccc(F)cc2)CC[C@@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638970	phase I
BRD-K11097458	OC[C@H]1O[C@H](CCNC(=O)c2ccc(F)cc2)CC[C@@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638971	phase I
BRD-K34898196	OC[C@@H]1O[C@H](CCNC(=O)c2ccc(F)cc2)CC[C@H]1NC(=O)Nc1ccc(Cl)c(Cl)c1	CID:54638972	phase I
BRD-K88968415	COc1ccccc1NC(=O)N[C@@H]1CC[C@@H](CCNS(=O)(=O)c2ccccc2)O[C@@H]1CO	CID:54638973	phase I
BRD-K71799397	COc1ccccc1NC(=O)N[C@H]1CC[C@H](CCNS(=O)(=O)c2ccccc2)O[C@H]1CO	CID:54638974	phase I
BRD-K63211622	COc1ccccc1NC(=O)N[C@H]1CC[C@@H](CCNS(=O)(=O)c2ccccc2)O[C@@H]1CO	CID:54638975	phase I
BRD-K26128727	COc1ccccc1NC(=O)N[C@@H]1CC[C@H](CCNS(=O)(=O)c2ccccc2)O[C@H]1CO	CID:54638976	phase I
BRD-K44547539	COc1ccccc1NC(=O)N[C@H]1CC[C@H](CCNS(=O)(=O)c2ccccc2)O[C@@H]1CO	CID:54638977	phase I
BRD-K10721194	COc1ccccc1NC(=O)N[C@@H]1CC[C@H](CCNS(=O)(=O)c2ccccc2)O[C@@H]1CO	CID:54638978	phase I
BRD-K63269129	COc1ccccc1NC(=O)N[C@H]1CC[C@@H](CCNS(=O)(=O)c2ccccc2)O[C@H]1CO	CID:54638979	phase I
BRD-K99700039	COc1ccccc1NC(=O)N[C@@H]1CC[C@@H](CCNS(=O)(=O)c2ccccc2)O[C@H]1CO	CID:54638980	phase I
BRD-K64556793	OC[C@H]1O[C@H](CC(=O)NCCN2CCCC2)CC[C@H]1NC(=O)c1cccc(F)c1	CID:54638981	phase I
BRD-K98881366	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCC2)CC[C@@H]1NC(=O)c1cccc(F)c1	CID:54638982	phase I
BRD-K04585040	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCC2)CC[C@H]1NC(=O)c1cccc(F)c1	CID:54638983	phase I
BRD-K32068846	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCC2)CC[C@@H]1NC(=O)c1cccc(F)c1	CID:54638984	phase I
BRD-K42960483	OC[C@H]1O[C@H](CC(=O)NCCN2CCCC2)CC[C@@H]1NC(=O)c1cccc(F)c1	CID:54638985	phase I
BRD-K22562809	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCC2)CC[C@H]1NC(=O)c1cccc(F)c1	CID:54638986	phase I
BRD-K72261411	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCC2)CC[C@@H]1NC(=O)c1cccc(F)c1	CID:54638987	phase I
BRD-K36160951	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCC2)CC[C@H]1NC(=O)c1cccc(F)c1	CID:54638988	phase I
BRD-K98830854	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccncc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638989	phase I
BRD-K62143565	OC[C@H]1O[C@H](CC(=O)NCCc2ccncc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638990	phase I
BRD-K10645566	OC[C@H]1O[C@@H](CC(=O)NCCc2ccncc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638991	phase I
BRD-K85861721	OC[C@@H]1O[C@H](CC(=O)NCCc2ccncc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638992	phase I
BRD-K41863121	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccncc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638993	phase I
BRD-K60360711	OC[C@H]1O[C@H](CC(=O)NCCc2ccncc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638994	phase I
BRD-K01352631	OC[C@H]1O[C@@H](CC(=O)NCCc2ccncc2)CC[C@@H]1NC(=O)Cc1ccccn1	CID:54638995	phase I
BRD-K74009886	OC[C@@H]1O[C@H](CC(=O)NCCc2ccncc2)CC[C@H]1NC(=O)Cc1ccccn1	CID:54638996	phase I
BRD-K45383509	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)C2CCCCC2)O[C@@H]1CO	CID:54638997	phase I
BRD-K82830100	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@H](CCn2cc(nn2)C2CCCCC2)O[C@H]1CO	CID:54638998	phase I
BRD-K67518269	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@H](CCn2cc(nn2)C2CCCCC2)O[C@@H]1CO	CID:54638999	phase I
BRD-K31487253	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@@H](CCn2cc(nn2)C2CCCCC2)O[C@H]1CO	CID:54639000	phase I
BRD-K32453902	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@H](CCn2cc(nn2)C2CCCCC2)O[C@@H]1CO	CID:54639001	phase I
BRD-K90233481	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@@H](CCn2cc(nn2)C2CCCCC2)O[C@H]1CO	CID:54639002	phase I
BRD-K90505752	OC[C@H]1O[C@H](CCNC(=O)CN2CCOCC2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639003	phase I
BRD-K59330510	OC[C@H]1O[C@@H](CCNC(=O)CN2CCOCC2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639004	phase I
BRD-K54980807	OC[C@@H]1O[C@@H](CCNC(=O)CN2CCOCC2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639005	phase I
BRD-K82925070	OC[C@@H]1O[C@@H](CCNC(=O)CN2CCOCC2)CC[C@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639006	phase I
BRD-K28421747	OC[C@H]1O[C@@H](CCNC(=O)CN2CCOCC2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639007	phase I
BRD-K45221651	OC[C@@H]1O[C@H](CCNC(=O)CN2CCOCC2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639008	phase I
BRD-K08995626	OC[C@H]1O[C@H](CCNC(=O)CN2CCOCC2)CC[C@@H]1NS(=O)(=O)c1ccc(F)cc1	CID:54639009	phase I
BRD-K67328514	OC[C@H]1O[C@H](CC(=O)NCC2CC2)CC[C@H]1NC(=O)C1CCC1	CID:54639010	phase I
BRD-K70765133	OC[C@@H]1O[C@@H](CC(=O)NCC2CC2)CC[C@@H]1NC(=O)C1CCC1	CID:54639011	phase I
BRD-K63366817	OC[C@H]1O[C@@H](CC(=O)NCC2CC2)CC[C@H]1NC(=O)C1CCC1	CID:54639012	phase I
BRD-K13002201	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)CC[C@@H]1NC(=O)C1CCC1	CID:54639013	phase I
BRD-K43249401	OC[C@H]1O[C@H](CC(=O)NCC2CC2)CC[C@@H]1NC(=O)C1CCC1	CID:54639014	phase I
BRD-K08039553	OC[C@@H]1O[C@@H](CC(=O)NCC2CC2)CC[C@H]1NC(=O)C1CCC1	CID:54639015	phase I
BRD-K22668950	OC[C@H]1O[C@@H](CC(=O)NCC2CC2)CC[C@@H]1NC(=O)C1CCC1	CID:54639016	phase I
BRD-K94317551	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)CC[C@H]1NC(=O)C1CCC1	CID:54639017	phase I
BRD-K31327364	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H](NC(=O)c2ccc3OCOc3c2)[C@@H](CO)O1	CID:54639018	phase I
BRD-K35196676	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H](NC(=O)c2ccc3OCOc3c2)[C@H](CO)O1	CID:54639019	phase I
BRD-K12884539	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H](NC(=O)c2ccc3OCOc3c2)[C@@H](CO)O1	CID:54639020	phase I
BRD-K24172839	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H](NC(=O)c2ccc3OCOc3c2)[C@H](CO)O1	CID:54639021	phase I
BRD-K03116835	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H](NC(=O)c2ccc3OCOc3c2)[C@@H](CO)O1	CID:54639022	phase I
BRD-K77709215	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H](NC(=O)c2ccc3OCOc3c2)[C@H](CO)O1	CID:54639023	phase I
BRD-K96431673	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H](NC(=O)c2ccc3OCOc3c2)[C@@H](CO)O1	CID:54639024	phase I
BRD-K00342680	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H](NC(=O)c2ccc3OCOc3c2)[C@H](CO)O1	CID:54639025	phase I
BRD-K08731287	OC[C@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639026	phase I
BRD-K16704189	OC[C@@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639027	phase I
BRD-K99268544	OC[C@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639028	phase I
BRD-K03807141	OC[C@@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639029	phase I
BRD-K51241952	OC[C@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639030	phase I
BRD-K73061717	OC[C@@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639031	phase I
BRD-K52653383	OC[C@H]1O[C@@H](CCn2cc(Cc3ccccc3)nn2)CC[C@@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639032	phase I
BRD-K94913400	OC[C@@H]1O[C@H](CCn2cc(Cc3ccccc3)nn2)CC[C@H]1NC(=O)Nc1cccc(Cl)c1	CID:54639033	phase I
BRD-K59958061	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)NCCN2CCCCC2)O[C@@H]1CO	CID:54639034	phase I
BRD-K34324287	Cc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)NCCN2CCCCC2)O[C@H]1CO	CID:54639035	phase I
BRD-K07359994	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)NCCN2CCCCC2)O[C@@H]1CO	CID:54639036	phase I
BRD-K68737064	Cc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)NCCN2CCCCC2)O[C@H]1CO	CID:54639037	phase I
BRD-K30033690	Cc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@@H](CC(=O)NCCN2CCCCC2)O[C@@H]1CO	CID:54639038	phase I
BRD-K56345641	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@H](CC(=O)NCCN2CCCCC2)O[C@H]1CO	CID:54639039	phase I
BRD-K28430035	Cc1ccc(cc1)S(=O)(=O)N[C@H]1C=C[C@H](CC(=O)NCCN2CCCCC2)O[C@@H]1CO	CID:54639040	phase I
BRD-K98638910	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1C=C[C@@H](CC(=O)NCCN2CCCCC2)O[C@H]1CO	CID:54639041	phase I
BRD-K46040098	COc1cccc(CNC(=O)C[C@@H]2CC[C@@H](NC(C)=O)[C@@H](CO)O2)c1	CID:54639042	phase I
BRD-K74083848	COc1cccc(CNC(=O)C[C@H]2CC[C@H](NC(C)=O)[C@H](CO)O2)c1	CID:54639043	phase I
BRD-K22181332	COc1cccc(CNC(=O)C[C@H]2CC[C@@H](NC(C)=O)[C@@H](CO)O2)c1	CID:54639044	phase I
BRD-K34839715	COc1cccc(CNC(=O)C[C@@H]2CC[C@H](NC(C)=O)[C@H](CO)O2)c1	CID:54639045	phase I
BRD-K27161987	COc1cccc(CNC(=O)C[C@@H]2CC[C@H](NC(C)=O)[C@@H](CO)O2)c1	CID:54639046	phase I
BRD-K54792609	COc1cccc(CNC(=O)C[C@H]2CC[C@@H](NC(C)=O)[C@H](CO)O2)c1	CID:54639047	phase I
BRD-K25644061	COc1cccc(CNC(=O)C[C@H]2CC[C@H](NC(C)=O)[C@@H](CO)O2)c1	CID:54639048	phase I
BRD-K67285049	COc1cccc(CNC(=O)C[C@@H]2CC[C@@H](NC(C)=O)[C@H](CO)O2)c1	CID:54639049	phase I
BRD-K91021522	OC[C@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@H]1NS(=O)(=O)Cc1ccccc1	CID:54639050	phase I
BRD-K14654869	OC[C@@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@@H]1NS(=O)(=O)Cc1ccccc1	CID:54639051	phase I
BRD-K71035792	OC[C@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@H]1NS(=O)(=O)Cc1ccccc1	CID:54639052	phase I
BRD-K62039221	OC[C@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@@H]1NS(=O)(=O)Cc1ccccc1	CID:54639053	phase I
BRD-K82822203	OC[C@@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@H]1NS(=O)(=O)Cc1ccccc1	CID:54639054	phase I
BRD-K13190592	OC[C@@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@@H]1NS(=O)(=O)Cc1ccccc1	CID:54639055	phase I
BRD-K36558227	OC[C@H]1O[C@@H](CCNC(=O)C2CCC2)CC[C@@H]1NS(=O)(=O)Cc1ccccc1	CID:54639056	phase I
BRD-K74900896	OC[C@@H]1O[C@H](CCNC(=O)C2CCC2)CC[C@H]1NS(=O)(=O)Cc1ccccc1	CID:54639057	phase I
BRD-K44760520	N[C@@H]1CC[C@H](CCn2cc(nn2)-c2ccccn2)O[C@H]1CO	CID:54639058	phase I
BRD-K55578148	N[C@H]1CC[C@@H](CCn2cc(nn2)-c2ccccn2)O[C@H]1CO	CID:54639059	phase I
BRD-K26606423	N[C@H]1CC[C@H](CCn2cc(nn2)-c2ccccn2)O[C@@H]1CO	CID:54639060	phase I
BRD-K29911749	N[C@@H]1CC[C@@H](CCn2cc(nn2)-c2ccccn2)O[C@H]1CO	CID:54639061	phase I
BRD-K19203541	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C=C[C@H]1NC(=O)c1ccccc1	CID:54639062	phase I
BRD-K12791594	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C=C[C@@H]1NC(=O)c1ccccc1	CID:54639063	phase I
BRD-K82399474	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C=C[C@@H]1NC(=O)c1ccccc1	CID:54639064	phase I
BRD-K76896049	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C=C[C@H]1NC(=O)c1ccccc1	CID:54639065	phase I
BRD-K53421673	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C=C[C@@H]1NC(=O)c1ccccc1	CID:54639066	phase I
BRD-K69006460	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C=C[C@H]1NC(=O)c1ccccc1	CID:54639067	phase I
BRD-K29452018	COCC(=O)N[C@@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54639068	phase I
BRD-K61649900	COCC(=O)N[C@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54639069	phase I
BRD-K13539834	COCC(=O)N[C@@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54639070	phase I
BRD-K44029853	COCC(=O)N[C@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54639071	phase I
BRD-K08173649	COCC(=O)N[C@@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54639072	phase I
BRD-K29063218	COCC(=O)N[C@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54639073	phase I
BRD-K62130095	COCC(=O)N[C@H]1C=C[C@H](CC(=O)N2CCCCC2)O[C@@H]1CO	CID:54639074	phase I
BRD-K75395214	COCC(=O)N[C@@H]1C=C[C@@H](CC(=O)N2CCCCC2)O[C@H]1CO	CID:54639075	phase I
BRD-K08926145	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2cccc(F)c2)O[C@@H]1CO	CID:54639076	phase I
BRD-K62456065	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@H](CC(=O)NCc2cccc(F)c2)O[C@H]1CO	CID:54639077	phase I
BRD-K45919129	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)NCc2cccc(F)c2)O[C@@H]1CO	CID:54639078	phase I
BRD-K76285876	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)NCc2cccc(F)c2)O[C@@H]1CO	CID:54639079	phase I
BRD-K05645732	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)NCc2cccc(F)c2)O[C@H]1CO	CID:54639080	phase I
BRD-K73127443	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)NCc2cccc(F)c2)O[C@H]1CO	CID:54639081	phase I
BRD-K61388502	COc1ccccc1S(=O)(=O)N[C@H]1CC[C@H](CC(=O)NCc2cccc(F)c2)O[C@@H]1CO	CID:54639082	phase I
BRD-K40985138	COc1ccccc1S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)NCc2cccc(F)c2)O[C@H]1CO	CID:54639083	phase I
BRD-K22778942	OC[C@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54639084	phase I
BRD-K10927790	OC[C@@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54639085	phase I
BRD-K68095812	OC[C@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54639086	phase I
BRD-K70581786	OC[C@@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54639087	phase I
BRD-K56943062	OC[C@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54639088	phase I
BRD-K79596575	OC[C@@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54639089	phase I
BRD-K94454791	OC[C@H]1O[C@@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@@H]1NC(=O)CCN1CCCCC1	CID:54639090	phase I
BRD-K25165092	OC[C@@H]1O[C@H](CC(=O)N2CCC(Cc3ccccc3)CC2)CC[C@H]1NC(=O)CCN1CCCCC1	CID:54639091	phase I
BRD-K38481268	OC[C@H]1O[C@H](CCNC(=O)c2cnccn2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54639092	phase I
BRD-K04395157	OC[C@@H]1O[C@@H](CCNC(=O)c2cnccn2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54639093	phase I
BRD-K83325143	OC[C@@H]1O[C@@H](CCNC(=O)c2cnccn2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54639094	phase I
BRD-K50149017	OC[C@H]1O[C@@H](CCNC(=O)c2cnccn2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54639095	phase I
BRD-K73483999	OC[C@H]1O[C@@H](CCNC(=O)c2cnccn2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54639096	phase I
BRD-K82765406	OC[C@@H]1O[C@H](CCNC(=O)c2cnccn2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54639097	phase I
BRD-K49931834	OC[C@H]1O[C@H](CCNC(=O)c2cnccn2)CC[C@@H]1NC(=O)c1ccc2OCOc2c1	CID:54639098	phase I
BRD-K17742539	OC[C@@H]1O[C@H](CCNC(=O)c2cnccn2)CC[C@H]1NC(=O)c1ccc2OCOc2c1	CID:54639099	phase I
BRD-K19890875	COc1ccc(NC(=O)N[C@@H]2CC[C@@H](CC(=O)NC3CCC3)O[C@@H]2CO)cc1	CID:54639100	phase I
BRD-K28649344	COc1ccc(NC(=O)N[C@H]2CC[C@H](CC(=O)NC3CCC3)O[C@H]2CO)cc1	CID:54639101	phase I
BRD-K31462841	COc1ccc(NC(=O)N[C@@H]2CC[C@H](CC(=O)NC3CCC3)O[C@@H]2CO)cc1	CID:54639102	phase I
BRD-K31774852	COc1ccc(NC(=O)N[C@H]2CC[C@@H](CC(=O)NC3CCC3)O[C@H]2CO)cc1	CID:54639103	phase I
BRD-K73118655	COc1ccc(NC(=O)N[C@H]2CC[C@H](CC(=O)NC3CCC3)O[C@@H]2CO)cc1	CID:54639104	phase I
BRD-K97829610	COc1ccc(NC(=O)N[C@@H]2CC[C@H](CC(=O)NC3CCC3)O[C@H]2CO)cc1	CID:54639105	phase I
BRD-K01979737	COc1ccc(NC(=O)N[C@@H]2CC[C@@H](CC(=O)NC3CCC3)O[C@H]2CO)cc1	CID:54639106	phase I
BRD-K24277661	OC[C@H]1O[C@H](CC(O)=O)CC[C@H]1NC(=O)c1ccncc1	CID:54639107	phase I
BRD-K77429897	OC[C@@H]1O[C@@H](CC(O)=O)CC[C@@H]1NC(=O)c1ccncc1	CID:54639108	phase I
BRD-K24017250	OC[C@H]1O[C@@H](CC(O)=O)CC[C@H]1NC(=O)c1ccncc1	CID:54639109	phase I
BRD-K95286989	OC[C@H]1O[C@H](CC(O)=O)CC[C@@H]1NC(=O)c1ccncc1	CID:54639110	phase I
BRD-K65368843	OC[C@H]1O[C@@H](CC(O)=O)CC[C@@H]1NC(=O)c1ccncc1	CID:54639111	phase I
BRD-K95265783	OC[C@@H]1O[C@H](CC(O)=O)CC[C@H]1NC(=O)c1ccncc1	CID:54639112	phase I
BRD-K75809222	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CCNC(=O)c2ccccc2F)O[C@@H]1CO	CID:54639113	phase I
BRD-K06163447	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CCNC(=O)c2ccccc2F)O[C@H]1CO	CID:54639114	phase I
BRD-K94241935	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CCNC(=O)c2ccccc2F)O[C@@H]1CO	CID:54639115	phase I
BRD-K19965545	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CCNC(=O)c2ccccc2F)O[C@H]1CO	CID:54639116	phase I
BRD-K70689011	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CCNC(=O)c2ccccc2F)O[C@@H]1CO	CID:54639117	phase I
BRD-K77053153	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CCNC(=O)c2ccccc2F)O[C@H]1CO	CID:54639118	phase I
BRD-K50657769	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CCNC(=O)c2ccccc2F)O[C@@H]1CO	CID:54639119	phase I
BRD-K12564766	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CCNC(=O)c2ccccc2F)O[C@H]1CO	CID:54639120	phase I
BRD-K20121890	CN1CCN(CC1)C(=O)C[C@H]1O[C@H](CO)[C@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639121	phase I
BRD-K74830065	CN1CCN(CC1)C(=O)C[C@@H]1O[C@@H](CO)[C@@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639122	phase I
BRD-K97045804	CN1CCN(CC1)C(=O)C[C@@H]1O[C@H](CO)[C@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639123	phase I
BRD-K59598504	CN1CCN(CC1)C(=O)C[C@H]1O[C@@H](CO)[C@@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639124	phase I
BRD-K26127000	CN1CCN(CC1)C(=O)C[C@@H]1O[C@@H](CO)[C@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639125	phase I
BRD-K02492147	CN1CCN(CC1)C(=O)C[C@@H]1O[C@H](CO)[C@@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639126	phase I
BRD-K20342806	CN1CCN(CC1)C(=O)C[C@H]1O[C@@H](CO)[C@H](NS(=O)(=O)c2cccc(F)c2)C=C1	CID:54639127	phase I
BRD-K27635561	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)N2CCc3ccccc3C2)O[C@@H]1CO	CID:54639128	phase I
BRD-K37106459	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CC(=O)N2CCc3ccccc3C2)O[C@H]1CO	CID:54639129	phase I
BRD-K96977391	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)N2CCc3ccccc3C2)O[C@@H]1CO	CID:54639130	phase I
BRD-K21660676	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)N2CCc3ccccc3C2)O[C@H]1CO	CID:54639131	phase I
BRD-K45138525	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@@H](CC(=O)N2CCc3ccccc3C2)O[C@@H]1CO	CID:54639132	phase I
BRD-K04402444	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@H](CC(=O)N2CCc3ccccc3C2)O[C@H]1CO	CID:54639133	phase I
BRD-K31830316	Cc1ccc(cc1)S(=O)(=O)N[C@H]1CC[C@H](CC(=O)N2CCc3ccccc3C2)O[C@@H]1CO	CID:54639134	phase I
BRD-K04937680	Cc1ccc(cc1)S(=O)(=O)N[C@@H]1CC[C@@H](CC(=O)N2CCc3ccccc3C2)O[C@H]1CO	CID:54639135	phase I
BRD-K64706654	OC[C@H]1O[C@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@H]1NC(=O)Cc1cccnc1	CID:54639136	phase I
BRD-K77603027	OC[C@@H]1O[C@@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54639137	phase I
BRD-K25955619	OC[C@H]1O[C@@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@H]1NC(=O)Cc1cccnc1	CID:54639138	phase I
BRD-K93569571	OC[C@@H]1O[C@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54639139	phase I
BRD-K73261664	OC[C@H]1O[C@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@@H]1NC(=O)Cc1cccnc1	CID:54639140	phase I
BRD-K36250651	OC[C@@H]1O[C@@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@H]1NC(=O)Cc1cccnc1	CID:54639141	phase I
BRD-K24656059	OC[C@@H]1O[C@H](CC(=O)Nc2ccc(cc2)-c2ccccc2)CC[C@H]1NC(=O)Cc1cccnc1	CID:54639142	phase I
BRD-K27757818	OC[C@H]1O[C@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@H]1NC(=O)c1ccncc1	CID:54639143	phase I
BRD-K36618106	OC[C@@H]1O[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54639144	phase I
BRD-K55078218	OC[C@H]1O[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@H]1NC(=O)c1ccncc1	CID:54639145	phase I
BRD-K83546471	OC[C@@H]1O[C@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54639146	phase I
BRD-K83407176	OC[C@H]1O[C@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54639147	phase I
BRD-K07601300	OC[C@@H]1O[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@H]1NC(=O)c1ccncc1	CID:54639148	phase I
BRD-K24742410	OC[C@H]1O[C@@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@@H]1NC(=O)c1ccncc1	CID:54639149	phase I
BRD-K96660315	OC[C@@H]1O[C@H](CC(=O)N2CCN(CC2)c2ccccc2)C=C[C@H]1NC(=O)c1ccncc1	CID:54639150	phase I
BRD-K19466708	OC[C@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NC(=O)c1cnccn1	CID:54639151	phase I
BRD-K41096823	OC[C@@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NC(=O)c1cnccn1	CID:54639152	phase I
BRD-K33711030	OC[C@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NC(=O)c1cnccn1	CID:54639153	phase I
BRD-K88045846	OC[C@@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NC(=O)c1cnccn1	CID:54639154	phase I
BRD-K40892926	OC[C@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NC(=O)c1cnccn1	CID:54639155	phase I
BRD-K23911230	OC[C@@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NC(=O)c1cnccn1	CID:54639156	phase I
BRD-K10270435	OC[C@H]1O[C@@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@@H]1NC(=O)c1cnccn1	CID:54639157	phase I
BRD-K22173650	OC[C@@H]1O[C@H](CCNS(=O)(=O)Cc2ccccc2)CC[C@H]1NC(=O)c1cnccn1	CID:54639158	phase I
BRD-K12857449	OC[C@H]1O[C@H](CC(=O)NCc2ccccc2Cl)CC[C@H]1NC(=O)C1CCOCC1	CID:54639159	phase I
BRD-K94025757	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccc2Cl)CC[C@@H]1NC(=O)C1CCOCC1	CID:54639160	phase I
BRD-K03727241	OC[C@H]1O[C@@H](CC(=O)NCc2ccccc2Cl)CC[C@H]1NC(=O)C1CCOCC1	CID:54639161	phase I
BRD-K46155530	OC[C@@H]1O[C@H](CC(=O)NCc2ccccc2Cl)CC[C@@H]1NC(=O)C1CCOCC1	CID:54639162	phase I
BRD-K28540419	OC[C@H]1O[C@H](CC(=O)NCc2ccccc2Cl)CC[C@@H]1NC(=O)C1CCOCC1	CID:54639163	phase I
BRD-K43776433	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645798	phase I
BRD-K19416218	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1	CID:54645799	phase I
BRD-K74639017	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1	CID:54645800	phase I
BRD-K94136966	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1	CID:54645801	phase I
BRD-K49906853	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1	CID:54645802	phase I
BRD-K49948755	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1	CID:54645803	phase I
BRD-K74287511	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1	CID:54645804	phase I
BRD-K82204596	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1	CID:54645805	phase I
BRD-K24502634	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1	CID:54645806	phase I
BRD-K21384842	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cccc(F)c4)O[C@H]3CO)c2c1	CID:54645807	phase I
BRD-K34336958	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cccc(F)c4)O[C@H]3CO)c2c1	CID:54645808	phase I
BRD-K40442760	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cccc(F)c4)O[C@@H]3CO)c2c1	CID:54645809	phase I
BRD-K42383812	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cccc(F)c4)O[C@H]3CO)c2c1	CID:54645810	phase I
BRD-K10680649	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cccc(F)c4)O[C@@H]3CO)c2c1	CID:54645811	phase I
BRD-K67788404	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cccc(F)c4)O[C@H]3CO)c2c1	CID:54645812	phase I
BRD-K75750101	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645813	phase I
BRD-K00959946	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645814	phase I
BRD-K65981470	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645815	phase I
BRD-K70868272	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645816	phase I
BRD-K03496708	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645817	phase I
BRD-K60700659	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645818	phase I
BRD-K32681593	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645819	phase I
BRD-K75819331	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645820	phase I
BRD-K04682465	CCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@@H](CO)O1	CID:54645821	phase I
BRD-K19629349	CCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@H](CO)O1	CID:54645822	phase I
BRD-K37300049	CCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@H](CO)O1	CID:54645823	phase I
BRD-K81109082	CCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@@H](CO)O1	CID:54645824	phase I
BRD-K99882679	CCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@H](CO)O1	CID:54645825	phase I
BRD-K43357772	CCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@@H](CO)O1	CID:54645826	phase I
BRD-K58358247	CCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccccc4F)cc23)[C@H](CO)O1	CID:54645827	phase I
BRD-K76578350	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645828	phase I
BRD-K01520595	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645829	phase I
BRD-K73500089	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645830	phase I
BRD-K23018071	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645831	phase I
BRD-K64645183	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645832	phase I
BRD-K58703114	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645833	phase I
BRD-K12483497	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645834	phase I
BRD-K79498538	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54645835	phase I
BRD-K34435836	COc1ccc(CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2)cc1	CID:54645836	phase I
BRD-K68494763	COc1ccc(CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2)cc1	CID:54645837	phase I
BRD-K32889681	COc1ccc(CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2)cc1	CID:54645838	phase I
BRD-K75091523	COc1ccc(CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2)cc1	CID:54645839	phase I
BRD-K83644384	COc1ccc(CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2)cc1	CID:54645840	phase I
BRD-K68701561	COc1ccc(CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2)cc1	CID:54645841	phase I
BRD-K10287818	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(N)cc23)[C@H](CO)O1	CID:54645842	phase I
BRD-K73334096	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(N)cc23)[C@@H](CO)O1	CID:54645843	phase I
BRD-K69792693	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(N)cc23)[C@H](CO)O1	CID:54645844	phase I
BRD-K29474997	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NC4CCCCC4)O[C@H]3CO)c2c1	CID:54645845	phase I
BRD-K56452877	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645846	phase I
BRD-K80777319	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645847	phase I
BRD-K55082119	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645848	phase I
BRD-K61123818	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645849	phase I
BRD-K85433055	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645850	phase I
BRD-K24465470	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645851	phase I
BRD-K09563163	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645852	phase I
BRD-K21558506	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645853	phase I
BRD-K89585847	OC[C@H]1O[C@@H](CC(=O)NCC2CC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645854	phase I
BRD-K53148273	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645855	phase I
BRD-K19825378	OC[C@H]1O[C@H](CC(=O)NCC2CC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645856	phase I
BRD-K47826846	OC[C@@H]1O[C@@H](CC(=O)NCC2CC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645857	phase I
BRD-K22356478	OC[C@H]1O[C@@H](CC(=O)NCC2CC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645858	phase I
BRD-K61741250	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645859	phase I
BRD-K98259048	OC[C@H]1O[C@H](CC(=O)NCC2CC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645860	phase I
BRD-K39144966	OC[C@@H]1O[C@@H](CC(=O)NCC2CC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54645861	phase I
BRD-K75576199	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54645862	phase I
BRD-K71674109	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54645863	phase I
BRD-K89735991	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54645864	phase I
BRD-K41667061	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54645865	phase I
BRD-K89076662	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54645866	phase I
BRD-K01248935	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54645867	phase I
BRD-K89627562	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54645868	phase I
BRD-K45475981	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54645869	phase I
BRD-K78761249	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645870	phase I
BRD-K15778794	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645871	phase I
BRD-K59830209	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645872	phase I
BRD-K77100270	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645873	phase I
BRD-K24550549	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645874	phase I
BRD-K43820987	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645875	phase I
BRD-K28851694	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645876	phase I
BRD-K22676415	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645877	phase I
BRD-K02280251	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCC(F)(F)F)O[C@@H]4CO)c3c2)cc1	CID:54645878	phase I
BRD-K15650895	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCC(F)(F)F)O[C@H]4CO)c3c2)cc1	CID:54645879	phase I
BRD-K54729370	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCC(F)(F)F)O[C@H]4CO)c3c2)cc1	CID:54645880	phase I
BRD-K88092133	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCC(F)(F)F)O[C@H]4CO)c3c2)cc1	CID:54645881	phase I
BRD-K74796495	OC[C@H]1O[C@@H](CC(=O)NCc2ccccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645882	phase I
BRD-K38122103	OC[C@@H]1O[C@H](CC(=O)NCc2ccccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645883	phase I
BRD-K71334452	OC[C@H]1O[C@H](CC(=O)NCc2ccccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645884	phase I
BRD-K02311587	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645885	phase I
BRD-K14652476	OC[C@@H]1O[C@H](CC(=O)NCc2ccccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645886	phase I
BRD-K65922289	OC[C@H]1O[C@H](CC(=O)NCc2ccccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645887	phase I
BRD-K66328731	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54645888	phase I
BRD-K16792691	CN(C)C(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@@H](CO)O1	CID:54645889	phase I
BRD-K78891011	CN(C)C(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@H](CO)O1	CID:54645890	phase I
BRD-K26484639	CN(C)C(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@@H](CO)O1	CID:54645891	phase I
BRD-K51126488	CN(C)C(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@H](CO)O1	CID:54645892	phase I
BRD-K74625930	CN(C)C(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@@H](CO)O1	CID:54645893	phase I
BRD-K13583181	CN(C)C(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@H](CO)O1	CID:54645894	phase I
BRD-K91123606	CN(C)C(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@@H](CO)O1	CID:54645895	phase I
BRD-K53406626	CN(C)C(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(F)cc4)cc23)[C@H](CO)O1	CID:54645896	phase I
BRD-K09935385	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645897	phase I
BRD-K84639586	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645898	phase I
BRD-K52460145	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645899	phase I
BRD-K37255594	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645900	phase I
BRD-K32234234	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645901	phase I
BRD-K81658952	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645902	phase I
BRD-K31680744	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645903	phase I
BRD-K81678234	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54645904	phase I
BRD-K72081524	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCCc4ccccc4)O[C@@H]3CO)c2c1	CID:54645905	phase I
BRD-K26594332	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCCc4ccccc4)O[C@H]3CO)c2c1	CID:54645906	phase I
BRD-K27706744	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCCc4ccccc4)O[C@@H]3CO)c2c1	CID:54645907	phase I
BRD-K42729412	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCCc4ccccc4)O[C@H]3CO)c2c1	CID:54645908	phase I
BRD-K65456352	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCCc4ccccc4)O[C@@H]3CO)c2c1	CID:54645909	phase I
BRD-K93612606	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCCc4ccccc4)O[C@H]3CO)c2c1	CID:54645910	phase I
BRD-K96165286	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCCc4ccccc4)O[C@@H]3CO)c2c1	CID:54645911	phase I
BRD-K64380185	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCCc4ccccc4)O[C@H]3CO)c2c1	CID:54645912	phase I
BRD-K34781184	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645913	phase I
BRD-K60334624	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645914	phase I
BRD-K16956545	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645915	phase I
BRD-K67774729	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645916	phase I
BRD-K42960120	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645917	phase I
BRD-K10837204	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645918	phase I
BRD-K67862512	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645919	phase I
BRD-K52184420	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6ccc7OCOc7c6)cc45	CID:54645920	phase I
BRD-K62014585	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645921	phase I
BRD-K67780580	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645922	phase I
BRD-K63233328	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645923	phase I
BRD-K37482798	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645924	phase I
BRD-K28169522	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645925	phase I
BRD-K88239034	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645926	phase I
BRD-K82284120	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645927	phase I
BRD-K60109523	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54645928	phase I
BRD-K07408742	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645929	phase I
BRD-K60776198	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645930	phase I
BRD-K23822091	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645931	phase I
BRD-K83486374	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645932	phase I
BRD-K60873020	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645933	phase I
BRD-K77425389	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645934	phase I
BRD-K28508449	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54645935	phase I
BRD-K19108281	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54645936	phase I
BRD-K30436233	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645937	phase I
BRD-K82365559	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54645938	phase I
BRD-K88908047	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645939	phase I
BRD-K86846131	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645940	phase I
BRD-K59176197	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54645941	phase I
BRD-K31556224	C[C@@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645942	phase I
BRD-K96900359	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645943	phase I
BRD-K55713064	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54645944	phase I
BRD-K66646581	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54645945	phase I
BRD-K82794234	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54645946	phase I
BRD-K13691358	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645947	phase I
BRD-K08306736	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54645948	phase I
BRD-K06228572	OC[C@H]1O[C@@H](CC(=O)NC2CCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645949	phase I
BRD-K97101742	OC[C@@H]1O[C@H](CC(=O)NC2CCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645950	phase I
BRD-K39504007	OC[C@H]1O[C@H](CC(=O)NC2CCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645951	phase I
BRD-K80789291	OC[C@@H]1O[C@@H](CC(=O)NC2CCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645952	phase I
BRD-K00347265	OC[C@H]1O[C@@H](CC(=O)NC2CCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645953	phase I
BRD-K25994126	OC[C@@H]1O[C@H](CC(=O)NC2CCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645954	phase I
BRD-K83920942	OC[C@H]1O[C@H](CC(=O)NC2CCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645955	phase I
BRD-K35868313	OC[C@@H]1O[C@@H](CC(=O)NC2CCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54645956	phase I
BRD-K35188965	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCOCC4)O[C@@H]3CO)c2c1	CID:54645957	phase I
BRD-K76904146	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCOCC4)O[C@H]3CO)c2c1	CID:54645958	phase I
BRD-K98993678	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCOCC4)O[C@@H]3CO)c2c1	CID:54645959	phase I
BRD-K37434018	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCOCC4)O[C@H]3CO)c2c1	CID:54645960	phase I
BRD-K52309792	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCOCC4)O[C@@H]3CO)c2c1	CID:54645961	phase I
BRD-K33451389	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCOCC4)O[C@H]3CO)c2c1	CID:54645962	phase I
BRD-K47102646	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCOCC4)O[C@@H]3CO)c2c1	CID:54645963	phase I
BRD-K99785919	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCOCC4)O[C@H]3CO)c2c1	CID:54645964	phase I
BRD-K00935206	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@@H](CO)O2	CID:54645965	phase I
BRD-K81736443	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@H](CO)O2	CID:54645966	phase I
BRD-K24077273	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@H](CO)O2	CID:54645967	phase I
BRD-K51971121	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@@H](CO)O2	CID:54645968	phase I
BRD-K22253301	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@H](CO)O2	CID:54645969	phase I
BRD-K15414305	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@@H](CO)O2	CID:54645970	phase I
BRD-K76662562	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34)[C@H](CO)O2	CID:54645971	phase I
BRD-K49911380	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645972	phase I
BRD-K10894258	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645973	phase I
BRD-K56176052	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645974	phase I
BRD-K46192888	OC[C@@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645975	phase I
BRD-K61979066	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645976	phase I
BRD-K22013971	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54645977	phase I
BRD-K40694355	OC[C@H]1O[C@H](CC(=O)NCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54645980	phase I
BRD-K59191656	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54645981	phase I
BRD-K61499353	OC[C@H]1O[C@@H](CC(=O)NCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54645982	phase I
BRD-K63602071	OC[C@@H]1O[C@H](CC(=O)NCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54645983	phase I
BRD-K49597140	OC[C@H]1O[C@H](CC(=O)NCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54645984	phase I
BRD-K53183074	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54645985	phase I
BRD-K54589358	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCOCC4)O[C@H]3CO)c2c1	CID:54645986	phase I
BRD-K45723650	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645987	phase I
BRD-K44341698	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645988	phase I
BRD-K98240084	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645989	phase I
BRD-K94694331	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645990	phase I
BRD-K09301754	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645991	phase I
BRD-K68368772	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645992	phase I
BRD-K25566775	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54645993	phase I
BRD-K72066167	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NC5CCCCC5)O[C@@H]4CO)c3c2	CID:54645994	phase I
BRD-K03864628	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NC5CCCCC5)O[C@H]4CO)c3c2	CID:54645995	phase I
BRD-K26666618	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NC5CCCCC5)O[C@@H]4CO)c3c2	CID:54645996	phase I
BRD-K57054528	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NC5CCCCC5)O[C@H]4CO)c3c2	CID:54645997	phase I
BRD-K86631008	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NC5CCCCC5)O[C@@H]4CO)c3c2	CID:54645998	phase I
BRD-K49434056	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NC5CCCCC5)O[C@H]4CO)c3c2	CID:54645999	phase I
BRD-K06532738	CN(C)C(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1	CID:54646002	phase I
BRD-K58180017	CN(C)C(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1	CID:54646003	phase I
BRD-K38289428	CN(C)C(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1	CID:54646004	phase I
BRD-K10821756	CN(C)C(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1	CID:54646005	phase I
BRD-K68682056	CN(C)C(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1	CID:54646006	phase I
BRD-K77106209	CN(C)C(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1	CID:54646007	phase I
BRD-K59704843	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1	CID:54646008	phase I
BRD-K26785978	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1	CID:54646009	phase I
BRD-K50174388	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1	CID:54646010	phase I
BRD-K78948132	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1	CID:54646011	phase I
BRD-K28223745	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1	CID:54646012	phase I
BRD-K88686946	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1	CID:54646013	phase I
BRD-K62990480	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646014	phase I
BRD-K06804050	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646015	phase I
BRD-K82502275	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646016	phase I
BRD-K56719502	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646017	phase I
BRD-K61825138	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646018	phase I
BRD-K60011163	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646019	phase I
BRD-K74458364	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646020	phase I
BRD-K65778372	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646021	phase I
BRD-K86979665	OC[C@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646022	phase I
BRD-K01326303	OC[C@@H]1O[C@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646023	phase I
BRD-K90830329	OC[C@H]1O[C@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646024	phase I
BRD-K62836687	OC[C@@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646025	phase I
BRD-K81543190	OC[C@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646026	phase I
BRD-K23396987	OC[C@@H]1O[C@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646027	phase I
BRD-K96634415	OC[C@H]1O[C@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646028	phase I
BRD-K69845975	OC[C@@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646029	phase I
BRD-K88187036	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646030	phase I
BRD-K76988892	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646031	phase I
BRD-K70783031	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646032	phase I
BRD-K22387508	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646033	phase I
BRD-K71346068	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646034	phase I
BRD-K64537516	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646035	phase I
BRD-K13891716	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646036	phase I
BRD-K65730939	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646037	phase I
BRD-K83859448	OC[C@H]1O[C@@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NC(=O)Cc4ccncc4)cc23	CID:54646038	phase I
BRD-K74659043	OC[C@@H]1O[C@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NC(=O)Cc4ccncc4)cc23	CID:54646039	phase I
BRD-K42959654	COCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@@H](CO)O1	CID:54646040	phase I
BRD-K84787606	COCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646041	phase I
BRD-K31108633	COCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@@H](CO)O1	CID:54646042	phase I
BRD-K45440108	COCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646043	phase I
BRD-K30781800	COCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@@H](CO)O1	CID:54646044	phase I
BRD-K27817736	COCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646045	phase I
BRD-K80940272	COCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@@H](CO)O1	CID:54646046	phase I
BRD-K98320434	COCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646047	phase I
BRD-K79664955	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(cc34)N(C)C)[C@@H](CO)O2	CID:54646048	phase I
BRD-K69719543	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(cc34)N(C)C)[C@@H](CO)O2	CID:54646049	phase I
BRD-K60548400	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(cc34)N(C)C)[C@H](CO)O2	CID:54646050	phase I
BRD-K61533941	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(cc34)N(C)C)[C@@H](CO)O2	CID:54646051	phase I
BRD-K16121755	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(cc34)N(C)C)[C@H](CO)O2	CID:54646052	phase I
BRD-K29326878	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646053	phase I
BRD-K89952884	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N[C@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646054	phase I
BRD-K75383594	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646055	phase I
BRD-K87304811	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N[C@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646056	phase I
BRD-K33057338	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646057	phase I
BRD-K29737933	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N[C@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646058	phase I
BRD-K57275439	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N[C@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646059	phase I
BRD-K18132838	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646060	phase I
BRD-K30822915	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N[C@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646061	phase I
BRD-K46241566	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646062	phase I
BRD-K58469266	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N[C@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646063	phase I
BRD-K11468724	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646064	phase I
BRD-K62943397	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N[C@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646065	phase I
BRD-K96121225	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@@H]3CO)c2c1	CID:54646066	phase I
BRD-K98716460	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N[C@@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646067	phase I
BRD-K67502058	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N[C@H](C)c4ccccc4)O[C@H]3CO)c2c1	CID:54646068	phase I
BRD-K66836247	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NS(=O)(=O)c4ccccc4)cc23	CID:54646069	phase I
BRD-K36110199	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NS(=O)(=O)c4ccccc4)cc23	CID:54646070	phase I
BRD-K74455073	OC[C@@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NS(=O)(=O)c4ccccc4)cc23	CID:54646071	phase I
BRD-K20200700	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NS(=O)(=O)c4ccccc4)cc23	CID:54646072	phase I
BRD-K03935278	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NS(=O)(=O)c4ccccc4)cc23	CID:54646073	phase I
BRD-K17713237	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@@H](CO)O2	CID:54646074	phase I
BRD-K16705018	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@H](CO)O2	CID:54646075	phase I
BRD-K93763244	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@@H](CO)O2	CID:54646076	phase I
BRD-K77953075	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@H](CO)O2	CID:54646077	phase I
BRD-K84625203	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@@H](CO)O2	CID:54646078	phase I
BRD-K73171326	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@H](CO)O2	CID:54646079	phase I
BRD-K44953633	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@@H](CO)O2	CID:54646080	phase I
BRD-K98376600	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)C)cc34)[C@H](CO)O2	CID:54646081	phase I
BRD-K78939963	OC[C@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646082	phase I
BRD-K28043081	OC[C@@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646083	phase I
BRD-K61907493	OC[C@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646084	phase I
BRD-K00740489	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646085	phase I
BRD-K93667957	OC[C@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646086	phase I
BRD-K48306626	OC[C@@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646087	phase I
BRD-K64147688	OC[C@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646088	phase I
BRD-K74149575	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646089	phase I
BRD-K08668362	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646090	phase I
BRD-K18001731	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646091	phase I
BRD-K11833731	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646092	phase I
BRD-K45098285	OC[C@@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646093	phase I
BRD-K86800060	OC[C@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646094	phase I
BRD-K92925409	OC[C@@H]1O[C@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646095	phase I
BRD-K65504774	OC[C@H]1O[C@H](CC(=O)N2CCOCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646096	phase I
BRD-K03210181	OC[C@@H]1O[C@@H](CC(=O)N2CCOCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646097	phase I
BRD-K74636477	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)N(C)C)O[C@@H]4CO)c3c2	CID:54646098	phase I
BRD-K23897871	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)N(C)C)O[C@H]4CO)c3c2	CID:54646099	phase I
BRD-K00199686	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)N(C)C)O[C@H]4CO)c3c2	CID:54646100	phase I
BRD-K80324403	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)N(C)C)O[C@@H]4CO)c3c2	CID:54646101	phase I
BRD-K42170810	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)N(C)C)O[C@H]4CO)c3c2	CID:54646102	phase I
BRD-K09170549	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)N(C)C)O[C@@H]4CO)c3c2	CID:54646103	phase I
BRD-K17088043	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)N(C)C)O[C@H]4CO)c3c2	CID:54646104	phase I
BRD-K94843767	OC[C@H]1O[C@@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646105	phase I
BRD-K43786699	OC[C@@H]1O[C@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646106	phase I
BRD-K24325779	OC[C@H]1O[C@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646107	phase I
BRD-K07877451	OC[C@@H]1O[C@@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646108	phase I
BRD-K54166087	OC[C@H]1O[C@@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646109	phase I
BRD-K15260875	OC[C@@H]1O[C@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646110	phase I
BRD-K90466405	OC[C@H]1O[C@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646111	phase I
BRD-K19061245	OC[C@@H]1O[C@@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23	CID:54646112	phase I
BRD-K31230167	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(N)cc23)[C@H](CO)O1	CID:54646113	phase I
BRD-K05315233	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(N)cc23)[C@@H](CO)O1	CID:54646114	phase I
BRD-K02125996	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(N)cc23)[C@H](CO)O1	CID:54646115	phase I
BRD-K68864067	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(N)cc23)[C@@H](CO)O1	CID:54646116	phase I
BRD-K76269493	CCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)COC)cc23)[C@@H](CO)O1	CID:54646117	phase I
BRD-K91359405	CCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)COC)cc23)[C@H](CO)O1	CID:54646118	phase I
BRD-K98834499	CCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)COC)cc23)[C@@H](CO)O1	CID:54646119	phase I
BRD-K40263565	CCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)COC)cc23)[C@H](CO)O1	CID:54646120	phase I
BRD-K84856528	CCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)COC)cc23)[C@@H](CO)O1	CID:54646121	phase I
BRD-K43650237	CCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)COC)cc23)[C@H](CO)O1	CID:54646122	phase I
BRD-K03735855	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1)c6ccccc6	CID:54646123	phase I
BRD-K64021372	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1)c6ccccc6	CID:54646124	phase I
BRD-K98869108	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1)c6ccccc6	CID:54646125	phase I
BRD-K42536980	C[C@@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1)c6ccccc6	CID:54646126	phase I
BRD-K48927563	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@@H](CO)O1)c6ccccc6	CID:54646127	phase I
BRD-K64551656	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23)[C@H](CO)O1)c6ccccc6	CID:54646128	phase I
BRD-K06912584	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646129	phase I
BRD-K22318001	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646130	phase I
BRD-K08508488	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646131	phase I
BRD-K86771738	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646132	phase I
BRD-K76087404	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646133	phase I
BRD-K97235918	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646134	phase I
BRD-K68178066	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646135	phase I
BRD-K91811806	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646136	phase I
BRD-K31903015	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646137	phase I
BRD-K95133676	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646138	phase I
BRD-K86997557	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646139	phase I
BRD-K23293459	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646140	phase I
BRD-K82989800	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646141	phase I
BRD-K34869284	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NC4CCCC4)O[C@@H]3CO)c2c1	CID:54646142	phase I
BRD-K65766198	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NC4CCCC4)O[C@H]3CO)c2c1	CID:54646143	phase I
BRD-K96707093	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NC4CCCC4)O[C@@H]3CO)c2c1	CID:54646144	phase I
BRD-K51368089	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NC4CCCC4)O[C@H]3CO)c2c1	CID:54646145	phase I
BRD-K51201721	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NC4CCCC4)O[C@@H]3CO)c2c1	CID:54646146	phase I
BRD-K84832762	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NC4CCCC4)O[C@H]3CO)c2c1	CID:54646147	phase I
BRD-K04371509	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NC4CCCC4)O[C@@H]3CO)c2c1	CID:54646148	phase I
BRD-K02876750	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NC4CCCC4)O[C@H]3CO)c2c1	CID:54646149	phase I
BRD-K94554079	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCCc4ccccc4)O[C@@H]3CO)c2c1	CID:54646150	phase I
BRD-K65077386	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCCc4ccccc4)O[C@H]3CO)c2c1	CID:54646151	phase I
BRD-K88487973	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCCc4ccccc4)O[C@@H]3CO)c2c1	CID:54646152	phase I
BRD-K36618304	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCCc4ccccc4)O[C@H]3CO)c2c1	CID:54646153	phase I
BRD-K90957289	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646154	phase I
BRD-K14649905	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646155	phase I
BRD-K36596745	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646156	phase I
BRD-K97364711	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646157	phase I
BRD-K75964914	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646158	phase I
BRD-K57476317	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646159	phase I
BRD-K16149503	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646160	phase I
BRD-K38589987	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646161	phase I
BRD-K39900015	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2	CID:54646162	phase I
BRD-K02206783	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2	CID:54646163	phase I
BRD-K72966614	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2	CID:54646164	phase I
BRD-K59099734	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2	CID:54646165	phase I
BRD-K86516784	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2	CID:54646166	phase I
BRD-K38998914	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2	CID:54646167	phase I
BRD-K34015625	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@@H](CO)O2	CID:54646168	phase I
BRD-K26799408	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCC5)cc34)[C@H](CO)O2	CID:54646169	phase I
BRD-K61655210	OC[C@H]1O[C@@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23	CID:54646170	phase I
BRD-K90982895	OC[C@@H]1O[C@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23	CID:54646171	phase I
BRD-K77631079	OC[C@H]1O[C@H](CC(=O)O)C[C@@H]2[C@H]1Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23	CID:54646172	phase I
BRD-K24338558	OC[C@@H]1O[C@@H](CC(=O)O)C[C@H]2[C@@H]1Oc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc23	CID:54646173	phase I
BRD-K11721480	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)C4CCOCC4)cc23	CID:54646174	phase I
BRD-K58227367	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)C4CCOCC4)cc23	CID:54646175	phase I
BRD-K27263987	OC[C@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)C4CCOCC4)cc23	CID:54646176	phase I
BRD-K32782699	OC[C@@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)C4CCOCC4)cc23	CID:54646177	phase I
BRD-K63523728	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@@H](CO)O2	CID:54646178	phase I
BRD-K80686631	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@H](CO)O2	CID:54646179	phase I
BRD-K10225826	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@@H](CO)O2	CID:54646180	phase I
BRD-K57766779	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@H](CO)O2	CID:54646181	phase I
BRD-K53914319	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@@H](CO)O2	CID:54646182	phase I
BRD-K45501379	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@H](CO)O2	CID:54646183	phase I
BRD-K82370171	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@@H](CO)O2	CID:54646184	phase I
BRD-K16030225	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)C5CCOCC5)cc34)[C@H](CO)O2	CID:54646185	phase I
BRD-K27066819	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@@H](CO)O2	CID:54646186	phase I
BRD-K11724909	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@H](CO)O2	CID:54646187	phase I
BRD-K06373442	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@@H](CO)O2	CID:54646188	phase I
BRD-K89567872	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@H](CO)O2	CID:54646189	phase I
BRD-K51266459	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@@H](CO)O2	CID:54646190	phase I
BRD-K37369665	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@H](CO)O2	CID:54646191	phase I
BRD-K57218099	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@@H](CO)O2	CID:54646192	phase I
BRD-K81582767	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34)[C@H](CO)O2	CID:54646193	phase I
BRD-K01594854	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4)cc23)[C@H](CO)O1	CID:54646194	phase I
BRD-K36360168	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccccc4)cc23)[C@@H](CO)O1	CID:54646195	phase I
BRD-K80576525	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4)cc23)[C@H](CO)O1	CID:54646196	phase I
BRD-K69438871	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4)cc23)[C@@H](CO)O1	CID:54646197	phase I
BRD-K94878334	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccccc4)cc23)[C@@H](CO)O1	CID:54646198	phase I
BRD-K86344535	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccccc4)cc23)[C@H](CO)O1	CID:54646199	phase I
BRD-K06559861	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccccn4)O[C@@H]3CO)c2c1	CID:54646200	phase I
BRD-K18713590	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@@H]3CO)c2c1	CID:54646201	phase I
BRD-K62657501	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@H]3CO)c2c1	CID:54646202	phase I
BRD-K50641952	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccccn4)O[C@H]3CO)c2c1	CID:54646203	phase I
BRD-K86154664	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccccn4)O[C@@H]3CO)c2c1	CID:54646204	phase I
BRD-K56417931	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@H]3CO)c2c1	CID:54646205	phase I
BRD-K10768305	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@@H]3CO)c2c1	CID:54646206	phase I
BRD-K23960714	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccccn4)O[C@H]3CO)c2c1	CID:54646207	phase I
BRD-K20822925	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23	CID:54646208	phase I
BRD-K08593711	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23	CID:54646209	phase I
BRD-K20469405	OC[C@@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23	CID:54646210	phase I
BRD-K36209664	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23	CID:54646211	phase I
BRD-K09845534	OC[C@@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)c4ccc5OCOc5c4)cc23	CID:54646212	phase I
BRD-K11088254	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)O)O[C@@H]3CO)c2c1	CID:54646213	phase I
BRD-K47890395	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)O)O[C@H]3CO)c2c1	CID:54646214	phase I
BRD-K90848748	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)O)O[C@H]3CO)c2c1	CID:54646215	phase I
BRD-K61339519	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)O)O[C@@H]3CO)c2c1	CID:54646216	phase I
BRD-K18748400	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)O)O[C@H]3CO)c2c1	CID:54646217	phase I
BRD-K57064803	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@@H]3CO)c2c1	CID:54646218	phase I
BRD-K16410418	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@H]3CO)c2c1	CID:54646219	phase I
BRD-K95880106	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@H]3CO)c2c1	CID:54646220	phase I
BRD-K66205522	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@@H]3CO)c2c1	CID:54646221	phase I
BRD-K61519793	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@H]3CO)c2c1	CID:54646222	phase I
BRD-K07967120	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@@H]3CO)c2c1	CID:54646223	phase I
BRD-K71031872	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc(Oc5ccccc5)cc4)O[C@H]3CO)c2c1	CID:54646224	phase I
BRD-K84994827	OC[C@H]1O[C@@H](CC(=O)NCc2ccncc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646225	phase I
BRD-K71611609	OC[C@@H]1O[C@H](CC(=O)NCc2ccncc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646226	phase I
BRD-K84239628	OC[C@H]1O[C@@H](CC(=O)NCc2ccncc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646227	phase I
BRD-K37020290	OC[C@@H]1O[C@H](CC(=O)NCc2ccncc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646228	phase I
BRD-K27679491	OC[C@H]1O[C@H](CC(=O)NCc2ccncc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646229	phase I
BRD-K20517870	OC[C@@H]1O[C@@H](CC(=O)NCc2ccncc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)NC5CCCC5)cc34	CID:54646230	phase I
BRD-K68323967	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646231	phase I
BRD-K51825814	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1)c5ccccc5	CID:54646232	phase I
BRD-K00259552	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646233	phase I
BRD-K17686770	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1)c5ccccc5	CID:54646234	phase I
BRD-K66131980	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646235	phase I
BRD-K10654753	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1)c5ccccc5	CID:54646236	phase I
BRD-K72375447	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646237	phase I
BRD-K10120618	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1)c5ccccc5	CID:54646238	phase I
BRD-K44777226	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccccn5)O[C@@H]4CO)c3c2)cc1	CID:54646239	phase I
BRD-K13185593	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCc5ccccn5)O[C@H]4CO)c3c2)cc1	CID:54646240	phase I
BRD-K96625719	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCc5ccccn5)O[C@@H]4CO)c3c2)cc1	CID:54646241	phase I
BRD-K62846431	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCc5ccccn5)O[C@H]4CO)c3c2)cc1	CID:54646242	phase I
BRD-K96922741	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCc5ccccn5)O[C@@H]4CO)c3c2)cc1	CID:54646243	phase I
BRD-K46319090	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCc5ccccn5)O[C@H]4CO)c3c2)cc1	CID:54646244	phase I
BRD-K51894281	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCc5ccccn5)O[C@@H]4CO)c3c2)cc1	CID:54646245	phase I
BRD-K67094066	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccccn5)O[C@H]4CO)c3c2)cc1	CID:54646246	phase I
BRD-K84120458	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccccc6F)cc45	CID:54646247	phase I
BRD-K36899442	OC[C@@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccccc6F)cc45	CID:54646248	phase I
BRD-K65485797	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccccc6F)cc45	CID:54646249	phase I
BRD-K02638906	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccccc6F)cc45	CID:54646250	phase I
BRD-K84047740	OC[C@@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccccc6F)cc45	CID:54646251	phase I
BRD-K39177148	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccccc6F)cc45	CID:54646252	phase I
BRD-K12441425	OC[C@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646253	phase I
BRD-K38121247	OC[C@@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646254	phase I
BRD-K97468443	OC[C@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646255	phase I
BRD-K41885374	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646256	phase I
BRD-K42083897	OC[C@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646257	phase I
BRD-K88968998	OC[C@@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646258	phase I
BRD-K82249256	OC[C@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646259	phase I
BRD-K52373488	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646260	phase I
BRD-K47064511	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646261	phase I
BRD-K33065959	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646262	phase I
BRD-K45124535	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646263	phase I
BRD-K56167818	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646264	phase I
BRD-K54971989	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646265	phase I
BRD-K40959762	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646266	phase I
BRD-K79750489	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646267	phase I
BRD-K85684641	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5)cc34	CID:54646268	phase I
BRD-K87850000	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@@H]4CO)c3c2)cc1	CID:54646269	phase I
BRD-K73558711	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2)cc1	CID:54646270	phase I
BRD-K20148542	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2)cc1	CID:54646271	phase I
BRD-K18024110	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@@H]4CO)c3c2)cc1	CID:54646272	phase I
BRD-K39148257	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2)cc1	CID:54646273	phase I
BRD-K40173185	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@@H]4CO)c3c2)cc1	CID:54646274	phase I
BRD-K43396185	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2)cc1	CID:54646275	phase I
BRD-K80059205	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCC4CC4)O[C@@H]3CO)c2c1	CID:54646276	phase I
BRD-K52356070	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646277	phase I
BRD-K37654434	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646278	phase I
BRD-K67348888	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCC4CC4)O[C@@H]3CO)c2c1	CID:54646279	phase I
BRD-K98463649	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646280	phase I
BRD-K60983473	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646281	phase I
BRD-K38493380	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646282	phase I
BRD-K13059597	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646283	phase I
BRD-K14261052	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646284	phase I
BRD-K69696272	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646285	phase I
BRD-K32799329	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646286	phase I
BRD-K17450769	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646287	phase I
BRD-K66689236	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646288	phase I
BRD-K99339232	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54646289	phase I
BRD-K68536005	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646290	phase I
BRD-K43006764	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646291	phase I
BRD-K07017100	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646292	phase I
BRD-K46003436	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646293	phase I
BRD-K12362628	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646294	phase I
BRD-K58052247	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646295	phase I
BRD-K37060179	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646296	phase I
BRD-K12868556	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646299	phase I
BRD-K87340398	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646300	phase I
BRD-K36671795	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646301	phase I
BRD-K86894923	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646302	phase I
BRD-K23058957	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646303	phase I
BRD-K20604601	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646304	phase I
BRD-K24427824	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Cc6ccncc6)cc45	CID:54646305	phase I
BRD-K23775758	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@@H](CO)O2	CID:54646306	phase I
BRD-K77125349	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@H](CO)O2	CID:54646307	phase I
BRD-K30438246	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@@H](CO)O2	CID:54646308	phase I
BRD-K07616985	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@H](CO)O2	CID:54646309	phase I
BRD-K22002407	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccccc5F)O[C@@H]4CO)c3c2	CID:54646310	phase I
BRD-K72739597	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCc5ccccc5F)O[C@H]4CO)c3c2	CID:54646311	phase I
BRD-K97972197	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCc5ccccc5F)O[C@@H]4CO)c3c2	CID:54646312	phase I
BRD-K73809982	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCc5ccccc5F)O[C@H]4CO)c3c2	CID:54646313	phase I
BRD-K77093925	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCc5ccccc5F)O[C@@H]4CO)c3c2	CID:54646314	phase I
BRD-K30613842	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCc5ccccc5F)O[C@H]4CO)c3c2	CID:54646315	phase I
BRD-K02813113	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCc5ccccc5F)O[C@@H]4CO)c3c2	CID:54646316	phase I
BRD-K59248941	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccccc5F)O[C@H]4CO)c3c2	CID:54646317	phase I
BRD-K52403446	OC[C@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646318	phase I
BRD-K10491285	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646321	phase I
BRD-K52780420	OC[C@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646322	phase I
BRD-K14509209	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646323	phase I
BRD-K22500599	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646324	phase I
BRD-K58719548	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646325	phase I
BRD-K55681488	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646326	phase I
BRD-K21047238	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646327	phase I
BRD-K19742528	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646328	phase I
BRD-K08432506	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646329	phase I
BRD-K71732099	OC[C@@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646330	phase I
BRD-K96238295	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCCN4CCCCC4)O[C@@H]3CO)c2c1	CID:54646331	phase I
BRD-K82768800	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCCN4CCCCC4)O[C@H]3CO)c2c1	CID:54646332	phase I
BRD-K13697129	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCCN4CCCCC4)O[C@@H]3CO)c2c1	CID:54646333	phase I
BRD-K24977302	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCCN4CCCCC4)O[C@@H]3CO)c2c1	CID:54646334	phase I
BRD-K94446761	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCCN4CCCCC4)O[C@H]3CO)c2c1	CID:54646335	phase I
BRD-K16075454	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646336	phase I
BRD-K52012504	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646337	phase I
BRD-K85774994	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646338	phase I
BRD-K50938873	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646339	phase I
BRD-K62299351	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646340	phase I
BRD-K33666425	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646341	phase I
BRD-K19084671	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646342	phase I
BRD-K10501200	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646343	phase I
BRD-K85200143	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)N5CCN(C)CC5)O[C@@H]4CO)c3c2)cc1	CID:54646344	phase I
BRD-K26095155	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)N5CCN(C)CC5)O[C@H]4CO)c3c2)cc1	CID:54646345	phase I
BRD-K96190924	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)N5CCN(C)CC5)O[C@@H]4CO)c3c2)cc1	CID:54646346	phase I
BRD-K11631766	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)N5CCN(C)CC5)O[C@H]4CO)c3c2)cc1	CID:54646347	phase I
BRD-K65913932	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)N5CCN(C)CC5)O[C@@H]4CO)c3c2)cc1	CID:54646348	phase I
BRD-K63585449	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)N5CCN(C)CC5)O[C@H]4CO)c3c2)cc1	CID:54646349	phase I
BRD-K30891382	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)N5CCN(C)CC5)O[C@@H]4CO)c3c2)cc1	CID:54646350	phase I
BRD-K75061326	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)N5CCN(C)CC5)O[C@H]4CO)c3c2)cc1	CID:54646351	phase I
BRD-K16063494	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646352	phase I
BRD-K53959928	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646353	phase I
BRD-K99723587	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646354	phase I
BRD-K13131627	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646355	phase I
BRD-K91449148	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646356	phase I
BRD-K07986943	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646357	phase I
BRD-K51998640	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccccn4)O[C@@H]3CO)c2c1	CID:54646358	phase I
BRD-K46473681	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@H]3CO)c2c1	CID:54646359	phase I
BRD-K36467636	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@H]3CO)c2c1	CID:54646360	phase I
BRD-K74823284	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccccn4)O[C@@H]3CO)c2c1	CID:54646361	phase I
BRD-K72785431	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc(Cl)cc4)O[C@@H]3CO)c2c1	CID:54646362	phase I
BRD-K89379568	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc(Cl)cc4)O[C@H]3CO)c2c1	CID:54646363	phase I
BRD-K61496587	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc(Cl)cc4)O[C@@H]3CO)c2c1	CID:54646364	phase I
BRD-K64700664	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc(Cl)cc4)O[C@H]3CO)c2c1	CID:54646365	phase I
BRD-K59611835	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc(Cl)cc4)O[C@@H]3CO)c2c1	CID:54646366	phase I
BRD-K95647562	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc(Cl)cc4)O[C@H]3CO)c2c1	CID:54646367	phase I
BRD-K94924347	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc(Cl)cc4)O[C@@H]3CO)c2c1	CID:54646368	phase I
BRD-K39236054	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc(Cl)cc4)O[C@H]3CO)c2c1	CID:54646369	phase I
BRD-K68103836	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@@H]3CO)c2c1	CID:54646370	phase I
BRD-K71963262	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@H]3CO)c2c1	CID:54646371	phase I
BRD-K00436546	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@@H]3CO)c2c1	CID:54646372	phase I
BRD-K88095357	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@H]3CO)c2c1	CID:54646373	phase I
BRD-K27935463	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@@H]3CO)c2c1	CID:54646374	phase I
BRD-K82246602	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@H]3CO)c2c1	CID:54646375	phase I
BRD-K40971145	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@@H]3CO)c2c1	CID:54646376	phase I
BRD-K53067088	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc(cc4)c5ccccc5)O[C@H]3CO)c2c1	CID:54646377	phase I
BRD-K24242444	CCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1	CID:54646378	phase I
BRD-K39007840	CCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1	CID:54646379	phase I
BRD-K22123421	CCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1	CID:54646380	phase I
BRD-K19529619	CCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1	CID:54646381	phase I
BRD-K71249580	CCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1	CID:54646382	phase I
BRD-K84098240	CCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1	CID:54646383	phase I
BRD-K05207940	CCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1	CID:54646384	phase I
BRD-K02544589	CCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1	CID:54646385	phase I
BRD-K89599747	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@@H](CO)O1	CID:54646386	phase I
BRD-K77621546	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@@H](CO)O1	CID:54646387	phase I
BRD-K96061818	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@H](CO)O1	CID:54646388	phase I
BRD-K24329506	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@@H](CO)O1	CID:54646389	phase I
BRD-K06086334	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@H](CO)O1	CID:54646390	phase I
BRD-K15980298	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@@H](CO)O1	CID:54646391	phase I
BRD-K62342148	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)C)cc23)[C@H](CO)O1	CID:54646392	phase I
BRD-K00349278	OC[C@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646393	phase I
BRD-K63843509	OC[C@@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646394	phase I
BRD-K06733952	OC[C@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646395	phase I
BRD-K01335708	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646396	phase I
BRD-K93468393	OC[C@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646397	phase I
BRD-K67851959	OC[C@@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646398	phase I
BRD-K62117749	OC[C@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646399	phase I
BRD-K32480492	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646400	phase I
BRD-K12187358	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(cc23)N(C)C)[C@@H](CO)O1)c4ccccc4	CID:54646401	phase I
BRD-K09085062	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(cc23)N(C)C)[C@H](CO)O1)c4ccccc4	CID:54646402	phase I
BRD-K94184760	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(cc23)N(C)C)[C@H](CO)O1)c4ccccc4	CID:54646403	phase I
BRD-K50587003	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(cc23)N(C)C)[C@@H](CO)O1)c4ccccc4	CID:54646404	phase I
BRD-K25094041	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(cc23)N(C)C)[C@H](CO)O1)c4ccccc4	CID:54646405	phase I
BRD-K99383477	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(cc23)N(C)C)[C@@H](CO)O1)c4ccccc4	CID:54646406	phase I
BRD-K98998964	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(cc23)N(C)C)[C@@H](CO)O1)c4ccccc4	CID:54646407	phase I
BRD-K78792702	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(cc23)N(C)C)[C@H](CO)O1)c4ccccc4	CID:54646408	phase I
BRD-K99915395	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(cc23)N(C)C)[C@H](CO)O1)c4ccccc4	CID:54646409	phase I
BRD-K40708745	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646410	phase I
BRD-K82758569	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646411	phase I
BRD-K74291148	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@@H]3CO)c2c1	CID:54646412	phase I
BRD-K24992635	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646413	phase I
BRD-K60697955	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@@H]3CO)c2c1	CID:54646414	phase I
BRD-K16506804	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646415	phase I
BRD-K60804903	OC[C@H]1O[C@H](CC(=O)NCc2cccc(F)c2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646416	phase I
BRD-K33881003	OC[C@@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646417	phase I
BRD-K25577594	OC[C@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646418	phase I
BRD-K21796872	OC[C@@H]1O[C@H](CC(=O)NCc2cccc(F)c2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646419	phase I
BRD-K82736385	OC[C@H]1O[C@H](CC(=O)NCc2cccc(F)c2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646420	phase I
BRD-K23701529	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCCCC4)O[C@@H]3CO)c2c1	CID:54646421	phase I
BRD-K29809218	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCCCC4)O[C@H]3CO)c2c1	CID:54646422	phase I
BRD-K35995762	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCCCC4)O[C@@H]3CO)c2c1	CID:54646423	phase I
BRD-K29258520	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCCCC4)O[C@H]3CO)c2c1	CID:54646424	phase I
BRD-K53665713	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCCCC4)O[C@@H]3CO)c2c1	CID:54646425	phase I
BRD-K00892322	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCCCC4)O[C@H]3CO)c2c1	CID:54646426	phase I
BRD-K54161818	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCCCC4)O[C@@H]3CO)c2c1	CID:54646427	phase I
BRD-K72373843	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCCCC4)O[C@H]3CO)c2c1	CID:54646428	phase I
BRD-K48911375	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NC5CCCCC5)O[C@@H]4CO)c3c2)cc1	CID:54646429	phase I
BRD-K98042112	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NC5CCCCC5)O[C@H]4CO)c3c2)cc1	CID:54646430	phase I
BRD-K56916873	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NC5CCCCC5)O[C@@H]4CO)c3c2)cc1	CID:54646431	phase I
BRD-K01825565	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NC5CCCCC5)O[C@H]4CO)c3c2)cc1	CID:54646432	phase I
BRD-K15476875	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NC5CCCCC5)O[C@@H]4CO)c3c2)cc1	CID:54646433	phase I
BRD-K39674306	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NC5CCCCC5)O[C@H]4CO)c3c2)cc1	CID:54646434	phase I
BRD-K93691156	CCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)COC)cc23)[C@@H](CO)O1	CID:54646435	phase I
BRD-K15318079	CCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)COC)cc23)[C@H](CO)O1	CID:54646436	phase I
BRD-K21707058	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646439	phase I
BRD-K57022684	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646440	phase I
BRD-K52045590	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646441	phase I
BRD-K47121420	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646442	phase I
BRD-K71259673	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646443	phase I
BRD-K44781836	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646444	phase I
BRD-K34898609	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646445	phase I
BRD-K19808762	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646446	phase I
BRD-K04776289	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646447	phase I
BRD-K69806016	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646448	phase I
BRD-K18932682	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646449	phase I
BRD-K07523222	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646450	phase I
BRD-K09521750	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646451	phase I
BRD-K51360326	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646452	phase I
BRD-K33017576	OC[C@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646453	phase I
BRD-K26212796	OC[C@@H]1O[C@H](CC(=O)NCc2cccc(F)c2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646454	phase I
BRD-K92650863	OC[C@H]1O[C@H](CC(=O)NCc2cccc(F)c2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646455	phase I
BRD-K19865807	OC[C@@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646456	phase I
BRD-K43526306	OC[C@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646457	phase I
BRD-K36888933	OC[C@@H]1O[C@H](CC(=O)NCc2cccc(F)c2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCC5)cc34	CID:54646458	phase I
BRD-K91809691	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccccc4F)O[C@H]3CO)c2c1	CID:54646461	phase I
BRD-K59196623	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccccc4F)O[C@@H]3CO)c2c1	CID:54646462	phase I
BRD-K01911039	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccccc4F)O[C@H]3CO)c2c1	CID:54646463	phase I
BRD-K67959996	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccccc4F)O[C@@H]3CO)c2c1	CID:54646464	phase I
BRD-K12159290	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccccc4F)O[C@H]3CO)c2c1	CID:54646465	phase I
BRD-K40389399	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccccc4F)O[C@@H]3CO)c2c1	CID:54646466	phase I
BRD-K61751605	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccccc4F)O[C@H]3CO)c2c1	CID:54646467	phase I
BRD-K56977200	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646468	phase I
BRD-K07558380	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646469	phase I
BRD-K51186655	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646470	phase I
BRD-K25469705	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646471	phase I
BRD-K26622714	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646472	phase I
BRD-K92079660	C[C@@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646473	phase I
BRD-K53934736	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646474	phase I
BRD-K37623909	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646475	phase I
BRD-K37510840	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646476	phase I
BRD-K63025696	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646477	phase I
BRD-K61437861	C[C@@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646478	phase I
BRD-K97112539	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646479	phase I
BRD-K66618978	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646480	phase I
BRD-K36150982	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646481	phase I
BRD-K94761446	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646482	phase I
BRD-K26077185	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)C4CCOCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646483	phase I
BRD-K83745732	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646484	phase I
BRD-K59913769	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646485	phase I
BRD-K14573341	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646486	phase I
BRD-K57207769	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646487	phase I
BRD-K12309677	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646488	phase I
BRD-K44657322	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646489	phase I
BRD-K79927100	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646490	phase I
BRD-K71485313	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCCC4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646491	phase I
BRD-K52656828	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NC4CCCCC4)O[C@@H]3CO)c2c1	CID:54646492	phase I
BRD-K01310096	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NC4CCCCC4)O[C@H]3CO)c2c1	CID:54646493	phase I
BRD-K77933659	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NC4CCCCC4)O[C@@H]3CO)c2c1	CID:54646494	phase I
BRD-K72988703	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NC4CCCCC4)O[C@H]3CO)c2c1	CID:54646495	phase I
BRD-K09404826	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NC4CCCCC4)O[C@@H]3CO)c2c1	CID:54646496	phase I
BRD-K10666842	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NC4CCCCC4)O[C@H]3CO)c2c1	CID:54646497	phase I
BRD-K43184721	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NC4CCCCC4)O[C@@H]3CO)c2c1	CID:54646498	phase I
BRD-K91423746	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NC4CCCCC4)O[C@H]3CO)c2c1	CID:54646499	phase I
BRD-K27948561	COCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1	CID:54646500	phase I
BRD-K11454759	COCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1	CID:54646501	phase I
BRD-K97630236	COCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1	CID:54646502	phase I
BRD-K99927461	COCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1	CID:54646503	phase I
BRD-K36970122	COCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1	CID:54646504	phase I
BRD-K33799929	COCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1	CID:54646505	phase I
BRD-K84497718	COCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@@H](CO)O1	CID:54646506	phase I
BRD-K56916068	COCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc23)[C@H](CO)O1	CID:54646507	phase I
BRD-K69873182	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646508	phase I
BRD-K43626867	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646509	phase I
BRD-K21163701	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646510	phase I
BRD-K58631614	OC[C@@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646511	phase I
BRD-K04267190	OC[C@H]1O[C@@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646512	phase I
BRD-K48431707	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646513	phase I
BRD-K16332856	OC[C@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646514	phase I
BRD-K16306049	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646515	phase I
BRD-K19876534	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646516	phase I
BRD-K35860134	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646517	phase I
BRD-K75627148	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646518	phase I
BRD-K18187596	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646519	phase I
BRD-K40045948	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@@H]4[C@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646520	phase I
BRD-K57345537	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Oc3ccccc3)cc2)C[C@H]4[C@@H]1Oc5ccc(NS(=O)(=O)c6ccc(F)cc6)cc45	CID:54646521	phase I
BRD-K13137954	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646522	phase I
BRD-K76257309	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646523	phase I
BRD-K87314084	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646524	phase I
BRD-K28648950	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646525	phase I
BRD-K03028122	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646526	phase I
BRD-K17299182	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646527	phase I
BRD-K27993001	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@@H](CO)O2	CID:54646528	phase I
BRD-K85242441	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34)[C@H](CO)O2	CID:54646529	phase I
BRD-K59731570	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cccnc4)O[C@@H]3CO)c2c1	CID:54646530	phase I
BRD-K56240103	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cccnc4)O[C@H]3CO)c2c1	CID:54646531	phase I
BRD-K86198141	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cccnc4)O[C@@H]3CO)c2c1	CID:54646532	phase I
BRD-K47105955	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cccnc4)O[C@H]3CO)c2c1	CID:54646533	phase I
BRD-K51392039	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cccnc4)O[C@@H]3CO)c2c1	CID:54646534	phase I
BRD-K82166043	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cccnc4)O[C@H]3CO)c2c1	CID:54646535	phase I
BRD-K85258806	COCC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cccnc4)O[C@@H]3CO)c2c1	CID:54646536	phase I
BRD-K13517531	COCC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cccnc4)O[C@H]3CO)c2c1	CID:54646537	phase I
BRD-K06852269	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54646538	phase I
BRD-K89551737	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54646539	phase I
BRD-K80226949	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54646540	phase I
BRD-K40414902	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54646541	phase I
BRD-K86483825	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54646542	phase I
BRD-K82935485	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@@H](CO)O2	CID:54646543	phase I
BRD-K89621861	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@@H](CO)O2	CID:54646544	phase I
BRD-K46300014	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@H](CO)O2	CID:54646545	phase I
BRD-K33544525	CN1CCN(CC1)C(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@@H](CO)O2	CID:54646546	phase I
BRD-K83544582	CN1CCN(CC1)C(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@H](CO)O2	CID:54646547	phase I
BRD-K87618551	CN1CCN(CC1)C(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@@H](CO)O2	CID:54646548	phase I
BRD-K64409112	CN1CCN(CC1)C(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Cc5ccncc5)cc34)[C@H](CO)O2	CID:54646549	phase I
BRD-K42482401	CN(C)C(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@@H](CO)O1	CID:54646550	phase I
BRD-K71271296	CN(C)C(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@H](CO)O1	CID:54646551	phase I
BRD-K36081737	CN(C)C(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@@H](CO)O1	CID:54646552	phase I
BRD-K09879686	CN(C)C(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@H](CO)O1	CID:54646553	phase I
BRD-K90556238	CN(C)C(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@@H](CO)O1	CID:54646554	phase I
BRD-K97102829	CN(C)C(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@H](CO)O1	CID:54646555	phase I
BRD-K09051149	CN(C)C(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@@H](CO)O1	CID:54646556	phase I
BRD-K97758158	CN(C)C(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CC4CC4)cc23)[C@H](CO)O1	CID:54646557	phase I
BRD-K29201528	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)N5CCCCC5)O[C@@H]4CO)c3c2	CID:54646558	phase I
BRD-K48562666	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)N5CCCCC5)O[C@H]4CO)c3c2	CID:54646559	phase I
BRD-K25734452	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)N5CCCCC5)O[C@@H]4CO)c3c2	CID:54646560	phase I
BRD-K51034923	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)N5CCCCC5)O[C@H]4CO)c3c2	CID:54646561	phase I
BRD-K68302437	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)N5CCCCC5)O[C@@H]4CO)c3c2	CID:54646562	phase I
BRD-K42074118	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)N5CCCCC5)O[C@H]4CO)c3c2	CID:54646563	phase I
BRD-K10210954	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)N5CCCCC5)O[C@@H]4CO)c3c2	CID:54646564	phase I
BRD-K06624861	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)N5CCCCC5)O[C@H]4CO)c3c2	CID:54646565	phase I
BRD-K66344816	OC[C@@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646566	phase I
BRD-K48714854	OC[C@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646567	phase I
BRD-K72875756	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646568	phase I
BRD-K24050338	OC[C@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646569	phase I
BRD-K38498143	OC[C@@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646570	phase I
BRD-K33263026	OC[C@H]1O[C@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646571	phase I
BRD-K09787095	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646572	phase I
BRD-K30635390	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646573	phase I
BRD-K82971022	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646574	phase I
BRD-K57607987	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646575	phase I
BRD-K78310246	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646576	phase I
BRD-K91745259	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646577	phase I
BRD-K02089646	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646578	phase I
BRD-K83933044	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646579	phase I
BRD-K45601310	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646580	phase I
BRD-K09864793	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)O)O[C@@H]4CO)c3c2)cc1	CID:54646581	phase I
BRD-K69724418	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)O)O[C@H]4CO)c3c2)cc1	CID:54646582	phase I
BRD-K39902590	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)O)O[C@H]4CO)c3c2)cc1	CID:54646583	phase I
BRD-K86438619	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)O)O[C@H]4CO)c3c2)cc1	CID:54646584	phase I
BRD-K20065144	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646585	phase I
BRD-K02445831	OC[C@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646586	phase I
BRD-K17783155	OC[C@@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Cc5ccncc5)cc34	CID:54646587	phase I
BRD-K63091163	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@@H]4CO)c3c2	CID:54646588	phase I
BRD-K43499440	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2	CID:54646589	phase I
BRD-K61416896	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@@H]4CO)c3c2	CID:54646590	phase I
BRD-K80362711	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2	CID:54646591	phase I
BRD-K00865615	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2	CID:54646592	phase I
BRD-K49830011	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCCc5ccccc5)O[C@@H]4CO)c3c2	CID:54646593	phase I
BRD-K27661070	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCCc5ccccc5)O[C@H]4CO)c3c2	CID:54646594	phase I
BRD-K01211710	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCC5CC5)O[C@@H]4CO)c3c2	CID:54646595	phase I
BRD-K89376450	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCC5CC5)O[C@H]4CO)c3c2	CID:54646596	phase I
BRD-K67765874	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCC5CC5)O[C@@H]4CO)c3c2	CID:54646597	phase I
BRD-K93320447	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCC5CC5)O[C@H]4CO)c3c2	CID:54646598	phase I
BRD-K60861723	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCC5CC5)O[C@@H]4CO)c3c2	CID:54646599	phase I
BRD-K29041589	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCC5CC5)O[C@H]4CO)c3c2	CID:54646600	phase I
BRD-K59755197	COc1ccc(cc1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCC5CC5)O[C@@H]4CO)c3c2	CID:54646601	phase I
BRD-K70550435	COCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@@H](CO)O1	CID:54646602	phase I
BRD-K95926324	COCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@H](CO)O1	CID:54646603	phase I
BRD-K96721928	COCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@@H](CO)O1	CID:54646604	phase I
BRD-K87089311	COCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@H](CO)O1	CID:54646605	phase I
BRD-K77827548	COCCNC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@@H](CO)O1	CID:54646606	phase I
BRD-K76882503	COCCNC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@H](CO)O1	CID:54646607	phase I
BRD-K08260539	COCCNC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@@H](CO)O1	CID:54646608	phase I
BRD-K00598313	COCCNC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NS(=O)(=O)c4ccccc4)cc23)[C@H](CO)O1	CID:54646609	phase I
BRD-K25237268	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6cccnc6)cc45	CID:54646610	phase I
BRD-K36418235	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6cccnc6)cc45	CID:54646611	phase I
BRD-K29475732	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6cccnc6)cc45	CID:54646612	phase I
BRD-K58438506	OC[C@H]1O[C@@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6cccnc6)cc45	CID:54646613	phase I
BRD-K73310446	OC[C@@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)c6cccnc6)cc45	CID:54646614	phase I
BRD-K83301268	OC[C@H]1O[C@H](CC(=O)N2CCc3ccccc3C2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)c6cccnc6)cc45	CID:54646615	phase I
BRD-K41182633	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646616	phase I
BRD-K16934333	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646617	phase I
BRD-K09444102	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646618	phase I
BRD-K25031780	OC[C@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646619	phase I
BRD-K94778363	OC[C@@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646620	phase I
BRD-K75405605	OC[C@H]1O[C@H](CC(=O)NCc2cccnc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646621	phase I
BRD-K48849176	OC[C@@H]1O[C@@H](CC(=O)NCc2cccnc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646622	phase I
BRD-K63926219	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCC4)cc23)[C@H](CO)O1	CID:54646623	phase I
BRD-K65974287	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCC4)cc23)[C@@H](CO)O1	CID:54646624	phase I
BRD-K38786629	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCC4)cc23)[C@H](CO)O1	CID:54646625	phase I
BRD-K47094330	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCC4)cc23)[C@H](CO)O1	CID:54646626	phase I
BRD-K03548778	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)NC4CCCC4)cc23)[C@@H](CO)O1	CID:54646627	phase I
BRD-K64997042	COC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)NC4CCCC4)cc23)[C@H](CO)O1	CID:54646628	phase I
BRD-K88641895	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)c4cccnc4)cc23	CID:54646629	phase I
BRD-K35589880	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)c4cccnc4)cc23	CID:54646630	phase I
BRD-K99517495	OC[C@@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)c4cccnc4)cc23	CID:54646631	phase I
BRD-K79339982	OC[C@H]1O[C@@H](CC(=O)NCC(F)(F)F)C[C@@H]2[C@H]1Oc3ccc(NC(=O)c4cccnc4)cc23	CID:54646632	phase I
BRD-K34383440	OC[C@@H]1O[C@H](CC(=O)NCC(F)(F)F)C[C@H]2[C@@H]1Oc3ccc(NC(=O)c4cccnc4)cc23	CID:54646633	phase I
BRD-K21281680	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646634	phase I
BRD-K23407460	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646635	phase I
BRD-K81943679	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646636	phase I
BRD-K46232974	C[C@@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646637	phase I
BRD-K50667779	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646638	phase I
BRD-K88119020	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646639	phase I
BRD-K68120955	C[C@@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646640	phase I
BRD-K63336416	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646641	phase I
BRD-K48038858	C[C@@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646642	phase I
BRD-K70231266	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646643	phase I
BRD-K02516751	C[C@@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646644	phase I
BRD-K46184370	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646645	phase I
BRD-K71742963	C[C@@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)c4cccnc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646646	phase I
BRD-K66757832	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Cc4ccncc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646647	phase I
BRD-K96079261	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Cc4ccncc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646648	phase I
BRD-K92023938	C[C@H](NC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Cc4ccncc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646649	phase I
BRD-K31703908	C[C@H](NC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Cc4ccncc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646650	phase I
BRD-K55134387	C[C@H](NC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)Cc4ccncc4)cc23)[C@@H](CO)O1)c5ccccc5	CID:54646651	phase I
BRD-K73650939	C[C@H](NC(=O)C[C@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)Cc4ccncc4)cc23)[C@H](CO)O1)c5ccccc5	CID:54646652	phase I
BRD-K58154162	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@@H](CO)O2	CID:54646653	phase I
BRD-K46498981	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@H](CO)O2	CID:54646654	phase I
BRD-K92897514	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@@H](CO)O2	CID:54646655	phase I
BRD-K09059649	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@H](CO)O2	CID:54646656	phase I
BRD-K70899691	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@@H](CO)O2	CID:54646657	phase I
BRD-K20381303	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@H](CO)O2	CID:54646658	phase I
BRD-K19549004	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@@H](CO)O2	CID:54646659	phase I
BRD-K45090628	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)c5cccnc5)cc34)[C@H](CO)O2	CID:54646660	phase I
BRD-K86824573	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4ccncc4)O[C@@H]3CO)c2c1	CID:54646661	phase I
BRD-K96021399	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccncc4)O[C@H]3CO)c2c1	CID:54646662	phase I
BRD-K11133230	CN(C)c1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccncc4)O[C@H]3CO)c2c1	CID:54646663	phase I
BRD-K13019660	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccncc4)O[C@@H]3CO)c2c1	CID:54646664	phase I
BRD-K13558526	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646665	phase I
BRD-K83025131	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646666	phase I
BRD-K86379744	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646667	phase I
BRD-K01632787	OC[C@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646668	phase I
BRD-K29956297	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646669	phase I
BRD-K86323620	OC[C@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646670	phase I
BRD-K26792953	OC[C@@H]1O[C@@H](CC(=O)NC2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NS(=O)(=O)c5ccc(F)cc5)cc34	CID:54646671	phase I
BRD-K27827760	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@@H](CO)O2	CID:54646672	phase I
BRD-K68504618	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@H](CO)O2	CID:54646673	phase I
BRD-K22345692	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@@H](CO)O2	CID:54646674	phase I
BRD-K31378663	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@H](CO)O2	CID:54646675	phase I
BRD-K08911251	COc1ccccc1CNC(=O)C[C@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@@H](CO)O2	CID:54646676	phase I
BRD-K12668859	COc1ccccc1CNC(=O)C[C@@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@H](CO)O2	CID:54646677	phase I
BRD-K71585748	COc1ccccc1CNC(=O)C[C@@H]2C[C@@H]3[C@@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@@H](CO)O2	CID:54646678	phase I
BRD-K01359264	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)CN(C)C)cc34)[C@H](CO)O2	CID:54646679	phase I
BRD-K40280267	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@@H]3CO)c2c1	CID:54646680	phase I
BRD-K27839561	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646681	phase I
BRD-K66052559	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@@H]3CO)c2c1	CID:54646682	phase I
BRD-K10856568	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646683	phase I
BRD-K06127304	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@@H]3CO)c2c1	CID:54646684	phase I
BRD-K79522563	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646685	phase I
BRD-K61885905	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)N4CCc5ccccc5C4)O[C@@H]3CO)c2c1	CID:54646686	phase I
BRD-K57072576	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)N4CCc5ccccc5C4)O[C@H]3CO)c2c1	CID:54646687	phase I
BRD-K93164329	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646688	phase I
BRD-K48230737	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646689	phase I
BRD-K32381042	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646690	phase I
BRD-K46920162	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646691	phase I
BRD-K21629388	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646692	phase I
BRD-K20332840	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646693	phase I
BRD-K89697623	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646694	phase I
BRD-K07373355	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646695	phase I
BRD-K80301668	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646696	phase I
BRD-K09945302	OC[C@@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646697	phase I
BRD-K68731139	OC[C@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646698	phase I
BRD-K28105726	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646699	phase I
BRD-K71254586	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646700	phase I
BRD-K03815046	OC[C@@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646701	phase I
BRD-K98370172	OC[C@H]1O[C@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646702	phase I
BRD-K92205342	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)C6CCOCC6)cc45	CID:54646703	phase I
BRD-K37991633	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCC4CC4)O[C@@H]3CO)c2c1	CID:54646704	phase I
BRD-K82004089	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646705	phase I
BRD-K28739456	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCC4CC4)O[C@@H]3CO)c2c1	CID:54646706	phase I
BRD-K95899688	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646707	phase I
BRD-K54822582	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCC4CC4)O[C@@H]3CO)c2c1	CID:54646708	phase I
BRD-K66413861	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646709	phase I
BRD-K35915475	CS(=O)(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCC4CC4)O[C@@H]3CO)c2c1	CID:54646710	phase I
BRD-K38524184	CS(=O)(=O)Nc1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCC4CC4)O[C@H]3CO)c2c1	CID:54646711	phase I
BRD-K59519347	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646712	phase I
BRD-K09547783	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646713	phase I
BRD-K44755254	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646714	phase I
BRD-K54737430	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646715	phase I
BRD-K25970159	OC[C@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646716	phase I
BRD-K59941784	OC[C@@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646717	phase I
BRD-K06790322	OC[C@H]1O[C@H](CC(=O)NCc2ccc(Cl)cc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646718	phase I
BRD-K53046450	OC[C@@H]1O[C@@H](CC(=O)NCc2ccc(Cl)cc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)CC5CC5)cc34	CID:54646719	phase I
BRD-K98842254	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccc(Cl)cc5)O[C@@H]4CO)c3c2	CID:54646720	phase I
BRD-K74902280	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCc5ccc(Cl)cc5)O[C@@H]4CO)c3c2	CID:54646721	phase I
BRD-K54595917	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCc5ccc(Cl)cc5)O[C@H]4CO)c3c2	CID:54646722	phase I
BRD-K59534645	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@H](CC(=O)NCc5ccc(Cl)cc5)O[C@@H]4CO)c3c2	CID:54646723	phase I
BRD-K26205424	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@@H](CC(=O)NCc5ccc(Cl)cc5)O[C@H]4CO)c3c2	CID:54646724	phase I
BRD-K39921641	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCc5ccc(Cl)cc5)O[C@@H]4CO)c3c2	CID:54646725	phase I
BRD-K53873629	COc1cccc(c1)S(=O)(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccc(Cl)cc5)O[C@H]4CO)c3c2	CID:54646726	phase I
BRD-K37822854	OC[C@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646727	phase I
BRD-K22307331	OC[C@@H]1O[C@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646728	phase I
BRD-K66566233	OC[C@H]1O[C@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646729	phase I
BRD-K80831196	OC[C@@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646730	phase I
BRD-K97636821	OC[C@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646731	phase I
BRD-K62768599	OC[C@@H]1O[C@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646732	phase I
BRD-K02548021	OC[C@H]1O[C@H](CC(=O)N2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646733	phase I
BRD-K67029063	OC[C@@H]1O[C@@H](CC(=O)N2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)C5CCOCC5)cc34	CID:54646734	phase I
BRD-K85770991	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646735	phase I
BRD-K80621614	CN(C)c1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cc(F)ccc4F)O[C@@H]3CO)c2c1	CID:54646736	phase I
BRD-K97424742	CN(C)c1ccc2O[C@H]3[C@H](C[C@H](CC(=O)NCc4cc(F)ccc4F)O[C@H]3CO)c2c1	CID:54646737	phase I
BRD-K80807816	OC[C@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646738	phase I
BRD-K71386122	OC[C@@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646739	phase I
BRD-K51287451	OC[C@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646740	phase I
BRD-K38545029	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646741	phase I
BRD-K32240700	OC[C@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646742	phase I
BRD-K91786278	OC[C@@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646743	phase I
BRD-K16782770	OC[C@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646744	phase I
BRD-K84284503	OC[C@@H]1O[C@@H](CC(=O)NCCc2ccccc2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54646745	phase I
BRD-K63428678	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646746	phase I
BRD-K27919582	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646747	phase I
BRD-K92789454	OC[C@@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646748	phase I
BRD-K49076793	OC[C@H]1O[C@@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646749	phase I
BRD-K68047011	OC[C@@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646750	phase I
BRD-K48047626	OC[C@H]1O[C@H](CC(=O)NCCN2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)c5cccnc5)cc34	CID:54646751	phase I
BRD-K36994929	COC(=O)C[C@@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646752	phase I
BRD-K00998404	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@@H](CO)O1	CID:54646753	phase I
BRD-K91589308	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646754	phase I
BRD-K19056919	COC(=O)C[C@H]1C[C@@H]2[C@@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@@H](CO)O1	CID:54646755	phase I
BRD-K02275742	COC(=O)C[C@@H]1C[C@H]2[C@H](Oc3ccc(NC(=O)CN(C)C)cc23)[C@H](CO)O1	CID:54646756	phase I
BRD-K26508045	COc1ccc(NC(=O)Nc2ccc3O[C@H]4[C@H](C[C@H](CC(=O)NCc5ccncc5)O[C@@H]4CO)c3c2)cc1	CID:54646779	phase I
BRD-K28615450	COc1ccc(NC(=O)Nc2ccc3O[C@@H]4[C@@H](C[C@@H](CC(=O)NCc5ccncc5)O[C@H]4CO)c3c2)cc1	CID:54646780	phase I
BRD-K78438907	OC[C@@H]1O[C@H](CC(=O)NCC2CC2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54646948	phase I
BRD-K32628102	OC[C@@H]1O[C@H](CC(=O)NCc2cc(F)ccc2F)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccccc5F)cc34	CID:54647052	phase I
BRD-K74667984	OC[C@H]1O[C@@H](CC(=O)NCc2cccc(F)c2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)c5ccc6OCOc6c5)cc34	CID:54647077	phase I
BRD-K99692850	COc1ccccc1CNC(=O)C[C@H]2C[C@H]3[C@H](Oc4ccc(NC(=O)Nc5ccccc5F)cc34)[C@H](CO)O2	CID:54647099	phase I
BRD-K17712926	OC[C@@H]1O[C@H](CC(=O)NCCc2ccccc2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54647107	phase I
BRD-K12360898	OC[C@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@H]3[C@@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54647195	phase I
BRD-K03883227	OC[C@@H]1O[C@@H](CC(=O)NCc2ccccn2)C[C@@H]3[C@H]1Oc4ccc(NC(=O)Nc5ccc(cc5)C(F)(F)F)cc34	CID:54647198	phase I
BRD-K06296238	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4ccncc4)O[C@@H]3CO)c2c1	CID:54647209	phase I
BRD-K24946412	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@H]4[C@@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54647362	phase I
BRD-K35616093	OC[C@H]1O[C@@H](CC(=O)NCc2ccc3OCOc3c2)C[C@@H]4[C@H]1Oc5ccc(NC(=O)Nc6ccc(cc6)C(F)(F)F)cc45	CID:54647366	phase I
BRD-K49988555	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54647487	phase I
BRD-K52047117	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@H](CC(=O)NCc4ccc5OCOc5c4)O[C@@H]3CO)c2c1	CID:54647489	phase I
BRD-K25388406	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4ccc5OCOc5c4)O[C@H]3CO)c2c1	CID:54647490	phase I
BRD-K33932270	CN(C)CC(=O)Nc1ccc2O[C@H]3[C@H](C[C@@H](CC(=O)NCc4cccnc4)O[C@H]3CO)c2c1	CID:54647772	phase I
BRD-K40690989	CN(C)CC(=O)Nc1ccc2O[C@@H]3[C@@H](C[C@@H](CC(=O)NCc4cccnc4)O[C@@H]3CO)c2c1	CID:54647773	phase I
BRD-K23438281	OC[C@@H]1O[C@H](CC(=O)NC2CCCCC2)C[C@@H]3[C@H]1Oc4ccc(NS(=O)(=O)c5ccccc5)cc34	CID:54648908	phase I
BRD-K30752405	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648972	phase I
BRD-K95434109	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648973	phase I
BRD-K48307191	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648974	phase I
BRD-K41844882	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648975	phase I
BRD-K56747890	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648976	phase I
BRD-K45494661	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648977	phase I
BRD-K27610514	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54648978	phase I
BRD-K76251313	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648979	phase I
BRD-K86097224	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648980	phase I
BRD-K91581849	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648981	phase I
BRD-K36516410	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648982	phase I
BRD-K23628394	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648983	phase I
BRD-K30218805	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648984	phase I
BRD-K17381515	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648985	phase I
BRD-K51141297	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54648986	phase I
BRD-K23233872	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54648987	phase I
BRD-K63968737	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54648988	phase I
BRD-K15579005	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54648989	phase I
BRD-K87804315	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54648990	phase I
BRD-K96425583	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54648991	phase I
BRD-K86879226	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54648992	phase I
BRD-K55522920	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54648993	phase I
BRD-K94940283	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54648994	phase I
BRD-K59633080	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54648995	phase I
BRD-K27962962	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54648996	phase I
BRD-K74078391	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54648997	phase I
BRD-K57408604	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54648998	phase I
BRD-K76261045	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54648999	phase I
BRD-K40543019	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649000	phase I
BRD-K30446755	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649001	phase I
BRD-K89388769	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649002	phase I
BRD-K68423398	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649003	phase I
BRD-K57766599	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649004	phase I
BRD-K50648023	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649005	phase I
BRD-K99161484	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649006	phase I
BRD-K11019021	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649007	phase I
BRD-K88943141	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649008	phase I
BRD-K18009761	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649009	phase I
BRD-K73196232	CO[C@H](CN(C)CC1CCOCC1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649010	phase I
BRD-K23727664	CO[C@@H](CN(C)CC1CCOCC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649011	phase I
BRD-K07020505	CO[C@@H](CN(C)CC1CCOCC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649012	phase I
BRD-K28709114	CO[C@H](CN(C)CC1CCOCC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649013	phase I
BRD-K61960033	CO[C@H](CN(C)CC1CCOCC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649014	phase I
BRD-K74257705	CO[C@H](CN(C)CC1CCOCC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649015	phase I
BRD-K23901007	CO[C@@H](CN(C)CC1CCOCC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649016	phase I
BRD-K79828436	CO[C@@H](CN(C)CC1CCOCC1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649017	phase I
BRD-K43963447	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649018	phase I
BRD-K10275859	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649019	phase I
BRD-K56211108	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649020	phase I
BRD-K73255556	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649021	phase I
BRD-K68361061	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649022	phase I
BRD-K58023987	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649023	phase I
BRD-K58042174	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649024	phase I
BRD-K68219508	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649025	phase I
BRD-K35440877	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649026	phase I
BRD-K72787581	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649027	phase I
BRD-K71197999	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649028	phase I
BRD-K83620070	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649029	phase I
BRD-K15222491	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649030	phase I
BRD-K08993600	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649031	phase I
BRD-K45853775	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649032	phase I
BRD-K67335820	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649033	phase I
BRD-K15811513	CO[C@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649034	phase I
BRD-K12767001	CO[C@@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649035	phase I
BRD-K29636459	CO[C@@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649036	phase I
BRD-K81899744	CO[C@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649037	phase I
BRD-K97163189	CO[C@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649038	phase I
BRD-K71892893	CO[C@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649039	phase I
BRD-K30113303	CO[C@@H](CN(C)C(=O)Nc1ccc(cc1)C(F)(F)F)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649040	phase I
BRD-K49919280	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649041	phase I
BRD-K03346868	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649042	phase I
BRD-K93490141	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649043	phase I
BRD-K37993296	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649044	phase I
BRD-K14487280	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649045	phase I
BRD-K19613760	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649046	phase I
BRD-K50085158	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649047	phase I
BRD-K12936425	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649048	phase I
BRD-K12425451	CO[C@H](CN(C)Cc1nccs1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649049	phase I
BRD-K89427926	CO[C@@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649050	phase I
BRD-K69556935	CO[C@@H](CN(C)Cc1nccs1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649051	phase I
BRD-K70871724	CO[C@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649052	phase I
BRD-K67241457	CO[C@H](CN(C)Cc1nccs1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649053	phase I
BRD-K25090764	CO[C@@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649054	phase I
BRD-K53272350	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649055	phase I
BRD-K06457057	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649056	phase I
BRD-K86986995	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649057	phase I
BRD-K82155738	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649058	phase I
BRD-K25323340	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649059	phase I
BRD-K72867209	CO[C@@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649060	phase I
BRD-K23931095	CO[C@H](CN(C)S(=O)(=O)c1cn(C)cn1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649061	phase I
BRD-K25498394	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649062	phase I
BRD-K51844455	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649063	phase I
BRD-K53345186	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649064	phase I
BRD-K59392211	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649065	phase I
BRD-K80253007	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649066	phase I
BRD-K04718515	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649067	phase I
BRD-K77596635	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649068	phase I
BRD-K04073989	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649069	phase I
BRD-K14061746	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649070	phase I
BRD-K16344244	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649071	phase I
BRD-K65354878	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649072	phase I
BRD-K45184415	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649073	phase I
BRD-K67798781	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649074	phase I
BRD-K88179544	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649075	phase I
BRD-K67933714	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649076	phase I
BRD-K64178462	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649077	phase I
BRD-K32162437	CO[C@H](CN(C)Cc1nccs1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649078	phase I
BRD-K93177490	CO[C@@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649079	phase I
BRD-K97737065	CO[C@@H](CN(C)Cc1nccs1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649080	phase I
BRD-K73109344	CO[C@H](CN(C)Cc1nccs1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649081	phase I
BRD-K55380358	CO[C@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649082	phase I
BRD-K42558476	CO[C@@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649083	phase I
BRD-K63865470	CO[C@@H](CN(C)Cc1nccs1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649084	phase I
BRD-K10814161	CO[C@H](CN(C)Cc1nccs1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649085	phase I
BRD-K97327508	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649086	phase I
BRD-K57490754	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649087	phase I
BRD-K41190238	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649088	phase I
BRD-K32894756	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649089	phase I
BRD-K64478813	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649090	phase I
BRD-K36014883	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649091	phase I
BRD-K45147071	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649092	phase I
BRD-K22010555	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649093	phase I
BRD-K30403168	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649094	phase I
BRD-K87893855	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649095	phase I
BRD-K21547311	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649096	phase I
BRD-K37920059	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649097	phase I
BRD-K65350890	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649098	phase I
BRD-K97722965	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649099	phase I
BRD-K63216438	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649100	phase I
BRD-K50832163	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649101	phase I
BRD-K31147434	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649102	phase I
BRD-K69091193	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649103	phase I
BRD-K87728132	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649104	phase I
BRD-K53813421	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649105	phase I
BRD-K79255795	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649106	phase I
BRD-K98742259	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649107	phase I
BRD-K11667974	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649108	phase I
BRD-K38678832	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649109	phase I
BRD-K68380056	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649110	phase I
BRD-K40597283	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649111	phase I
BRD-K21139275	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649112	phase I
BRD-K56398628	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649113	phase I
BRD-K71095875	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649114	phase I
BRD-K46178029	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649115	phase I
BRD-K61873333	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649116	phase I
BRD-K08813275	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649117	phase I
BRD-K86757617	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649118	phase I
BRD-K89109315	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649119	phase I
BRD-K23744058	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649120	phase I
BRD-K90613621	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649121	phase I
BRD-K05640282	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649122	phase I
BRD-K07003080	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649123	phase I
BRD-K52898544	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649124	phase I
BRD-K78011385	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649125	phase I
BRD-K67540261	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649126	phase I
BRD-K02132857	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649127	phase I
BRD-K75092094	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649128	phase I
BRD-K21386069	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649129	phase I
BRD-K56601439	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649130	phase I
BRD-K52457887	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649131	phase I
BRD-K22595386	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649132	phase I
BRD-K55193076	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649133	phase I
BRD-K32277249	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649134	phase I
BRD-K67921699	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649135	phase I
BRD-K94365199	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649136	phase I
BRD-K38991762	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649137	phase I
BRD-K89146275	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649138	phase I
BRD-K32563579	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649139	phase I
BRD-K85498716	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649140	phase I
BRD-K55624132	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649141	phase I
BRD-K67689741	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649142	phase I
BRD-K64266734	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649143	phase I
BRD-K74546480	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649144	phase I
BRD-K24986598	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649145	phase I
BRD-K49545421	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649146	phase I
BRD-K85739307	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649147	phase I
BRD-K44478610	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649148	phase I
BRD-K79258593	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649149	phase I
BRD-K87123346	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649150	phase I
BRD-K74211371	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649151	phase I
BRD-K00256608	CO[C@@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649152	phase I
BRD-K47240178	CO[C@@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649153	phase I
BRD-K18144986	CO[C@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649154	phase I
BRD-K01435720	CO[C@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649155	phase I
BRD-K00671069	CO[C@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649156	phase I
BRD-K06550805	CO[C@@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649157	phase I
BRD-K90140894	CO[C@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649158	phase I
BRD-K17863985	CO[C@@H](CN(C)C(=O)Nc1ccc(F)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649159	phase I
BRD-K92864945	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649160	phase I
BRD-K94685656	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649161	phase I
BRD-K98938228	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649162	phase I
BRD-K96267517	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649163	phase I
BRD-K42620042	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649164	phase I
BRD-K03016409	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649165	phase I
BRD-K50929556	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649166	phase I
BRD-K57667228	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649167	phase I
BRD-K06022983	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649168	phase I
BRD-K85773425	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649169	phase I
BRD-K96005107	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649170	phase I
BRD-K55659732	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649171	phase I
BRD-K03643699	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649172	phase I
BRD-K02341205	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649173	phase I
BRD-K74750574	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649174	phase I
BRD-K16004461	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649175	phase I
BRD-K05078233	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649176	phase I
BRD-K43857354	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649177	phase I
BRD-K00223956	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649178	phase I
BRD-K85805864	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649179	phase I
BRD-K48040318	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649180	phase I
BRD-K58835910	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649181	phase I
BRD-K68312364	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649182	phase I
BRD-K53803963	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649183	phase I
BRD-K41125638	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649184	phase I
BRD-K15418616	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649185	phase I
BRD-K60860515	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649186	phase I
BRD-K28276103	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649187	phase I
BRD-K56261447	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649188	phase I
BRD-K35554380	CO[C@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649189	phase I
BRD-K19616315	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649190	phase I
BRD-K93291781	CO[C@@H](CN(C)S(=O)(=O)c1ccccc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649191	phase I
BRD-K64290134	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649192	phase I
BRD-K95877457	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649193	phase I
BRD-K84739463	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649194	phase I
BRD-K35829399	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649195	phase I
BRD-K72451078	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649196	phase I
BRD-K04521490	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649197	phase I
BRD-K77588167	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649198	phase I
BRD-K99763083	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649199	phase I
BRD-K73096266	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649200	phase I
BRD-K80394569	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649201	phase I
BRD-K06877934	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649202	phase I
BRD-K67480908	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649203	phase I
BRD-K96752633	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649204	phase I
BRD-K86985145	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649205	phase I
BRD-K04922291	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649206	phase I
BRD-K13141487	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649207	phase I
BRD-K87373784	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649208	phase I
BRD-K09761560	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649209	phase I
BRD-K44549295	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649210	phase I
BRD-K96855280	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649211	phase I
BRD-K85827194	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649212	phase I
BRD-K38177488	CO[C@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649213	phase I
BRD-K73083114	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649214	phase I
BRD-K17566112	CO[C@@H](CN(C)C(=O)c1ccccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649215	phase I
BRD-K02442093	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649218	phase I
BRD-K97717522	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649219	phase I
BRD-K99737029	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649220	phase I
BRD-K65763571	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649221	phase I
BRD-K42553302	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649222	phase I
BRD-K63279176	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649223	phase I
BRD-K08472586	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649224	phase I
BRD-K47926873	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649225	phase I
BRD-K09725203	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649226	phase I
BRD-K16068142	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649227	phase I
BRD-K76931353	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649228	phase I
BRD-K09555199	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649229	phase I
BRD-K13400061	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649230	phase I
BRD-K49183852	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@H](C)CO)C(=O)c1ccccc1	CID:54649231	phase I
BRD-K61620767	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)C(=O)c1ccccc1	CID:54649232	phase I
BRD-K90552071	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)C(=O)c1ccccc1	CID:54649233	phase I
BRD-K98303739	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)C(=O)c1ccccc1	CID:54649234	phase I
BRD-K78386654	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)C(=O)c1ccccc1	CID:54649235	phase I
BRD-K29388838	CO[C@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@@H](C)CO)C(=O)c1ccccc1	CID:54649236	phase I
BRD-K07357513	CO[C@@H](CN(C)Cc1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)C(=O)c1ccccc1	CID:54649237	phase I
BRD-K00636532	CO[C@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649240	phase I
BRD-K42605934	CO[C@@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649241	phase I
BRD-K69954048	CO[C@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649242	phase I
BRD-K99155518	CO[C@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649243	phase I
BRD-K62761144	CO[C@@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649244	phase I
BRD-K16514883	CO[C@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@@H](C)CN(Cc1ccccc1Cl)[C@@H](C)CO	CID:54649245	phase I
BRD-K92986986	CO[C@@H](CN(C)C(=O)Nc1ccc(Cl)cc1)[C@H](C)CN(Cc1ccccc1Cl)[C@H](C)CO	CID:54649246	phase I
BRD-K76084102	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649247	phase I
BRD-K65470727	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649248	phase I
BRD-K34122000	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649249	phase I
BRD-K04575404	CO[C@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649250	phase I
BRD-K05803357	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649251	phase I
BRD-K44225498	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649252	phase I
BRD-K29276696	CO[C@H](CN(C)C(=O)c1cnccn1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649253	phase I
BRD-K47885451	CO[C@@H](CN(C)C(=O)c1cnccn1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649254	phase I
BRD-K86059888	CO[C@@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649255	phase I
BRD-K82993704	CO[C@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649256	phase I
BRD-K60624482	CO[C@@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649257	phase I
BRD-K62820230	CO[C@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649258	phase I
BRD-K76732672	CO[C@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649259	phase I
BRD-K30151357	CO[C@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649260	phase I
BRD-K35930698	CO[C@@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649261	phase I
BRD-K67555693	CO[C@@H](CN(C)Cc1ccc(cc1)-c1ccccn1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649262	phase I
BRD-K23770948	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649263	phase I
BRD-K08002976	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649264	phase I
BRD-K64860117	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649265	phase I
BRD-K36261261	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649266	phase I
BRD-K06794322	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649267	phase I
BRD-K77265816	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649268	phase I
BRD-K94521200	CO[C@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649269	phase I
BRD-K02732091	CO[C@@H](CN(C)S(=O)(=O)c1ccc(C)cc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649270	phase I
BRD-K53931115	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649271	phase I
BRD-K12272248	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649272	phase I
BRD-K21498250	CO[C@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649273	phase I
BRD-K77003912	CO[C@@H](CN(C)C(=O)c1ccc2OCOc2c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649274	phase I
BRD-K33039006	CO[C@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649275	phase I
BRD-K45339826	CO[C@@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649276	phase I
BRD-K86571176	CO[C@@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649277	phase I
BRD-K60705848	CO[C@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649278	phase I
BRD-K99100793	CO[C@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649279	phase I
BRD-K39107373	CO[C@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649280	phase I
BRD-K32434708	CO[C@@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649281	phase I
BRD-K22041611	CO[C@@H](CN(C)C(=O)c1cc(Cl)cc(Cl)c1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(F)cc1	CID:54649282	phase I
BRD-K00445923	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649283	phase I
BRD-K10813758	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649284	phase I
BRD-K86250735	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649285	phase I
BRD-K85229892	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649286	phase I
BRD-K68300134	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649287	phase I
BRD-K88676137	CO[C@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649288	phase I
BRD-K08703292	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649289	phase I
BRD-K16372954	CO[C@@H](CN(C)C(=O)C1CCOCC1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccccc1	CID:54649290	phase I
BRD-K22629238	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(C)cc1	CID:54649291	phase I
BRD-K36462169	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649294	phase I
BRD-K00381581	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649295	phase I
BRD-K77316712	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649296	phase I
BRD-K10558099	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649297	phase I
BRD-K68774060	CO[C@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccccc1F	CID:54649298	phase I
BRD-K57061210	CO[C@@H](CN(C)S(=O)(=O)c1ccc(F)cc1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccccc1F	CID:54649299	phase I
BRD-K18246949	CO[C@@H](CN(C)C(=O)C1CC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649300	phase I
BRD-K49480198	CO[C@H](CN(C)C(=O)C1CC1)[C@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649301	phase I
BRD-K57962577	CO[C@@H](CN(C)C(=O)C1CC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649302	phase I
BRD-K92137277	CO[C@H](CN(C)C(=O)C1CC1)[C@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649303	phase I
BRD-K42733037	CO[C@H](CN(C)C(=O)C1CC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649304	phase I
BRD-K20721504	CO[C@@H](CN(C)C(=O)C1CC1)[C@@H](C)CN([C@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649305	phase I
BRD-K96586144	CO[C@H](CN(C)C(=O)C1CC1)[C@@H](C)CN([C@@H](C)CO)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54649306	phase I
BRD-K67433929	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649307	phase I
BRD-K93894185	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649308	phase I
BRD-K03416270	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649309	phase I
BRD-K37766746	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649310	phase I
BRD-K25164076	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649311	phase I
BRD-K76636716	CO[C@@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649312	phase I
BRD-K71387353	CO[C@H](CN(C)Cc1cc(F)ccc1F)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(F)cc1	CID:54649313	phase I
BRD-K16636143	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649316	phase I
BRD-K36777393	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649317	phase I
BRD-K55100062	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649318	phase I
BRD-K18440865	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649319	phase I
BRD-K45336346	CO[C@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649320	phase I
BRD-K44993940	CO[C@@H](CN(C)S(=O)(=O)c1cccc(Cl)c1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1ccc(Cl)cc1	CID:54649321	phase I
BRD-K08373870	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649322	phase I
BRD-K05733208	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649323	phase I
BRD-K69705756	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649324	phase I
BRD-K82328933	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649325	phase I
BRD-K69586787	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649326	phase I
BRD-K72694250	CO[C@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649327	phase I
BRD-K64649040	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649328	phase I
BRD-K10449938	CO[C@@H](CN(C)S(=O)(=O)c1ccc(Cl)cc1)[C@H](C)CN([C@H](C)CO)S(=O)(=O)c1cccc(Cl)c1	CID:54649329	phase I
BRD-K84935204	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCc1ccncc1	CID:54649330	phase I
BRD-K45883686	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCc1ccncc1	CID:54649331	phase I
BRD-K14535500	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)N1CCOCC1	CID:54649332	phase I
BRD-K01478916	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)N1CCOCC1	CID:54649333	phase I
BRD-K06718821	C\C=C\c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649334	phase I
BRD-K08663380	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NC1CCCCC1	CID:54649335	phase I
BRD-K76784707	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NC1CCCCC1	CID:54649336	phase I
BRD-K51041684	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)N1CCc2ccccc2C1	CID:54649337	phase I
BRD-K84567604	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)N1CCc2ccccc2C1	CID:54649338	phase I
BRD-K64920356	CN1CCN(CC1)C(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1ccc(cc1)C#N)[S@@](=O)C(C)(C)C	CID:54649339	phase I
BRD-K73575094	CN1CCN(CC1)C(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1ccc(cc1)C#N)[S@](=O)C(C)(C)C	CID:54649340	phase I
BRD-K55038865	COCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@](=O)C(C)(C)C	CID:54649341	phase I
BRD-K63521250	COCCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@@](=O)C(C)(C)C	CID:54649342	phase I
BRD-K55896440	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCCN1CCCCC1	CID:54649343	phase I
BRD-K37638153	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCCN1CCCCC1	CID:54649344	phase I
BRD-K05791917	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)NCc1ccccn1	CID:54649345	phase I
BRD-K45340761	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)NCc1ccccn1	CID:54649346	phase I
BRD-K47570616	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccc(F)c1)C(=O)NCC(F)(F)F	CID:54649347	phase I
BRD-K14002526	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccc(F)c1)C(=O)NCC(F)(F)F	CID:54649348	phase I
BRD-K15453459	COc1cccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(c2)-c2ccc(cc2)C#N)[S@@](=O)C(C)(C)C)c1	CID:54649349	phase I
BRD-K16348047	COc1cccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(c2)-c2ccc(cc2)C#N)[S@](=O)C(C)(C)C)c1	CID:54649350	phase I
BRD-K35535652	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cncnc1)C(=O)NCc1ccccc1F	CID:54649351	phase I
BRD-K01594626	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cncnc1)C(=O)NCc1ccccc1F	CID:54649352	phase I
BRD-K73104592	COc1ccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(\C=C\C)c2)[S@](=O)C(C)(C)C)cc1	CID:54649353	phase I
BRD-K05961870	COc1ccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(\C=C\C)c2)[S@@](=O)C(C)(C)C)cc1	CID:54649354	phase I
BRD-K49685495	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCCCC1	CID:54649355	phase I
BRD-K64801282	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCCCC1	CID:54649356	phase I
BRD-K02785641	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)NC1CCC1	CID:54649357	phase I
BRD-K98419480	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)NC1CCC1	CID:54649358	phase I
BRD-K77811363	CN(C)C(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1ccc(F)cc1)[S@](=O)C(C)(C)C	CID:54649359	phase I
BRD-K50358328	CN(C)C(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1ccc(F)cc1)[S@@](=O)C(C)(C)C	CID:54649360	phase I
BRD-K62732912	CN1CCN(CC1)C(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@@](=O)C(C)(C)C	CID:54649361	phase I
BRD-K79781870	CN1CCN(CC1)C(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@](=O)C(C)(C)C	CID:54649362	phase I
BRD-K63374765	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCCc1ccncc1	CID:54649363	phase I
BRD-K17525686	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCCc1ccncc1	CID:54649364	phase I
BRD-K70201679	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NCc1ccccc1	CID:54649365	phase I
BRD-K78918239	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCc1ccccc1	CID:54649366	phase I
BRD-K31829694	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NCc1ccc2OCOc2c1	CID:54649367	phase I
BRD-K77596469	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NCc1ccc2OCOc2c1	CID:54649368	phase I
BRD-K37434447	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCOCC1	CID:54649369	phase I
BRD-K70469022	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCOCC1	CID:54649370	phase I
BRD-K33013391	C\C=C\c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCc1ccccn1	CID:54649371	phase I
BRD-K83675132	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1	CID:54649372	phase I
BRD-K61431779	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1	CID:54649373	phase I
BRD-K54410116	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1	CID:54649374	phase I
BRD-K70179603	CCCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1ccc(F)cc1)[S@@](=O)C(C)(C)C	CID:54649375	phase I
BRD-K93210686	CCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1ccc(F)cc1)[S@](=O)C(C)(C)C	CID:54649376	phase I
BRD-K71795383	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)N1CCCCC1	CID:54649377	phase I
BRD-K19106401	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)N1CCCCC1	CID:54649378	phase I
BRD-K78097639	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NCCc1ccncc1	CID:54649379	phase I
BRD-K04759195	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NCCc1ccncc1	CID:54649380	phase I
BRD-K50799972	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCc1ccncc1	CID:54649381	phase I
BRD-K32310489	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NCc1ccncc1	CID:54649382	phase I
BRD-K20834925	COc1ccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(c2)-c2cccc(c2)C#N)[S@@](=O)C(C)(C)C)cc1	CID:54649383	phase I
BRD-K95666496	COc1ccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(c2)-c2cccc(c2)C#N)[S@](=O)C(C)(C)C)cc1	CID:54649384	phase I
BRD-K36928794	COc1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NCC(F)(F)F	CID:54649385	phase I
BRD-K60242118	COc1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCC(F)(F)F	CID:54649386	phase I
BRD-K40521754	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCN(C)CC1	CID:54649387	phase I
BRD-K85650383	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCN(C)CC1	CID:54649388	phase I
BRD-K36835942	COc1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649389	phase I
BRD-K88306467	COc1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649390	phase I
BRD-K92014112	CCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@@](=O)C(C)(C)C	CID:54649391	phase I
BRD-K92685052	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(F)cc1)C(=O)N1CCCCC1	CID:54649392	phase I
BRD-K44235509	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(F)cc1)C(=O)N1CCCCC1	CID:54649393	phase I
BRD-K57206606	C\C=C\c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCc1ccncc1	CID:54649394	phase I
BRD-K16778485	CCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(c1)C(=O)N(C)C)[S@@](=O)C(C)(C)C	CID:54649395	phase I
BRD-K01568615	CCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(c1)C(=O)N(C)C)[S@](=O)C(C)(C)C	CID:54649396	phase I
BRD-K60391168	COCCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(F)c1)[S@@](=O)C(C)(C)C	CID:54649397	phase I
BRD-K50194167	COCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(F)c1)[S@](=O)C(C)(C)C	CID:54649398	phase I
BRD-K36313546	COc1cccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(c2)-c2ccncc2)[S@](=O)C(C)(C)C)c1	CID:54649399	phase I
BRD-K74094800	COc1cccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(c2)-c2ccncc2)[S@@](=O)C(C)(C)C)c1	CID:54649400	phase I
BRD-K55808012	CN(C)C(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@](=O)C(C)(C)C	CID:54649401	phase I
BRD-K68849294	CN(C)C(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCC1)[S@@](=O)C(C)(C)C	CID:54649402	phase I
BRD-K67236950	CCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(OC)c1)[S@@](=O)C(C)(C)C	CID:54649403	phase I
BRD-K41721791	CCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(OC)c1)[S@](=O)C(C)(C)C	CID:54649404	phase I
BRD-K76439996	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCc1ccncc1	CID:54649405	phase I
BRD-K60558875	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCc1ccncc1	CID:54649406	phase I
BRD-K87182158	CN1CCN(CC1)C(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1ccccc1F)[S@](=O)C(C)(C)C	CID:54649407	phase I
BRD-K85426712	CN1CCN(CC1)C(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1ccccc1F)[S@@](=O)C(C)(C)C	CID:54649408	phase I
BRD-K39507473	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)N1CCOCC1	CID:54649409	phase I
BRD-K37405154	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)N1CCOCC1	CID:54649410	phase I
BRD-K54432046	CCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(F)c1)[S@](=O)C(C)(C)C	CID:54649411	phase I
BRD-K93112400	CCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(F)c1)[S@@](=O)C(C)(C)C	CID:54649412	phase I
BRD-K85134515	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCc1ccccc1F	CID:54649413	phase I
BRD-K25379780	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCc1ccccc1F	CID:54649414	phase I
BRD-K36656125	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCCCC1	CID:54649415	phase I
BRD-K02159117	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCCCC1	CID:54649416	phase I
BRD-K05356589	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)N1CCc2ccccc2C1	CID:54649417	phase I
BRD-K86326967	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)N1CCc2ccccc2C1	CID:54649418	phase I
BRD-K50576452	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCOCC1	CID:54649419	phase I
BRD-K43519318	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCOCC1	CID:54649420	phase I
BRD-K68085828	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NC1CCC1	CID:54649421	phase I
BRD-K21107294	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NC1CCC1	CID:54649422	phase I
BRD-K97554220	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649423	phase I
BRD-K65862059	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649424	phase I
BRD-K19167425	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)N1CCCCC1	CID:54649425	phase I
BRD-K61051532	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccccc1F)C(=O)N1CCCCC1	CID:54649426	phase I
BRD-K63809549	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCc1ccc2OCOc2c1	CID:54649427	phase I
BRD-K88937432	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCc1ccc2OCOc2c1	CID:54649428	phase I
BRD-K04753511	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cncnc1)C(=O)N1CCc2ccccc2C1	CID:54649429	phase I
BRD-K11068374	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cncnc1)C(=O)N1CCc2ccccc2C1	CID:54649430	phase I
BRD-K99913693	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCN(C)CC1	CID:54649431	phase I
BRD-K68796015	COc1ccccc1-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCN(C)CC1	CID:54649432	phase I
BRD-K74951051	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NCc1ccccc1F	CID:54649433	phase I
BRD-K36721554	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NCc1ccccc1F	CID:54649434	phase I
BRD-K29736077	CCCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(OC)c1)[S@@](=O)C(C)(C)C	CID:54649435	phase I
BRD-K34160774	CCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(OC)c1)[S@](=O)C(C)(C)C	CID:54649436	phase I
BRD-K71401720	COc1cccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(\C=C\C)c2)[S@@](=O)C(C)(C)C)c1	CID:54649437	phase I
BRD-K28305693	COc1cccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(\C=C\C)c2)[S@](=O)C(C)(C)C)c1	CID:54649438	phase I
BRD-K71631401	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCCc1ccncc1	CID:54649439	phase I
BRD-K06370852	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccncc1)C(=O)NCCc1ccncc1	CID:54649440	phase I
BRD-K00449983	C\C=C\c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NCc1ccccc1	CID:54649441	phase I
BRD-K00541818	C\C=C\c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCc1ccccc1	CID:54649442	phase I
BRD-K97473407	COc1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649443	phase I
BRD-K42654448	COc1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N(C)C	CID:54649444	phase I
BRD-K49441594	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCCN1CCCC1	CID:54649445	phase I
BRD-K54805796	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCCN1CCCC1	CID:54649446	phase I
BRD-K73837493	CCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(F)c1)[S@](=O)C(C)(C)C	CID:54649447	phase I
BRD-K80881992	CCCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)-c1cccc(F)c1)[S@@](=O)C(C)(C)C	CID:54649448	phase I
BRD-K70435062	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)N1CCN(C)CC1	CID:54649449	phase I
BRD-K66521855	CN(C)C(=O)c1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)N1CCN(C)CC1	CID:54649450	phase I
BRD-K29547084	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)N1CCCCC1	CID:54649451	phase I
BRD-K20099363	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)N1CCCCC1	CID:54649452	phase I
BRD-K63521663	COc1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NCC(F)(F)F	CID:54649453	phase I
BRD-K78133682	COc1cccc(c1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCC(F)(F)F	CID:54649454	phase I
BRD-K55194575	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NCc1ccccc1	CID:54649455	phase I
BRD-K92773691	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NCc1ccccc1	CID:54649456	phase I
BRD-K56583519	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCc1ccncc1	CID:54649457	phase I
BRD-K45114520	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCc1ccncc1	CID:54649458	phase I
BRD-K62917576	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccccc1)C(=O)NCc1ccc2OCOc2c1	CID:54649459	phase I
BRD-K31103241	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCCc1ccncc1	CID:54649460	phase I
BRD-K70074151	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCCc1ccncc1	CID:54649461	phase I
BRD-K36741877	COc1ccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(c2)-c2ccc(cc2)C#N)[S@@](=O)C(C)(C)C)cc1	CID:54649462	phase I
BRD-K64034190	COc1ccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(c2)-c2ccc(cc2)C#N)[S@](=O)C(C)(C)C)cc1	CID:54649463	phase I
BRD-K46343228	COc1cccc(CNC(=O)c2cc3CN([C@@H](CCO)c3c(n2)-c2cccc(c2)-c2cccc(c2)C#N)[S@@](=O)C(C)(C)C)c1	CID:54649464	phase I
BRD-K51361049	COc1cccc(CNC(=O)c2cc3CN([C@H](CCO)c3c(n2)-c2cccc(c2)-c2cccc(c2)C#N)[S@](=O)C(C)(C)C)c1	CID:54649465	phase I
BRD-K72382350	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NC1CCCCC1	CID:54649466	phase I
BRD-K89606138	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NC1CCCCC1	CID:54649467	phase I
BRD-K26277326	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@@H](CCO)c12)[S@@](=O)C(C)(C)C)C(=O)NC1CCCC1	CID:54649468	phase I
BRD-K71552321	CN(C)C(=O)c1ccc(cc1)-c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)[S@](=O)C(C)(C)C)C(=O)NC1CCCC1	CID:54649469	phase I
BRD-K81156227	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCCN1CCCC1	CID:54649470	phase I
BRD-K13299110	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccc(c1)C#N)C(=O)NCCN1CCCC1	CID:54649471	phase I
BRD-K79657514	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCCN1CCCCC1	CID:54649472	phase I
BRD-K37299375	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1ccc(cc1)C#N)C(=O)NCCN1CCCCC1	CID:54649473	phase I
BRD-K42595694	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649474	phase I
BRD-K72282141	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649475	phase I
BRD-K33620583	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649476	phase I
BRD-K95919017	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649477	phase I
BRD-K18982118	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649478	phase I
BRD-K89676402	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649479	phase I
BRD-K11238413	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649480	phase I
BRD-K38186418	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649481	phase I
BRD-K13118793	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649482	phase I
BRD-K43460092	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649483	phase I
BRD-K59015387	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649484	phase I
BRD-K84238725	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649485	phase I
BRD-K78386932	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649486	phase I
BRD-K31262969	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649487	phase I
BRD-K98471960	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649488	phase I
BRD-K53674232	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649489	phase I
BRD-K81527737	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649490	phase I
BRD-K15935695	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649491	phase I
BRD-K29054201	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649492	phase I
BRD-K75179331	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649493	phase I
BRD-K18925740	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649494	phase I
BRD-K88899439	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649495	phase I
BRD-K81438250	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649496	phase I
BRD-K89222451	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649497	phase I
BRD-K40073746	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)OC	CID:54649498	phase I
BRD-K19969523	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649499	phase I
BRD-K86535717	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649500	phase I
BRD-K52971552	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649501	phase I
BRD-K65373229	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649502	phase I
BRD-K07796595	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649503	phase I
BRD-K69174517	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649504	phase I
BRD-K45409613	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)OC	CID:54649505	phase I
BRD-K17507122	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649506	phase I
BRD-K42704273	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649507	phase I
BRD-K96551169	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649508	phase I
BRD-K96534186	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649509	phase I
BRD-K41763142	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649510	phase I
BRD-K02665621	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649511	phase I
BRD-K80841398	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649512	phase I
BRD-K03354784	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649513	phase I
BRD-K80976693	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649514	phase I
BRD-K87536251	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649515	phase I
BRD-K16331350	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649516	phase I
BRD-K04237106	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649517	phase I
BRD-K87167564	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649518	phase I
BRD-K54839171	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649519	phase I
BRD-K35571012	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)OC	CID:54649520	phase I
BRD-K07700224	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649521	phase I
BRD-K28513938	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649522	phase I
BRD-K51088127	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649523	phase I
BRD-K63607326	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649524	phase I
BRD-K98850601	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649525	phase I
BRD-K95631838	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649526	phase I
BRD-K11977286	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649527	phase I
BRD-K95367721	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649528	phase I
BRD-K71151012	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649529	phase I
BRD-K33591392	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649530	phase I
BRD-K70918484	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649531	phase I
BRD-K66857873	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649532	phase I
BRD-K96451524	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649533	phase I
BRD-K16813995	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649534	phase I
BRD-K72760455	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649535	phase I
BRD-K62320150	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)OC	CID:54649536	phase I
BRD-K35743871	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649537	phase I
BRD-K99307487	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649538	phase I
BRD-K69649444	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649539	phase I
BRD-K95779464	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649540	phase I
BRD-K86786416	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649541	phase I
BRD-K37014875	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649542	phase I
BRD-K99628932	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649543	phase I
BRD-K45850755	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649544	phase I
BRD-K45929778	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649545	phase I
BRD-K06935006	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649546	phase I
BRD-K52225919	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649547	phase I
BRD-K19011062	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649548	phase I
BRD-K36471847	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649549	phase I
BRD-K24106654	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649550	phase I
BRD-K31060354	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649551	phase I
BRD-K76243603	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649552	phase I
BRD-K05713002	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649553	phase I
BRD-K95275773	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649554	phase I
BRD-K07481948	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649555	phase I
BRD-K30214283	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649556	phase I
BRD-K77328005	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649557	phase I
BRD-K46597784	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649558	phase I
BRD-K28437309	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649559	phase I
BRD-K82005490	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649560	phase I
BRD-K68907515	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@@H]1O2)C#N	CID:54649561	phase I
BRD-K93602295	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@H]1O2)C#N	CID:54649562	phase I
BRD-K96006237	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@@H]1O2)C#N	CID:54649563	phase I
BRD-K93410778	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@H]1O2)C#N	CID:54649564	phase I
BRD-K22174526	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@H]1O2)C#N	CID:54649565	phase I
BRD-K79841204	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@H]1O2)C#N	CID:54649566	phase I
BRD-K40555995	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649567	phase I
BRD-K60879194	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649568	phase I
BRD-K07568447	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649569	phase I
BRD-K54636101	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649570	phase I
BRD-K87920375	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649571	phase I
BRD-K04206413	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649572	phase I
BRD-K36070105	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649573	phase I
BRD-K18102341	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649574	phase I
BRD-K27887926	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649575	phase I
BRD-K65065275	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649576	phase I
BRD-K13079805	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649577	phase I
BRD-K69073546	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649578	phase I
BRD-K73716473	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649579	phase I
BRD-K85297660	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649580	phase I
BRD-K07442049	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649581	phase I
BRD-K61484514	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649582	phase I
BRD-K81658138	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649583	phase I
BRD-K79333016	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649584	phase I
BRD-K60477597	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649585	phase I
BRD-K81940726	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649586	phase I
BRD-K60073229	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649587	phase I
BRD-K78420710	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649588	phase I
BRD-K60836534	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649589	phase I
BRD-K94217081	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649590	phase I
BRD-K65603160	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649591	phase I
BRD-K26873914	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649592	phase I
BRD-K70072942	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649593	phase I
BRD-K25923961	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649594	phase I
BRD-K45177540	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649595	phase I
BRD-K24734706	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649596	phase I
BRD-K75621129	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649597	phase I
BRD-K43781861	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649598	phase I
BRD-K25098415	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649599	phase I
BRD-K39284479	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649600	phase I
BRD-K13839830	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649601	phase I
BRD-K16421840	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649602	phase I
BRD-K50413145	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649605	phase I
BRD-K84233319	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649606	phase I
BRD-K74299234	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649607	phase I
BRD-K18979455	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649608	phase I
BRD-K85114251	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649609	phase I
BRD-K78719595	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649610	phase I
BRD-K15485967	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649611	phase I
BRD-K99856384	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649612	phase I
BRD-K74314059	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649613	phase I
BRD-K57441129	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649614	phase I
BRD-K43692189	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649615	phase I
BRD-K31575862	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649616	phase I
BRD-K67344967	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649617	phase I
BRD-K56826759	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649618	phase I
BRD-K15769121	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649619	phase I
BRD-K33868913	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649620	phase I
BRD-K16633334	CO[C@@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649621	phase I
BRD-K99546030	CO[C@@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649622	phase I
BRD-K41423946	CO[C@H]1CC[C@@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649623	phase I
BRD-K41915268	CO[C@H]1CC[C@H]2CCOc3c(cccc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649624	phase I
BRD-K72356321	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649625	phase I
BRD-K37280550	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649626	phase I
BRD-K10812716	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649627	phase I
BRD-K81897236	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649628	phase I
BRD-K35421408	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649629	phase I
BRD-K24671931	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649630	phase I
BRD-K01975855	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649631	phase I
BRD-K95457967	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649632	phase I
BRD-K66641352	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649633	phase I
BRD-K56339035	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649634	phase I
BRD-K88321606	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649635	phase I
BRD-K52463977	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649636	phase I
BRD-K38481376	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649637	phase I
BRD-K84015265	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649638	phase I
BRD-K31479060	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649639	phase I
BRD-K16244298	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649640	phase I
BRD-K23123734	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649641	phase I
BRD-K80761414	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649642	phase I
BRD-K25161864	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649643	phase I
BRD-K79937035	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649644	phase I
BRD-K40513181	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649645	phase I
BRD-K95125640	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649646	phase I
BRD-K36716113	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649647	phase I
BRD-K44925448	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649648	phase I
BRD-K30600059	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649649	phase I
BRD-K86452395	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649650	phase I
BRD-K93923246	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](OC)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649651	phase I
BRD-K26910201	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](OC)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649652	phase I
BRD-K05377469	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649653	phase I
BRD-K61974010	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649654	phase I
BRD-K07497357	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649655	phase I
BRD-K03163743	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649656	phase I
BRD-K53783288	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649657	phase I
BRD-K30111752	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649658	phase I
BRD-K89674009	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649659	phase I
BRD-K66226084	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649660	phase I
BRD-K49910674	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649661	phase I
BRD-K22907310	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649662	phase I
BRD-K98245381	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649663	phase I
BRD-K50876388	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649664	phase I
BRD-K43915000	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649665	phase I
BRD-K38748890	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649666	phase I
BRD-K80568112	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649667	phase I
BRD-K16605233	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649668	phase I
BRD-K99338550	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649669	phase I
BRD-K27843502	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649670	phase I
BRD-K21161559	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649671	phase I
BRD-K01208204	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649672	phase I
BRD-K23499378	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649673	phase I
BRD-K31589685	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649674	phase I
BRD-K87865520	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@@H]1O2)C#N	CID:54649675	phase I
BRD-K22135724	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649676	phase I
BRD-K73688688	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649677	phase I
BRD-K16539011	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)[C@@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649678	phase I
BRD-K06062006	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)[C@H](C)C(=O)N(C)C[C@H]1O2)C#N	CID:54649679	phase I
BRD-K59207957	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649680	phase I
BRD-K29609299	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649681	phase I
BRD-K02953825	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649682	phase I
BRD-K45237033	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649683	phase I
BRD-K48875630	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649684	phase I
BRD-K64976146	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649685	phase I
BRD-K30106607	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649686	phase I
BRD-K82585779	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649687	phase I
BRD-K70751829	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649688	phase I
BRD-K99953989	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649689	phase I
BRD-K13069055	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649690	phase I
BRD-K86813544	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649691	phase I
BRD-K62803063	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649692	phase I
BRD-K90239051	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649693	phase I
BRD-K35429561	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649694	phase I
BRD-K44258506	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649695	phase I
BRD-K78269577	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649696	phase I
BRD-K60203832	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649697	phase I
BRD-K10055064	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649698	phase I
BRD-K97086358	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649699	phase I
BRD-K47492310	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649700	phase I
BRD-K62714735	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649701	phase I
BRD-K43456220	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649702	phase I
BRD-K83567669	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649703	phase I
BRD-K30797133	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649704	phase I
BRD-K18454119	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649705	phase I
BRD-K57138551	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649706	phase I
BRD-K25329768	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649707	phase I
BRD-K87931030	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649708	phase I
BRD-K31921933	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)N(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649709	phase I
BRD-K38787519	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649710	phase I
BRD-K28641265	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649711	phase I
BRD-K66907139	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649712	phase I
BRD-K11392157	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649713	phase I
BRD-K67090914	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649714	phase I
BRD-K71155312	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649715	phase I
BRD-K15947051	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649716	phase I
BRD-K12313989	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649717	phase I
BRD-K61059900	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649718	phase I
BRD-K66115910	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649719	phase I
BRD-K60144139	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649720	phase I
BRD-K91648652	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649721	phase I
BRD-K12880737	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649722	phase I
BRD-K34695725	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649723	phase I
BRD-K03209844	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649724	phase I
BRD-K04321001	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649725	phase I
BRD-K68036990	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649726	phase I
BRD-K36090848	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649727	phase I
BRD-K04873321	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@@H]1O2)c1ccccc1)C#N	CID:54649728	phase I
BRD-K12441550	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649729	phase I
BRD-K18561719	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649730	phase I
BRD-K60170940	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649731	phase I
BRD-K54067509	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649732	phase I
BRD-K41731469	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)C[C@@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649733	phase I
BRD-K19390761	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)C[C@H](CC(=O)N(C)C[C@H]1O2)c1ccccc1)C#N	CID:54649734	phase I
BRD-K61676471	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649735	phase I
BRD-K53632480	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649736	phase I
BRD-K00046588	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649737	phase I
BRD-K36021765	CO[C@H]1CC[C@H]2CCN(C)C(=O)[C@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649738	phase I
BRD-K19203549	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649739	phase I
BRD-K82050323	CO[C@@H]1CC[C@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649740	phase I
BRD-K28329571	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649741	phase I
BRD-K29379469	CO[C@H]1CC[C@@H]2CCN(C)C(=O)[C@@H](C)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649742	phase I
BRD-K07928515	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649743	phase I
BRD-K94243450	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649744	phase I
BRD-K55446881	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649745	phase I
BRD-K66632266	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649746	phase I
BRD-K19302998	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649747	phase I
BRD-K12251642	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649748	phase I
BRD-K37252182	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649749	phase I
BRD-K36940835	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649750	phase I
BRD-K40735917	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649751	phase I
BRD-K60363992	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2)c1ccccc1	CID:54649752	phase I
BRD-K19981693	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649753	phase I
BRD-K97370549	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649754	phase I
BRD-K96093221	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649755	phase I
BRD-K24259871	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649756	phase I
BRD-K52106083	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649757	phase I
BRD-K87947740	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2)c1ccccc1	CID:54649758	phase I
BRD-K04006812	CO[C@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649759	phase I
BRD-K82815491	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649760	phase I
BRD-K50943704	CO[C@@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649761	phase I
BRD-K92269212	CO[C@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649762	phase I
BRD-K23453536	CO[C@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649763	phase I
BRD-K44480322	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649764	phase I
BRD-K82325043	CO[C@@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649765	phase I
BRD-K50435683	CO[C@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649766	phase I
BRD-K58087285	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649767	phase I
BRD-K33204746	CO[C@@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649768	phase I
BRD-K50462936	CO[C@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649769	phase I
BRD-K45495870	CO[C@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649770	phase I
BRD-K38265819	CO[C@@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649771	phase I
BRD-K48263651	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649772	phase I
BRD-K45888106	CO[C@H]1CC[C@@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649773	phase I
BRD-K89230185	CO[C@H]1CC[C@H]2CCN(C)C(=O)CCCN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649774	phase I
BRD-K15160697	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649775	phase I
BRD-K97729706	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649776	phase I
BRD-K57351233	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649777	phase I
BRD-K68365891	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649778	phase I
BRD-K71575663	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649779	phase I
BRD-K68743686	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649780	phase I
BRD-K54785440	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649781	phase I
BRD-K47593849	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N)c1ccccc1	CID:54649782	phase I
BRD-K99016279	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649783	phase I
BRD-K84879982	CO[C@@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649784	phase I
BRD-K95935686	CO[C@H]1CC[C@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649785	phase I
BRD-K16276539	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649786	phase I
BRD-K58941403	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649787	phase I
BRD-K59831227	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649788	phase I
BRD-K23220665	CO[C@H]1CC[C@@H]2CCN(C)C(=O)C[C@H](CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N)c1ccccc1	CID:54649789	phase I
BRD-K18554416	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)CC3(CCCCC3)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649790	phase I
BRD-K01071579	CO[C@H]1CC[C@H]2CCN(C)C(=O)CC3(CCCCC3)CN(C)C(=O)c3cc(ccc3OC[C@H]1O2)C#N	CID:54649791	phase I
BRD-K79324911	CO[C@H]1CC[C@@H]2CCN(C)C(=O)CC3(CCCCC3)CN(C)C(=O)c3cc(ccc3OC[C@@H]1O2)C#N	CID:54649792	phase I
BRD-K68408385	CO[C@@H]1CC[C@@H]2CCN(C)C(=O)CC3(CCCCC3)CN(C)C(=O)c3cccc(C#N)c3OC[C@@H]1O2	CID:54649793	phase I
BRD-K61866431	CO[C@H]1CC[C@@H]2CCN(C)C(=O)CC3(CCCCC3)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649794	phase I
BRD-K52764062	CO[C@H]1CC[C@H]2CCN(C)C(=O)CC3(CCCCC3)CN(C)C(=O)c3cccc(C#N)c3OC[C@H]1O2	CID:54649795	phase I
BRD-K70235890	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649796	phase I
BRD-K43653210	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649797	phase I
BRD-K47538257	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649798	phase I
BRD-K74132270	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@@H]1O2)C#N	CID:54649799	phase I
BRD-K73213708	CO[C@@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649800	phase I
BRD-K08817808	CO[C@@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649801	phase I
BRD-K20023110	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649802	phase I
BRD-K64922699	CO[C@H]1CC[C@@H]2CCOc3ccc(cc3C(=O)N(C)CCCC(=O)N(C)C[C@H]1O2)C#N	CID:54649803	phase I
BRD-K87554792	CO[C@H]1CC[C@H]2CCOc3ccc(cc3C(=O)N(C)CC3(CCCCC3)CC(=O)N(C)C[C@H]1O2)C#N	CID:54649804	phase I
BRD-K79529972	C[C@@H]1CCn2cc(COC[C@@H](NC1=O)c1ccccc1)nn2	CID:54649805	phase I
BRD-K01757377	C[C@@H]1CCn2cc(COC[C@H](NC1=O)c1ccccc1)nn2	CID:54649806	phase I
BRD-K70558234	O=C1CCCn2cc(COC[C@H](N1)c1ccccc1)nn2	CID:54649807	phase I
BRD-K41645779	O=C1CCCn2cc(COC[C@@H](N1)c1ccccc1)nn2	CID:54649808	phase I
BRD-K12873970	O=C1N[C@H](Cc2ccccc2)COCc2cn(CC[C@H]1Cc1ccccc1)nn2	CID:54649809	phase I
BRD-K61185334	O=C1N[C@@H](Cc2ccccc2)COCc2cn(CC[C@H]1Cc1ccccc1)nn2	CID:54649810	phase I
BRD-K10923439	O=C1N[C@@H](Cc2ccccc2)COCc2cn(CC[C@@H]1Cc1ccccc1)nn2	CID:54649811	phase I
BRD-K51670762	O=C1N[C@H](Cc2ccccc2)COCc2cn(CC[C@@H]1Cc1ccccc1)nn2	CID:54649812	phase I
BRD-K14992578	O=C1N[C@@H](COCc2cn(CC[C@@H]1Cc1ccccc1)nn2)c1ccccc1	CID:54649813	phase I
BRD-K77540020	O=C1N[C@H](COCc2cn(CC[C@@H]1Cc1ccccc1)nn2)c1ccccc1	CID:54649814	phase I
BRD-K10421834	O=C1N[C@@H](COCc2cn(CC[C@H]1Cc1ccccc1)nn2)c1ccccc1	CID:54649815	phase I
BRD-K47971885	COc1ccc(C[C@H]2CCn3cc(COC[C@H](Cc4ccccc4)NC2=O)nn3)cc1	CID:54649816	phase I
BRD-K31487236	COc1ccc(C[C@@H]2CCn3cc(COC[C@H](Cc4ccccc4)NC2=O)nn3)cc1	CID:54649817	phase I
BRD-K35789946	COc1ccc(C[C@@H]2CCc3cnnn3COC[C@H](Cc3ccccc3)NC2=O)cc1	CID:54649818	phase I
BRD-K23424219	COc1ccc(C[C@@H]2CCc3cnnn3COC[C@@H](Cc3ccccc3)NC2=O)cc1	CID:54649819	phase I
BRD-K55793776	COc1ccc(C[C@H]2CCc3cnnn3COC[C@H](Cc3ccccc3)NC2=O)cc1	CID:54649820	phase I
BRD-K82335556	COc1ccc(C[C@H]2CCc3cnnn3COC[C@@H](Cc3ccccc3)NC2=O)cc1	CID:54649821	phase I
BRD-K89219015	O=C1N[C@H](Cc2ccccc2)COCn2nncc2CC[C@H]1Cc1ccccc1	CID:54649822	phase I
BRD-K28187112	O=C1N[C@@H](Cc2ccccc2)COCn2nncc2CC[C@@H]1Cc1ccccc1	CID:54649823	phase I
BRD-K23886631	O=C1N[C@H](Cc2ccccc2)COCn2nncc2CC[C@@H]1Cc1ccccc1	CID:54649824	phase I
BRD-K99803997	COc1ccc(C[C@@H]2CCc3cnnn3COC[C@H](NC2=O)c2ccccc2)cc1	CID:54649825	phase I
BRD-K65568947	COc1ccc(C[C@@H]2CCc3cnnn3COC[C@@H](NC2=O)c2ccccc2)cc1	CID:54649826	phase I
BRD-K26016896	COc1ccc(C[C@H]2CCc3cnnn3COC[C@@H](NC2=O)c2ccccc2)cc1	CID:54649827	phase I
BRD-K83836941	Clc1ccc(C[C@@H]2CCn3cc(COC[C@@H](NC2=O)c2ccccc2)nn3)cc1	CID:54649828	phase I
BRD-K60064462	Clc1cccc(C[C@H]2CCn3cc(COC[C@H](NC2=O)c2ccccc2)nn3)c1	CID:54649829	phase I
BRD-K95422706	O=C1N[C@@H](COCn2nncc2CC[C@H]1Cc1ccccc1)c1ccccc1	CID:54649830	phase I
BRD-K86253182	O=C1N[C@H](COCn2nncc2CC[C@@H]1Cc1ccccc1)c1ccccc1	CID:54649831	phase I
BRD-K95901503	C[C@@H]1CCc2cnnn2COC[C@H](NC1=O)c1ccccc1	CID:54649832	phase I
BRD-K86629698	O=C1CCCc2cnnn2COC[C@H](N1)c1ccccc1	CID:54649833	phase I
BRD-K44320761	C[C@@H]1CCc2cnnn2COC[C@@H](Cc2ccccc2)NC1=O	CID:54649834	phase I
BRD-K27417269	COc1ccc(C[C@@H]2CCn3cc(COC[C@H](NC2=O)C(C)C)nn3)cc1	CID:54649835	phase I
BRD-K92202681	COc1ccc(C[C@H]2CCn3cc(COC[C@H](NC2=O)C(C)C)nn3)cc1	CID:54649836	phase I
BRD-K36517203	COc1ccc(C[C@H]2CCn3cc(COC[C@@H](NC2=O)C(C)C)nn3)cc1	CID:54649837	phase I
BRD-K43992612	COc1ccc(C[C@@H]2CCn3cc(COC[C@@H](NC2=O)C(C)C)nn3)cc1	CID:54649838	phase I
BRD-K28997108	CC(C)[C@@H]1COCc2cn(CC[C@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649839	phase I
BRD-K60024977	CC(C)[C@@H]1COCc2cn(CC[C@@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649840	phase I
BRD-K49525275	CC(C)[C@H]1COCc2cn(CC[C@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649841	phase I
BRD-K87592402	CC(C)[C@H]1COCc2cn(CC[C@@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649842	phase I
BRD-K29768655	CC(C)C[C@@H]1COCc2cn(CC[C@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649843	phase I
BRD-K38244121	CC(C)C[C@@H]1COCc2cn(CC[C@@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649844	phase I
BRD-K73515365	CC(C)C[C@H]1COCc2cn(CC[C@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649845	phase I
BRD-K14768034	CC(C)C[C@H]1COCc2cn(CC[C@@H](Cc3ccccc3)C(=O)N1)nn2	CID:54649846	phase I
BRD-K29660619	COc1ccc(C[C@H]2CCn3cc(COC[C@@H](CC(C)C)NC2=O)nn3)cc1	CID:54649847	phase I
BRD-K32401097	COc1ccc(C[C@@H]2CCn3cc(COC[C@@H](CC(C)C)NC2=O)nn3)cc1	CID:54649848	phase I
BRD-K46730958	COc1ccc(C[C@@H]2CCn3cc(COC[C@H](CC(C)C)NC2=O)nn3)cc1	CID:54649849	phase I
BRD-K46549154	COc1ccc(C[C@H]2CCn3cc(COC[C@H](CC(C)C)NC2=O)nn3)cc1	CID:54649850	phase I
BRD-K13674694	CC(C)C[C@@H]1COCc2cn(CC[C@H](C)C(=O)N1)nn2	CID:54649851	phase I
BRD-K81690566	CC(C)C[C@H]1COCc2cn(CC[C@H](C)C(=O)N1)nn2	CID:54649852	phase I
BRD-K64728664	CC(C)C[C@@H]1COCc2cn(CCCC(=O)N1)nn2	CID:54649853	phase I
BRD-A26583774	Clc1cccc(CC2COCc3cnnn3CCC(c3ccccc3)C(=O)N2)c1	CID:54649854	phase I
BRD-A92729194	Clc1ccc(CC2COCc3cnnn3CCC(c3ccccc3)C(=O)N2)cc1	CID:54649855	phase I
BRD-K66729666	COc1ccc(C[C@H]2CCc3cnnn3COC[C@H](CC(C)C)NC2=O)cc1	CID:54649856	phase I
BRD-K57308809	COc1ccc(C[C@@H]2CCc3cnnn3COC[C@H](CC(C)C)NC2=O)cc1	CID:54649857	phase I
BRD-K22248406	CC(C)C[C@H]1COCn2nncc2CC[C@H](Cc2ccccc2)C(=O)N1	CID:54649858	phase I
BRD-K64568504	CC(C)C[C@H]1COCn2nncc2CC[C@@H](Cc2ccccc2)C(=O)N1	CID:54649859	phase I
BRD-K95202918	CC(C)C[C@@H]1COCn2nncc2CCCC(=O)N1	CID:54649860	phase I
BRD-K24561725	CC(C)[C@@H]1COCn2nncc2CCCC(=O)N1	CID:54649861	phase I
BRD-K14350179	CC(C)[C@H]1COCn2nncc2CCCC(=O)N1	CID:54649862	phase I
BRD-K34462187	CC(C)[C@H]1COCn2nncc2CC[C@H](C)C(=O)N1	CID:54649863	phase I
BRD-K30719410	CC(C)C[C@H]1COCn2nncc2CC[C@H](C)C(=O)N1	CID:54649864	phase I
BRD-K98170574	COc1ccc(C[C@H]2CCc3cnnn3COC[C@@H](NC2=O)C(C)C)cc1	CID:54649865	phase I
BRD-K98384558	COc1ccc(C[C@@H]2CCc3cnnn3COC[C@@H](NC2=O)C(C)C)cc1	CID:54649866	phase I
BRD-K15259924	COc1ccc(C[C@H]2CCc3cnnn3COC[C@H](NC2=O)C(C)C)cc1	CID:54649867	phase I
BRD-K67693903	CC(C)[C@H]1COCn2nncc2CC[C@@H](Cc2ccccc2)C(=O)N1	CID:54649868	phase I
BRD-K18298066	CC(C)[C@@H]1COCn2nncc2CC[C@H](Cc2ccccc2)C(=O)N1	CID:54649869	phase I
BRD-A03684405	O=C1[C@H](Cc2ccccc2)CCn2cc(COCC3CCCN13)nn2	CID:54649870	phase I
BRD-A95489119	O=C1[C@@H](Cc2ccccc2)CCn2cc(COCC3CCCN13)nn2	CID:54649871	phase I
BRD-K16588281	COc1ccc(C[C@H]2CCn3cc(COC[C@@H](NC2=O)c2ccccc2)nn3)cc1	CID:54649872	phase I
BRD-K90136643	COc1ccc(C[C@@H]2CCn3cc(COC[C@H](NC2=O)c2ccccc2)nn3)cc1	CID:54649873	phase I
BRD-K66670355	C[C@@H]1CCn2cc(COC[C@@H](Cc3ccccc3)NC1=O)nn2	CID:54649874	phase I
BRD-K22229373	O=C1CCCc2cnnn2COC[C@H](Cc2ccccc2)N1	CID:54649875	phase I
BRD-K43326597	O=C1CCCn2cc(COC[C@@H](Cc3ccccc3)N1)nn2	CID:54649876	phase I
BRD-K42411085	O=C1CCCn2cc(COC[C@H](Cc3ccccc3)N1)nn2	CID:54649877	phase I
BRD-K22854278	CC(C)[C@H]1COCc2cn(CCCC(=O)N1)nn2	CID:54649878	phase I
BRD-K87081268	CC(C)[C@@H]1COCc2cn(CC[C@H](C)C(=O)N1)nn2	CID:54649879	phase I
BRD-K89304832	C\C=C\c1cccc(c1)-c1nc(cc2CN([C@H](CCO)c12)C(=O)NC(C)C)C(=O)Nc1nccs1	CID:54649880	phase I
BRD-K88449712	OCC[C@H]1N(Cc2cc(nc(c12)-c1cccc(c1)-c1ccc(F)cc1)C(=O)N1CCOCC1)C(=O)c1ccc2OCOc2c1	CID:54649881	phase I
BRD-K69330446	CCOC(=O)c1cc2CN([C@H](CCO)c2c(n1)-c1cccc(Br)c1)C(=O)NC(C)C	CID:54649882	phase I
BRD-K10775155	CCOC(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(Br)c1)C(=O)NC(C)C	CID:54649883	phase I
BRD-K05710256	CC(C)NC(=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NC1Cc2ccccc2C1	CID:54649884	phase I
BRD-K65006048	CC(C)NC(=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(c1)-c1cccnc1)C(=O)NC1Cc2ccccc2C1	CID:54649885	phase I
BRD-K72773830	CN(C)C(=O)c1cc2CN([C@@H](CCO)c2c(n1)-c1cccc(c1)C1=CCCCC1)S(C)(=O)=O	CID:54649886	phase I
BRD-K71424148	CC(C)(C)[S@](=O)N1Cc2cc(nc(c2[C@@H]1CCO)-c1cccc(Br)c1)C(=O)NC1CCCCC1	CID:54649887	phase I
BRD-K60861976	CC(C)(C)[S@@](=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(Br)c1)C(=O)NC1CCCCC1	CID:54649888	phase I
BRD-K47471281	CCC(=O)N1Cc2cc(nc(c2[C@H]1CCO)-c1cccc(c1)-c1cncnc1)C(=O)N(C)C	CID:54649889	phase I
BRD-K47234370	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)C1CCCC1)c1ccccc1	CID:54649892	phase I
BRD-K46446437	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)C1CCCC1)c1ccccc1	CID:54649893	phase I
BRD-K11401713	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)C1CCCC1)c1ccccc1	CID:54649894	phase I
BRD-K31000214	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)C1CCCC1)c1ccccc1	CID:54649895	phase I
BRD-K51800846	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)C1CCCC1)c1ccccc1	CID:54649896	phase I
BRD-K28530075	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)C1CCCC1)c1ccccc1	CID:54649897	phase I
BRD-K15600521	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N[C@@H]1C#N	CID:54649898	phase I
BRD-K08123737	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N[C@H]1C#N	CID:54649899	phase I
BRD-K54375254	COc1cccc(c1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N[C@@H]1C#N	CID:54649900	phase I
BRD-K57611352	CCc1cnc(s1)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649901	phase I
BRD-K79947616	CCc1cnc(s1)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649902	phase I
BRD-K82560670	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649903	phase I
BRD-K36078054	CCc1cnc(s1)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649904	phase I
BRD-K25018652	CCc1cnc(s1)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649905	phase I
BRD-K81956993	CCc1cnc(s1)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649906	phase I
BRD-K19833084	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649907	phase I
BRD-K77233343	CCc1cnc(s1)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CC(C)C	CID:54649908	phase I
BRD-K36232701	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)S(=O)(=O)c1cccc(F)c1	CID:54649909	phase I
BRD-K67514995	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)S(=O)(=O)c1cccc(F)c1	CID:54649910	phase I
BRD-K45371861	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)S(=O)(=O)c1cccc(F)c1	CID:54649911	phase I
BRD-K88684430	OC[C@H]1[C@@H]([C@@H](C#N)N1c1nc(cs1)-c1ccccc1)c1ccc(cc1)C1=CCCC1	CID:54649913	phase I
BRD-K29322455	OC[C@@H]1[C@H]([C@H](C#N)N1c1nc(cs1)-c1ccccc1)c1ccc(cc1)C1=CCCC1	CID:54649914	phase I
BRD-K18778674	OC[C@H]1[C@H]([C@H](C#N)N1c1nc(cs1)-c1ccccc1)c1ccc(cc1)C1=CCCC1	CID:54649915	phase I
BRD-K07107626	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)Cc2ccncc2)[C@@H]1C#N	CID:54649916	phase I
BRD-K37357652	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)Cc2ccncc2)[C@H]1C#N	CID:54649917	phase I
BRD-K68554461	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)Cc2ccncc2)[C@H]1C#N	CID:54649918	phase I
BRD-K45319854	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(=O)Cc2ccncc2)[C@@H]1C#N	CID:54649919	phase I
BRD-K64305210	CCS(=O)(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54649920	phase I
BRD-K03785392	CCS(=O)(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54649921	phase I
BRD-K05931533	CCS(=O)(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54649922	phase I
BRD-K89348354	CCS(=O)(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54649923	phase I
BRD-K89141537	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54649924	phase I
BRD-K41539131	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54649925	phase I
BRD-K64582453	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54649926	phase I
BRD-K16667431	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54649927	phase I
BRD-K43830653	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54649928	phase I
BRD-K71777270	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54649929	phase I
BRD-K07799833	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649930	phase I
BRD-K36065557	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649931	phase I
BRD-K36200934	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649932	phase I
BRD-K52981369	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649933	phase I
BRD-K09329774	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649934	phase I
BRD-K15108654	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649935	phase I
BRD-K43621195	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)c1cccnc1)c1ccc(cc1)C#Cc1ccccc1F	CID:54649936	phase I
BRD-K86838317	OC[C@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C1=CCCCC1	CID:54649937	phase I
BRD-K14974894	OC[C@@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)C1=CCCCC1	CID:54649938	phase I
BRD-K28884887	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)CN1CCOCC1	CID:54649939	phase I
BRD-K45033698	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)C(=O)CN1CCOCC1	CID:54649940	phase I
BRD-K41344641	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)CN1CCOCC1	CID:54649941	phase I
BRD-K63724542	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)CN1CCOCC1	CID:54649942	phase I
BRD-K66642908	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)CN1CCOCC1	CID:54649943	phase I
BRD-K44916273	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:54649944	phase I
BRD-K20827004	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:54649945	phase I
BRD-K36008374	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:54649946	phase I
BRD-K51993206	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:54649947	phase I
BRD-K65968843	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:54649948	phase I
BRD-K76005262	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:54649949	phase I
BRD-K99795671	CCc1csc(n1)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649950	phase I
BRD-K58307544	CCc1csc(n1)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649951	phase I
BRD-K14023438	CCc1csc(n1)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649952	phase I
BRD-K55749829	CCc1csc(n1)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649953	phase I
BRD-K30563708	CCc1csc(n1)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649954	phase I
BRD-K42886157	CCc1csc(n1)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649955	phase I
BRD-K60703528	CCc1csc(n1)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)\C=C\C	CID:54649956	phase I
BRD-K52403701	CCCNC(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649957	phase I
BRD-K02076218	CCCNC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649958	phase I
BRD-K81164606	CCCNC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649959	phase I
BRD-K78094112	CCCNC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649960	phase I
BRD-K00069117	CCCNC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649961	phase I
BRD-K50014464	CCCNC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649962	phase I
BRD-K88402291	CCCNC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649963	phase I
BRD-K52221985	CCCNC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1ccccc1F	CID:54649964	phase I
BRD-K68325500	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)Cc1ccccn1)c1ccc(cc1)C#CC1CC1	CID:54649965	phase I
BRD-K19194092	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)Cc1ccccn1)c1ccc(cc1)C#CC1CC1	CID:54649966	phase I
BRD-K00124439	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)Cc1ccccn1)c1ccc(cc1)C#CC1CC1	CID:54649967	phase I
BRD-K05273600	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)Cc1ccccn1)c1ccc(cc1)C#CC1CC1	CID:54649968	phase I
BRD-K62732905	Cc1nc(sc1C)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccccc1	CID:54649969	phase I
BRD-K15626512	Cc1nc(sc1C)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccccc1	CID:54649970	phase I
BRD-K80999199	Cc1nc(sc1C)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccccc1	CID:54649971	phase I
BRD-K73769216	OC[C@@H]1[C@@H]([C@@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649972	phase I
BRD-K69661816	OC[C@@H]1[C@@H]([C@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649973	phase I
BRD-K37197256	OC[C@H]1[C@@H]([C@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649974	phase I
BRD-K06589837	OC[C@@H]1[C@H]([C@@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649975	phase I
BRD-K13701195	OC[C@H]1[C@H]([C@@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649976	phase I
BRD-K60151881	OC[C@H]1[C@H]([C@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649977	phase I
BRD-K55854370	OC[C@@H]1[C@H]([C@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649978	phase I
BRD-K82014438	OC[C@H]1[C@@H]([C@@H](C#N)N1S(=O)(=O)Cc1ccccc1)c1ccccc1	CID:54649979	phase I
BRD-K30724479	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)NC1CCCCC1	CID:54649980	phase I
BRD-K16413530	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)NC1CCCCC1	CID:54649981	phase I
BRD-K67863009	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)NC1CCCCC1	CID:54649982	phase I
BRD-K96482472	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@H]1C#N)C(=O)NC1CCCCC1	CID:54649983	phase I
BRD-K35702939	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)NC1CCCCC1	CID:54649984	phase I
BRD-K39376673	OC[C@H]1N[C@H](C#N)[C@H]1c1ccc(\C=C\c2ccccc2)cc1	CID:54649985	phase I
BRD-K96098018	OC[C@H]1N[C@@H](C#N)[C@H]1c1ccc(\C=C\c2ccccc2)cc1	CID:54649986	phase I
BRD-K99344911	Cc1ccccc1S(=O)(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CC1CC1	CID:54649987	phase I
BRD-K68185250	Cc1ccccc1S(=O)(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CC1CC1	CID:54649988	phase I
BRD-K63301075	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@H]1C#N)C(=O)CN(C)C	CID:54649989	phase I
BRD-K37225211	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)CN(C)C	CID:54649990	phase I
BRD-K58660339	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)C(=O)CN(C)C	CID:54649991	phase I
BRD-K65481562	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)CN(C)C	CID:54649992	phase I
BRD-K58826089	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)CN(C)C	CID:54649993	phase I
BRD-K59605310	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)CN(C)C	CID:54649994	phase I
BRD-K64190282	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)C(=O)c1ccccn1	CID:54649995	phase I
BRD-K66084396	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)c1ccccn1	CID:54649996	phase I
BRD-K04588345	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)c1ccccn1	CID:54649997	phase I
BRD-K61082257	COc1cccc(c1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)c1ccccn1	CID:54649998	phase I
BRD-K32986110	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)c1ccccn1	CID:54649999	phase I
BRD-K13942440	COc1cccc(c1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)C(=O)c1ccccn1	CID:54650000	phase I
BRD-K93584503	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)Cc1ccccc1	CID:54650001	phase I
BRD-K64513711	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)Cc1ccccc1	CID:54650002	phase I
BRD-K21590495	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)Cc1ccccc1	CID:54650003	phase I
BRD-K41547297	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)Nc1ccccc1F)c1ccc(\C=C\c2ccccc2)cc1	CID:54650004	phase I
BRD-K45932120	OC[C@@H]1[C@@H]([C@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650005	phase I
BRD-K64326023	OC[C@@H]1[C@@H]([C@@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650006	phase I
BRD-K47407883	OC[C@@H]1[C@H]([C@@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650007	phase I
BRD-K26903971	OC[C@H]1[C@@H]([C@@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650008	phase I
BRD-K24776817	OC[C@H]1[C@H]([C@@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650009	phase I
BRD-K66729212	OC[C@@H]1[C@H]([C@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650010	phase I
BRD-K67236726	OC[C@H]1[C@@H]([C@H](C#N)N1S(=O)(=O)c1ccccc1)c1ccc(cc1)C1=CCCCC1	CID:54650011	phase I
BRD-K24062021	OC[C@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650012	phase I
BRD-K33217566	OC[C@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650013	phase I
BRD-K87304961	OC[C@@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650014	phase I
BRD-K37879473	OC[C@@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650015	phase I
BRD-K80044001	OC[C@H]1N[C@@H](C#N)[C@@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650016	phase I
BRD-K25362512	OC[C@@H]1N[C@@H](C#N)[C@@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650017	phase I
BRD-K99644669	OC[C@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)-c1cccc(F)c1	CID:54650018	phase I
BRD-K31220088	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650019	phase I
BRD-K05688054	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650020	phase I
BRD-K48593692	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650021	phase I
BRD-K01011412	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650022	phase I
BRD-K25006240	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650023	phase I
BRD-K80732408	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650024	phase I
BRD-K70470333	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650025	phase I
BRD-K26537262	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccc2OCOc2c1)c1ccccc1	CID:54650026	phase I
BRD-K28576143	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)C1CCOCC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:54650027	phase I
BRD-K35801592	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)C1CCOCC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:54650028	phase I
BRD-K49071649	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)C1CCOCC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:54650029	phase I
BRD-K95042038	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N[C@H]1C#N	CID:54650030	phase I
BRD-K30954716	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N[C@@H]1C#N	CID:54650031	phase I
BRD-K40123546	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N[C@H]1C#N	CID:54650032	phase I
BRD-K38385428	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N[C@@H]1C#N	CID:54650033	phase I
BRD-K50739913	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N[C@H]1C#N	CID:54650034	phase I
BRD-K29499344	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N[C@@H]1C#N	CID:54650035	phase I
BRD-K25300451	CCS(=O)(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650036	phase I
BRD-K97024014	CCS(=O)(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650037	phase I
BRD-K01570637	CCS(=O)(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650038	phase I
BRD-K12395425	CCS(=O)(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650039	phase I
BRD-K43580610	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N[C@@H]1C#N	CID:54650040	phase I
BRD-K15525634	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N[C@H]1C#N	CID:54650041	phase I
BRD-K37316675	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650042	phase I
BRD-K29746329	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650043	phase I
BRD-K37530005	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650044	phase I
BRD-K93896332	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650045	phase I
BRD-K93730701	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650046	phase I
BRD-K94655951	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650047	phase I
BRD-K21400342	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650048	phase I
BRD-K45151011	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)C1CCOCC1)c1ccc(cc1)C1=CCCC1	CID:54650049	phase I
BRD-K29611469	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)C1CCOCC1)c1ccc(cc1)C1=CCCC1	CID:54650050	phase I
BRD-K83473338	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)C1CCOCC1)c1ccc(cc1)C1=CCCC1	CID:54650051	phase I
BRD-K77943850	CN(C)CC(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#Cc1cccnc1	CID:54650052	phase I
BRD-K20725229	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650053	phase I
BRD-K99496840	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650054	phase I
BRD-K68735643	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650055	phase I
BRD-K28250273	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650056	phase I
BRD-K49689003	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650057	phase I
BRD-K07431800	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650058	phase I
BRD-K60132930	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)Nc1cccc(F)c1)c1ccccc1	CID:54650059	phase I
BRD-K28568387	CS(=O)(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(\C=C\c2ccccc2)cc1	CID:54650060	phase I
BRD-K42931788	COCC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1cccnc1	CID:54650061	phase I
BRD-K93054014	COCC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1cccnc1	CID:54650062	phase I
BRD-K90064059	COCC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1cccnc1	CID:54650063	phase I
BRD-K27586026	COCC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1cccnc1	CID:54650064	phase I
BRD-K71805031	COCC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1cccnc1	CID:54650065	phase I
BRD-K02694971	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650066	phase I
BRD-K71477834	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650067	phase I
BRD-K60784115	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650068	phase I
BRD-K99524324	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650069	phase I
BRD-K85630885	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650070	phase I
BRD-K69735552	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650071	phase I
BRD-K61362569	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650072	phase I
BRD-K97008061	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)c1ccccc1F)c1ccccc1	CID:54650073	phase I
BRD-K98866561	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650074	phase I
BRD-K90259550	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650075	phase I
BRD-K73843002	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650076	phase I
BRD-K08340668	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650077	phase I
BRD-K06541323	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650078	phase I
BRD-K67769696	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)C1CC1	CID:54650079	phase I
BRD-K07458582	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650080	phase I
BRD-K01594737	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)C1CC1	CID:54650081	phase I
BRD-K08831772	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54650082	phase I
BRD-K12216461	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54650083	phase I
BRD-K37957394	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54650084	phase I
BRD-K03130528	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54650085	phase I
BRD-K78655498	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54650086	phase I
BRD-K85632805	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)S(C)(=O)=O	CID:54650087	phase I
BRD-K50986888	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54650088	phase I
BRD-K39894071	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)S(C)(=O)=O	CID:54650089	phase I
BRD-K46088987	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C#Cc1ccc(F)cc1	CID:54650090	phase I
BRD-K77229182	CC(C)NC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650091	phase I
BRD-K04367289	CC(C)NC(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650092	phase I
BRD-K63898109	CC(C)NC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650093	phase I
BRD-K50791983	CC(C)NC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650094	phase I
BRD-K45295352	CC(C)NC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650095	phase I
BRD-K97910278	CC(C)NC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650096	phase I
BRD-K60993486	CC(C)NC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650097	phase I
BRD-K03969729	CC(C)NC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1ccc(F)cc1	CID:54650098	phase I
BRD-K04133968	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)Cc1ccccc1)c1ccc(cc1)-c1cncnc1	CID:54650099	phase I
BRD-K98367121	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)Cc1ccccc1)c1ccc(cc1)-c1cncnc1	CID:54650100	phase I
BRD-K54046891	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)Cc1ccccc1)c1ccc(cc1)-c1cncnc1	CID:54650101	phase I
BRD-K30628839	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)Cc1ccccc1)c1ccc(cc1)-c1cncnc1	CID:54650102	phase I
BRD-K06716139	COc1ccccc1NC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccccc1	CID:54650103	phase I
BRD-K80065513	COc1ccccc1NC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccccc1	CID:54650104	phase I
BRD-K43349989	COc1ccccc1NC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccccc1	CID:54650105	phase I
BRD-K96713754	COc1ccccc1NC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccccc1	CID:54650106	phase I
BRD-K16533918	COc1ccccc1NC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccccc1	CID:54650107	phase I
BRD-K37957530	COc1ccccc1NC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccccc1	CID:54650108	phase I
BRD-K64641861	COc1ccccc1NC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccccc1	CID:54650109	phase I
BRD-K13944250	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)C1CC1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54650110	phase I
BRD-K96741939	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)C1CC1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54650111	phase I
BRD-K52651393	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)C1CC1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54650112	phase I
BRD-K06663546	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)C1CC1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54650113	phase I
BRD-K85976669	COCC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650114	phase I
BRD-K03034193	COCC(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650115	phase I
BRD-K89860739	COCC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650116	phase I
BRD-K95526045	COCC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650117	phase I
BRD-K48030215	COCC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650118	phase I
BRD-K48492265	COCC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650119	phase I
BRD-K06202986	COCC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CCC1CCCC1	CID:54650120	phase I
BRD-K71166745	CCS(=O)(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#Cc1ccccc1F	CID:54650121	phase I
BRD-K81123598	CCS(=O)(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#Cc1ccccc1F	CID:54650122	phase I
BRD-K96935347	CCS(=O)(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#Cc1ccccc1F	CID:54650123	phase I
BRD-K80926963	CCS(=O)(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#Cc1ccccc1F	CID:54650124	phase I
BRD-K88334823	CCS(=O)(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#Cc1ccccc1F	CID:54650125	phase I
BRD-K33713995	OC[C@@H]1[C@@H]([C@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650126	phase I
BRD-K63030439	OC[C@@H]1[C@@H]([C@@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650127	phase I
BRD-K89079417	OC[C@H]1[C@@H]([C@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650128	phase I
BRD-K47029744	OC[C@H]1[C@H]([C@@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650129	phase I
BRD-K52682771	OC[C@H]1[C@@H]([C@@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650130	phase I
BRD-K66814954	OC[C@@H]1[C@H]([C@@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650131	phase I
BRD-K48598367	OC[C@@H]1[C@H]([C@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650132	phase I
BRD-K03258328	OC[C@H]1[C@H]([C@H](C#N)N1S(=O)(=O)c1ccc(F)cc1)c1ccccc1	CID:54650133	phase I
BRD-K31970894	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C1=CCCCC1	CID:54650134	phase I
BRD-K29181432	OC[C@@H]1[C@@H]([C@@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C1=CCCCC1	CID:54650135	phase I
BRD-K89961851	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C1=CCCCC1	CID:54650136	phase I
BRD-K18746324	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C1=CCCCC1	CID:54650137	phase I
BRD-K21109208	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C1=CCCCC1	CID:54650138	phase I
BRD-K97924168	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)Cc1ccncc1)c1ccc(cc1)C1=CCCCC1	CID:54650139	phase I
BRD-K71225733	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)CCN1CCCCC1)c1ccccc1	CID:54650140	phase I
BRD-K89895693	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)CCN1CCCCC1)c1ccccc1	CID:54650141	phase I
BRD-K62957477	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)CCN1CCCCC1)c1ccccc1	CID:54650142	phase I
BRD-K35224528	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)CCN1CCCCC1)c1ccccc1	CID:54650143	phase I
BRD-K02952507	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)c1cccc(F)c1	CID:54650144	phase I
BRD-K46766834	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)C(=O)c1cccc(F)c1	CID:54650145	phase I
BRD-K99481965	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)c1cccc(F)c1	CID:54650146	phase I
BRD-K43209476	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1C#N)C(=O)c1cccc(F)c1	CID:54650147	phase I
BRD-K46574442	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)c1cccc(F)c1	CID:54650148	phase I
BRD-K25866499	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)c1cccc(F)c1	CID:54650149	phase I
BRD-K69936629	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N([C@@H]1C#N)C(=O)c1cccc(F)c1	CID:54650150	phase I
BRD-K01608965	CCc1cnc(s1)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650151	phase I
BRD-K31427141	CCc1cnc(s1)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650152	phase I
BRD-K19914944	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650153	phase I
BRD-K63944563	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650154	phase I
BRD-K47977047	CCc1cnc(s1)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650155	phase I
BRD-K43194109	CCc1cnc(s1)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650156	phase I
BRD-K70399291	CCc1cnc(s1)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650157	phase I
BRD-K07004447	OC[C@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650158	phase I
BRD-K28035139	OC[C@@H]1N[C@@H](C#N)[C@@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650159	phase I
BRD-K29102147	OC[C@@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650160	phase I
BRD-K74656908	OC[C@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650161	phase I
BRD-K86961442	OC[C@@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650162	phase I
BRD-K74260000	OC[C@H]1N[C@@H](C#N)[C@@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650163	phase I
BRD-K37612077	OC[C@@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)C#CC1CCCCC1	CID:54650164	phase I
BRD-K53039836	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCC1	CID:54650165	phase I
BRD-K72972600	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCC1	CID:54650166	phase I
BRD-K58761147	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCC1	CID:54650167	phase I
BRD-K34382714	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCC1	CID:54650168	phase I
BRD-K42156657	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCC1	CID:54650169	phase I
BRD-K27005217	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1C#N)C(=O)c1cccnc1	CID:54650170	phase I
BRD-K17745445	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)c1cccnc1	CID:54650171	phase I
BRD-K94067270	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1C#N)C(=O)c1cccnc1	CID:54650172	phase I
BRD-K37461197	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1C#N)C(=O)c1cccnc1	CID:54650173	phase I
BRD-K88856990	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1C#N)C(=O)c1cccnc1	CID:54650174	phase I
BRD-K15464148	OC[C@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650175	phase I
BRD-K60539617	OC[C@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650176	phase I
BRD-K11309655	OC[C@@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650177	phase I
BRD-K53867540	OC[C@@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650178	phase I
BRD-K80648041	OC[C@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650179	phase I
BRD-K94781393	OC[C@@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650180	phase I
BRD-K96635690	OC[C@@H]1N[C@@H](C#N)[C@@H]1c1ccc(cc1)C#Cc1ccccc1F	CID:54650181	phase I
BRD-K76856691	CCCNC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650182	phase I
BRD-K26909795	CCCNC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650183	phase I
BRD-K52785744	CCCNC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650184	phase I
BRD-K19362120	CCCNC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650185	phase I
BRD-K48296029	CCCNC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650186	phase I
BRD-K80400482	CCCNC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650187	phase I
BRD-K46381939	CCCNC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650188	phase I
BRD-K86354270	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccnc1	CID:54650189	phase I
BRD-K46267071	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccnc1	CID:54650190	phase I
BRD-K19516543	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccnc1	CID:54650191	phase I
BRD-K02446652	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccnc1	CID:54650192	phase I
BRD-K69664985	CC(C)NC(=O)N1[C@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650193	phase I
BRD-K65506786	CC(C)NC(=O)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650194	phase I
BRD-K17135741	CC(C)NC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650195	phase I
BRD-K31126514	CC(C)NC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650196	phase I
BRD-K24272049	CC(C)NC(=O)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650197	phase I
BRD-K48864121	CC(C)NC(=O)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650198	phase I
BRD-K99999497	CC(C)NC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650199	phase I
BRD-K50314382	CC(C)NC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C#CC1CCCCC1	CID:54650200	phase I
BRD-K38622866	CCc1cnc(s1)N1[C@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650201	phase I
BRD-K90805324	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650202	phase I
BRD-K30934140	CCc1cnc(s1)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650203	phase I
BRD-K51895259	CCc1cnc(s1)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650204	phase I
BRD-K44410738	CCc1cnc(s1)N1[C@@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650205	phase I
BRD-K56379651	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650206	phase I
BRD-K76820571	CCc1cnc(s1)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)-c1cccc(F)c1	CID:54650207	phase I
BRD-K72354054	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:54650208	phase I
BRD-K24118943	OC[C@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C#Cc1cccnc1	CID:54650391	phase I
BRD-K35128023	OC[C@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)C#Cc1cccnc1	CID:54650392	phase I
BRD-K85580817	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650440	phase I
BRD-K95710843	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650441	phase I
BRD-K48019220	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650442	phase I
BRD-K90361987	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650443	phase I
BRD-K13005651	OC[C@H]1[C@@H]([C@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650444	phase I
BRD-K03496358	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650445	phase I
BRD-K51862446	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:54650446	phase I
BRD-K90469014	CCc1csc(n1)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCC1	CID:54650542	phase I
BRD-K06896230	CCc1csc(n1)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C1=CCCC1	CID:54650543	phase I
BRD-K02208014	OC[C@@H]1[C@H]([C@H](C#N)N1C(=O)C1CCC1)c1ccc(cc1)-c1cccnc1	CID:54650751	phase I
BRD-K86372560	OC[C@H]1[C@H]([C@H](C#N)N1C(=O)NC1CCCCC1)c1ccc(cc1)C1=CCCCC1	CID:54650953	phase I
BRD-K78847404	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)NC1CCCCC1)c1ccc(cc1)C1=CCCCC1	CID:54650957	phase I
BRD-K82364958	OC[C@H]1N[C@@H](C#N)[C@@H]1c1ccc(cc1)C1=CCCC1	CID:54650960	phase I
BRD-K23429973	OC[C@@H]1N[C@@H](C#N)[C@H]1c1ccc(cc1)C1=CCCC1	CID:54650962	phase I
BRD-K81605832	OC[C@@H]1N[C@H](C#N)[C@H]1c1ccc(cc1)C1=CCCC1	CID:54650963	phase I
BRD-K08805764	OC[C@H]1N[C@H](C#N)[C@@H]1c1ccc(cc1)C1=CCCC1	CID:54650964	phase I
BRD-K63305270	COCC(=O)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54650998	phase I
BRD-K21652416	COCC(=O)N1[C@H](CO)[C@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54651000	phase I
BRD-K37145632	COCC(=O)N1[C@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54651001	phase I
BRD-K15358569	COCC(=O)N1[C@@H](CO)[C@@H]([C@H]1C#N)c1ccc(cc1)C1=CCCCC1	CID:54651002	phase I
BRD-K83720640	OC[C@@H]1[C@@H]([C@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCCC1	CID:54651043	phase I
BRD-K62841356	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)c1ccccn1)c1ccc(cc1)C1=CCCCC1	CID:54651044	phase I
BRD-K07536006	CCc1cnc(s1)N1[C@@H](CO)[C@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCC1	CID:54651052	phase I
BRD-K30013099	CCc1cnc(s1)N1[C@@H](CO)[C@@H]([C@@H]1C#N)c1ccc(cc1)C1=CCCC1	CID:54651053	phase I
BRD-K62472719	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:54651064	phase I
BRD-K05885800	CCc1csc(n1)N1[C@@H](CO)[C@@H]([C@@H]1CNC(C)C)c1ccc(cc1)\C=C\C	CID:54651171	phase I
BRD-K17530818	CCc1csc(n1)N1[C@H](CO)[C@@H]([C@@H]1CNC(C)C)c1ccc(cc1)\C=C\C	CID:54651172	phase I
BRD-K43683841	CCc1csc(n1)N1[C@H](CO)[C@H]([C@H]1CNC(C)C)c1ccc(cc1)\C=C\C	CID:54651173	phase I
BRD-K39561037	OC[C@@H]1N(Cc2ccccn2)[C@H](CN(C)S(C)(=O)=O)[C@H]1c1ccccc1	CID:54651174	phase I
BRD-K86449639	OC[C@@H]1N(Cc2ccccn2)[C@H](CN(C)S(C)(=O)=O)[C@@H]1c1ccccc1	CID:54651175	phase I
BRD-K96747266	OC[C@@H]1N(Cc2ccccn2)[C@@H](CN(C)S(C)(=O)=O)[C@@H]1c1ccccc1	CID:54651176	phase I
BRD-K60850440	OC[C@H]1N(Cc2ccccn2)[C@H](CN(C)S(C)(=O)=O)[C@@H]1c1ccccc1	CID:54651177	phase I
BRD-K55288106	OC[C@H]1N(Cc2ccccn2)[C@@H](CN(C)S(C)(=O)=O)[C@H]1c1ccccc1	CID:54651178	phase I
BRD-K91652715	OC[C@@H]1N(Cc2ccccn2)[C@@H](CN(C)S(C)(=O)=O)[C@H]1c1ccccc1	CID:54651179	phase I
BRD-K76252019	OC[C@H]1N(Cc2ccccn2)[C@H](CN(C)S(C)(=O)=O)[C@H]1c1ccccc1	CID:54651180	phase I
BRD-K93594354	OC[C@H]1N(Cc2ccccn2)[C@@H](CN(C)S(C)(=O)=O)[C@@H]1c1ccccc1	CID:54651181	phase I
BRD-K22416922	OC[C@@H]1N[C@@H](CNC(=O)c2ccccc2F)[C@@H]1c1ccccc1	CID:54651182	phase I
BRD-K80724940	OC[C@H]1N[C@H](CNC(=O)c2ccccc2F)[C@H]1c1ccccc1	CID:54651183	phase I
BRD-K29373549	OC[C@@H]1N[C@@H](CNC(=O)c2ccccc2F)[C@H]1c1ccccc1	CID:54651184	phase I
BRD-K40813780	OC[C@H]1N[C@H](CNC(=O)c2ccccc2F)[C@@H]1c1ccccc1	CID:54651185	phase I
BRD-K58642524	CCN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)CC)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651186	phase I
BRD-K93996655	CCN(C[C@H]1[C@@H]([C@H](CO)N1C(=O)CC)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651187	phase I
BRD-K92824836	CCN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)CC)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651188	phase I
BRD-K30649361	CCN(C[C@@H]1[C@H]([C@@H](CO)N1C(=O)CC)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651189	phase I
BRD-K98968761	CCN(C[C@H]1[C@H]([C@@H](CO)N1C(=O)CC)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651190	phase I
BRD-K39014631	COCC(=O)N(C)C[C@H]1[C@@H]([C@H](CO)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651195	phase I
BRD-K44878051	COCC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651196	phase I
BRD-K52874783	COCC(=O)N(C)C[C@H]1[C@@H]([C@@H](CO)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651197	phase I
BRD-K15262863	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(CC2CC2)[C@@H]1CNS(C)(=O)=O	CID:54651198	phase I
BRD-K16026816	CCNC[C@@H]1[C@@H]([C@H](CO)N1S(C)(=O)=O)c1ccc(cc1)-c1ccc(F)cc1	CID:54651199	phase I
BRD-K30296979	CN(C[C@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1ccc(F)cc1)C(=O)C1CCC1	CID:54651200	phase I
BRD-K23410901	CC(C)CN(C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651201	phase I
BRD-K47597660	CC(C)CN(C[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651202	phase I
BRD-K78714545	CC(C)CN(C[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651203	phase I
BRD-K50302985	CC(C)CN(C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651204	phase I
BRD-K75048204	CC(C)CN(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651205	phase I
BRD-K20097363	CC(C)CN(C[C@@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651206	phase I
BRD-K99265073	CC(C)CN(C[C@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccccn1	CID:54651207	phase I
BRD-K54445308	CC(C)N(C[C@@H]1N[C@@H](CO)[C@H]1c1ccccc1)C(=O)CN1CCOCC1	CID:54651208	phase I
BRD-K63455741	CC(C)N(C[C@H]1N[C@H](CO)[C@@H]1c1ccccc1)C(=O)CN1CCOCC1	CID:54651209	phase I
BRD-K28073457	OC[C@@H]1[C@H]([C@@H](CNC(=O)c2ccccn2)N1Cc1cccnc1)c1ccccc1	CID:54651210	phase I
BRD-K78717223	OC[C@@H]1[C@H]([C@H](CNC(=O)c2ccccn2)N1Cc1cccnc1)c1ccccc1	CID:54651211	phase I
BRD-K30936057	OC[C@H]1[C@@H]([C@@H](CNC(=O)c2ccccn2)N1Cc1cccnc1)c1ccccc1	CID:54651212	phase I
BRD-K75264577	OC[C@H]1[C@H]([C@H](CNC(=O)c2ccccn2)N1Cc1cccnc1)c1ccccc1	CID:54651213	phase I
BRD-K48914099	OC[C@H]1[C@@H]([C@H](CNC(=O)c2ccccn2)N1Cc1cccnc1)c1ccccc1	CID:54651214	phase I
BRD-K90424352	OC[C@@H]1[C@@H]([C@@H](CNC(=O)c2ccccn2)N1Cc1cccnc1)c1ccccc1	CID:54651215	phase I
BRD-K83727172	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N[C@H]1CNS(=O)(=O)c1ccccc1	CID:54651216	phase I
BRD-K38596298	CCCNC(=O)N1[C@@H](CO)[C@H]([C@H]1CNC(=O)c1ccc(F)cc1)c1ccccc1	CID:54651217	phase I
BRD-K75636693	CCCNC(=O)N1[C@@H](CO)[C@@H]([C@H]1CNC(=O)c1ccc(F)cc1)c1ccccc1	CID:54651218	phase I
BRD-K29812154	CCN(C[C@@H]1[C@H]([C@@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)C1CC1	CID:54651219	phase I
BRD-K32354807	CCN(C[C@H]1[C@@H]([C@@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)C1CC1	CID:54651220	phase I
BRD-K90705468	CCN(C[C@@H]1[C@H]([C@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)C1CC1	CID:54651221	phase I
BRD-K62436804	COCCN(C[C@@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(C)=O	CID:54651222	phase I
BRD-K40496631	COCCN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(C)=O	CID:54651223	phase I
BRD-K20079620	COCCN(C[C@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(C)=O	CID:54651224	phase I
BRD-K13012097	COCCN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(C)=O	CID:54651225	phase I
BRD-K76896099	CCN(C[C@@H]1N[C@H](CO)[C@H]1c1ccccc1)C(=O)c1ccncc1	CID:54651226	phase I
BRD-K73642355	CCN(C[C@@H]1N[C@@H](CO)[C@H]1c1ccccc1)C(=O)c1ccncc1	CID:54651227	phase I
BRD-K32516224	CCN(C[C@H]1N[C@H](CO)[C@H]1c1ccccc1)C(=O)c1ccncc1	CID:54651228	phase I
BRD-K21622447	CCN(C[C@H]1N[C@@H](CO)[C@@H]1c1ccccc1)C(=O)c1ccncc1	CID:54651229	phase I
BRD-K81921806	CCN(C[C@@H]1N[C@@H](CO)[C@@H]1c1ccccc1)C(=O)c1ccncc1	CID:54651230	phase I
BRD-K37879871	CCN(C[C@H]1N[C@H](CO)[C@@H]1c1ccccc1)C(=O)c1ccncc1	CID:54651231	phase I
BRD-K03808778	CCNC[C@H]1[C@H]([C@@H](CO)N1C(=O)Cc1ccccn1)c1ccccc1	CID:54651232	phase I
BRD-K26952068	CCNC[C@@H]1[C@@H]([C@H](CO)N1C(=O)Cc1ccccn1)c1ccccc1	CID:54651233	phase I
BRD-K13036885	CCNC[C@@H]1[C@H]([C@@H](CO)N1C(=O)Cc1ccccn1)c1ccccc1	CID:54651234	phase I
BRD-K25989007	CC(C)NC(=O)N1[C@@H](CO)[C@@H]([C@H]1CN(C)C(=O)c1ccccc1)c1ccccc1	CID:54651235	phase I
BRD-K22127625	CCC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1F	CID:54651236	phase I
BRD-K11095531	CCC(=O)N(C)C[C@@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1F	CID:54651237	phase I
BRD-K94516855	CCC(=O)N(C)C[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1F	CID:54651238	phase I
BRD-K57337567	CCC(=O)N(C)C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1F	CID:54651239	phase I
BRD-K92038420	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N([C@@H]1CNC(=O)NC(C)C)C(=O)C1CC1	CID:54651240	phase I
BRD-K39151515	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1CNC(=O)NC(C)C)C(=O)C1CC1	CID:54651241	phase I
BRD-K69894866	CN(C[C@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)C1=CCCC1)C(=O)c1ccccn1	CID:54651242	phase I
BRD-K59261663	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N[C@H]1CN(C(C)C)C(=O)c1ccccc1F	CID:54651243	phase I
BRD-K52413350	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N[C@@H]1CN(C(C)C)C(=O)c1ccccc1F	CID:54651244	phase I
BRD-K32550888	CCN(C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651245	phase I
BRD-K01604352	CCN(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651246	phase I
BRD-K80579245	CCN(C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651247	phase I
BRD-K80991460	CCN(C[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651248	phase I
BRD-K40274786	COCC(=O)NC[C@@H]1[C@@H]([C@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651249	phase I
BRD-K21374126	COCC(=O)NC[C@@H]1[C@H]([C@@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651250	phase I
BRD-K11719436	COCC(=O)NC[C@@H]1[C@@H]([C@@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651251	phase I
BRD-K94064112	COCC(=O)NC[C@H]1[C@H]([C@@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651252	phase I
BRD-K12227848	COCC(=O)NC[C@H]1[C@@H]([C@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651253	phase I
BRD-K51733045	COCC(=O)NC[C@@H]1[C@H]([C@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651254	phase I
BRD-K58985339	COCC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651255	phase I
BRD-K73679670	CCN(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)-c1cccc(F)c1)C(=O)CN(C)C	CID:54651256	phase I
BRD-K22496535	CCN(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1cccc(F)c1)C(=O)CN(C)C	CID:54651257	phase I
BRD-K48001367	CCC(=O)N1[C@@H](CO)[C@@H]([C@H]1CNC(=O)c1ccncc1)c1ccc(cc1)\C=C\C	CID:54651258	phase I
BRD-K56040287	CCC(=O)N1[C@@H](CO)[C@H]([C@H]1CNC(=O)c1ccncc1)c1ccc(cc1)\C=C\C	CID:54651259	phase I
BRD-K70252286	CCN(C[C@@H]1[C@H]([C@@H](CO)N1CC1CC1)c1ccc(cc1)C1=CCCCC1)C(C)=O	CID:54651260	phase I
BRD-K47686314	CCN(C[C@H]1[C@@H]([C@H](CO)N1CC1CC1)c1ccc(cc1)C1=CCCCC1)C(C)=O	CID:54651261	phase I
BRD-K87562020	OC[C@H]1[C@H]([C@@H](CNC(=O)c2ccncc2)N1CC1CCCC1)c1ccccc1	CID:54651262	phase I
BRD-K20554239	OC[C@@H]1[C@@H]([C@@H](CNC(=O)c2ccncc2)N1CC1CCCC1)c1ccccc1	CID:54651263	phase I
BRD-K50893227	OC[C@@H]1[C@@H]([C@H](CNC(=O)c2ccncc2)N1CC1CCCC1)c1ccccc1	CID:54651264	phase I
BRD-K52921974	OC[C@H]1[C@H]([C@H](CNC(=O)c2ccncc2)N1CC1CCCC1)c1ccccc1	CID:54651265	phase I
BRD-K85862256	CCC(=O)N1[C@@H](CO)[C@@H]([C@@H]1CN(C)C(=O)CN1CCOCC1)c1ccccc1	CID:54651266	phase I
BRD-K01777999	CCC(=O)N1[C@H](CO)[C@H]([C@@H]1CN(C)C(=O)CN1CCOCC1)c1ccccc1	CID:54651267	phase I
BRD-K01912493	CCC(=O)N1[C@H](CO)[C@H]([C@H]1CN(C)C(=O)CN1CCOCC1)c1ccccc1	CID:54651268	phase I
BRD-K30644784	CCN(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)NC1CCCC1	CID:54651270	phase I
BRD-K82048228	CCN(C[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)NC1CCCC1	CID:54651271	phase I
BRD-K05928130	CCN(C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)NC1CCCC1	CID:54651272	phase I
BRD-K76415725	CC(C)N(C[C@H]1N[C@H](CO)[C@H]1c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651273	phase I
BRD-K17508599	CC(C)N(C[C@@H]1N[C@@H](CO)[C@@H]1c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651274	phase I
BRD-K21120783	CC(C)N(C[C@@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccc(F)cc1	CID:54651275	phase I
BRD-K99335646	CC(C)N(C[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccc(F)cc1	CID:54651276	phase I
BRD-K49907349	CC(C)N(C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccc(F)cc1	CID:54651277	phase I
BRD-K98065679	CC(C)N(C[C@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccc(F)cc1	CID:54651278	phase I
BRD-K49294047	CC(C)N(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1ccc(F)cc1	CID:54651279	phase I
BRD-K92277566	CN(C(C)=O)C[C@@H]1N(C(C)=O)[C@H](CO)[C@H]1c1ccc(cc1)-c1cccc(C#N)c1	CID:54651280	phase I
BRD-K37140349	CN(C(C)=O)C[C@H]1N(C(C)=O)[C@@H](CO)[C@@H]1c1ccc(cc1)-c1cccc(C#N)c1	CID:54651281	phase I
BRD-K36353158	CCN(C[C@@H]1[C@@H]([C@@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651282	phase I
BRD-K27539817	CCN(C[C@H]1[C@@H]([C@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651283	phase I
BRD-K88942732	CCN(C[C@H]1[C@H]([C@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651284	phase I
BRD-K80284099	CCN(C[C@@H]1[C@@H]([C@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651285	phase I
BRD-K55543534	CCN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651286	phase I
BRD-K05778745	CCN(C[C@H]1[C@H]([C@@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651287	phase I
BRD-K56076713	CCN(C[C@@H]1[C@H]([C@@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651288	phase I
BRD-K28082924	CCN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)COC)c1ccccc1)S(C)(=O)=O	CID:54651289	phase I
BRD-K35760166	COCC(=O)NC[C@@H]1[C@@H]([C@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651290	phase I
BRD-K57397611	COCC(=O)NC[C@@H]1[C@H]([C@@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651291	phase I
BRD-K30934336	COCC(=O)NC[C@H]1[C@H]([C@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651292	phase I
BRD-K41200351	COCC(=O)NC[C@@H]1[C@@H]([C@@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651293	phase I
BRD-K65716211	COCC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651294	phase I
BRD-K89447773	COCC(=O)NC[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651295	phase I
BRD-K39108047	COCC(=O)NC[C@H]1[C@@H]([C@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651296	phase I
BRD-K89793018	COCC(=O)NC[C@H]1[C@H]([C@@H](CO)N1C(=O)C1CC1)c1ccc(cc1)C1=CCCC1	CID:54651297	phase I
BRD-K40973428	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N[C@@H]1CNC(=O)CC1CC1	CID:54651298	phase I
BRD-K07933458	CCc1csc(n1)N1[C@@H](CO)[C@H]([C@H]1CNCCOC)c1ccccc1	CID:54651299	phase I
BRD-K96343889	OC[C@@H]1N[C@H](CNC(=O)c2ccccn2)[C@@H]1c1ccc(cc1)-c1ccc(F)cc1	CID:54651300	phase I
BRD-K75884310	CC(=O)NC[C@@H]1[C@H]([C@H](CO)N1Cc1cccnc1)c1ccc(cc1)C1=CCCC1	CID:54651301	phase I
BRD-K40862820	CC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1Cc1cccnc1)c1ccc(cc1)C1=CCCC1	CID:54651302	phase I
BRD-K50005301	OC[C@H]1[C@H]([C@H](CNC(=O)C2CCC2)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651303	phase I
BRD-K85444001	OC[C@@H]1[C@H]([C@H](CNC(=O)C2CCC2)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651304	phase I
BRD-K51372689	OC[C@@H]1[C@@H]([C@@H](CNC(=O)C2CCC2)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651305	phase I
BRD-K90974935	OC[C@@H]1[C@H]([C@@H](CNC(=O)C2CCC2)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651306	phase I
BRD-K66390767	OC[C@H]1[C@@H]([C@@H](CNC(=O)C2CCC2)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651307	phase I
BRD-K95470847	OC[C@H]1[C@@H]([C@H](CNC(=O)C2CCC2)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651308	phase I
BRD-K32159948	CN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(=O)c1ccccn1	CID:54651309	phase I
BRD-K25768791	CN(C[C@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(=O)c1ccccn1	CID:54651310	phase I
BRD-K87511374	CN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(=O)c1ccccn1	CID:54651311	phase I
BRD-K18692529	CN(C[C@@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1)C(=O)c1ccccn1	CID:54651312	phase I
BRD-K41444660	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1CNC(C)C)C(=O)c1ccccc1	CID:54651313	phase I
BRD-K02636305	CCC(=O)NC[C@@H]1[C@H]([C@@H](CO)N1Cc1ccccn1)c1ccc(\C=C\C)cc1	CID:54651314	phase I
BRD-K38172414	CCC(=O)NC[C@H]1[C@H]([C@@H](CO)N1Cc1ccccn1)c1ccc(\C=C\C)cc1	CID:54651315	phase I
BRD-K33483445	CCC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1Cc1ccccn1)c1ccc(\C=C\C)cc1	CID:54651316	phase I
BRD-K88626416	CCC(=O)NC[C@@H]1[C@H]([C@H](CO)N1Cc1ccccn1)c1ccc(\C=C\C)cc1	CID:54651317	phase I
BRD-K26886657	CCC(=O)NC[C@H]1[C@@H]([C@H](CO)N1Cc1ccccn1)c1ccc(\C=C\C)cc1	CID:54651318	phase I
BRD-K48427969	CCC(=O)NC[C@@H]1[C@@H]([C@H](CO)N1Cc1ccccn1)c1ccc(\C=C\C)cc1	CID:54651319	phase I
BRD-K89949395	CCN(C[C@@H]1[C@H]([C@H](CO)N1Cc1cccnc1)c1ccc(\C=C\C)cc1)C(C)=O	CID:54651320	phase I
BRD-K72827150	CCNC[C@@H]1[C@@H]([C@H](CO)N1c1nc(C)c(C)s1)c1ccc(cc1)\C=C\C	CID:54651321	phase I
BRD-K27837783	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N[C@@H]1CN(CC(C)C)C(=O)c1ccccn1	CID:54651322	phase I
BRD-K51871563	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N[C@@H]1CN(CC(C)C)C(=O)c1ccccn1	CID:54651323	phase I
BRD-K97516320	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N[C@H]1CN(CC(C)C)C(=O)c1ccccn1	CID:54651324	phase I
BRD-K75265760	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N[C@H]1CN(CC(C)C)C(=O)c1ccccn1	CID:54651325	phase I
BRD-K81631939	CCC(=O)NC[C@H]1[C@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651326	phase I
BRD-K01558205	CCC(=O)NC[C@@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651327	phase I
BRD-K24387065	CCC(=O)NC[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651328	phase I
BRD-K04696500	CCC(=O)NC[C@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651329	phase I
BRD-K37795187	CCC(=O)NC[C@@H]1[C@@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651330	phase I
BRD-K36961201	CCC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651331	phase I
BRD-K61242732	CCC(=O)NC[C@H]1[C@@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651332	phase I
BRD-K71169857	CCC(=O)NC[C@@H]1[C@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651333	phase I
BRD-K08138210	OC[C@@H]1N[C@H](CN(CC2CCC2)C(=O)c2ccc(F)cc2)[C@@H]1c1ccccc1	CID:54651334	phase I
BRD-K51218228	OC[C@H]1N[C@@H](CN(CC2CCC2)C(=O)c2ccc(F)cc2)[C@H]1c1ccccc1	CID:54651335	phase I
BRD-K76423693	CCN(C[C@H]1N[C@H](CO)[C@H]1c1ccc(cc1)\C=C\C)C(=O)CN1CCOCC1	CID:54651336	phase I
BRD-K66271478	CCN(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)\C=C\C)C(=O)CN1CCOCC1	CID:54651337	phase I
BRD-K68730107	CCN(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)\C=C\C)C(=O)CN1CCOCC1	CID:54651338	phase I
BRD-K07001848	OC[C@H]1N[C@H](CNC(=O)CN2CCOCC2)[C@H]1c1ccc(cc1)-c1ccccc1	CID:54651339	phase I
BRD-K90665148	OC[C@@H]1N[C@@H](CNC(=O)CN2CCOCC2)[C@@H]1c1ccc(cc1)-c1ccccc1	CID:54651340	phase I
BRD-K69681876	OC[C@@H]1N[C@@H](CNC(=O)CN2CCOCC2)[C@H]1c1ccc(cc1)-c1ccccc1	CID:54651341	phase I
BRD-K52342362	CC(C)CN(C[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCC1)C(C)=O	CID:54651342	phase I
BRD-K58250123	CC(C)N(C[C@@H]1[C@H]([C@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)CN(C)C	CID:54651343	phase I
BRD-K23838495	CC(C)N(C[C@H]1[C@@H]([C@@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)CN(C)C	CID:54651344	phase I
BRD-K72967213	CC(C)N(C[C@H]1[C@H]([C@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)CN(C)C	CID:54651345	phase I
BRD-K49005570	CC(C)N(C[C@@H]1[C@H]([C@@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)CN(C)C	CID:54651346	phase I
BRD-K62209432	CC(C)N(C[C@@H]1[C@@H]([C@@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)CN(C)C	CID:54651347	phase I
BRD-K06514792	CC(C)N(C[C@H]1[C@@H]([C@H](CO)N1S(C)(=O)=O)c1ccccc1)C(=O)CN(C)C	CID:54651348	phase I
BRD-K67188562	COCC(=O)N1[C@H](CO)[C@@H]([C@@H]1CNC(=O)c1ccccn1)c1ccccc1	CID:54651349	phase I
BRD-K75297646	COCC(=O)N1[C@H](CO)[C@H]([C@@H]1CNC(=O)c1ccccn1)c1ccccc1	CID:54651350	phase I
BRD-K32859585	COCC(=O)N1[C@@H](CO)[C@H]([C@@H]1CNC(=O)c1ccccn1)c1ccccc1	CID:54651351	phase I
BRD-K02065962	COCC(=O)N1[C@H](CO)[C@H]([C@H]1CNC(=O)c1ccccn1)c1ccccc1	CID:54651352	phase I
BRD-K01626580	COCC(=O)N1[C@@H](CO)[C@@H]([C@@H]1CNC(=O)c1ccccn1)c1ccccc1	CID:54651353	phase I
BRD-K87449690	COCC(=O)N1[C@H](CO)[C@@H]([C@H]1CNC(=O)c1ccccn1)c1ccccc1	CID:54651354	phase I
BRD-K32301393	CC(=O)N1[C@@H](CO)[C@@H]([C@@H]1CNC(=O)CN1CCOCC1)c1ccccc1	CID:54651355	phase I
BRD-K50269042	CC(=O)N1[C@H](CO)[C@H]([C@@H]1CNC(=O)CN1CCOCC1)c1ccccc1	CID:54651356	phase I
BRD-K50472386	CC(=O)N1[C@H](CO)[C@H]([C@H]1CNC(=O)CN1CCOCC1)c1ccccc1	CID:54651357	phase I
BRD-K40695780	CC(=O)N1[C@H](CO)[C@@H]([C@@H]1CNC(=O)CN1CCOCC1)c1ccccc1	CID:54651358	phase I
BRD-K17343593	CC(=O)N1[C@@H](CO)[C@H]([C@@H]1CNC(=O)CN1CCOCC1)c1ccccc1	CID:54651359	phase I
BRD-K75085700	CC(=O)N1[C@H](CO)[C@@H]([C@H]1CNC(=O)CN1CCOCC1)c1ccccc1	CID:54651360	phase I
BRD-K22643697	CN(C[C@@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651361	phase I
BRD-K26526202	CN(C[C@@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651362	phase I
BRD-K12524159	CN(C[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651363	phase I
BRD-K25038599	CN(C[C@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651364	phase I
BRD-K91859707	CN(C[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651365	phase I
BRD-K88051295	CN(C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccccc1)S(=O)(=O)c1ccccc1	CID:54651366	phase I
BRD-K55640577	COCCN(C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1cccnc1	CID:54651367	phase I
BRD-K69768745	COCCN(C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1cccnc1	CID:54651368	phase I
BRD-K06614363	COCCN(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1cccnc1	CID:54651369	phase I
BRD-K63559825	COCCN(C[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C(=O)c1cccnc1	CID:54651370	phase I
BRD-K40332746	CC(C)N(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)-c1ccccc1)C(C)=O	CID:54651371	phase I
BRD-K55160246	CC(C)N(C[C@H]1N[C@H](CO)[C@H]1c1ccc(cc1)-c1ccccc1)C(C)=O	CID:54651372	phase I
BRD-K23629581	CC(C)N(C[C@@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)-c1ccccc1)C(C)=O	CID:54651373	phase I
BRD-K05896800	CC(C)N(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1ccccc1)C(C)=O	CID:54651374	phase I
BRD-K95285735	CN(C[C@@H]1[C@H]([C@H](CO)N1CC1CC1)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651375	phase I
BRD-K72636868	CN(C[C@H]1[C@@H]([C@@H](CO)N1CC1CC1)c1ccccc1)C(=O)c1cccc(F)c1	CID:54651376	phase I
BRD-K39887954	CCCNC(=O)N1[C@@H](CO)[C@H]([C@H]1CNC(C)=O)c1ccc(cc1)C1=CCCC1	CID:54651377	phase I
BRD-K13997553	CCCNC(=O)N1[C@@H](CO)[C@@H]([C@H]1CNC(C)=O)c1ccc(cc1)C1=CCCC1	CID:54651378	phase I
BRD-K52914297	CCC(=O)N1[C@@H](CO)[C@H]([C@@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651379	phase I
BRD-K93841862	CCC(=O)N1[C@@H](CO)[C@@H]([C@@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651380	phase I
BRD-K57364182	CCC(=O)N1[C@H](CO)[C@@H]([C@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651381	phase I
BRD-K44568925	CCC(=O)N1[C@H](CO)[C@@H]([C@@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651382	phase I
BRD-K74144927	CCC(=O)N1[C@@H](CO)[C@H]([C@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651383	phase I
BRD-K40961223	CCC(=O)N1[C@@H](CO)[C@@H]([C@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651384	phase I
BRD-K31647448	CCC(=O)N1[C@H](CO)[C@H]([C@@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651385	phase I
BRD-K61172568	CCC(=O)N1[C@H](CO)[C@H]([C@H]1CN(C(C)C)S(C)(=O)=O)c1ccccc1	CID:54651386	phase I
BRD-K77871059	CCC(=O)N1[C@@H](CO)[C@H]([C@@H]1CN(C)C(=O)c1ccccc1F)c1ccccc1	CID:54651387	phase I
BRD-K70588377	CCC(=O)N1[C@H](CO)[C@@H]([C@H]1CN(C)C(=O)c1ccccc1F)c1ccccc1	CID:54651388	phase I
BRD-K44366812	CCC(=O)N1[C@H](CO)[C@H]([C@@H]1CN(C)C(=O)c1ccccc1F)c1ccccc1	CID:54651389	phase I
BRD-K14196440	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N([C@H]1CNC(C)=O)C(=O)Cc1cccnc1	CID:54651390	phase I
BRD-K79746073	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1CNC(C)=O)C(=O)Cc1cccnc1	CID:54651391	phase I
BRD-K15384215	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1CNC(C)=O)C(=O)Cc1cccnc1	CID:54651392	phase I
BRD-K58606467	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@@H]1CNC(C)=O)C(=O)Cc1cccnc1	CID:54651393	phase I
BRD-K94373167	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1CN(C)C(=O)CC1CC1)C(=O)C1CC1	CID:54651394	phase I
BRD-K59475795	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1CN(C)C(=O)CC1CC1)C(=O)C1CC1	CID:54651395	phase I
BRD-K45576003	OC[C@@H]1N[C@@H](CNC(=O)c2cccc(F)c2)[C@@H]1c1ccc(cc1)C1=CCCCC1	CID:54651396	phase I
BRD-K23077259	OC[C@H]1N[C@H](CNC(=O)c2cccc(F)c2)[C@H]1c1ccc(cc1)C1=CCCCC1	CID:54651397	phase I
BRD-K97400656	CCC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1Cc1cccnc1)c1ccccc1	CID:54651398	phase I
BRD-K46385262	CCN(C[C@@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)C1=CCCC1)C(=O)c1cccnc1	CID:54651399	phase I
BRD-K49090949	CCN(C[C@H]1N[C@H](CO)[C@H]1c1ccc(cc1)C1=CCCC1)C(=O)c1cccnc1	CID:54651400	phase I
BRD-K74316684	CCN(C[C@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)C1=CCCC1)C(=O)c1cccnc1	CID:54651401	phase I
BRD-K96103953	CCNC[C@H]1[C@@H]([C@@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)C1=CCCCC1	CID:54651402	phase I
BRD-K85079349	OC[C@@H]1[C@@H]([C@H](CNCC2CCC2)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651403	phase I
BRD-K84331602	OC[C@@H]1[C@@H]([C@@H](CNCC2CCC2)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651404	phase I
BRD-K91070947	OC[C@H]1[C@H]([C@@H](CNCC2CCC2)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651405	phase I
BRD-K37282474	OC[C@H]1[C@@H]([C@H](CNCC2CCC2)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651406	phase I
BRD-K06359153	OC[C@H]1[C@H]([C@H](CNCC2CCC2)N1C(=O)Cc1cccnc1)c1ccccc1	CID:54651407	phase I
BRD-K83833567	CN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)c1ccccc1)c1ccccc1)C(=O)C1CCC1	CID:54651408	phase I
BRD-K32718105	CN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)c1ccccc1)c1ccccc1)C(=O)C1CCC1	CID:54651409	phase I
BRD-K53111504	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1CN(C)C(=O)c1ccccn1)C(C)=O	CID:54651410	phase I
BRD-K69075782	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N([C@H]1CN(C)C(=O)c1ccccn1)C(C)=O	CID:54651411	phase I
BRD-K85804197	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@@H]1CN(C)C(=O)c1ccccn1)C(C)=O	CID:54651412	phase I
BRD-K95142134	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N([C@H]1CN(C)C(=O)c1ccccn1)C(C)=O	CID:54651413	phase I
BRD-K26045715	OC[C@H]1[C@H]([C@H](CNCC2CCC2)N1CC1CC1)c1ccccc1	CID:54651414	phase I
BRD-K74206117	OC[C@@H]1[C@H]([C@@H](CNCC2CCC2)N1CC1CC1)c1ccccc1	CID:54651415	phase I
BRD-K83315952	OC[C@H]1[C@H]([C@@H](CNCC2CCC2)N1CC1CC1)c1ccccc1	CID:54651416	phase I
BRD-K86997406	OC[C@@H]1[C@@H]([C@@H](CNCC2CCC2)N1CC1CC1)c1ccccc1	CID:54651417	phase I
BRD-K95434676	CC(=O)N(CC1CCC1)C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)C1=CCCC1	CID:54651418	phase I
BRD-K28208028	CC(=O)N(CC1CCC1)C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)C1=CCCC1	CID:54651419	phase I
BRD-K44833108	CN(C)CC(=O)NC[C@@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651420	phase I
BRD-K80076202	CN(C)CC(=O)NC[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651421	phase I
BRD-K87501901	CN(C)CC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651422	phase I
BRD-K81469015	CN(C)CC(=O)NC[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651423	phase I
BRD-K65617817	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N([C@H]1CN(C)C(=O)NC1CCCC1)C(C)=O	CID:54651424	phase I
BRD-K92135888	COCC(=O)NC[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1ccccc1F	CID:54651425	phase I
BRD-K73276569	COCC(=O)NC[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)-c1ccccc1F	CID:54651426	phase I
BRD-K33236383	COCC(=O)NC[C@H]1N[C@H](CO)[C@H]1c1ccc(cc1)-c1ccccc1F	CID:54651427	phase I
BRD-K29834680	CCC(=O)N(CC(C)C)C[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651428	phase I
BRD-K73994412	CCC(=O)N(CC(C)C)C[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccccc1	CID:54651429	phase I
BRD-K87339026	CC(C)NC[C@@H]1[C@@H]([C@H](CO)N1S(C)(=O)=O)c1ccc(cc1)C1=CCCCC1	CID:54651430	phase I
BRD-K40349140	CC(C)NC(=O)N(C[C@@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccccc1)C1CCCC1	CID:54651431	phase I
BRD-K39092862	CC(C)NC(=O)N(C[C@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccccc1)C1CCCC1	CID:54651432	phase I
BRD-K54930318	COCC(=O)N(C[C@@H]1[C@H]([C@H](CO)N1C(=O)NC(C)C)c1ccccc1)C(C)C	CID:54651433	phase I
BRD-K01780082	COCC(=O)N(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)NC(C)C)c1ccccc1)C(C)C	CID:54651434	phase I
BRD-K83981181	COCC(=O)N(C[C@H]1[C@@H]([C@H](CO)N1C(=O)NC(C)C)c1ccccc1)C(C)C	CID:54651435	phase I
BRD-K25199340	COCC(=O)N(C[C@@H]1[C@H]([C@@H](CO)N1C(=O)NC(C)C)c1ccccc1)C(C)C	CID:54651436	phase I
BRD-K98374785	CCC(=O)N(C)C[C@@H]1[C@@H]([C@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)\C=C\C	CID:54651437	phase I
BRD-K81284476	CCC(=O)N(C)C[C@H]1[C@H]([C@@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)\C=C\C	CID:54651438	phase I
BRD-K64122011	CCC(=O)N(C)C[C@H]1[C@@H]([C@@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)\C=C\C	CID:54651439	phase I
BRD-K46932228	CCC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)\C=C\C	CID:54651440	phase I
BRD-K33066317	CCN(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)-c1ccc(F)cc1)C(=O)COC	CID:54651441	phase I
BRD-K32460251	CCN(C[C@@H]1N[C@H](CO)[C@H]1c1ccc(cc1)-c1ccc(F)cc1)C(=O)COC	CID:54651442	phase I
BRD-K41405597	CCN(C[C@H]1N[C@H](CO)[C@H]1c1ccc(cc1)-c1ccc(F)cc1)C(=O)COC	CID:54651443	phase I
BRD-K88114291	CCN(C[C@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)-c1ccc(F)cc1)C(=O)COC	CID:54651444	phase I
BRD-K90154335	CCN(C[C@@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)-c1ccc(F)cc1)C(=O)COC	CID:54651445	phase I
BRD-K97318829	CCCNC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651446	phase I
BRD-K89624539	CCCNC(=O)N(C)C[C@H]1[C@@H]([C@@H](CO)N1C(=O)c1ccccc1)c1ccccc1	CID:54651447	phase I
BRD-K92847204	CCCN(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651448	phase I
BRD-K69040870	CCCN(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651449	phase I
BRD-K33452357	COCC(=O)N(C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)\C=C\C)C(C)C	CID:54651450	phase I
BRD-K96063588	COCC(=O)N(C[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)\C=C\C)C(C)C	CID:54651451	phase I
BRD-K60595964	COCC(=O)N(C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)\C=C\C)C(C)C	CID:54651452	phase I
BRD-K63446165	COCC(=O)N(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)\C=C\C)C(C)C	CID:54651453	phase I
BRD-K97182575	COCC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1	CID:54651454	phase I
BRD-K37708631	COCC(=O)N(C)C[C@@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1	CID:54651455	phase I
BRD-K46004847	COCC(=O)N(C)C[C@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccccc1	CID:54651456	phase I
BRD-K10471793	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N[C@H]1CN(C(C)C)C(=O)C1CCC1	CID:54651457	phase I
BRD-K51394868	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N[C@@H]1CN(C(C)C)C(=O)C1CCC1	CID:54651458	phase I
BRD-K56244259	CCNC[C@@H]1[C@@H]([C@H](CO)N1c1nc(C)c(C)s1)c1ccc(cc1)C1=CCCC1	CID:54651459	phase I
BRD-K65134227	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(Cc2cccnc2)[C@@H]1CNC(C)C	CID:54651460	phase I
BRD-K15277331	CCC(=O)N(C)C[C@H]1[C@@H]([C@@H](CO)N1C(=O)Cc1ccncc1)c1ccccc1	CID:54651461	phase I
BRD-K97878521	CN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CC1)c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651462	phase I
BRD-K21503128	CN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CC1)c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651463	phase I
BRD-K17003857	CCN(C[C@@H]1[C@H]([C@H](CO)N1C(=O)C1CCC1)c1ccc(cc1)\C=C\C)C(=O)CC	CID:54651464	phase I
BRD-K14352739	CCN(C[C@H]1[C@@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccc(cc1)\C=C\C)C(=O)CC	CID:54651465	phase I
BRD-K91745830	COCC(=O)N1[C@@H](CO)[C@@H]([C@@H]1CN(C)C(=O)c1ccncc1)c1ccccc1	CID:54651466	phase I
BRD-K53390234	COCC(=O)N1[C@H](CO)[C@H]([C@H]1CN(C)C(=O)c1ccncc1)c1ccccc1	CID:54651467	phase I
BRD-K51579714	COCC(=O)N1[C@H](CO)[C@H]([C@@H]1CN(C)C(=O)c1ccncc1)c1ccccc1	CID:54651468	phase I
BRD-K96041907	CCCNC(=O)N(C)C[C@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)C1=CCCCC1	CID:54651469	phase I
BRD-K12177722	CN(C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccc(F)cc1)C(C)=O	CID:54651470	phase I
BRD-K88581223	CN(C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccc(F)cc1)C(C)=O	CID:54651471	phase I
BRD-K45760843	CN(C[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)-c1ccc(F)cc1)C(C)=O	CID:54651472	phase I
BRD-K19272295	CCC(=O)N(C)C[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651473	phase I
BRD-K57036336	CCC(=O)N(C)C[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651474	phase I
BRD-K44204702	CN(C[C@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1cccc(F)c1)C(=O)CC1CC1	CID:54651475	phase I
BRD-K65367823	OC[C@H]1N[C@H](CNC(=O)C2CCCC2)[C@H]1c1ccccc1	CID:54651476	phase I
BRD-K01275558	OC[C@@H]1N[C@@H](CNC(=O)C2CCCC2)[C@@H]1c1ccccc1	CID:54651477	phase I
BRD-K30758067	OC[C@H]1[C@@H]([C@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651478	phase I
BRD-K09957764	OC[C@H]1[C@H]([C@@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651479	phase I
BRD-K60994540	OC[C@@H]1[C@@H]([C@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651480	phase I
BRD-K18655724	OC[C@H]1[C@H]([C@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651481	phase I
BRD-K34532593	OC[C@@H]1[C@@H]([C@@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651482	phase I
BRD-K93570498	OC[C@H]1[C@@H]([C@@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651483	phase I
BRD-K60202553	OC[C@@H]1[C@H]([C@@H](CNC(=O)NC2CCCC2)N1C(=O)C1CC1)c1ccccc1	CID:54651484	phase I
BRD-K56219428	CN(C)CC(=O)NC[C@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1cccc(c1)C#N	CID:54651525	phase I
BRD-K45058329	CCCNC(=O)NC[C@@H]1[C@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651600	phase I
BRD-K87967738	CCCNC(=O)NC[C@@H]1[C@@H]([C@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651601	phase I
BRD-K07627743	CCCNC(=O)NC[C@H]1[C@@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651602	phase I
BRD-K44123761	CCCNC(=O)NC[C@@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651603	phase I
BRD-K70264850	CCCNC(=O)NC[C@H]1[C@H]([C@@H](CO)N1C(C)=O)c1ccc(cc1)C1=CCCCC1	CID:54651605	phase I
BRD-K62358627	COCC(=O)N(C[C@H]1N[C@H](CO)[C@H]1c1ccc(cc1)C1=CCCCC1)C(C)C	CID:54651702	phase I
BRD-K61599229	COCC(=O)N(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)C1=CCCCC1)C(C)C	CID:54651703	phase I
BRD-K65290386	COCC(=O)N(C[C@@H]1N[C@@H](CO)[C@@H]1c1ccc(cc1)C1=CCCCC1)C(C)C	CID:54651704	phase I
BRD-K96170115	COCC(=O)N(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)C1=CCCCC1)C(C)C	CID:54651705	phase I
BRD-K72869385	CN(C[C@H]1[C@@H]([C@H](CO)N1CC1CC1)c1ccc(cc1)C1=CCCCC1)C(C)=O	CID:54651752	phase I
BRD-K85352360	CN(C[C@@H]1[C@H]([C@@H](CO)N1CC1CC1)c1ccc(cc1)C1=CCCCC1)C(C)=O	CID:54651753	phase I
BRD-K58480962	COCCN(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)-c1cccnc1)C(C)=O	CID:54651984	phase I
BRD-K85646123	CC(C)NC[C@H]1[C@H]([C@@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)C1=CCCCC1	CID:54652075	phase I
BRD-K53640012	CC(C)NC[C@@H]1[C@@H]([C@H](CO)N1C(=O)NC(C)C)c1ccc(cc1)C1=CCCCC1	CID:54652077	phase I
BRD-K55857083	CCN(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)C1=CCCC1)C(=O)c1ccncc1	CID:54652101	phase I
BRD-K78787424	CCN(C[C@@H]1N[C@@H](CO)[C@H]1c1ccc(cc1)C1=CCCC1)C(=O)c1ccncc1	CID:54652102	phase I
BRD-K35468072	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1Cc1cccnc1	CID:54652405	phase I
BRD-K68831362	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1Cc1cccnc1	CID:54652406	phase I
BRD-K29946363	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1Cc1cccnc1	CID:54652407	phase I
BRD-K47771675	OC[C@@H]1[C@H]2[C@H](CNc3ccccc23)N1Cc1cccnc1	CID:54652408	phase I
BRD-K87313043	OC[C@@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccc2OCOc2c1	CID:54652409	phase I
BRD-K30098855	OC[C@H]1[C@H]2[C@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccc2OCOc2c1	CID:54652410	phase I
BRD-K32407455	OC[C@@H]1[C@H]2[C@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccc2OCOc2c1	CID:54652411	phase I
BRD-K61102260	OC[C@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccc2OCOc2c1	CID:54652412	phase I
BRD-K06898795	CN1C[C@H]2[C@H]([C@@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652413	phase I
BRD-K59085546	CN1C[C@@H]2[C@@H]([C@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652414	phase I
BRD-K71479066	CN1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652415	phase I
BRD-K30507268	CN1C[C@H]2[C@H]([C@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652416	phase I
BRD-K99569179	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1CC1CCOCC1	CID:54652417	phase I
BRD-K88373420	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1CC1CCOCC1	CID:54652418	phase I
BRD-K15168329	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1CC1CCOCC1	CID:54652419	phase I
BRD-K75648471	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1CC1CCOCC1	CID:54652420	phase I
BRD-K32162676	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3cccc(F)c3)c3ccccc23)N1Cc1cocn1	CID:54652421	phase I
BRD-K62050953	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3cccc(F)c3)c3ccccc23)N1Cc1cocn1	CID:54652422	phase I
BRD-K57346283	CCCNC(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2cccc(OC)c2)c2ccccc12	CID:54652427	phase I
BRD-K69480620	CCCNC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2cccc(OC)c2)c2ccccc12	CID:54652428	phase I
BRD-K53728687	CCCNC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2cccc(OC)c2)c2ccccc12	CID:54652429	phase I
BRD-K43952716	CCCNC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2cccc(OC)c2)c2ccccc12	CID:54652430	phase I
BRD-K71672626	Cc1cccc(c1)S(=O)(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C2CC2)c2ccccc12	CID:54652431	phase I
BRD-K36619075	Cc1cccc(c1)S(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C2CC2)c2ccccc12	CID:54652432	phase I
BRD-K12515921	Cc1cccc(c1)S(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C2CC2)c2ccccc12	CID:54652433	phase I
BRD-K15886574	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccc(F)cc3)c3ccccc23)N1C(=O)c1cccnc1	CID:54652434	phase I
BRD-K66333474	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccc(F)cc3)c3ccccc23)N1C(=O)c1cccnc1	CID:54652435	phase I
BRD-K08011922	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3ccc(F)cc3)c3ccccc23)N1C(=O)c1cccnc1	CID:54652436	phase I
BRD-K26694002	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3ccc(F)cc3)c3ccccc23)N1C(=O)c1cccnc1	CID:54652437	phase I
BRD-K97599743	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3cnccn3)c3ccccc23)N1CC1CCCC1	CID:54652438	phase I
BRD-K67763841	OC[C@@H]1[C@H]2[C@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652439	phase I
BRD-K82276852	OC[C@H]1[C@H]2[C@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652440	phase I
BRD-K38385119	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652441	phase I
BRD-K56367200	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652442	phase I
BRD-K46643133	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652443	phase I
BRD-K29785890	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652444	phase I
BRD-K36961456	COc1ccccc1CN1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)C1CCCCC1)c1ccccc21	CID:54652445	phase I
BRD-K76351896	COc1ccccc1CN1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)C1CCCCC1)c1ccccc21	CID:54652446	phase I
BRD-K94385551	COc1ccccc1CN1[C@@H](CO)[C@H]2[C@@H]1CN(C(=O)C1CCCCC1)c1ccccc21	CID:54652447	phase I
BRD-K74152472	COc1ccccc1CN1[C@H](CO)[C@@H]2[C@H]1CN(C(=O)C1CCCCC1)c1ccccc21	CID:54652448	phase I
BRD-K89148860	CN1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)Nc2cccc(F)c2)c2ccccc12	CID:54652449	phase I
BRD-K61181530	CN1C[C@H]2[C@H]([C@@H](CO)N2C(=O)Nc2cccc(F)c2)c2ccccc12	CID:54652450	phase I
BRD-K62153980	CN1C[C@H]2[C@H]([C@H](CO)N2C(=O)Nc2cccc(F)c2)c2ccccc12	CID:54652451	phase I
BRD-K27141795	CN1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)Nc2cccc(F)c2)c2ccccc12	CID:54652452	phase I
BRD-K35307739	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccccc3Cl)c3ccccc23)N1Cc1ccncc1	CID:54652453	phase I
BRD-K06833365	CN(C)CC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2cc(F)ccc2F)c2ccccc12	CID:54652454	phase I
BRD-K24011082	OC[C@H]1[C@H]2[C@H](CN(c3ccccc23)S(=O)(=O)c2ccccc2F)N1C(=O)CC1CC1	CID:54652455	phase I
BRD-K54711075	OC[C@@H]1[C@H]2[C@H](CN(c3ccccc23)S(=O)(=O)c2ccccc2F)N1C(=O)CC1CC1	CID:54652456	phase I
BRD-K61635139	OC[C@@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccccc2F)N1C(=O)CC1CC1	CID:54652457	phase I
BRD-K96535153	OC[C@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccccc2F)N1C(=O)CC1CC1	CID:54652458	phase I
BRD-K54408195	COc1ccccc1C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)Cc2cccnc2)c2ccccc12	CID:54652459	phase I
BRD-K40494872	COc1ccccc1C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)Cc2cccnc2)c2ccccc12	CID:54652460	phase I
BRD-K38176517	COc1ccccc1C(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)Cc2cccnc2)c2ccccc12	CID:54652461	phase I
BRD-K30437804	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3ccc4OCOc4c3)c3ccccc23)N1C(=O)CC1CC1	CID:54652462	phase I
BRD-K69803214	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3ccc4OCOc4c3)c3ccccc23)N1C(=O)CC1CC1	CID:54652463	phase I
BRD-K84449870	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3ccc4OCOc4c3)c3ccccc23)N1C(=O)CC1CC1	CID:54652464	phase I
BRD-K16827660	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3ccc4OCOc4c3)c3ccccc23)N1C(=O)CC1CC1	CID:54652465	phase I
BRD-K58952483	COc1ccc(cc1)C(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)NC(C)C)c2ccccc12	CID:54652466	phase I
BRD-K29311288	COc1ccc(cc1)C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)NC(C)C)c2ccccc12	CID:54652467	phase I
BRD-K41641213	COc1ccc(cc1)C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)NC(C)C)c2ccccc12	CID:54652468	phase I
BRD-K22357409	COc1ccc(cc1)C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)NC(C)C)c2ccccc12	CID:54652469	phase I
BRD-K67392692	OC[C@H]1[C@H]2[C@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652470	phase I
BRD-K55004655	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652471	phase I
BRD-K05001416	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652472	phase I
BRD-K59722258	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1S(=O)(=O)c1ccccc1	CID:54652473	phase I
BRD-K06328518	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3ccncc3)c3ccccc23)N1C(=O)c1ccccn1	CID:54652474	phase I
BRD-K73423421	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3ccncc3)c3ccccc23)N1C(=O)c1ccccn1	CID:54652475	phase I
BRD-K20429911	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3ccncc3)c3ccccc23)N1C(=O)c1ccccn1	CID:54652476	phase I
BRD-K03559171	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3ccncc3)c3ccccc23)N1C(=O)c1ccccn1	CID:54652477	phase I
BRD-K71038516	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1Cc1cccnc1	CID:54652478	phase I
BRD-K99638197	OC[C@@H]1[C@H]2[C@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1Cc1cccnc1	CID:54652479	phase I
BRD-K93181983	OC[C@H]1[C@H]2[C@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1Cc1cccnc1	CID:54652480	phase I
BRD-K30267135	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1Cc1cccnc1	CID:54652481	phase I
BRD-K15466057	COCC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CN(C(=O)Nc1cc(F)ccc1F)c1ccccc21	CID:54652482	phase I
BRD-K51975159	COCC(=O)N1[C@H](CO)[C@@H]2[C@H]1CN(C(=O)Nc1cc(F)ccc1F)c1ccccc21	CID:54652483	phase I
BRD-K31765411	COCC(=O)N1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)Nc1cc(F)ccc1F)c1ccccc21	CID:54652484	phase I
BRD-K56505861	COCC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)Nc1cc(F)ccc1F)c1ccccc21	CID:54652485	phase I
BRD-K19944193	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)C3CCCCC3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652486	phase I
BRD-K20081026	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)C3CCCCC3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652487	phase I
BRD-K24169646	OC[C@H]1[C@H]2[C@H](CN(C(=O)C3CCCCC3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652488	phase I
BRD-K82726072	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1CC1CCOCC1	CID:54652489	phase I
BRD-K82963710	OC[C@@H]1[C@H]2[C@H](CNc3ccccc23)N1CC1CCOCC1	CID:54652490	phase I
BRD-K56775501	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1CC1CCOCC1	CID:54652491	phase I
BRD-K40963786	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1CC1CCOCC1	CID:54652492	phase I
BRD-K67099101	CC(C)NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2ccccn2)c2ccccc12	CID:54652493	phase I
BRD-K48165980	CC(C)NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2ccccn2)c2ccccc12	CID:54652494	phase I
BRD-K26766547	CC(C)NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2ccccn2)c2ccccc12	CID:54652495	phase I
BRD-K47924474	CC(C)NC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2ccccn2)c2ccccc12	CID:54652496	phase I
BRD-K17645417	CN1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)c1ccc(F)cc1)c1ccccc21	CID:54652497	phase I
BRD-K79527000	CN1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)c1ccc(F)cc1)c1ccccc21	CID:54652498	phase I
BRD-K56046253	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1C(=O)Nc1ccc(F)cc1	CID:54652499	phase I
BRD-K18814836	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1C(=O)Nc1ccc(F)cc1	CID:54652500	phase I
BRD-K24009388	OC[C@@H]1[C@H]2[C@H](CNc3ccccc23)N1C(=O)Nc1ccc(F)cc1	CID:54652501	phase I
BRD-K78246556	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1C(=O)Nc1ccc(F)cc1	CID:54652502	phase I
BRD-K25295874	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2ccc3OCOc3c2)c2ccccc12	CID:54652503	phase I
BRD-K56593426	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2ccc3OCOc3c2)c2ccccc12	CID:54652504	phase I
BRD-K59397033	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2ccc3OCOc3c2)c2ccccc12	CID:54652505	phase I
BRD-K05789716	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccc(Cl)cc3)c3ccccc23)N1C(=O)C1CC1	CID:54652506	phase I
BRD-K45966720	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccc(Cl)cc3)c3ccccc23)N1C(=O)C1CC1	CID:54652507	phase I
BRD-K44413293	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3ccc(Cl)cc3)c3ccccc23)N1C(=O)C1CC1	CID:54652508	phase I
BRD-K86781204	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3ccc(Cl)cc3)c3ccccc23)N1C(=O)C1CC1	CID:54652509	phase I
BRD-K55702567	Cc1ccc(cc1)S(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2cccnc2)c2ccccc12	CID:54652510	phase I
BRD-K15882173	Cc1ccc(cc1)S(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2cccnc2)c2ccccc12	CID:54652511	phase I
BRD-K43624311	Cc1ccc(cc1)S(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2cccnc2)c2ccccc12	CID:54652512	phase I
BRD-K43624963	Cc1ccc(cc1)S(=O)(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2cccnc2)c2ccccc12	CID:54652513	phase I
BRD-K01477275	OC[C@@H]1[C@H]2[C@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1Cc1ccc(Cl)cc1	CID:54652514	phase I
BRD-K18381522	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1Cc1ccc(Cl)cc1	CID:54652515	phase I
BRD-K92912836	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1Cc1ccc(Cl)cc1	CID:54652516	phase I
BRD-K90004840	OC[C@H]1[C@H]2[C@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1Cc1ccc(Cl)cc1	CID:54652517	phase I
BRD-K53674027	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3ccccc3F)c3ccccc23)N1C(=O)C1CCCC1	CID:54652518	phase I
BRD-K10013730	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3ccccc3F)c3ccccc23)N1C(=O)C1CCCC1	CID:54652519	phase I
BRD-K97824883	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3ccccc3F)c3ccccc23)N1C(=O)C1CCCC1	CID:54652520	phase I
BRD-K48551077	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3ccccc3F)c3ccccc23)N1C(=O)C1CCCC1	CID:54652521	phase I
BRD-K44802959	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1C(=O)c1cccc(F)c1	CID:54652522	phase I
BRD-K93538891	OC[C@H]1[C@H]2[C@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1C(=O)c1cccc(F)c1	CID:54652523	phase I
BRD-K64273758	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1C(=O)c1cccc(F)c1	CID:54652524	phase I
BRD-K07360484	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Cc3ccccc3)c3ccccc23)N1C(=O)c1cccc(F)c1	CID:54652525	phase I
BRD-K20857608	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3cccnc3)c3ccccc23)N1C(=O)CN1CCOCC1	CID:54652526	phase I
BRD-K79422060	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3cccnc3)c3ccccc23)N1C(=O)CN1CCOCC1	CID:54652527	phase I
BRD-K08058167	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3cccnc3)c3ccccc23)N1C(=O)CN1CCOCC1	CID:54652528	phase I
BRD-K40471863	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3cccnc3)c3ccccc23)N1C(=O)CN1CCOCC1	CID:54652529	phase I
BRD-K93186542	COc1ccccc1C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652530	phase I
BRD-K39222404	COc1ccccc1C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652531	phase I
BRD-K43349162	COc1ccccc1C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652532	phase I
BRD-K05978741	COc1cccc(c1)C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652533	phase I
BRD-K53740124	COc1cccc(c1)C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652534	phase I
BRD-K37478894	COc1cccc(c1)C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652535	phase I
BRD-K16838397	COc1cccc(c1)C(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2ccccc2Cl)c2ccccc12	CID:54652536	phase I
BRD-K16772343	CCCNC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)C1CCC1)c1ccccc21	CID:54652537	phase I
BRD-K50010596	CCCNC(=O)N1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)C1CCC1)c1ccccc21	CID:54652538	phase I
BRD-K17122788	CN1[C@@H](CO)[C@H]2[C@@H]1CNc1ccccc21	CID:54652539	phase I
BRD-K14246967	CN1[C@@H](CO)[C@@H]2[C@H]1CNc1ccccc21	CID:54652540	phase I
BRD-K05814022	CN1[C@H](CO)[C@@H]2[C@H]1CNc1ccccc21	CID:54652541	phase I
BRD-K22642889	CN1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C2CCOCC2)c2ccccc12	CID:54652542	phase I
BRD-K96834740	CN1C[C@H]2[C@H]([C@H](CO)N2C(=O)C2CCOCC2)c2ccccc12	CID:54652543	phase I
BRD-K95607309	CN1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C2CCOCC2)c2ccccc12	CID:54652544	phase I
BRD-K69510809	CN1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C2CCOCC2)c2ccccc12	CID:54652545	phase I
BRD-K03157318	COCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2ccccc2)c2ccccc12	CID:54652546	phase I
BRD-K85312201	COCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2ccccc2)c2ccccc12	CID:54652547	phase I
BRD-K25822929	COCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2ccccc2)c2ccccc12	CID:54652548	phase I
BRD-K48433912	COCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2ccccc2)c2ccccc12	CID:54652549	phase I
BRD-K25380050	CC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(c1ccccc21)S(=O)(=O)c1ccc(F)cc1	CID:54652550	phase I
BRD-K37562700	CC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CN(c1ccccc21)S(=O)(=O)c1ccc(F)cc1	CID:54652551	phase I
BRD-K80738071	CC(=O)N1[C@H](CO)[C@@H]2[C@H]1CN(c1ccccc21)S(=O)(=O)c1ccc(F)cc1	CID:54652552	phase I
BRD-K20216424	CC(=O)N1[C@H](CO)[C@H]2[C@@H]1CN(c1ccccc21)S(=O)(=O)c1ccc(F)cc1	CID:54652553	phase I
BRD-K30910503	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1C(=O)C1CCCCC1	CID:54652554	phase I
BRD-K11577993	OC[C@@H]1[C@H]2[C@H](CNc3ccccc23)N1C(=O)C1CCCCC1	CID:54652555	phase I
BRD-K10702894	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1C(=O)C1CCCCC1	CID:54652556	phase I
BRD-K41419164	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1C(=O)C1CCCCC1	CID:54652557	phase I
BRD-K59204160	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3ccccc3)c3ccccc23)N1C(=O)Nc1ccccc1Cl	CID:54652558	phase I
BRD-K52689785	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3ccccc3)c3ccccc23)N1C(=O)Nc1ccccc1Cl	CID:54652559	phase I
BRD-K57490099	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3ccccc3)c3ccccc23)N1C(=O)Nc1ccccc1Cl	CID:54652560	phase I
BRD-K75101679	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3ccccc3)c3ccccc23)N1C(=O)Nc1ccccc1Cl	CID:54652561	phase I
BRD-K06902141	OC[C@@H]1[C@H]2[C@H](CNc3ccccc23)N1C(=O)Cc1ccccn1	CID:54652562	phase I
BRD-K53373965	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1C(=O)Cc1ccccn1	CID:54652563	phase I
BRD-K79035462	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1C(=O)Cc1ccccn1	CID:54652564	phase I
BRD-K15014572	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1C(=O)Cc1ccccn1	CID:54652565	phase I
BRD-K99369826	COc1ccc(CN2[C@H](CO)[C@@H]3[C@H]2CN(C(=O)Nc2ccc(F)cc2)c2ccccc32)cc1	CID:54652566	phase I
BRD-K43533284	COc1ccc(CN2[C@H](CO)[C@H]3[C@@H]2CN(C(=O)Nc2ccc(F)cc2)c2ccccc32)cc1	CID:54652567	phase I
BRD-K58869442	COc1ccc(CN2[C@@H](CO)[C@@H]3[C@H]2CN(C(=O)Nc2ccc(F)cc2)c2ccccc32)cc1	CID:54652568	phase I
BRD-K24698610	COc1ccc(CN2[C@@H](CO)[C@H]3[C@@H]2CN(C(=O)Nc2ccc(F)cc2)c2ccccc32)cc1	CID:54652569	phase I
BRD-K83577967	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3ccncc3)c3ccccc23)N1Cc1ccccc1F	CID:54652570	phase I
BRD-K87801302	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3ccncc3)c3ccccc23)N1Cc1ccccc1F	CID:54652571	phase I
BRD-K65750468	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3ccncc3)c3ccccc23)N1Cc1ccccc1F	CID:54652572	phase I
BRD-K92800455	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3ccncc3)c3ccccc23)N1Cc1ccccc1F	CID:54652573	phase I
BRD-K32100931	OC[C@@H]1[C@H]2[C@H](CNc3ccccc23)N1Cc1ccccc1Cl	CID:54652574	phase I
BRD-K98062050	OC[C@@H]1[C@@H]2[C@@H](CNc3ccccc23)N1Cc1ccccc1Cl	CID:54652575	phase I
BRD-K60895709	OC[C@H]1[C@@H]2[C@@H](CNc3ccccc23)N1Cc1ccccc1Cl	CID:54652576	phase I
BRD-K38444262	OC[C@H]1[C@H]2[C@H](CNc3ccccc23)N1Cc1ccccc1Cl	CID:54652577	phase I
BRD-K96703623	OC[C@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccccc2)N1Cc1ccccn1	CID:54652578	phase I
BRD-K49736551	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3cccnc3)c3ccccc23)N1Cc1ccc2OCOc2c1	CID:54652580	phase I
BRD-K42470309	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3cccnc3)c3ccccc23)N1Cc1ccc2OCOc2c1	CID:54652581	phase I
BRD-K79609340	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3cccnc3)c3ccccc23)N1Cc1ccc2OCOc2c1	CID:54652582	phase I
BRD-K39151995	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3cccnc3)c3ccccc23)N1Cc1ccc2OCOc2c1	CID:54652583	phase I
BRD-K59937136	CCCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)Nc2ccc(F)cc2)c2ccccc12	CID:54652584	phase I
BRD-K22599598	CCCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)Nc2ccc(F)cc2)c2ccccc12	CID:54652585	phase I
BRD-K55030454	CCCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)Nc2ccc(F)cc2)c2ccccc12	CID:54652586	phase I
BRD-K38373714	CCCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)Nc2ccc(F)cc2)c2ccccc12	CID:54652587	phase I
BRD-K98675009	OC[C@@H]1[C@H]2[C@H](CN(C(=O)C3CC3)c3ccccc23)N1C(=O)c1ccccc1	CID:54652588	phase I
BRD-K88099061	OC[C@H]1[C@H]2[C@H](CN(C(=O)C3CC3)c3ccccc23)N1C(=O)c1ccccc1	CID:54652589	phase I
BRD-K33928422	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)C3CC3)c3ccccc23)N1C(=O)c1ccccc1	CID:54652590	phase I
BRD-K31869770	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)C3CC3)c3ccccc23)N1C(=O)c1ccccc1	CID:54652591	phase I
BRD-K48441067	COCC(=O)N1[C@H](CO)[C@@H]2[C@H]1CN(C)c1ccccc21	CID:54652592	phase I
BRD-K55633328	COCC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(C)c1ccccc21	CID:54652593	phase I
BRD-K01823914	COCC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CN(C)c1ccccc21	CID:54652594	phase I
BRD-K88595392	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1C(=O)c1ccncc1	CID:54652595	phase I
BRD-K27477764	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1C(=O)c1ccncc1	CID:54652596	phase I
BRD-K45429601	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1C(=O)c1ccncc1	CID:54652597	phase I
BRD-K21699764	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cccc(Cl)c3)c3ccccc23)N1C(=O)c1ccncc1	CID:54652598	phase I
BRD-K22905567	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(C)=O)c2ccccc12	CID:54652599	phase I
BRD-K75034919	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(C)=O)c2ccccc12	CID:54652600	phase I
BRD-K81146041	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(C)=O)c2ccccc12	CID:54652601	phase I
BRD-K24789695	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(C)=O)c2ccccc12	CID:54652602	phase I
BRD-K80110842	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3cccc(F)c3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652603	phase I
BRD-K81812196	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cccc(F)c3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652604	phase I
BRD-K05906947	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3cccc(F)c3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652605	phase I
BRD-K76355933	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cccc(F)c3)c3ccccc23)N1C(=O)Cc1ccccn1	CID:54652606	phase I
BRD-K46092809	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3ccccc3F)c3ccccc23)N1C(=O)Cc1cccnc1	CID:54652607	phase I
BRD-K24896023	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccccc3F)c3ccccc23)N1C(=O)Cc1cccnc1	CID:54652608	phase I
BRD-K76779710	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccccc3F)c3ccccc23)N1C(=O)Cc1cccnc1	CID:54652609	phase I
BRD-K47037681	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3ccccc3F)c3ccccc23)N1C(=O)Cc1cccnc1	CID:54652610	phase I
BRD-K52189832	COc1ccc(CN2[C@@H](CO)[C@H]3[C@@H]2CNc2ccccc32)cc1	CID:54652611	phase I
BRD-K28513058	COc1ccc(CN2[C@@H](CO)[C@@H]3[C@H]2CNc2ccccc32)cc1	CID:54652612	phase I
BRD-K34231294	COc1ccc(CN2[C@H](CO)[C@H]3[C@@H]2CNc2ccccc32)cc1	CID:54652613	phase I
BRD-K20902354	COc1ccc(CN2[C@H](CO)[C@@H]3[C@H]2CNc2ccccc32)cc1	CID:54652614	phase I
BRD-K73005792	CN1[C@@H](CO)[C@H]2[C@@H]1CN(C(=O)Nc1ccccc1F)c1ccccc21	CID:54652615	phase I
BRD-K67015214	CN1[C@H](CO)[C@@H]2[C@H]1CN(C(=O)Nc1ccccc1F)c1ccccc21	CID:54652616	phase I
BRD-K24230322	CN1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)Nc1ccccc1F)c1ccccc21	CID:54652617	phase I
BRD-K08351986	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1C(=O)C1CC1	CID:54652618	phase I
BRD-K52071480	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1C(=O)C1CC1	CID:54652619	phase I
BRD-K87341885	OC[C@H]1[C@H]2[C@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1C(=O)C1CC1	CID:54652620	phase I
BRD-K38914331	OC[C@@H]1[C@H]2[C@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1C(=O)C1CC1	CID:54652621	phase I
BRD-K96113587	CCCNC(=O)N1C[C@H]2[C@H]([C@H](CO)N2CC2CCCCC2)c2ccccc12	CID:54652622	phase I
BRD-K63764020	CCCNC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2CC2CCCCC2)c2ccccc12	CID:54652623	phase I
BRD-K18390187	CCCNC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2CC2CCCCC2)c2ccccc12	CID:54652624	phase I
BRD-K43337737	CCCNC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2CC2CCCCC2)c2ccccc12	CID:54652625	phase I
BRD-K60737413	CCCNC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)CN2CCOCC2)c2ccccc12	CID:54652626	phase I
BRD-K43025837	CCCNC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)CN2CCOCC2)c2ccccc12	CID:54652627	phase I
BRD-K01751906	CCCNC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)CN2CCOCC2)c2ccccc12	CID:54652628	phase I
BRD-K73919378	CCCNC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)CN2CCOCC2)c2ccccc12	CID:54652629	phase I
BRD-K33226370	COc1ccccc1C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)Nc2ccccc2)c2ccccc12	CID:54652630	phase I
BRD-K82158149	COc1ccccc1C(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)Nc2ccccc2)c2ccccc12	CID:54652631	phase I
BRD-K62771975	COc1ccccc1C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)Nc2ccccc2)c2ccccc12	CID:54652632	phase I
BRD-K42543764	COc1ccccc1C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)Nc2ccccc2)c2ccccc12	CID:54652633	phase I
BRD-K72114074	COCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)c2ccccc2F)c2ccccc12	CID:54652634	phase I
BRD-K97864534	COCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)c2ccccc2F)c2ccccc12	CID:54652635	phase I
BRD-K69306987	COCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)c2ccccc2F)c2ccccc12	CID:54652636	phase I
BRD-K80204885	COCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)c2ccccc2F)c2ccccc12	CID:54652637	phase I
BRD-K76786157	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3cccc(F)c3)c3ccccc23)N1C(=O)C1CCOCC1	CID:54652638	phase I
BRD-K04288183	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3cccc(F)c3)c3ccccc23)N1C(=O)C1CCOCC1	CID:54652639	phase I
BRD-K37249103	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3cccc(F)c3)c3ccccc23)N1C(=O)C1CCOCC1	CID:54652640	phase I
BRD-K73838803	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3cccc(F)c3)c3ccccc23)N1C(=O)C1CCOCC1	CID:54652641	phase I
BRD-K85950149	COCC(=O)N1[C@H](CO)[C@@H]2[C@H]1CNc1ccccc21	CID:54652642	phase I
BRD-K03272554	COCC(=O)N1[C@H](CO)[C@H]2[C@@H]1CNc1ccccc21	CID:54652643	phase I
BRD-K65633533	COCC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CNc1ccccc21	CID:54652644	phase I
BRD-K58350294	COCC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CNc1ccccc21	CID:54652645	phase I
BRD-K07073046	CCC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CN(c1ccccc21)S(=O)(=O)c1ccccc1C	CID:54652646	phase I
BRD-K83441480	CCC(=O)N1[C@H](CO)[C@H]2[C@@H]1CN(c1ccccc21)S(=O)(=O)c1ccccc1C	CID:54652647	phase I
BRD-K35900085	CCC(=O)N1[C@H](CO)[C@@H]2[C@H]1CN(c1ccccc21)S(=O)(=O)c1ccccc1C	CID:54652648	phase I
BRD-K46028776	CCC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(c1ccccc21)S(=O)(=O)c1ccccc1C	CID:54652649	phase I
BRD-K75117691	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccccc3)c3ccccc23)N1Cc1ccccc1Cl	CID:54652650	phase I
BRD-K10225413	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3ccccc3)c3ccccc23)N1Cc1ccccc1Cl	CID:54652651	phase I
BRD-K25042903	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3ccccc3)c3ccccc23)N1Cc1ccccc1Cl	CID:54652652	phase I
BRD-K23784811	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3ccccc3)c3ccccc23)N1Cc1ccccc1Cl	CID:54652653	phase I
BRD-K44564943	OC[C@@H]1[C@H]2[C@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1CC1CCOCC1	CID:54652654	phase I
BRD-K24306712	OC[C@H]1[C@H]2[C@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1CC1CCOCC1	CID:54652655	phase I
BRD-K73451477	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1CC1CCOCC1	CID:54652656	phase I
BRD-K05639721	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)CC(F)(F)F)c3ccccc23)N1CC1CCOCC1	CID:54652657	phase I
BRD-K28452359	Cc1cccc(c1)S(=O)(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652658	phase I
BRD-K67601479	Cc1cccc(c1)S(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652659	phase I
BRD-K69510309	Cc1cccc(c1)S(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652660	phase I
BRD-K69200251	Cc1cccc(c1)S(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2CC2CCOCC2)c2ccccc12	CID:54652661	phase I
BRD-K89499048	COc1ccc(cc1)C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2ccc(Cl)cc2)c2ccccc12	CID:54652662	phase I
BRD-K35306330	COc1ccc(cc1)C(=O)N1C[C@H]2[C@H]([C@H](CO)N2Cc2ccc(Cl)cc2)c2ccccc12	CID:54652663	phase I
BRD-K67733357	COc1ccc(cc1)C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2Cc2ccc(Cl)cc2)c2ccccc12	CID:54652664	phase I
BRD-K01576758	COc1ccc(cc1)C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2ccc(Cl)cc2)c2ccccc12	CID:54652665	phase I
BRD-K34811324	COc1cccc(c1)C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)c2ccc(F)cc2)c2ccccc12	CID:54652666	phase I
BRD-K61127355	COc1cccc(c1)C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)c2ccc(F)cc2)c2ccccc12	CID:54652667	phase I
BRD-K48548528	COc1cccc(c1)C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)c2ccc(F)cc2)c2ccccc12	CID:54652668	phase I
BRD-K66750772	COc1cccc(c1)C(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)c2ccc(F)cc2)c2ccccc12	CID:54652669	phase I
BRD-K34856675	CN1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)c2cccnc2)c2ccccc12	CID:54652670	phase I
BRD-K75000753	CN1C[C@H]2[C@H]([C@@H](CO)N2C(=O)c2cccnc2)c2ccccc12	CID:54652671	phase I
BRD-K47543154	CN1C[C@@H]2[C@@H]([C@@H](CO)N2S(=O)(=O)c2ccccc2)c2ccccc12	CID:54652672	phase I
BRD-K80597067	CN1C[C@H]2[C@H]([C@H](CO)N2S(=O)(=O)c2ccccc2)c2ccccc12	CID:54652673	phase I
BRD-K78757578	CN1C[C@H]2[C@H]([C@@H](CO)N2S(=O)(=O)c2ccccc2)c2ccccc12	CID:54652674	phase I
BRD-K72713245	CN1C[C@@H]2[C@@H]([C@H](CO)N2S(=O)(=O)c2ccccc2)c2ccccc12	CID:54652675	phase I
BRD-K19417837	OC[C@@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccccc1Cl	CID:54652676	phase I
BRD-K40138205	OC[C@H]1[C@H]2[C@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccccc1Cl	CID:54652677	phase I
BRD-K98168260	OC[C@@H]1[C@H]2[C@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccccc1Cl	CID:54652678	phase I
BRD-K39911750	OC[C@H]1[C@@H]2[C@@H](CN(c3ccccc23)S(=O)(=O)c2ccc(F)cc2)N1Cc1ccccc1Cl	CID:54652679	phase I
BRD-K08852751	CN1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)C1CCCCC1)c1ccccc21	CID:54652680	phase I
BRD-K89584002	CN1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)C1CCCCC1)c1ccccc21	CID:54652681	phase I
BRD-K28623651	OC[C@H]1[C@H]2[C@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Cc1ccccc1	CID:54652682	phase I
BRD-K21539100	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Cc1ccccc1	CID:54652683	phase I
BRD-K31949858	OC[C@@H]1[C@H]2[C@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Cc1ccccc1	CID:54652684	phase I
BRD-K26069906	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)C3CCOCC3)c3ccccc23)N1C(=O)Cc1ccccc1	CID:54652685	phase I
BRD-K45955794	CCCNC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)c1cccnc1)c1ccccc21	CID:54652686	phase I
BRD-K37246443	CCCNC(=O)N1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)c1cccnc1)c1ccccc21	CID:54652687	phase I
BRD-K91504630	CC(C)NC(=O)N1[C@H](CO)[C@H]2[C@@H]1CN(C)c1ccccc21	CID:54652688	phase I
BRD-K62744999	CC(C)NC(=O)N1[C@H](CO)[C@@H]2[C@H]1CN(C)c1ccccc21	CID:54652689	phase I
BRD-K06518099	CC(C)NC(=O)N1[C@@H](CO)[C@@H]2[C@H]1CN(C)c1ccccc21	CID:54652690	phase I
BRD-K85916563	CC(C)NC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CN(C)c1ccccc21	CID:54652691	phase I
BRD-K58869323	OC[C@@H]1[C@H]2[C@H](CN(C(=O)c3ccccn3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652692	phase I
BRD-K37251488	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)c3ccccn3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652693	phase I
BRD-K55308802	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)c3ccccn3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652694	phase I
BRD-K59523333	OC[C@H]1[C@H]2[C@H](CN(C(=O)c3ccccn3)c3ccccc23)N1C(=O)Nc1ccccc1F	CID:54652695	phase I
BRD-K64402699	COc1ccccc1CN1[C@@H](CO)[C@H]2[C@@H]1CN(C(=O)c1cccnc1)c1ccccc21	CID:54652696	phase I
BRD-K45759060	COc1ccccc1CN1[C@@H](CO)[C@@H]2[C@H]1CN(C(=O)c1cccnc1)c1ccccc21	CID:54652697	phase I
BRD-K39301663	COc1ccccc1CN1[C@H](CO)[C@H]2[C@@H]1CN(C(=O)c1cccnc1)c1ccccc21	CID:54652698	phase I
BRD-K37277634	COc1ccccc1CN1[C@H](CO)[C@@H]2[C@H]1CN(C(=O)c1cccnc1)c1ccccc21	CID:54652699	phase I
BRD-K74185228	OC[C@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cc(F)ccc3F)c3ccccc23)N1Cc1cccnc1	CID:54652700	phase I
BRD-K15918270	OC[C@@H]1[C@@H]2[C@@H](CN(C(=O)Nc3cc(F)ccc3F)c3ccccc23)N1Cc1cccnc1	CID:54652701	phase I
BRD-K51050139	OC[C@H]1[C@H]2[C@H](CN(C(=O)Nc3cc(F)ccc3F)c3ccccc23)N1Cc1cccnc1	CID:54652702	phase I
BRD-K38400632	OC[C@@H]1[C@H]2[C@H](CN(C(=O)Nc3cc(F)ccc3F)c3ccccc23)N1Cc1cccnc1	CID:54652703	phase I
BRD-K52252091	CC(C)NC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C2CCCC2)c2ccccc12	CID:54652704	phase I
BRD-K58898119	CC(C)NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C2CCCC2)c2ccccc12	CID:54652705	phase I
BRD-K24824043	CC(C)NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C2CCCC2)c2ccccc12	CID:54652706	phase I
BRD-K75744810	CC(C)NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C2CCCC2)c2ccccc12	CID:54652707	phase I
BRD-K77984885	CCCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2Cc2cocn2)c2ccccc12	CID:54652708	phase I
BRD-K07702264	CCCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2Cc2cocn2)c2ccccc12	CID:54652709	phase I
BRD-K47727686	CN(C)CC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CN(C(=O)Cc1ccccc1)c1ccccc21	CID:54652710	phase I
BRD-K21898148	COc1ccc(cc1)C(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)Cc2ccccn2)c2ccccc12	CID:54652711	phase I
BRD-K03406275	COc1ccc(cc1)C(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)Cc2ccccn2)c2ccccc12	CID:54652712	phase I
BRD-K13582094	COc1ccc(cc1)C(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)Cc2ccccn2)c2ccccc12	CID:54652713	phase I
BRD-K36616116	COc1ccc(cc1)C(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)Cc2ccccn2)c2ccccc12	CID:54652714	phase I
BRD-K57883133	CC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)CC2CC2)c2ccccc12	CID:54652715	phase I
BRD-K06614049	CC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)CC2CC2)c2ccccc12	CID:54652716	phase I
BRD-K44218307	CC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)CC2CC2)c2ccccc12	CID:54652717	phase I
BRD-K19308316	CC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)CC2CC2)c2ccccc12	CID:54652718	phase I
BRD-K73184677	CC(C)NC(=O)N1[C@@H](CO)[C@H]2[C@@H]1CNc1ccccc21	CID:54652719	phase I
BRD-K82927587	CC(C)NC(=O)N1[C@H](CO)[C@H]2[C@@H]1CNc1ccccc21	CID:54652720	phase I
BRD-K91440401	COc1cccc(CN2[C@H](CO)[C@@H]3[C@H]2CN(C(=O)c2ccncc2)c2ccccc32)c1	CID:54652942	phase I
BRD-K79219981	CN1[C@@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54653977	phase I
BRD-K14346766	CN1[C@@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54653978	phase I
BRD-K38540783	CN1[C@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54653979	phase I
BRD-K44887903	CN1[C@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54653980	phase I
BRD-K45480436	CN1[C@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54653981	phase I
BRD-K42752188	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653982	phase I
BRD-K24572125	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653983	phase I
BRD-K09557852	CN1[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653984	phase I
BRD-K39367499	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653985	phase I
BRD-K25765811	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653986	phase I
BRD-K86981020	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653987	phase I
BRD-K80998388	CN1[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653988	phase I
BRD-K15104539	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54653989	phase I
BRD-K86843304	CN1[C@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NS(=O)(=O)CC(F)(F)F)cc2C1=O	CID:54653990	phase I
BRD-K32652655	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)O[C@@H]2COc2ccc(NC(=O)c3cscn3)cc2C1=O	CID:54653991	phase I
BRD-K58493165	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)O[C@H]2COc2ccc(NC(=O)c3cscn3)cc2C1=O	CID:54653992	phase I
BRD-K46810582	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)O[C@@H]2COc2ccc(NC(=O)c3cscn3)cc2C1=O	CID:54653993	phase I
BRD-K31314139	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)O[C@H]2COc2ccc(NC(=O)c3cscn3)cc2C1=O	CID:54653994	phase I
BRD-K20441249	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N4CCN(C)CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54653995	phase I
BRD-K77729938	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N4CCN(C)CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54653996	phase I
BRD-K31027517	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N4CCN(C)CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54653997	phase I
BRD-K85549762	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N4CCN(C)CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54653998	phase I
BRD-K69980290	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N4CCN(C)CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54653999	phase I
BRD-K74429632	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N4CCN(C)CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654000	phase I
BRD-K50230035	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N4CCN(C)CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654001	phase I
BRD-K54743934	COC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cncs4)cc3C(=O)N2C)O1	CID:54654002	phase I
BRD-K94797630	COc1cccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654003	phase I
BRD-K69449918	COc1cccc(NC(=O)C[C@@H]2CC[C@@H]3[C@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654004	phase I
BRD-K07594626	COc1cccc(NC(=O)C[C@@H]2CC[C@H]3[C@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654005	phase I
BRD-K58282082	COc1cccc(NC(=O)C[C@@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654006	phase I
BRD-K15513102	COc1cccc(NC(=O)C[C@H]2CC[C@H]3[C@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654007	phase I
BRD-K13107877	COc1cccc(NC(=O)C[C@@H]2CC[C@@H]3[C@@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654008	phase I
BRD-K81641277	COc1cccc(NC(=O)C[C@H]2CC[C@@H]3[C@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654009	phase I
BRD-K96636466	COc1cccc(NC(=O)C[C@H]2CC[C@@H]3[C@@H](COc4ccc(NC(=O)C5CCOCC5)cc4C(=O)N3C)O2)c1	CID:54654010	phase I
BRD-K83980681	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4ccno4)cc3C(=O)N2C)O1	CID:54654011	phase I
BRD-K41888384	CN1[C@H]2CC[C@@H](CC(=O)NC3CCCC3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654012	phase I
BRD-K06188347	CN1[C@@H]2CC[C@H](CC(=O)NC3CCCC3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654013	phase I
BRD-K50845321	CN1[C@H]2CC[C@@H](CC(=O)NC3CCCC3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654014	phase I
BRD-K39839350	CN1[C@H]2CC[C@H](CC(=O)NC3CCCC3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654015	phase I
BRD-K35493431	CN1[C@@H]2CC[C@@H](CC(=O)NC3CCCC3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654016	phase I
BRD-K95773671	CN1[C@@H]2CC[C@@H](CC(=O)NC3CCCC3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654017	phase I
BRD-K09002810	CN1[C@@H]2CC[C@H](CC(=O)NC3CCCC3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654018	phase I
BRD-K98383296	CN1[C@H]2CC[C@H](CC(=O)Nc3ccc4CCCc4c3)O[C@@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654019	phase I
BRD-K97408390	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654020	phase I
BRD-K61387428	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654021	phase I
BRD-K35193027	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654022	phase I
BRD-K54586093	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654023	phase I
BRD-K62219715	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654024	phase I
BRD-K45887240	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654025	phase I
BRD-K89637659	CN1[C@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3C)cc2C1=O	CID:54654026	phase I
BRD-K95880052	CN(C)C(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654027	phase I
BRD-K03679890	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654028	phase I
BRD-K10388622	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654029	phase I
BRD-K35131740	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654030	phase I
BRD-K57027181	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654031	phase I
BRD-K50572265	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654032	phase I
BRD-K78128989	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654033	phase I
BRD-K87377799	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)NCc4ccccc4)cc3C(=O)N2C)O1	CID:54654034	phase I
BRD-K98092496	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccccc3Cl)O[C@@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654035	phase I
BRD-K55252655	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccccc3Cl)O[C@@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654036	phase I
BRD-K42216874	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccccc3Cl)O[C@@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654037	phase I
BRD-K82582276	CN1[C@H]2CC[C@H](CC(=O)NCc3ccccc3Cl)O[C@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654038	phase I
BRD-K17654006	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccccc3Cl)O[C@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654039	phase I
BRD-K44150994	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccccc3Cl)O[C@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654040	phase I
BRD-K08666983	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccccc3Cl)O[C@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654041	phase I
BRD-K00812396	CN1[C@H]2CC[C@H](CC(=O)NCc3ccccc3Cl)O[C@@H]2COc2ccc(NC(=O)Nc3cccc(C)c3)cc2C1=O	CID:54654042	phase I
BRD-K00611064	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654043	phase I
BRD-K30758351	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654044	phase I
BRD-K30468438	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654045	phase I
BRD-K13119088	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654046	phase I
BRD-K31641287	CN1[C@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654047	phase I
BRD-K49255961	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654048	phase I
BRD-K89520577	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654049	phase I
BRD-K86448961	CN1[C@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654050	phase I
BRD-K69317358	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654051	phase I
BRD-K82121314	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654052	phase I
BRD-K63964021	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654053	phase I
BRD-K35455895	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654054	phase I
BRD-K96646082	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654055	phase I
BRD-K46732958	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654056	phase I
BRD-K53283295	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654057	phase I
BRD-K71855031	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)c3ccccc3F)cc2C1=O	CID:54654058	phase I
BRD-K01547285	CN(C)CCCNC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654059	phase I
BRD-K22630074	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654060	phase I
BRD-K59611536	CN(C)CCCNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654061	phase I
BRD-K43325273	CN(C)CCCNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654062	phase I
BRD-K26962314	CN(C)CCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654063	phase I
BRD-K59108735	CN(C)CCCNC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654064	phase I
BRD-K33562246	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654065	phase I
BRD-K94846015	COC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654066	phase I
BRD-K71104315	COC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654067	phase I
BRD-K20820984	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654068	phase I
BRD-K86842803	COC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654069	phase I
BRD-K48054407	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654070	phase I
BRD-K35081088	COC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654071	phase I
BRD-K32053117	COC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654072	phase I
BRD-K31791559	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCC(F)(F)F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654073	phase I
BRD-K13960684	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCC(F)(F)F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654074	phase I
BRD-K95481773	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCC(F)(F)F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654075	phase I
BRD-K22608272	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCC(F)(F)F)CC[C@H]3N(C)C(=O)c2c1	CID:54654076	phase I
BRD-K56593673	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCC(F)(F)F)CC[C@H]3N(C)C(=O)c2c1	CID:54654077	phase I
BRD-K68167702	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCC(F)(F)F)CC[C@H]3N(C)C(=O)c2c1	CID:54654078	phase I
BRD-K87010644	CNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Nc4ccc(cc4)C#N)cc3C(=O)N2C)O1	CID:54654079	phase I
BRD-K43438744	COc1cccc(c1)S(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccc(cc4)C(C)C)CC[C@@H]3N(C)C(=O)c2c1	CID:54654080	phase I
BRD-K16954564	CCCNC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccccc4C)CC[C@@H]3N(C)C(=O)c2c1	CID:54654081	phase I
BRD-K39398102	CN1[C@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654082	phase I
BRD-K89087272	CN1[C@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654083	phase I
BRD-K39363780	CN1[C@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654084	phase I
BRD-K29110787	CN1[C@@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654085	phase I
BRD-K21082546	CN1[C@@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654086	phase I
BRD-K14487375	CN1[C@@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654087	phase I
BRD-K78853683	CN1[C@@H]2CC[C@@H](CC(=O)N3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654088	phase I
BRD-K76885481	CN1[C@H]2CC[C@H](CC(=O)N3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccs3)cc2C1=O	CID:54654089	phase I
BRD-K09861842	COCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654090	phase I
BRD-K35995122	COCCNC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654091	phase I
BRD-K48431409	COCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654092	phase I
BRD-K23728767	COCCNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654093	phase I
BRD-K83426260	COCCNC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654094	phase I
BRD-K81674214	COCCNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654095	phase I
BRD-K32735617	COCCNC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654096	phase I
BRD-K36446300	COCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Cc4ccccc4)cc3C(=O)N2C)O1	CID:54654097	phase I
BRD-K29674378	COc1ccc(CNC(=O)C[C@@H]2CC[C@H]3[C@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654098	phase I
BRD-K90410459	COc1ccc(CNC(=O)C[C@H]2CC[C@@H]3[C@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654099	phase I
BRD-K12511144	COc1ccc(CNC(=O)C[C@@H]2CC[C@@H]3[C@@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654100	phase I
BRD-K38955087	COc1ccc(CNC(=O)C[C@@H]2CC[C@@H]3[C@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654101	phase I
BRD-K57640948	COc1ccc(CNC(=O)C[C@H]2CC[C@H]3[C@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654102	phase I
BRD-K83726357	COc1ccc(CNC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654103	phase I
BRD-K71045429	COc1ccc(CNC(=O)C[C@H]2CC[C@@H]3[C@@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654104	phase I
BRD-K50791850	COc1ccc(CNC(=O)C[C@@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)C(C)C)cc4C(=O)N3C)O2)cc1	CID:54654105	phase I
BRD-K57851810	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccccc3F)O[C@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654106	phase I
BRD-K14030662	CN1[C@H]2CC[C@H](CC(=O)NCc3ccccc3F)O[C@@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654107	phase I
BRD-K70117295	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccccc3F)O[C@@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654108	phase I
BRD-K11627226	CN1[C@H]2CC[C@H](CC(=O)NCc3ccccc3F)O[C@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654109	phase I
BRD-K39066612	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccccc3F)O[C@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654110	phase I
BRD-K32388810	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccccc3F)O[C@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654111	phase I
BRD-K16980601	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccccc3F)O[C@@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654112	phase I
BRD-K92434936	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccccc3F)O[C@@H]2COc2ccc(NC(=O)C3CCCCC3)cc2C1=O	CID:54654113	phase I
BRD-K51908245	CCCC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCc4cccc(F)c4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654114	phase I
BRD-K95269843	CCCC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCc4cccc(F)c4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654115	phase I
BRD-K97614198	CCCC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCc4cccc(F)c4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654116	phase I
BRD-K95352880	CCCC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCc4cccc(F)c4)CC[C@H]3N(C)C(=O)c2c1	CID:54654117	phase I
BRD-K47943934	CCCC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCc4cccc(F)c4)CC[C@H]3N(C)C(=O)c2c1	CID:54654118	phase I
BRD-K91377183	CCCC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCc4cccc(F)c4)CC[C@H]3N(C)C(=O)c2c1	CID:54654119	phase I
BRD-K34929727	CCCC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCc4cccc(F)c4)CC[C@H]3N(C)C(=O)c2c1	CID:54654120	phase I
BRD-K81706693	CCCC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCc4cccc(F)c4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654121	phase I
BRD-K01800462	COCC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccc(F)cc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654122	phase I
BRD-K87252271	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654123	phase I
BRD-K83365001	CN1[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654124	phase I
BRD-K32784186	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654125	phase I
BRD-K87492806	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654126	phase I
BRD-K88901529	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654127	phase I
BRD-K72324716	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654128	phase I
BRD-K34604832	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2C1=O	CID:54654129	phase I
BRD-K68655663	CN1[C@H]2CC[C@H](CC(=O)NCC3CC3)O[C@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654130	phase I
BRD-K43842808	CN1[C@H]2CC[C@@H](CC(=O)NCC3CC3)O[C@@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654131	phase I
BRD-K81873565	CN1[C@@H]2CC[C@H](CC(=O)NCC3CC3)O[C@@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654132	phase I
BRD-K55362990	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CC3)O[C@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654133	phase I
BRD-K14417684	CN1[C@H]2CC[C@@H](CC(=O)NCC3CC3)O[C@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654134	phase I
BRD-K89347234	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CC3)O[C@@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654135	phase I
BRD-K19520352	CN1[C@@H]2CC[C@H](CC(=O)NCC3CC3)O[C@H]2COc2ccc(NC(=O)NC3CCCC3)cc2C1=O	CID:54654136	phase I
BRD-K43931839	CN1[C@H]2CC[C@H](CC(=O)Nc3ccc4CCCCc4c3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654137	phase I
BRD-K62993927	CN1[C@@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654138	phase I
BRD-K79116978	CN1[C@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654139	phase I
BRD-K64544620	CN1[C@@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654140	phase I
BRD-K90679612	CN1[C@@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654141	phase I
BRD-K92924609	CN1[C@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654142	phase I
BRD-K13667629	CN1[C@@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654143	phase I
BRD-K61045941	CN1[C@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654144	phase I
BRD-K85779012	CN1[C@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654145	phase I
BRD-K97029281	CC(C)c1cccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NS(=O)(=O)c5ccccc5Cl)cc4C(=O)N3C)O2)c1	CID:54654146	phase I
BRD-K49988102	CCCNC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654147	phase I
BRD-K95033227	CCCNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654148	phase I
BRD-K34038660	CCCNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654149	phase I
BRD-K43481697	CCCNC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654150	phase I
BRD-K85388022	CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654151	phase I
BRD-K88003242	CCCNC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654152	phase I
BRD-K38860595	CCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654153	phase I
BRD-K93754181	CCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4ccc5OCOc5c4)cc3C(=O)N2C)O1	CID:54654154	phase I
BRD-K60759206	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654155	phase I
BRD-K20950855	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654156	phase I
BRD-K56553629	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654157	phase I
BRD-K62689646	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654158	phase I
BRD-K70875408	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654159	phase I
BRD-K17883815	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654160	phase I
BRD-K84336022	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654161	phase I
BRD-K20342961	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4cscn4)cc3C(=O)N2C)O1	CID:54654162	phase I
BRD-K18319377	CC(C)NC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccccc4Cl)CC[C@@H]3N(C)C(=O)c2c1	CID:54654163	phase I
BRD-K16117792	CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654164	phase I
BRD-K88279116	CNC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654165	phase I
BRD-K00172657	CNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654166	phase I
BRD-K15690570	CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654167	phase I
BRD-K31815095	CNC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654168	phase I
BRD-K83873778	CNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654169	phase I
BRD-K34684441	CNC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654170	phase I
BRD-K09584219	CNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54654171	phase I
BRD-K36853464	COc1cccc(CNC(=O)C[C@H]2CC[C@@H]3[C@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654172	phase I
BRD-K46746423	COc1cccc(CNC(=O)C[C@@H]2CC[C@@H]3[C@@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654173	phase I
BRD-K67402106	COc1cccc(CNC(=O)C[C@@H]2CC[C@H]3[C@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654174	phase I
BRD-K12907790	COc1cccc(CNC(=O)C[C@@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654175	phase I
BRD-K46373821	COc1cccc(CNC(=O)C[C@H]2CC[C@H]3[C@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654176	phase I
BRD-K42702351	COc1cccc(CNC(=O)C[C@@H]2CC[C@@H]3[C@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654177	phase I
BRD-K78710535	COc1cccc(CNC(=O)C[C@H]2CC[C@@H]3[C@@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654178	phase I
BRD-K61004012	COc1cccc(CNC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)c5cccs5)cc4C(=O)N3C)O2)c1	CID:54654179	phase I
BRD-K03413212	COCC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N4CCc5ccccc5C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654180	phase I
BRD-K30851490	COCC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N4CCc5ccccc5C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654181	phase I
BRD-K90842913	COCC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N4CCc5ccccc5C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654182	phase I
BRD-K40518011	COCC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N4CCc5ccccc5C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654183	phase I
BRD-K15185037	COCC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N4CCc5ccccc5C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654184	phase I
BRD-K87507139	COCC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N4CCc5ccccc5C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654185	phase I
BRD-K23414424	COCC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N4CCc5ccccc5C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654186	phase I
BRD-K58415365	COCC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N4CCc5ccccc5C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654187	phase I
BRD-K40212960	CN1[C@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654188	phase I
BRD-K19873234	CN1[C@@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654189	phase I
BRD-K96274292	CN1[C@@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654190	phase I
BRD-K19204484	CN1[C@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654191	phase I
BRD-K48225424	CN1[C@@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654192	phase I
BRD-K65124350	CN1[C@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654193	phase I
BRD-K53808186	CN1[C@@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654194	phase I
BRD-K85314854	CN1[C@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc2C1=O	CID:54654195	phase I
BRD-K22827077	CN1[C@H]2CC[C@H](CC(=O)NC3CCC3)O[C@@H]2COc2ccc(NC(=O)CC(F)(F)F)cc2C1=O	CID:54654196	phase I
BRD-K18511213	CC(C)c1ccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)Nc5ccc(F)c(F)c5)cc4C(=O)N3C)O2)cc1	CID:54654197	phase I
BRD-K04577097	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654198	phase I
BRD-K86336638	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654199	phase I
BRD-K55082668	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654200	phase I
BRD-K55149044	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654201	phase I
BRD-K58980886	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654202	phase I
BRD-K84245233	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654203	phase I
BRD-K12974237	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654204	phase I
BRD-K36671358	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C(=O)N2C)O1	CID:54654205	phase I
BRD-K71361154	COc1ccccc1CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C(=O)N2C)O1	CID:54654206	phase I
BRD-K57330428	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C(=O)N2C)O1	CID:54654207	phase I
BRD-K67087978	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C(=O)N2C)O1	CID:54654208	phase I
BRD-K88392283	COc1ccccc1CNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C(=O)N2C)O1	CID:54654209	phase I
BRD-K16980308	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3C(=O)N2C)O1	CID:54654210	phase I
BRD-K06039860	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654211	phase I
BRD-K31618614	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654212	phase I
BRD-K35716266	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(C)=O)cc3C(=O)N2C)O1	CID:54654215	phase I
BRD-K77905217	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(C)=O)cc3C(=O)N2C)O1	CID:54654216	phase I
BRD-K77804886	CCNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(C)=O)cc3C(=O)N2C)O1	CID:54654217	phase I
BRD-K70802145	CCNC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(C)=O)cc3C(=O)N2C)O1	CID:54654218	phase I
BRD-K80563095	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(C)=O)cc3C(=O)N2C)O1	CID:54654219	phase I
BRD-K09645804	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(C)=O)cc3C(=O)N2C)O1	CID:54654220	phase I
BRD-K15707609	CN1[C@@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654221	phase I
BRD-K64694541	CN1[C@@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654222	phase I
BRD-K11424789	CN1[C@@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654223	phase I
BRD-K48809858	CN1[C@@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654224	phase I
BRD-K53283097	CN1[C@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654225	phase I
BRD-K28987821	CN1[C@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654226	phase I
BRD-K39014692	CN1[C@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654227	phase I
BRD-K47002284	CN1[C@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3cccc(F)c3)cc2C1=O	CID:54654228	phase I
BRD-K68200852	CN1[C@@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654229	phase I
BRD-K95611306	CN1[C@@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654230	phase I
BRD-K76379937	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654231	phase I
BRD-K82494270	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654232	phase I
BRD-K19390271	CN1[C@@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654233	phase I
BRD-K07660364	CN1[C@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654234	phase I
BRD-K26968526	CN1[C@@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654237	phase I
BRD-K32380923	CN1[C@@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654238	phase I
BRD-K05984448	CN1[C@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654239	phase I
BRD-K01922500	CN1[C@@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654240	phase I
BRD-K63860984	CN1[C@@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654241	phase I
BRD-K36623409	CN1[C@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654242	phase I
BRD-K00596708	CN1[C@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654243	phase I
BRD-K01221769	CN1[C@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654244	phase I
BRD-K79004751	COc1cccc(CNC(=O)C[C@H]2CC[C@@H]3[C@@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654245	phase I
BRD-K81699431	COc1cccc(CNC(=O)C[C@H]2CC[C@H]3[C@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654246	phase I
BRD-K91535031	COc1cccc(CNC(=O)C[C@@H]2CC[C@H]3[C@@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654247	phase I
BRD-K88560304	COc1cccc(CNC(=O)C[C@@H]2CC[C@H]3[C@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654248	phase I
BRD-K17289060	COc1cccc(CNC(=O)C[C@@H]2CC[C@@H]3[C@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654249	phase I
BRD-K20272026	COc1cccc(CNC(=O)C[C@H]2CC[C@@H]3[C@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654250	phase I
BRD-K37933621	COc1cccc(CNC(=O)C[C@@H]2CC[C@@H]3[C@@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654251	phase I
BRD-K17666351	COc1cccc(CNC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NS(=O)(=O)c5ccccc5F)cc4C(=O)N3C)O2)c1	CID:54654252	phase I
BRD-K31610599	CN1[C@@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654253	phase I
BRD-K39143839	CN1[C@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654254	phase I
BRD-K70077013	CN1[C@@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654255	phase I
BRD-K07686903	CN1[C@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654256	phase I
BRD-K40121369	CN1[C@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654257	phase I
BRD-K11857988	CN1[C@@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654258	phase I
BRD-K23664396	CN1[C@@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654259	phase I
BRD-K20121961	C[C@@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654260	phase I
BRD-K96003120	C[C@@H](NC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654261	phase I
BRD-K15955205	C[C@@H](NC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654262	phase I
BRD-K81662460	C[C@@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654263	phase I
BRD-K51812182	C[C@@H](NC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654264	phase I
BRD-K62265198	C[C@@H](NC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654265	phase I
BRD-K51703152	C[C@H](NC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654266	phase I
BRD-K46661156	C[C@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654267	phase I
BRD-K51471107	C[C@H](NC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654268	phase I
BRD-K74582039	C[C@H](NC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654269	phase I
BRD-K19995377	C[C@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654270	phase I
BRD-K45319476	C[C@H](NC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654271	phase I
BRD-K88281008	C[C@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654272	phase I
BRD-K60667054	C[C@@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654273	phase I
BRD-K93339435	C[C@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654274	phase I
BRD-K55345900	C[C@@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3C(=O)N2C)O1)c1ccccc1	CID:54654275	phase I
BRD-K61683215	CN1[C@@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654276	phase I
BRD-K93376546	CN1[C@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654277	phase I
BRD-K13007539	CN1[C@@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654278	phase I
BRD-K34502913	CN1[C@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654279	phase I
BRD-K46447740	CN1[C@@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654280	phase I
BRD-K12506756	CN1[C@@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654281	phase I
BRD-K67260071	CN1[C@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654282	phase I
BRD-K59983542	CN1[C@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654283	phase I
BRD-K83654676	CC(C)c1cccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)c5cnccn5)cc4C(=O)N3C)O2)c1	CID:54654284	phase I
BRD-K66732564	COc1ccccc1NC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccc5COCc5c4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654285	phase I
BRD-K91595583	CN1[C@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2C1=O	CID:54654286	phase I
BRD-K21665449	CN1[C@@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2C1=O	CID:54654287	phase I
BRD-K47533918	CN1[C@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2C1=O	CID:54654288	phase I
BRD-K35584941	CN1[C@@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2C1=O	CID:54654289	phase I
BRD-K24469697	CN1[C@@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2C1=O	CID:54654290	phase I
BRD-K64040351	CN1[C@@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2C1=O	CID:54654291	phase I
BRD-K09124072	CN1[C@H]2CC[C@H](CC(=O)NCCN3CCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccc(c3)C#N)cc2C1=O	CID:54654292	phase I
BRD-K07105437	CN1[C@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654293	phase I
BRD-K43568193	CN1[C@@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654294	phase I
BRD-K71943487	CN1[C@@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654295	phase I
BRD-K80045183	CN1[C@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654296	phase I
BRD-K16434151	CN1[C@@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654297	phase I
BRD-K48457318	CN1[C@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654298	phase I
BRD-K17884417	CN1[C@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654299	phase I
BRD-K41878610	CN1[C@@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654300	phase I
BRD-K96543798	CN1[C@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cccc(F)c3)cc2C1=O	CID:54654301	phase I
BRD-K10835142	CCNC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654302	phase I
BRD-K88327759	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654303	phase I
BRD-K25789307	CCNC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654304	phase I
BRD-K14215828	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654305	phase I
BRD-K26053980	CCNC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654306	phase I
BRD-K69276764	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654307	phase I
BRD-K28117690	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@H](C)c4ccccc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654308	phase I
BRD-K05833481	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N[C@@H](C)c4ccccc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654309	phase I
BRD-K38123135	CCNC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N[C@@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654310	phase I
BRD-K95488738	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@@H](C)c4ccccc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654311	phase I
BRD-K48659337	CCNC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654314	phase I
BRD-K36159233	CCNC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@@H](C)c4ccccc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654315	phase I
BRD-K79090110	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654316	phase I
BRD-K45230579	COC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654317	phase I
BRD-K20182751	COC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654318	phase I
BRD-K00967758	COC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654319	phase I
BRD-K97633445	COC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654320	phase I
BRD-K53833823	COC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654321	phase I
BRD-K51579715	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654322	phase I
BRD-K48923155	COC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Nc4cc(C)cc(C)c4)cc3C(=O)N2C)O1	CID:54654323	phase I
BRD-K55297678	CCC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4c(F)cccc4F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654324	phase I
BRD-K18918854	CN1[C@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654325	phase I
BRD-K81882789	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654326	phase I
BRD-K37010295	CN1[C@@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654327	phase I
BRD-K71571889	CN1[C@@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654328	phase I
BRD-K09722997	CN1[C@@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654329	phase I
BRD-K73408523	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654330	phase I
BRD-K57552429	CN1[C@@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654331	phase I
BRD-K09701578	CN1[C@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654332	phase I
BRD-K14357170	CN1[C@@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654333	phase I
BRD-K92947165	CN1[C@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654334	phase I
BRD-K03113036	CN1[C@@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654335	phase I
BRD-K14971087	CN1[C@@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654336	phase I
BRD-K17535604	CN1[C@@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654337	phase I
BRD-K45543414	CN1[C@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654338	phase I
BRD-K19399946	CN1[C@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654339	phase I
BRD-K72271119	CN1[C@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3ccc(F)c(F)c3)cc2C1=O	CID:54654340	phase I
BRD-K95422182	CN1[C@H]2CC[C@H](CC(=O)Nc3ccc(C)cc3)O[C@@H]2COc2ccc(NC(=O)C3CCC3)cc2C1=O	CID:54654341	phase I
BRD-K96663038	COc1cccc(NC(=O)Nc2ccc3OC[C@@H]4O[C@@H](CC(=O)NCCc5ccccc5)CC[C@H]4N(C)C(=O)c3c2)c1	CID:54654342	phase I
BRD-K33616265	COc1cccc(NC(=O)Nc2ccc3OC[C@@H]4O[C@H](CC(=O)NCCc5ccccc5)CC[C@@H]4N(C)C(=O)c3c2)c1	CID:54654343	phase I
BRD-K57950796	COc1cccc(NC(=O)Nc2ccc3OC[C@H]4O[C@@H](CC(=O)NCCc5ccccc5)CC[C@H]4N(C)C(=O)c3c2)c1	CID:54654344	phase I
BRD-K99169187	COc1cccc(NC(=O)Nc2ccc3OC[C@H]4O[C@H](CC(=O)NCCc5ccccc5)CC[C@@H]4N(C)C(=O)c3c2)c1	CID:54654345	phase I
BRD-K34462945	COc1cccc(NC(=O)Nc2ccc3OC[C@@H]4O[C@@H](CC(=O)NCCc5ccccc5)CC[C@@H]4N(C)C(=O)c3c2)c1	CID:54654346	phase I
BRD-K72118202	COc1cccc(NC(=O)Nc2ccc3OC[C@H]4O[C@H](CC(=O)NCCc5ccccc5)CC[C@H]4N(C)C(=O)c3c2)c1	CID:54654347	phase I
BRD-K48047846	COc1cccc(NC(=O)Nc2ccc3OC[C@@H]4O[C@H](CC(=O)NCCc5ccccc5)CC[C@H]4N(C)C(=O)c3c2)c1	CID:54654348	phase I
BRD-K90132168	COc1cccc(NC(=O)Nc2ccc3OC[C@H]4O[C@@H](CC(=O)NCCc5ccccc5)CC[C@@H]4N(C)C(=O)c3c2)c1	CID:54654349	phase I
BRD-K00422823	COC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654350	phase I
BRD-K26160077	COC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654351	phase I
BRD-K56635255	COC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654352	phase I
BRD-K36796217	COC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654353	phase I
BRD-K72267874	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654354	phase I
BRD-K85906476	COC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654355	phase I
BRD-K99808872	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cccc(Cl)c4)cc3C(=O)N2C)O1	CID:54654356	phase I
BRD-K73701691	CN1[C@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654357	phase I
BRD-K99452176	CN1[C@@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654358	phase I
BRD-K05722694	CN1[C@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654359	phase I
BRD-K58991610	CN1[C@@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654360	phase I
BRD-K57759735	CN1[C@@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654361	phase I
BRD-K34238482	CN1[C@@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654362	phase I
BRD-K43266948	CN1[C@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654363	phase I
BRD-K65824347	CN1[C@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccccc3F)cc2C1=O	CID:54654364	phase I
BRD-K86375847	CN1[C@H]2CC[C@H](CC(=O)Nc3ccc4COCc4c3)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2C1=O	CID:54654365	phase I
BRD-K87445406	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654366	phase I
BRD-K13199470	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654367	phase I
BRD-K27006579	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654368	phase I
BRD-K72064822	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654369	phase I
BRD-K43279914	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654370	phase I
BRD-K98403755	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654371	phase I
BRD-K24050458	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654372	phase I
BRD-K92707657	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)C4CCOCC4)cc3C(=O)N2C)O1	CID:54654373	phase I
BRD-K48005755	COc1ccccc1NC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NS(C)(=O)=O)cc3C(=O)N2C)O1	CID:54654374	phase I
BRD-K02317159	CC(C)NC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCc4ccc(F)cc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654375	phase I
BRD-K18401446	CC(C)NC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCc4ccc(F)cc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654376	phase I
BRD-K82602524	CC(C)NC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCc4ccc(F)cc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654377	phase I
BRD-K95518555	CC(C)NC(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCc4ccc(F)cc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654378	phase I
BRD-K20051162	CC(C)NC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCc4ccc(F)cc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654379	phase I
BRD-K26350615	CC(C)NC(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCc4ccc(F)cc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654380	phase I
BRD-K86156277	CC(C)NC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCc4ccc(F)cc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654381	phase I
BRD-K93653328	CC(C)NC(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCc4ccc(F)cc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654382	phase I
BRD-K07056593	CC(C)c1cccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)c5ccc(cc5)C#N)cc4C(=O)N3C)O2)c1	CID:54654383	phase I
BRD-K49909254	CN1[C@H]2CC[C@H](CC(=O)NCC(F)(F)F)O[C@H]2COc2ccc(NC(=O)Nc3ccc(C)cc3)cc2C1=O	CID:54654384	phase I
BRD-K69951274	CN1[C@@H]2CC[C@H](CC(=O)NCC(F)(F)F)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(C)cc3)cc2C1=O	CID:54654385	phase I
BRD-K00513921	CN1[C@@H]2CC[C@@H](CC(=O)NCC(F)(F)F)O[C@H]2COc2ccc(NC(=O)Nc3ccc(C)cc3)cc2C1=O	CID:54654386	phase I
BRD-K85237791	CN1[C@@H]2CC[C@@H](CC(=O)NCC(F)(F)F)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(C)cc3)cc2C1=O	CID:54654387	phase I
BRD-K36681355	CN1[C@H]2CC[C@H](CC(=O)NCC(F)(F)F)O[C@@H]2COc2ccc(NC(=O)Nc3ccc(C)cc3)cc2C1=O	CID:54654388	phase I
BRD-K50974880	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCCOC)CC[C@@H]3N(C)C(=O)c2c1	CID:54654389	phase I
BRD-K86728331	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCCOC)CC[C@@H]3N(C)C(=O)c2c1	CID:54654390	phase I
BRD-K02010139	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCCOC)CC[C@H]3N(C)C(=O)c2c1	CID:54654391	phase I
BRD-K68018568	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCCOC)CC[C@@H]3N(C)C(=O)c2c1	CID:54654392	phase I
BRD-K16910145	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCCOC)CC[C@H]3N(C)C(=O)c2c1	CID:54654393	phase I
BRD-K25277218	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCCOC)CC[C@H]3N(C)C(=O)c2c1	CID:54654394	phase I
BRD-K63337793	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCCOC)CC[C@H]3N(C)C(=O)c2c1	CID:54654395	phase I
BRD-K92334440	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCCOC)CC[C@@H]3N(C)C(=O)c2c1	CID:54654396	phase I
BRD-K94373667	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCC4CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654397	phase I
BRD-K04230416	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCC4CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654398	phase I
BRD-K02750843	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCC4CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654399	phase I
BRD-K06731779	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCC4CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654400	phase I
BRD-K16255194	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCC4CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654401	phase I
BRD-K46989099	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCC4CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654402	phase I
BRD-K67242881	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCC4CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654403	phase I
BRD-K87707378	COc1ccc(cc1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCC4CC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654404	phase I
BRD-K62307953	CN1[C@H]2CC[C@H](CC(=O)Nc3cccc(F)c3)O[C@@H]2COc2ccc(NS(=O)(=O)CC(F)(F)F)cc2C1=O	CID:54654405	phase I
BRD-K32803351	CN1[C@H]2CC[C@H](CC(=O)Nc3ccc4CCCc4c3)O[C@@H]2COc2ccc(NC(=O)Nc3cccc(c3)C#N)cc2C1=O	CID:54654406	phase I
BRD-K00663349	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654407	phase I
BRD-K89489862	CN1[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654408	phase I
BRD-K34466966	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654409	phase I
BRD-K57953517	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654410	phase I
BRD-K56812045	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654411	phase I
BRD-K12678780	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654412	phase I
BRD-K60354118	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654413	phase I
BRD-K36138091	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654414	phase I
BRD-K88897538	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654415	phase I
BRD-K49896210	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654416	phase I
BRD-K52123998	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654417	phase I
BRD-K60581054	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654418	phase I
BRD-K27049144	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654419	phase I
BRD-K03430401	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654420	phase I
BRD-K42626894	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654421	phase I
BRD-K99198153	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654422	phase I
BRD-K48076585	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654423	phase I
BRD-K35738777	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654424	phase I
BRD-K16775575	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654425	phase I
BRD-K65310032	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@H]3N(C)C(=O)c2c1	CID:54654426	phase I
BRD-K34106732	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)N[C@@H]4CCN(Cc5ccccc5)C4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654427	phase I
BRD-K29269418	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654428	phase I
BRD-K06499413	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654429	phase I
BRD-K84022666	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654430	phase I
BRD-K95062171	CN1[C@@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654431	phase I
BRD-K39669696	CN1[C@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654432	phase I
BRD-K72174974	CN1[C@@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654433	phase I
BRD-K25866514	CN1[C@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654434	phase I
BRD-K14091022	CN1[C@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654435	phase I
BRD-K68166950	CN1[C@@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654436	phase I
BRD-K33780441	CN1[C@@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654437	phase I
BRD-K95698191	CN1[C@@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654438	phase I
BRD-K69719681	CN1[C@@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654439	phase I
BRD-K47812430	CN1[C@H]2CC[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654440	phase I
BRD-K49452151	CN1[C@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654441	phase I
BRD-K41660807	CN1[C@H]2CC[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654442	phase I
BRD-K73680494	COC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654443	phase I
BRD-K33071234	COC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654444	phase I
BRD-K36057770	COC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654445	phase I
BRD-K56950192	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654446	phase I
BRD-K13499761	COC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654447	phase I
BRD-K46276961	COC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654448	phase I
BRD-K53410660	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NS(=O)(=O)c4ccccc4Cl)cc3C(=O)N2C)O1	CID:54654449	phase I
BRD-K01245760	CN1[C@@H]2CC[C@H](CC(=O)NCC(F)(F)F)O[C@@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654450	phase I
BRD-K60753740	CN1[C@@H]2CC[C@@H](CC(=O)NCC(F)(F)F)O[C@@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654451	phase I
BRD-K96957785	CN1[C@@H]2CC[C@H](CC(=O)NCC(F)(F)F)O[C@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654452	phase I
BRD-K09068728	CN1[C@@H]2CC[C@@H](CC(=O)NCC(F)(F)F)O[C@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654453	phase I
BRD-K07516181	CN1[C@H]2CC[C@H](CC(=O)NCC(F)(F)F)O[C@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654454	phase I
BRD-K85205404	CN1[C@H]2CC[C@@H](CC(=O)NCC(F)(F)F)O[C@@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654455	phase I
BRD-K20758354	CN1[C@H]2CC[C@@H](CC(=O)NCC(F)(F)F)O[C@H]2COc2ccc(NC(=O)c3ccccc3Cl)cc2C1=O	CID:54654456	phase I
BRD-K79917113	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654457	phase I
BRD-K17627845	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654458	phase I
BRD-K79929772	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654459	phase I
BRD-K78449133	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654460	phase I
BRD-K79153888	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654461	phase I
BRD-K97337381	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654462	phase I
BRD-K95498999	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654463	phase I
BRD-K12405591	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCc4ccccc4F)CC[C@H]3N(C)C(=O)c2c1	CID:54654464	phase I
BRD-K24427624	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCc4ccccc4F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654465	phase I
BRD-K17839088	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCc4ccccc4F)CC[C@H]3N(C)C(=O)c2c1	CID:54654466	phase I
BRD-K40034561	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCc4ccccc4F)CC[C@H]3N(C)C(=O)c2c1	CID:54654467	phase I
BRD-K88842895	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCc4ccccc4F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654468	phase I
BRD-K55743249	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCc4ccccc4F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654469	phase I
BRD-K95608631	CCS(=O)(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCc4ccccc4F)CC[C@H]3N(C)C(=O)c2c1	CID:54654470	phase I
BRD-K73522157	CCS(=O)(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCc4ccccc4F)CC[C@@H]3N(C)C(=O)c2c1	CID:54654471	phase I
BRD-K81331655	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)c3ccc(cc3)C#N)cc2C1=O	CID:54654472	phase I
BRD-K06772064	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654473	phase I
BRD-K40454949	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654474	phase I
BRD-K55851396	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654475	phase I
BRD-K62056344	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654476	phase I
BRD-K66383562	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654477	phase I
BRD-K35841161	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654478	phase I
BRD-K52846581	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54654479	phase I
BRD-K62638625	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654480	phase I
BRD-K94557542	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654481	phase I
BRD-K77640397	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654482	phase I
BRD-K62628154	CN1[C@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654483	phase I
BRD-K23149749	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654484	phase I
BRD-K57037989	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654485	phase I
BRD-K49378999	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654486	phase I
BRD-K70551857	CN1[C@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3)cc2C1=O	CID:54654487	phase I
BRD-K16472441	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)cc3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654488	phase I
BRD-K58649267	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)cc3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654489	phase I
BRD-K53923750	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(Cl)cc3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654490	phase I
BRD-K03250561	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(Cl)cc3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654491	phase I
BRD-K71361566	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)cc3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654492	phase I
BRD-K55437057	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc(Cl)cc3)O[C@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654493	phase I
BRD-K35637774	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc(Cl)cc3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654494	phase I
BRD-K97424427	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc(Cl)cc3)O[C@@H]2COc2ccc(NC(=O)Nc3c(C)noc3C)cc2C1=O	CID:54654495	phase I
BRD-K94293090	CN1[C@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654496	phase I
BRD-K83001027	CN1[C@@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654497	phase I
BRD-K08760804	CN1[C@@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654498	phase I
BRD-K81112982	CN1[C@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654499	phase I
BRD-K97251260	CN1[C@@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654500	phase I
BRD-K09059658	CN1[C@@H]2CC[C@@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654501	phase I
BRD-K88180879	CN1[C@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654502	phase I
BRD-K72199653	CN1[C@H]2CC[C@H](CC(=O)Nc3cn(C)nc3C)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654503	phase I
BRD-K71761811	CN1[C@H]2CC[C@@H](CC(=O)NC3CCCCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654504	phase I
BRD-K85099724	CN1[C@@H]2CC[C@H](CC(=O)NC3CCCCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654505	phase I
BRD-K14862006	CN1[C@H]2CC[C@H](CC(=O)NC3CCCCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654506	phase I
BRD-K97062166	CN1[C@@H]2CC[C@@H](CC(=O)NC3CCCCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654507	phase I
BRD-K23723926	CN1[C@H]2CC[C@@H](CC(=O)NC3CCCCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654508	phase I
BRD-K11749439	CN1[C@@H]2CC[C@H](CC(=O)NC3CCCCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654509	phase I
BRD-K53342443	CN1[C@@H]2CC[C@@H](CC(=O)NC3CCCCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654510	phase I
BRD-K86086755	CN1[C@H]2CC[C@H](CC(=O)NC3CCCCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654511	phase I
BRD-K43774268	CC(C)c1ccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)c5ccno5)cc4C(=O)N3C)O2)cc1	CID:54654512	phase I
BRD-K92659956	CN1[C@@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654513	phase I
BRD-K33328711	CN1[C@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654514	phase I
BRD-K12241427	CN1[C@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654515	phase I
BRD-K45924279	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654516	phase I
BRD-K27175304	CN1[C@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654517	phase I
BRD-K55641492	CN1[C@@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654518	phase I
BRD-K19036853	CN1[C@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654519	phase I
BRD-K03716420	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654520	phase I
BRD-K97373677	CC(C)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccc(Cl)cc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654521	phase I
BRD-K63731274	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4ccccc4F)cc3C(=O)N2C)O1	CID:54654522	phase I
BRD-K68522303	COC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4ccccc4F)cc3C(=O)N2C)O1	CID:54654523	phase I
BRD-K38052671	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4ccccc4F)cc3C(=O)N2C)O1	CID:54654524	phase I
BRD-K77411261	COC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4ccccc4F)cc3C(=O)N2C)O1	CID:54654525	phase I
BRD-K46734661	COC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4ccccc4F)cc3C(=O)N2C)O1	CID:54654526	phase I
BRD-K28112059	COC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4ccccc4F)cc3C(=O)N2C)O1	CID:54654527	phase I
BRD-K67190692	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654528	phase I
BRD-K43484121	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654529	phase I
BRD-K69014051	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654530	phase I
BRD-K84195635	CN1[C@@H]2CC[C@@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654531	phase I
BRD-K80193146	CN1[C@H]2CC[C@@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654532	phase I
BRD-K96329791	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654533	phase I
BRD-K96952717	CN1[C@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3cccc(c3)C(F)(F)F)cc2C1=O	CID:54654534	phase I
BRD-K48654093	CN1[C@@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654535	phase I
BRD-K22033393	CN1[C@@H]2CC[C@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654536	phase I
BRD-K29626061	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654537	phase I
BRD-K81826010	CN1[C@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654538	phase I
BRD-K16939073	CN1[C@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654539	phase I
BRD-K16401691	CN1[C@@H]2CC[C@@H](CC(=O)NCC3CCCCC3)O[C@@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654540	phase I
BRD-K95762279	CN1[C@H]2CC[C@H](CC(=O)Nc3cc(F)ccc3F)O[C@@H]2COc2ccc(NC(=O)c3ccc(cc3)C#N)cc2C1=O	CID:54654541	phase I
BRD-K40098720	CN1[C@@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654542	phase I
BRD-K78451750	CN1[C@@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654543	phase I
BRD-K88541752	CN1[C@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654544	phase I
BRD-K56482508	CN1[C@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654545	phase I
BRD-K18152229	CN1[C@@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654546	phase I
BRD-K41014695	CN1[C@@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654547	phase I
BRD-K17973355	CN1[C@H]2CC[C@@H](CC(=O)NCCCN3CCOCC3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654548	phase I
BRD-K59130924	CN1[C@H]2CC[C@H](CC(=O)NCCCN3CCOCC3)O[C@@H]2COc2ccc(NC(=O)Nc3ccccc3Cl)cc2C1=O	CID:54654549	phase I
BRD-K07760433	CN1[C@H]2CC[C@H](CC(=O)Nc3cccc4ccccc34)O[C@@H]2COc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2C1=O	CID:54654550	phase I
BRD-K06280926	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654551	phase I
BRD-K56731825	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654552	phase I
BRD-K07244661	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654553	phase I
BRD-K14415573	CN(C)C(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654554	phase I
BRD-K50266413	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654555	phase I
BRD-K37088230	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654556	phase I
BRD-K38796873	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654557	phase I
BRD-K07852637	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4ccc(F)cc4)cc3C(=O)N2C)O1	CID:54654558	phase I
BRD-K76765843	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654559	phase I
BRD-K07125273	COC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654560	phase I
BRD-K65851733	COC(=O)C[C@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654561	phase I
BRD-K39622686	COC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654562	phase I
BRD-K89953543	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654563	phase I
BRD-K69616553	COC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654564	phase I
BRD-K12382140	COC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654565	phase I
BRD-K10810699	COC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54654566	phase I
BRD-K39613698	COc1ccccc1C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4cccc(c4)C(C)C)CC[C@@H]3N(C)C(=O)c2c1	CID:54654567	phase I
BRD-K42173890	CN1[C@@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654568	phase I
BRD-K66740714	CN1[C@@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654569	phase I
BRD-K57696989	CN1[C@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654570	phase I
BRD-K24192521	CN1[C@@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654571	phase I
BRD-K03845749	CN1[C@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654572	phase I
BRD-K18309912	CN1[C@H]2CC[C@@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654573	phase I
BRD-K09503339	CN1[C@@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654574	phase I
BRD-K35440818	CN1[C@H]2CC[C@H](CC(=O)N3CCOCC3)O[C@@H]2COc2ccc(NS(C)(=O)=O)cc2C1=O	CID:54654575	phase I
BRD-K87159745	COc1ccccc1C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCCc4ccncc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654576	phase I
BRD-K47024121	COc1ccccc1C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCCc4ccncc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654577	phase I
BRD-K35769695	COc1ccccc1C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCCc4ccncc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654578	phase I
BRD-K51181663	COc1ccccc1C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCCc4ccncc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654579	phase I
BRD-K66142238	COc1ccccc1C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCCc4ccncc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654580	phase I
BRD-K12738359	COc1ccccc1C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCCc4ccncc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654581	phase I
BRD-K96020117	COc1ccccc1C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCCc4ccncc4)CC[C@H]3N(C)C(=O)c2c1	CID:54654582	phase I
BRD-K05025838	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCCCN4CCOCC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654583	phase I
BRD-K87865140	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCCCN4CCOCC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654584	phase I
BRD-K28582709	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCCCN4CCOCC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654585	phase I
BRD-K16466792	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCCCN4CCOCC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654586	phase I
BRD-K97993646	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)NCCCN4CCOCC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654587	phase I
BRD-K45431864	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@H](CC(=O)NCCCN4CCOCC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654588	phase I
BRD-K13807179	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCCCN4CCOCC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654589	phase I
BRD-K85724483	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)NCCCN4CCOCC4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654590	phase I
BRD-K33994902	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654591	phase I
BRD-K98123586	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654592	phase I
BRD-K43225681	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654593	phase I
BRD-K32755775	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654594	phase I
BRD-K88058683	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654595	phase I
BRD-K00248931	CN1[C@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654596	phase I
BRD-K30794866	CN1[C@@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654597	phase I
BRD-K88282487	CN1[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COc2ccc(NC(=O)C3CCOCC3)cc2C1=O	CID:54654598	phase I
BRD-K21913257	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654599	phase I
BRD-K87730884	CN1[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654600	phase I
BRD-K42361978	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654601	phase I
BRD-K35002913	CN1[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654602	phase I
BRD-K71718338	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654603	phase I
BRD-K94676520	CN1[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654604	phase I
BRD-K25991217	CN1[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654605	phase I
BRD-K83757561	CN1[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654606	phase I
BRD-K12980773	CN1[C@@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654607	phase I
BRD-K58788895	CN1[C@@H]2CC[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654608	phase I
BRD-K46255436	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)Cc3cccs3)cc2C1=O	CID:54654609	phase I
BRD-K68645163	CN1[C@H]2CC[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)O[C@H]2COc2ccc(NC(=O)c3cnccn3)cc2C1=O	CID:54654613	phase I
BRD-K31929173	CN1[C@@H]2CC[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)O[C@H]2COc2ccc(NC(=O)Nc3ccccc3F)cc2C1=O	CID:54654640	phase I
BRD-K35701136	COC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)c4ccc(cc4)C(F)(F)F)cc3C(=O)N2C)O1	CID:54654656	phase I
BRD-K16826857	COc1cccc(c1)C(=O)Nc1ccc2OC[C@@H]3O[C@@H](CC(=O)N[C@@H](C)c4ccccc4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654676	phase I
BRD-K65081680	COc1cccc(c1)C(=O)Nc1ccc2OC[C@H]3O[C@@H](CC(=O)Nc4ccc5CCCCc5c4)CC[C@@H]3N(C)C(=O)c2c1	CID:54654681	phase I
BRD-K10779199	COc1ccccc1CNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Nc4ccc(F)c(F)c4)cc3C(=O)N2C)O1	CID:54654700	phase I
BRD-K48508383	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)Nc4ccc(F)c(F)c4)cc3C(=O)N2C)O1	CID:54654703	phase I
BRD-K32761691	COc1cccc(c1)S(=O)(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCC4CCCCC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654715	phase I
BRD-K75828577	CN1[C@H]2CC[C@H](CC(=O)NC3CCCC3)O[C@H]2COc2ccc(NC(=O)c3ccccc3)cc2C1=O	CID:54654776	phase I
BRD-K19919069	CC(C)c1cccc(NC(=O)C[C@H]2CC[C@H]3[C@@H](COc4ccc(NC(=O)NCc5ccccc5)cc4C(=O)N3C)O2)c1	CID:54654798	phase I
BRD-K05702937	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)Nc4c(C)noc4C)cc3C(=O)N2C)O1	CID:54654805	phase I
BRD-K00816125	CCCNC(=O)C[C@H]1CC[C@@H]2[C@@H](COc3ccc(NC(=O)NC(C)C)cc3C(=O)N2C)O1	CID:54654898	phase I
BRD-K52542879	CCCC(=O)Nc1ccc2OC[C@@H]3O[C@H](CC(=O)NCC4CC4)CC[C@H]3N(C)C(=O)c2c1	CID:54654906	phase I
BRD-K57974008	C[C@@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cc(C)on4)cc3C(=O)N2C)O1)c1ccccc1	CID:54655268	phase I
BRD-K41141892	CCCNC(=O)C[C@@H]1CC[C@H]2[C@H](COc3ccc(NC(=O)Cc4cccs4)cc3C(=O)N2C)O1	CID:54655704	phase I
BRD-K16026651	COC(=O)C[C@H]1CC[C@H]2[C@@H](COc3ccc(NC(=O)c4cc(F)cc(F)c4)cc3C(=O)N2C)O1	CID:54655756	phase I
BRD-K80790879	CN1[C@@H]2CC[C@H](CC(O)=O)O[C@H]2COc2ccc(NC(=O)c3cc(C)on3)cc2C1=O	CID:54656096	phase I
BRD-K65736998	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cc(C)on4)cc3C(=O)N2C)O1	CID:54656566	phase I
BRD-K87423723	CCCNC(=O)C[C@H]1CC[C@@H]2[C@H](COc3ccc(NC(=O)c4cc(C)on4)cc3C(=O)N2C)O1	CID:54657141	phase I
BRD-K89056622	CS(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3)CC[C@H]12	CID:54657476	phase I
BRD-K20159808	CS(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3)CC[C@H]12	CID:54657477	phase I
BRD-K56206243	COC(=O)C[C@@H]1CC[C@@H]2NC[C@@H](O)COC[C@H]2O1	CID:54657478	phase I
BRD-K70810261	COC(=O)C[C@@H]1CC[C@H]2NC[C@@H](O)COC[C@@H]2O1	CID:54657479	phase I
BRD-K40597368	COC(=O)C[C@H]1CC[C@H]2NC[C@H](O)COC[C@@H]2O1	CID:54657480	phase I
BRD-K74245085	COC(=O)C[C@H]1CC[C@@H]2NC[C@@H](O)COC[C@H]2O1	CID:54657481	phase I
BRD-K82669795	COC(=O)C[C@H]1CC[C@@H]2NC[C@H](O)COC[C@H]2O1	CID:54657482	phase I
BRD-K79199685	COC(=O)C[C@@H]1CC[C@H]2NC[C@H](O)COC[C@@H]2O1	CID:54657483	phase I
BRD-K68614469	COC(=O)C[C@@H]1CC[C@@H]2NC[C@H](O)COC[C@H]2O1	CID:54657484	phase I
BRD-K64622657	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2CC2CCOCC2)O1	CID:54657485	phase I
BRD-K77786391	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2CC2CCOCC2)O1	CID:54657486	phase I
BRD-K19971276	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2CC2CCOCC2)O1	CID:54657487	phase I
BRD-K61284851	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2CC2CCOCC2)O1	CID:54657488	phase I
BRD-K84240784	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2CC2CCOCC2)O1	CID:54657489	phase I
BRD-K05856102	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2CC2CCOCC2)O1	CID:54657490	phase I
BRD-K83859302	Cc1noc(C)c1NC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]12	CID:54657491	phase I
BRD-K50716931	Cc1noc(C)c1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]12	CID:54657492	phase I
BRD-K74894470	Cc1noc(C)c1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]12	CID:54657493	phase I
BRD-K03568952	O[C@H]1COC[C@H]2O[C@@H](CC(=O)Nc3nccs3)CC[C@@H]2N(Cc2cc(F)cc(F)c2)C1	CID:54657494	phase I
BRD-K51068004	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)Nc3nccs3)CC[C@H]2N(Cc2cc(F)cc(F)c2)C1	CID:54657497	phase I
BRD-K98054202	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)Nc3nccs3)CC[C@H]2N(Cc2cc(F)cc(F)c2)C1	CID:54657498	phase I
BRD-K80278608	O[C@@H]1COC[C@H]2O[C@H](CC(=O)Nc3nccs3)CC[C@@H]2N(Cc2cc(F)cc(F)c2)C1	CID:54657499	phase I
BRD-K13883913	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)Nc3nccs3)CC[C@@H]2N(Cc2cc(F)cc(F)c2)C1	CID:54657500	phase I
BRD-K84455184	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)Nc3nccs3)CC[C@H]2N(Cc2cc(F)cc(F)c2)C1	CID:54657501	phase I
BRD-K14206468	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NC3CCCC3)CC[C@@H]2N(C1)C(=O)c1ccc2OCOc2c1	CID:54657502	phase I
BRD-K27915767	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCCC3)CC[C@H]2N(C1)C(=O)c1ccc2OCOc2c1	CID:54657503	phase I
BRD-K08616215	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NC3CCCC3)CC[C@H]2N(C1)C(=O)c1ccc2OCOc2c1	CID:54657504	phase I
BRD-K53187535	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCCC3)CC[C@H]2N(C1)C(=O)c1ccc2OCOc2c1	CID:54657505	phase I
BRD-K84636160	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NC3CCCC3)CC[C@@H]2N(C1)C(=O)c1ccc2OCOc2c1	CID:54657506	phase I
BRD-K96640402	Cn1cnc(CCNC(=O)C[C@@H]2CC[C@@H]3[C@H](COC[C@@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657507	phase I
BRD-K92656786	Cn1cnc(CCNC(=O)C[C@@H]2CC[C@@H]3[C@H](COC[C@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657508	phase I
BRD-K04574057	Cn1cnc(CCNC(=O)C[C@@H]2CC[C@H]3[C@@H](COC[C@@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657509	phase I
BRD-K88821227	Cn1cnc(CCNC(=O)C[C@@H]2CC[C@H]3[C@@H](COC[C@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657510	phase I
BRD-K51256476	Cn1cnc(CCNC(=O)C[C@H]2CC[C@H]3[C@@H](COC[C@@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657511	phase I
BRD-K39481055	Cn1cnc(CCNC(=O)C[C@H]2CC[C@@H]3[C@H](COC[C@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657512	phase I
BRD-K29326853	Cn1cnc(CCNC(=O)C[C@H]2CC[C@@H]3[C@H](COC[C@@H](O)CN3C(=O)Nc3ccc(cc3)C(F)(F)F)O2)c1	CID:54657513	phase I
BRD-K89010697	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657514	phase I
BRD-K26193607	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657515	phase I
BRD-K22787051	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657516	phase I
BRD-K11359987	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657517	phase I
BRD-K60637442	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657518	phase I
BRD-K94222931	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657519	phase I
BRD-K77774562	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657520	phase I
BRD-K52207968	CCCNC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(O)=O)CC[C@@H]12	CID:54657521	phase I
BRD-K62995317	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(O)=O)CC[C@H]12	CID:54657522	phase I
BRD-K17750548	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(O)=O)CC[C@H]12	CID:54657523	phase I
BRD-K47574438	CCCNC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(O)=O)CC[C@@H]12	CID:54657524	phase I
BRD-K32330804	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657525	phase I
BRD-K06619089	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657526	phase I
BRD-K29286627	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657527	phase I
BRD-K97595524	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657528	phase I
BRD-K83390709	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657529	phase I
BRD-K80223377	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657530	phase I
BRD-K70852733	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657531	phase I
BRD-K79260617	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657532	phase I
BRD-K03448064	C[C@@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657533	phase I
BRD-K51759637	C[C@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657534	phase I
BRD-K18238232	C[C@@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657535	phase I
BRD-K01055635	C[C@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657536	phase I
BRD-K30837577	C[C@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657537	phase I
BRD-K07164057	C[C@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657538	phase I
BRD-K91771673	C[C@@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657539	phase I
BRD-K43649826	C[C@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657540	phase I
BRD-K42986817	C[C@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657541	phase I
BRD-K27161555	C[C@@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657542	phase I
BRD-K12484704	C[C@@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657543	phase I
BRD-K91143067	C[C@@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657544	phase I
BRD-K43421680	C[C@@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657545	phase I
BRD-K35371149	C[C@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657546	phase I
BRD-K85322309	C[C@@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657547	phase I
BRD-K09292709	C[C@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2cccc(Cl)c2)O1)c1ccccc1	CID:54657548	phase I
BRD-K29253390	COC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657549	phase I
BRD-K48035058	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657550	phase I
BRD-K77287734	COC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657551	phase I
BRD-K09542523	COC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657552	phase I
BRD-K24932095	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657553	phase I
BRD-K75455321	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657554	phase I
BRD-K64418359	COC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657555	phase I
BRD-K75416754	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2cn(C)cn2)O1	CID:54657556	phase I
BRD-K48360530	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1cccc(Cl)c1	CID:54657557	phase I
BRD-K06161868	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1cccc(Cl)c1	CID:54657558	phase I
BRD-K88617912	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1cccc(Cl)c1	CID:54657559	phase I
BRD-K44420259	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1cccc(Cl)c1	CID:54657560	phase I
BRD-K65988431	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1cccc(Cl)c1	CID:54657561	phase I
BRD-K55596430	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1cccc(Cl)c1	CID:54657562	phase I
BRD-K60994920	COc1ccc(CN2C[C@@H](O)COC[C@@H]3O[C@@H](CC(=O)NCCN4CCCC4)CC[C@@H]23)cc1	CID:54657563	phase I
BRD-K63072081	COc1ccc(CN2C[C@H](O)COC[C@H]3O[C@@H](CC(=O)NCCN4CCCC4)CC[C@H]23)cc1	CID:54657564	phase I
BRD-K64873832	COc1ccc(CN2C[C@H](O)COC[C@@H]3O[C@H](CC(=O)NCCN4CCCC4)CC[C@@H]23)cc1	CID:54657565	phase I
BRD-K76369294	COc1ccc(CN2C[C@@H](O)COC[C@@H]3O[C@H](CC(=O)NCCN4CCCC4)CC[C@@H]23)cc1	CID:54657566	phase I
BRD-K25159388	COc1ccc(CN2C[C@H](O)COC[C@H]3O[C@H](CC(=O)NCCN4CCCC4)CC[C@H]23)cc1	CID:54657567	phase I
BRD-K18639483	COc1ccc(CN2C[C@@H](O)COC[C@H]3O[C@@H](CC(=O)NCCN4CCCC4)CC[C@H]23)cc1	CID:54657568	phase I
BRD-K52662613	COc1ccc(CN2C[C@@H](O)COC[C@H]3O[C@H](CC(=O)NCCN4CCCC4)CC[C@H]23)cc1	CID:54657569	phase I
BRD-K24717178	COc1ccc(CN2C[C@H](O)COC[C@@H]3O[C@@H](CC(=O)NCCN4CCCC4)CC[C@@H]23)cc1	CID:54657570	phase I
BRD-K58856256	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]2N(Cc2cocn2)C1	CID:54657571	phase I
BRD-K28636199	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@H]2N(C1)C(=O)c1ccccc1	CID:54657572	phase I
BRD-K24769439	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@H]2N(C1)C(=O)c1ccccc1	CID:54657573	phase I
BRD-K50868745	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]2N(C1)C(=O)c1ccccc1	CID:54657574	phase I
BRD-K31415071	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]2N(C1)C(=O)c1ccccc1	CID:54657575	phase I
BRD-K93852877	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@H]2N(C1)C(=O)c1ccccc1	CID:54657576	phase I
BRD-K65240553	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]2N(C1)C(=O)c1ccccc1	CID:54657577	phase I
BRD-K82234732	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657578	phase I
BRD-K99103407	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657579	phase I
BRD-K13693445	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657580	phase I
BRD-K35158088	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657581	phase I
BRD-K78316354	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657582	phase I
BRD-K97981711	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657583	phase I
BRD-K14886982	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657584	phase I
BRD-K58475709	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@@H]2N(Cc2cccc(c2)-c2ccncc2)C1	CID:54657585	phase I
BRD-K45375659	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COC1	CID:54657586	phase I
BRD-K28883735	O[C@@H]1CN[C@@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COC1	CID:54657587	phase I
BRD-K42142217	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COC1	CID:54657588	phase I
BRD-K80686274	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COC1	CID:54657589	phase I
BRD-K01971712	O[C@@H]1CN[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COC1	CID:54657590	phase I
BRD-K54179080	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COC1	CID:54657591	phase I
BRD-K50186544	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)NCc3ccc4OCOc4c3)O[C@H]2COC1	CID:54657592	phase I
BRD-K55561254	O[C@H]1CN[C@H]2CC[C@H](CC(=O)NCc3ccc4OCOc4c3)O[C@@H]2COC1	CID:54657593	phase I
BRD-K90431990	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]12	CID:54657594	phase I
BRD-K07269289	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]12	CID:54657595	phase I
BRD-K05543055	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]12	CID:54657596	phase I
BRD-K59340545	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]12	CID:54657597	phase I
BRD-K96555842	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]12	CID:54657598	phase I
BRD-K48306168	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]12	CID:54657599	phase I
BRD-K67655178	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]12	CID:54657600	phase I
BRD-K18542345	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]12	CID:54657601	phase I
BRD-K10211010	O[C@@H]1COC[C@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657602	phase I
BRD-K43570134	O[C@H]1COC[C@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657603	phase I
BRD-K63000292	O[C@H]1COC[C@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657604	phase I
BRD-K47551852	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657605	phase I
BRD-K76352755	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657606	phase I
BRD-K31224309	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657607	phase I
BRD-K92795064	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657608	phase I
BRD-K71504944	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54657609	phase I
BRD-K09388341	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cc(F)ccc2F)C1	CID:54657610	phase I
BRD-K38797319	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cc(F)ccc2F)C1	CID:54657611	phase I
BRD-K12411600	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@@H]2N(Cc2cc(F)ccc2F)C1	CID:54657612	phase I
BRD-K49998237	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@@H]2N(Cc2cc(F)ccc2F)C1	CID:54657613	phase I
BRD-K63818532	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cc(F)ccc2F)C1	CID:54657614	phase I
BRD-K35558120	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@@H]2N(Cc2cc(F)ccc2F)C1	CID:54657615	phase I
BRD-K66356233	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cc(F)ccc2F)C1	CID:54657616	phase I
BRD-K26583430	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)C2CCCC2)O1	CID:54657617	phase I
BRD-K89885223	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)C2CCCC2)O1	CID:54657618	phase I
BRD-K49070267	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)C2CCCC2)O1	CID:54657619	phase I
BRD-K68148111	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)C2CCCC2)O1	CID:54657620	phase I
BRD-K64136010	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)C2CCCC2)O1	CID:54657621	phase I
BRD-K15804688	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)C2CCCC2)O1	CID:54657622	phase I
BRD-K58033375	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)C2CCCC2)O1	CID:54657623	phase I
BRD-K06470746	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccncc3)CC[C@H]2N(C1)C(=O)CCN1CCCCC1	CID:54657624	phase I
BRD-K63933178	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NC3Cc4ccccc4C3)CC[C@@H]2N(C1)C(=O)Cc1ccccc1	CID:54657625	phase I
BRD-K04745699	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3Cc4ccccc4C3)CC[C@@H]2N(C1)C(=O)Cc1ccccc1	CID:54657626	phase I
BRD-K49283955	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NC3Cc4ccccc4C3)CC[C@H]2N(C1)C(=O)Cc1ccccc1	CID:54657627	phase I
BRD-K24855340	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NC3Cc4ccccc4C3)CC[C@H]2N(C1)C(=O)Cc1ccccc1	CID:54657628	phase I
BRD-K13757679	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NC3Cc4ccccc4C3)CC[C@H]2N(C1)C(=O)Cc1ccccc1	CID:54657629	phase I
BRD-K65482654	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NC3Cc4ccccc4C3)CC[C@H]2N(C1)C(=O)Cc1ccccc1	CID:54657630	phase I
BRD-K47228813	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NC3Cc4ccccc4C3)CC[C@@H]2N(C1)C(=O)Cc1ccccc1	CID:54657631	phase I
BRD-K23050218	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NC3Cc4ccccc4C3)CC[C@@H]2N(C1)C(=O)Cc1ccccc1	CID:54657632	phase I
BRD-K91729331	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657633	phase I
BRD-K18400716	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657634	phase I
BRD-K23618054	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657635	phase I
BRD-K12388484	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657636	phase I
BRD-K03262953	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657637	phase I
BRD-K65012833	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657638	phase I
BRD-K87838816	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657639	phase I
BRD-K91487294	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54657640	phase I
BRD-K90987254	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657641	phase I
BRD-K02055666	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657642	phase I
BRD-K79615119	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657643	phase I
BRD-K16323731	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657644	phase I
BRD-K85955502	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657645	phase I
BRD-K30684242	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657646	phase I
BRD-K35510956	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657647	phase I
BRD-K33776933	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54657648	phase I
BRD-K04326190	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccncn3)CC[C@H]2N(C1)S(=O)(=O)c1cccc(F)c1	CID:54657649	phase I
BRD-K99902401	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccncn3)CC[C@@H]2N(C1)S(=O)(=O)c1cccc(F)c1	CID:54657650	phase I
BRD-K26631510	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccncn3)CC[C@@H]2N(C1)S(=O)(=O)c1cccc(F)c1	CID:54657651	phase I
BRD-K98945308	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccncn3)CC[C@@H]2N(C1)S(=O)(=O)c1cccc(F)c1	CID:54657652	phase I
BRD-K91686310	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccncn3)CC[C@H]2N(C1)S(=O)(=O)c1cccc(F)c1	CID:54657653	phase I
BRD-K12575545	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657654	phase I
BRD-K74341727	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657655	phase I
BRD-K44925462	COc1ccccc1CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657656	phase I
BRD-K91156247	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657657	phase I
BRD-K11604106	COc1ccccc1CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657658	phase I
BRD-K37849751	COc1ccccc1CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657659	phase I
BRD-K32931486	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)Nc2ccc(F)cc2)O1	CID:54657660	phase I
BRD-K38672372	O[C@H]1COC[C@@H]2O[C@@H](CC(O)=O)CC[C@H]2N(C1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1	CID:54657661	phase I
BRD-K60362139	O[C@H]1COC[C@H]2O[C@@H](CC(O)=O)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1	CID:54657662	phase I
BRD-K78914942	O[C@@H]1COC[C@@H]2O[C@H](CC(O)=O)CC[C@H]2N(C1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1	CID:54657663	phase I
BRD-K61788733	O[C@@H]1COC[C@@H]2O[C@@H](CC(O)=O)CC[C@H]2N(C1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1	CID:54657664	phase I
BRD-K35060373	O[C@H]1COC[C@H]2O[C@H](CC(O)=O)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1	CID:54657665	phase I
BRD-K48624606	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54657666	phase I
BRD-K38126560	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54657667	phase I
BRD-K12365616	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54657668	phase I
BRD-K30697829	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54657669	phase I
BRD-K90871122	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54657670	phase I
BRD-K31566137	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54657671	phase I
BRD-K83826027	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2COC1	CID:54657672	phase I
BRD-K47261397	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2COC1	CID:54657673	phase I
BRD-K80496944	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2COC1	CID:54657674	phase I
BRD-K15752270	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2COC1	CID:54657675	phase I
BRD-K20433775	O[C@H]1CN[C@H]2CC[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2COC1	CID:54657676	phase I
BRD-K28460793	O[C@@H]1CN[C@@H]2CC[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2COC1	CID:54657677	phase I
BRD-K51583960	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@H]2COC1	CID:54657678	phase I
BRD-K03235359	O[C@@H]1CN[C@H]2CC[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)O[C@@H]2COC1	CID:54657679	phase I
BRD-K77909743	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2ccc(Cl)cc2)O1	CID:54657680	phase I
BRD-K97894266	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2ccc(Cl)cc2)O1	CID:54657681	phase I
BRD-K06780475	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@H]2N(Cc2nccs2)C1	CID:54657682	phase I
BRD-K82727027	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]2N(Cc2nccs2)C1	CID:54657683	phase I
BRD-K14758616	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@H]2N(Cc2nccs2)C1	CID:54657684	phase I
BRD-K56764633	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]2N(Cc2nccs2)C1	CID:54657685	phase I
BRD-K02460212	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]2N(Cc2nccs2)C1	CID:54657686	phase I
BRD-K51457407	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]2N(Cc2nccs2)C1	CID:54657687	phase I
BRD-K61260096	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@H]2N(Cc2nccs2)C1	CID:54657688	phase I
BRD-K35468722	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657689	phase I
BRD-K32581454	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657690	phase I
BRD-K03652504	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657691	phase I
BRD-K07339740	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657692	phase I
BRD-K66555347	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657693	phase I
BRD-K26676775	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657694	phase I
BRD-K45356824	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54657695	phase I
BRD-K03669312	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2ccccn2)O1	CID:54657696	phase I
BRD-K09458434	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2ccccn2)O1	CID:54657697	phase I
BRD-K43703651	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2ccccn2)O1	CID:54657698	phase I
BRD-K55875111	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2ccccn2)O1	CID:54657699	phase I
BRD-K04229162	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2ccccn2)O1	CID:54657700	phase I
BRD-K94029810	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2ccccn2)O1	CID:54657701	phase I
BRD-K47752932	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccccn2)O1	CID:54657702	phase I
BRD-K07100440	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccccn2)O1	CID:54657703	phase I
BRD-K44756290	CN1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@H]12	CID:54657704	phase I
BRD-K95545045	CN1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@@H]12	CID:54657705	phase I
BRD-K57087594	CN1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]12	CID:54657706	phase I
BRD-K52577250	CN1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@H]12	CID:54657707	phase I
BRD-K65465954	CN1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@@H]12	CID:54657708	phase I
BRD-K43031910	CN1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]12	CID:54657709	phase I
BRD-K46587586	CN1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]12	CID:54657710	phase I
BRD-K22563530	CN1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]12	CID:54657711	phase I
BRD-K10327449	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54657712	phase I
BRD-K23558120	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]2N(C1)C(=O)c1ccccc1F	CID:54657713	phase I
BRD-K79564569	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54657714	phase I
BRD-K62473229	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]2N(C1)C(=O)c1ccccc1F	CID:54657715	phase I
BRD-K95208083	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]2N(C1)C(=O)c1ccccc1F	CID:54657716	phase I
BRD-K61952473	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54657717	phase I
BRD-K66577472	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54657718	phase I
BRD-K08446710	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]2N(C1)C(=O)c1ccccc1F	CID:54657719	phase I
BRD-K20876879	O[C@@H]1CN[C@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COC1	CID:54657720	phase I
BRD-K84218095	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COC1	CID:54657721	phase I
BRD-K50366616	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@H]2COC1	CID:54657722	phase I
BRD-K75633187	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@H]2COC1	CID:54657723	phase I
BRD-K79064338	O[C@@H]1CN[C@@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@H]2COC1	CID:54657724	phase I
BRD-K26484692	O[C@H]1CN[C@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COC1	CID:54657725	phase I
BRD-K22080587	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)NCCN3CCCCC3)O[C@@H]2COC1	CID:54657726	phase I
BRD-K78483792	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)NCCN3CCCCC3)O[C@H]2COC1	CID:54657727	phase I
BRD-K94390774	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657728	phase I
BRD-K07569193	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657729	phase I
BRD-K84976438	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657730	phase I
BRD-K85605624	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657731	phase I
BRD-K75693278	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657732	phase I
BRD-K64930062	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657733	phase I
BRD-K89986699	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657734	phase I
BRD-K15392449	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54657735	phase I
BRD-K31830150	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54657736	phase I
BRD-K51363657	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cccnc1	CID:54657737	phase I
BRD-K75322905	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54657738	phase I
BRD-K70392319	O[C@@H]1COC[C@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cccnc1	CID:54657739	phase I
BRD-K16964495	O[C@H]1COC[C@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cccnc1	CID:54657740	phase I
BRD-K21572481	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54657741	phase I
BRD-K48945537	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54657742	phase I
BRD-K54546524	Cc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]12	CID:54657743	phase I
BRD-K14302652	Cc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]12	CID:54657744	phase I
BRD-K95154332	Cc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]12	CID:54657745	phase I
BRD-K80169513	Cc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]12	CID:54657746	phase I
BRD-K42677417	Cc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]12	CID:54657747	phase I
BRD-K89958315	Cc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]12	CID:54657748	phase I
BRD-K20197338	Cc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]12	CID:54657749	phase I
BRD-K58560613	Cc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]12	CID:54657750	phase I
BRD-K75368232	CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657751	phase I
BRD-K04701379	CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657752	phase I
BRD-K85797809	CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657753	phase I
BRD-K75813018	CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657754	phase I
BRD-K90163207	CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657755	phase I
BRD-K95567178	CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657756	phase I
BRD-K74671783	CNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657757	phase I
BRD-K24621485	CNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54657758	phase I
BRD-K36130407	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54657759	phase I
BRD-K72502177	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54657760	phase I
BRD-K93880770	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54657761	phase I
BRD-K06891569	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54657762	phase I
BRD-K78487432	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54657763	phase I
BRD-K09203309	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54657764	phase I
BRD-K96625837	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccccc1F	CID:54657765	phase I
BRD-K22052171	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]2N(C1)S(=O)(=O)c1ccccc1F	CID:54657766	phase I
BRD-K51257364	CCC(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@H]12	CID:54657767	phase I
BRD-K95487462	CCC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@@H]12	CID:54657768	phase I
BRD-K53407305	CCC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@H]12	CID:54657769	phase I
BRD-K86755654	CCC(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@H]12	CID:54657770	phase I
BRD-K41120089	CCC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@H]12	CID:54657771	phase I
BRD-K68782403	CCC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@@H]12	CID:54657772	phase I
BRD-K75413841	CCC(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@@H]12	CID:54657773	phase I
BRD-K64285892	CCC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@@H]12	CID:54657774	phase I
BRD-K74553461	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COC1	CID:54657775	phase I
BRD-K41430135	O[C@H]1CN[C@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COC1	CID:54657776	phase I
BRD-K86780816	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COC1	CID:54657777	phase I
BRD-K97194666	O[C@@H]1CN[C@@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COC1	CID:54657778	phase I
BRD-K29953802	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COC1	CID:54657779	phase I
BRD-K70821391	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COC1	CID:54657780	phase I
BRD-K60636255	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)N3CCc4ccccc4C3)O[C@H]2COC1	CID:54657781	phase I
BRD-K44699604	O[C@@H]1CN[C@H]2CC[C@H](CC(=O)N3CCc4ccccc4C3)O[C@@H]2COC1	CID:54657782	phase I
BRD-K83132555	COCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657783	phase I
BRD-K80398603	COCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657784	phase I
BRD-K06083657	COCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657785	phase I
BRD-K32897268	COCCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657786	phase I
BRD-K38643780	COCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657787	phase I
BRD-K99874282	COCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657788	phase I
BRD-K75843415	COCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2cc(Cl)cc(Cl)c2)O1	CID:54657789	phase I
BRD-K20281332	CN(C)CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2CC2CCCC2)O1	CID:54657790	phase I
BRD-K19933506	CN(C)CCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2CC2CCCC2)O1	CID:54657793	phase I
BRD-K05050883	CN(C)CCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2CC2CCCC2)O1	CID:54657794	phase I
BRD-K18767302	CN(C)CCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2CC2CCCC2)O1	CID:54657795	phase I
BRD-K27343142	CN(C)CCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2CC2CCCC2)O1	CID:54657796	phase I
BRD-K02058097	COc1cccc(NC(=O)N2C[C@H](O)COC[C@H]3O[C@@H](CC(=O)N(C)C)CC[C@H]23)c1	CID:54657797	phase I
BRD-K76358141	COc1cccc(NC(=O)N2C[C@@H](O)COC[C@H]3O[C@@H](CC(=O)N(C)C)CC[C@H]23)c1	CID:54657798	phase I
BRD-K70166659	COc1cccc(NC(=O)N2C[C@H](O)COC[C@H]3O[C@H](CC(=O)N(C)C)CC[C@H]23)c1	CID:54657799	phase I
BRD-K08078340	COc1cccc(NC(=O)N2C[C@@H](O)COC[C@@H]3O[C@@H](CC(=O)N(C)C)CC[C@@H]23)c1	CID:54657800	phase I
BRD-K66033125	COc1cccc(NC(=O)N2C[C@@H](O)COC[C@@H]3O[C@H](CC(=O)N(C)C)CC[C@@H]23)c1	CID:54657801	phase I
BRD-K92860459	COc1cccc(NC(=O)N2C[C@H](O)COC[C@@H]3O[C@@H](CC(=O)N(C)C)CC[C@@H]23)c1	CID:54657802	phase I
BRD-K07625901	COc1cccc(NC(=O)N2C[C@H](O)COC[C@@H]3O[C@H](CC(=O)N(C)C)CC[C@@H]23)c1	CID:54657803	phase I
BRD-K51322285	COc1cccc(NC(=O)N2C[C@@H](O)COC[C@H]3O[C@H](CC(=O)N(C)C)CC[C@H]23)c1	CID:54657804	phase I
BRD-K68445037	Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@@H]12	CID:54657805	phase I
BRD-K44029733	Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@H]12	CID:54657806	phase I
BRD-K76624532	Cc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@H]12	CID:54657807	phase I
BRD-K52831370	Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@@H]12	CID:54657808	phase I
BRD-K70861166	Cc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@@H]12	CID:54657809	phase I
BRD-K85930698	Cc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@@H]12	CID:54657810	phase I
BRD-K76665741	Cc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@H]12	CID:54657811	phase I
BRD-K16782389	Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCc3ccc4OCOc4c3)CC[C@H]12	CID:54657812	phase I
BRD-K94708051	O[C@H]1CN[C@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@@H]2COC1	CID:54657815	phase I
BRD-K02189204	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COC1	CID:54657816	phase I
BRD-K01202062	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@@H]2COC1	CID:54657817	phase I
BRD-K43108514	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COC1	CID:54657818	phase I
BRD-K89491100	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)NCCc3ccncc3)O[C@H]2COC1	CID:54657819	phase I
BRD-K43939579	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)NCCc3ccncc3)O[C@H]2COC1	CID:54657820	phase I
BRD-K40358966	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]2N(Cc2nccs2)C1	CID:54657821	phase I
BRD-K98668154	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]2N(Cc2nccs2)C1	CID:54657822	phase I
BRD-K19405573	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]2N(Cc2nccs2)C1	CID:54657823	phase I
BRD-K58439833	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]2N(Cc2nccs2)C1	CID:54657824	phase I
BRD-K88967430	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]2N(Cc2nccs2)C1	CID:54657825	phase I
BRD-K91758467	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]2N(Cc2nccs2)C1	CID:54657826	phase I
BRD-K89412540	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@@H]2N(Cc2nccs2)C1	CID:54657827	phase I
BRD-K06217925	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCC(Cc4ccccc4)CC3)CC[C@H]2N(Cc2nccs2)C1	CID:54657828	phase I
BRD-K38290133	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@H]2N(Cc2ccccc2F)C1	CID:54657829	phase I
BRD-K02222982	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]2N(Cc2ccccc2F)C1	CID:54657830	phase I
BRD-K96044609	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(Cc2ccccc2F)C1	CID:54657831	phase I
BRD-K71540580	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@H]2N(Cc2ccccc2F)C1	CID:54657832	phase I
BRD-K74428993	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@@H]2N(Cc2ccccc2F)C1	CID:54657833	phase I
BRD-K70617194	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(Cc2ccccc2F)C1	CID:54657834	phase I
BRD-K50171542	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@@H]2N(Cc2ccccc2F)C1	CID:54657835	phase I
BRD-K84391460	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]2N(Cc2ccccc2F)C1	CID:54657836	phase I
BRD-K50120786	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657837	phase I
BRD-K38210246	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657838	phase I
BRD-K33610498	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657839	phase I
BRD-K02322717	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657840	phase I
BRD-K07323881	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657841	phase I
BRD-K80806285	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657842	phase I
BRD-K03077507	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657843	phase I
BRD-K08247301	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(F)cc1	CID:54657844	phase I
BRD-K79490177	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657845	phase I
BRD-K58514045	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657846	phase I
BRD-K07572455	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657847	phase I
BRD-K97048125	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657848	phase I
BRD-K17139153	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657849	phase I
BRD-K06714535	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657850	phase I
BRD-K32882027	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657851	phase I
BRD-K41354272	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657852	phase I
BRD-K99615821	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657853	phase I
BRD-K63827443	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657854	phase I
BRD-K24133356	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657855	phase I
BRD-K36424197	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657856	phase I
BRD-K69548259	COc1ccc(cc1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657857	phase I
BRD-K07790303	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657858	phase I
BRD-K12858756	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54657859	phase I
BRD-K08936794	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54657860	phase I
BRD-K64619734	COCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2F)O1	CID:54657861	phase I
BRD-K14385562	COCCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2F)O1	CID:54657862	phase I
BRD-K07634536	COCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2F)O1	CID:54657863	phase I
BRD-K49283005	COCCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2F)O1	CID:54657864	phase I
BRD-K72352929	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657865	phase I
BRD-K72109199	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657866	phase I
BRD-K10844902	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657867	phase I
BRD-K76729250	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657868	phase I
BRD-K62455331	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657869	phase I
BRD-K20978396	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657870	phase I
BRD-K69178842	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657871	phase I
BRD-K45077070	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@@H]2N(C1)C(=O)Nc1cc(Cl)cc(Cl)c1	CID:54657872	phase I
BRD-K76637414	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657873	phase I
BRD-K81666293	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657874	phase I
BRD-K15535200	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657875	phase I
BRD-K30737452	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657876	phase I
BRD-K09936924	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657877	phase I
BRD-K43982847	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(C1)C(=O)c1cnccn1	CID:54657878	phase I
BRD-K44080306	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657879	phase I
BRD-K56805970	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(C1)C(=O)c1cnccn1	CID:54657880	phase I
BRD-K55009937	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@H]12	CID:54657881	phase I
BRD-K25963301	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]12	CID:54657882	phase I
BRD-K27798440	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@H]12	CID:54657883	phase I
BRD-K86265052	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]12	CID:54657884	phase I
BRD-K00411687	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]12	CID:54657885	phase I
BRD-K67983441	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@@H]12	CID:54657886	phase I
BRD-K88602713	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@H]12	CID:54657887	phase I
BRD-K61415682	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCCCN3CCOCC3)CC[C@H]12	CID:54657888	phase I
BRD-K88607897	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccncn3)CC[C@H]2N(C1)C(=O)Nc1ccccc1	CID:54657889	phase I
BRD-K78023266	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccncn3)CC[C@H]2N(C1)C(=O)Nc1ccccc1	CID:54657890	phase I
BRD-K88361133	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccncn3)CC[C@H]2N(C1)C(=O)Nc1ccccc1	CID:54657891	phase I
BRD-K29785053	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccncn3)CC[C@@H]2N(C1)C(=O)Nc1ccccc1	CID:54657892	phase I
BRD-K43862194	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccncn3)CC[C@@H]2N(C1)C(=O)Nc1ccccc1	CID:54657893	phase I
BRD-K49525301	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657894	phase I
BRD-K60298771	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657895	phase I
BRD-K71278614	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657896	phase I
BRD-K72217541	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657897	phase I
BRD-K99149118	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657898	phase I
BRD-K74548617	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657899	phase I
BRD-K96047861	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@@H]2N(CCC(F)(F)F)C1	CID:54657900	phase I
BRD-K31369513	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@H]2N(CCC(F)(F)F)C1	CID:54657901	phase I
BRD-K90305015	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(C1)C(=O)c1cc(Cl)cc(Cl)c1	CID:54657902	phase I
BRD-K92754298	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(C1)C(=O)c1cc(Cl)cc(Cl)c1	CID:54657903	phase I
BRD-K08377525	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(C1)C(=O)c1cc(Cl)cc(Cl)c1	CID:54657904	phase I
BRD-K56328447	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(C1)C(=O)c1cc(Cl)cc(Cl)c1	CID:54657905	phase I
BRD-K35400569	O[C@H]1CN[C@H]2CC[C@H](CC(=O)Nc3nccs3)O[C@@H]2COC1	CID:54657906	phase I
BRD-K59867372	O[C@@H]1CN[C@@H]2CC[C@H](CC(=O)Nc3nccs3)O[C@H]2COC1	CID:54657907	phase I
BRD-K15377376	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)Nc3nccs3)O[C@H]2COC1	CID:54657908	phase I
BRD-K97196700	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)Nc3nccs3)O[C@H]2COC1	CID:54657909	phase I
BRD-K26862321	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)Nc3nccs3)O[C@@H]2COC1	CID:54657910	phase I
BRD-K86619642	O[C@@H]1CN[C@H]2CC[C@H](CC(=O)Nc3nccs3)O[C@@H]2COC1	CID:54657911	phase I
BRD-K33909884	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)Nc3nccs3)O[C@@H]2COC1	CID:54657912	phase I
BRD-K04025047	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)Nc3nccs3)O[C@H]2COC1	CID:54657913	phase I
BRD-K70663894	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657914	phase I
BRD-K38405570	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657915	phase I
BRD-K87838487	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657916	phase I
BRD-K27744061	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657917	phase I
BRD-K15966733	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657918	phase I
BRD-K23154136	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657919	phase I
BRD-K62836482	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657920	phase I
BRD-K54327934	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)C2CCOCC2)O1	CID:54657921	phase I
BRD-K39988373	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657922	phase I
BRD-K86671899	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657923	phase I
BRD-K26041656	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657924	phase I
BRD-K19190776	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657925	phase I
BRD-K94646939	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657926	phase I
BRD-K55313038	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657927	phase I
BRD-K53181055	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657928	phase I
BRD-K95917977	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)c(Cl)c1	CID:54657929	phase I
BRD-K83600073	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657930	phase I
BRD-K24058148	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657931	phase I
BRD-K00224166	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657932	phase I
BRD-K29528387	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657933	phase I
BRD-K59725859	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657934	phase I
BRD-K50887310	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657935	phase I
BRD-K15230829	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657936	phase I
BRD-K83391808	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2ccccc2F)O1	CID:54657937	phase I
BRD-K44482328	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(Cc2cccc(Cl)c2)C1	CID:54657938	phase I
BRD-K71100175	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(Cc2cccc(Cl)c2)C1	CID:54657939	phase I
BRD-K94509791	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(Cc2cccc(Cl)c2)C1	CID:54657940	phase I
BRD-K02522894	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(Cc2cccc(Cl)c2)C1	CID:54657941	phase I
BRD-K51774400	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(Cc2cccc(Cl)c2)C1	CID:54657942	phase I
BRD-K29642180	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(Cc2cccc(Cl)c2)C1	CID:54657943	phase I
BRD-K63532493	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(Cc2cccc(Cl)c2)C1	CID:54657944	phase I
BRD-K37551767	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CCCCC3)CC[C@H]2N(Cc2cccc(Cl)c2)C1	CID:54657945	phase I
BRD-K25940840	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2ccncc2)O1	CID:54657946	phase I
BRD-K19995388	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2ccncc2)O1	CID:54657947	phase I
BRD-K14854082	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2ccncc2)O1	CID:54657948	phase I
BRD-K41540007	CN(C)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2C(=O)c2ccncc2)O1	CID:54657949	phase I
BRD-K68780601	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccncc2)O1	CID:54657950	phase I
BRD-K80852934	CN(C)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)c2ccncc2)O1	CID:54657951	phase I
BRD-K33490627	CN(C)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C(=O)c2ccncc2)O1	CID:54657952	phase I
BRD-K68749296	CN(C)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccncc2)O1	CID:54657953	phase I
BRD-K96569047	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@@H]12	CID:54657954	phase I
BRD-K23033683	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@@H]12	CID:54657955	phase I
BRD-K95204731	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@H]12	CID:54657956	phase I
BRD-K40219191	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@H]12	CID:54657957	phase I
BRD-K80559952	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@H]12	CID:54657958	phase I
BRD-K63987424	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@H]12	CID:54657959	phase I
BRD-K42207609	COc1ccccc1NC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCCc3ccncc3)CC[C@@H]12	CID:54657960	phase I
BRD-K97585006	COc1ccccc1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@@H]12	CID:54657961	phase I
BRD-K85616320	Cc1noc(C)c1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@@H]12	CID:54657962	phase I
BRD-K85932041	Cc1noc(C)c1NC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCC3CC3)CC[C@@H]12	CID:54657963	phase I
BRD-K24578841	Cc1noc(C)c1NC(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@H]12	CID:54657964	phase I
BRD-K99547414	Cc1noc(C)c1NC(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCC3CC3)CC[C@H]12	CID:54657965	phase I
BRD-K95650611	Cc1noc(C)c1NC(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCC3CC3)CC[C@@H]12	CID:54657966	phase I
BRD-K56864693	Cc1noc(C)c1NC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@H]12	CID:54657967	phase I
BRD-K80408519	Cc1noc(C)c1NC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCC3CC3)CC[C@H]12	CID:54657968	phase I
BRD-K98956791	Cc1noc(C)c1NC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@@H]12	CID:54657969	phase I
BRD-K23589333	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@H]2N(Cc2cocn2)C1	CID:54657970	phase I
BRD-K58679238	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(Cc2cocn2)C1	CID:54657971	phase I
BRD-K56763965	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:54657972	phase I
BRD-K83016905	COC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:54657973	phase I
BRD-K36962815	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:54657974	phase I
BRD-K22508185	COC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:54657975	phase I
BRD-K07157902	COC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:54657976	phase I
BRD-K88797027	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2OC)O1	CID:54657977	phase I
BRD-K10578928	COc1ccccc1CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657978	phase I
BRD-K62734359	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657979	phase I
BRD-K03601317	COc1ccccc1CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657980	phase I
BRD-K00113100	COc1ccccc1CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657981	phase I
BRD-K46065939	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657982	phase I
BRD-K79437423	COc1ccccc1CNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657983	phase I
BRD-K13983359	COc1ccccc1CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657984	phase I
BRD-K16724492	COc1ccccc1CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2cccc(c2)-c2ccncc2)O1	CID:54657985	phase I
BRD-K88786596	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2cccc(F)c2)O1	CID:54657986	phase I
BRD-K17906992	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2cccc(F)c2)O1	CID:54657987	phase I
BRD-K72620090	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2cccc(F)c2)O1	CID:54657988	phase I
BRD-K31920348	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2cccc(F)c2)O1	CID:54657989	phase I
BRD-K95021846	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2cccc(F)c2)O1	CID:54657990	phase I
BRD-K67058688	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2cccc(F)c2)O1	CID:54657991	phase I
BRD-K95328825	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2cccc(F)c2)O1	CID:54657992	phase I
BRD-K80741006	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657993	phase I
BRD-K07522124	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657994	phase I
BRD-K12279187	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657995	phase I
BRD-K93487374	CN1CCN(CC1)C(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657996	phase I
BRD-K57502578	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657997	phase I
BRD-K75732649	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657998	phase I
BRD-K00549983	CN1CCN(CC1)C(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54657999	phase I
BRD-K13782405	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2C)O1	CID:54658000	phase I
BRD-K53912655	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@@H]2N(CC2CCOCC2)C1	CID:54658001	phase I
BRD-K02217114	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@H]2N(CC2CCOCC2)C1	CID:54658002	phase I
BRD-K30199293	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCC3CC3)CC[C@@H]2N(CC2CCOCC2)C1	CID:54658003	phase I
BRD-K01607762	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CC3)CC[C@H]2N(CC2CCOCC2)C1	CID:54658004	phase I
BRD-K63270290	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@@H]2N(CC2CCOCC2)C1	CID:54658005	phase I
BRD-K65909937	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCC3CC3)CC[C@H]2N(CC2CCOCC2)C1	CID:54658006	phase I
BRD-K64391475	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCC3CC3)CC[C@@H]2N(CC2CCOCC2)C1	CID:54658007	phase I
BRD-K75425370	Cn1cnc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@H]12	CID:54658008	phase I
BRD-K29957577	Cn1cnc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]12	CID:54658009	phase I
BRD-K72772617	Cn1cnc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]12	CID:54658010	phase I
BRD-K61997144	Cn1cnc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]12	CID:54658011	phase I
BRD-K38870294	Cn1cnc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]12	CID:54658012	phase I
BRD-K75639577	Cn1cnc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@H]12	CID:54658013	phase I
BRD-K30270755	Cn1cnc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@H]12	CID:54658014	phase I
BRD-K42709418	Cn1cnc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@H]12	CID:54658015	phase I
BRD-K38232832	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]12	CID:54658016	phase I
BRD-K57754556	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]12	CID:54658017	phase I
BRD-K72780683	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]12	CID:54658018	phase I
BRD-K39447340	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]12	CID:54658019	phase I
BRD-K70003473	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]12	CID:54658020	phase I
BRD-K15793745	COc1cccc(c1)S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]12	CID:54658021	phase I
BRD-K56865671	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]12	CID:54658022	phase I
BRD-K23680395	COc1cccc(c1)S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]12	CID:54658023	phase I
BRD-K90680884	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCCN3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658024	phase I
BRD-K49634971	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCCN3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658025	phase I
BRD-K90141430	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCCN3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658026	phase I
BRD-K41389876	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCCN3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658027	phase I
BRD-K24123159	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCCN3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658028	phase I
BRD-K14395166	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCN3CCCCC3)CC[C@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658029	phase I
BRD-K73166612	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCCN3CCCCC3)CC[C@@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54658030	phase I
BRD-K72980353	O[C@H]1CN[C@@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COC1	CID:54658031	phase I
BRD-K13448237	O[C@H]1CN[C@@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COC1	CID:54658032	phase I
BRD-K70200040	O[C@@H]1CN[C@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COC1	CID:54658033	phase I
BRD-K21904592	O[C@@H]1CN[C@@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COC1	CID:54658034	phase I
BRD-K96707310	O[C@H]1CN[C@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COC1	CID:54658035	phase I
BRD-K89692527	O[C@H]1CN[C@H]2CC[C@@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COC1	CID:54658036	phase I
BRD-K32345392	O[C@@H]1CN[C@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@@H]2COC1	CID:54658037	phase I
BRD-K89266502	O[C@@H]1CN[C@@H]2CC[C@H](CC(=O)NC3Cc4ccccc4C3)O[C@H]2COC1	CID:54658038	phase I
BRD-K72150200	Cc1ccccc1S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]12	CID:54658039	phase I
BRD-K49512493	Cc1ccccc1S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@H]12	CID:54658040	phase I
BRD-K58945843	Cc1ccccc1S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@H]12	CID:54658041	phase I
BRD-K65657366	Cc1ccccc1S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@H]12	CID:54658042	phase I
BRD-K67697926	Cc1ccccc1S(=O)(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@H]12	CID:54658043	phase I
BRD-K50131741	Cc1ccccc1S(=O)(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]12	CID:54658044	phase I
BRD-K60595380	Cc1ccccc1S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]12	CID:54658045	phase I
BRD-K47284302	Cc1ccccc1S(=O)(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)NCc3ccccc3Cl)CC[C@@H]12	CID:54658046	phase I
BRD-K73627655	COC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2CCC(F)(F)F)O1	CID:54658047	phase I
BRD-K86162390	COC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2CCC(F)(F)F)O1	CID:54658048	phase I
BRD-K18351060	COC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2CCC(F)(F)F)O1	CID:54658049	phase I
BRD-K98036459	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2CCC(F)(F)F)O1	CID:54658050	phase I
BRD-K01383339	COC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2CCC(F)(F)F)O1	CID:54658051	phase I
BRD-K08371414	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2CCC(F)(F)F)O1	CID:54658052	phase I
BRD-K18456137	COC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2CCC(F)(F)F)O1	CID:54658053	phase I
BRD-K54652275	COC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2CCC(F)(F)F)O1	CID:54658054	phase I
BRD-K61881697	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccncc2)O1	CID:54658055	phase I
BRD-K48710616	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccncc2)O1	CID:54658056	phase I
BRD-K43851624	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccncc2)O1	CID:54658057	phase I
BRD-K66775134	CCNC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccncc2)O1	CID:54658058	phase I
BRD-K46965430	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccncc2)O1	CID:54658059	phase I
BRD-K03222452	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccncc2)O1	CID:54658060	phase I
BRD-K44787412	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccncc2)O1	CID:54658061	phase I
BRD-K47303556	CCNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccncc2)O1	CID:54658062	phase I
BRD-K63164430	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(CC2CCCCC2)C1	CID:54658063	phase I
BRD-K43283393	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(CC2CCCCC2)C1	CID:54658064	phase I
BRD-K70653194	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(CC2CCCCC2)C1	CID:54658065	phase I
BRD-K74702716	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(CC2CCCCC2)C1	CID:54658066	phase I
BRD-K42140123	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(CC2CCCCC2)C1	CID:54658067	phase I
BRD-K93301765	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(F)cc3)CC[C@@H]2N(CC2CCCCC2)C1	CID:54658068	phase I
BRD-K58958454	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCCc3ccccc3)CC[C@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658069	phase I
BRD-K89631978	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658070	phase I
BRD-K45595662	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658071	phase I
BRD-K99647384	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658072	phase I
BRD-K28738449	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCCc3ccccc3)CC[C@@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658073	phase I
BRD-K33778189	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658074	phase I
BRD-K16422757	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCCc3ccccc3)CC[C@@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658075	phase I
BRD-K25471349	CCCNC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658076	phase I
BRD-K41404328	CCCNC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658077	phase I
BRD-K03445781	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658078	phase I
BRD-K00918977	CCCNC(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658079	phase I
BRD-K70631162	CCCNC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658080	phase I
BRD-K94243176	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658081	phase I
BRD-K82154894	CCCNC(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658082	phase I
BRD-K66299073	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658083	phase I
BRD-K52203672	CCCNC(=O)N1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658084	phase I
BRD-K65418120	CCCNC(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658085	phase I
BRD-K13626871	CCCNC(=O)N1C[C@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658086	phase I
BRD-K56130969	CCCNC(=O)N1C[C@@H](O)COC[C@@H]2O[C@@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658087	phase I
BRD-K34392222	CCCNC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658088	phase I
BRD-K24781398	CCCNC(=O)N1C[C@@H](O)COC[C@@H]2O[C@H](CC(=O)N[C@@H]3CCN(Cc4ccccc4)C3)CC[C@@H]12	CID:54658089	phase I
BRD-K73082254	CCCNC(=O)N1C[C@@H](O)COC[C@H]2O[C@@H](CC(=O)N[C@H]3CCN(Cc4ccccc4)C3)CC[C@H]12	CID:54658090	phase I
BRD-K32655366	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658091	phase I
BRD-K76665419	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658092	phase I
BRD-K20763692	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658093	phase I
BRD-K41579429	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658094	phase I
BRD-K89644093	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658095	phase I
BRD-K56535275	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658096	phase I
BRD-K70797508	O[C@@H]1COC[C@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658097	phase I
BRD-K41723088	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCCCC3)CC[C@H]2N(Cc2ccc3OCOc3c2)C1	CID:54658098	phase I
BRD-K83341069	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54658099	phase I
BRD-K06418154	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(C1)C(=O)c1ccncc1	CID:54658100	phase I
BRD-K71650306	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(C1)C(=O)c1ccncc1	CID:54658101	phase I
BRD-K76436920	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(C1)C(=O)c1ccncc1	CID:54658102	phase I
BRD-K04630954	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54658103	phase I
BRD-K65927786	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(C1)C(=O)c1ccncc1	CID:54658104	phase I
BRD-K16034108	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54658105	phase I
BRD-K90546933	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3cccc(F)c3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54658106	phase I
BRD-K37916557	CN1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]12	CID:54658117	phase I
BRD-K83316435	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NC3Cc4ccccc4C3)CC[C@@H]2N(C1)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54658138	phase I
BRD-K21635943	COc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]12	CID:54658174	phase I
BRD-K38763121	C[C@H](NC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2C)O1)c1ccccc1	CID:54658205	phase I
BRD-K26899819	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(Cc2cc(F)ccc2F)C1	CID:54658212	phase I
BRD-K70153099	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2cc(F)ccc2F)C1	CID:54658214	phase I
BRD-K11852206	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2cc(F)ccc2F)C1	CID:54658215	phase I
BRD-K40445382	CCCNC(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]12	CID:54658318	phase I
BRD-K80012633	C[C@@H](NC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1)c1ccccc1	CID:54658324	phase I
BRD-K63947990	C[C@@H](NC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1)c1ccccc1	CID:54658327	phase I
BRD-K84807441	C[C@H](NC(=O)C[C@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1)c1ccccc1	CID:54658330	phase I
BRD-K58696649	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54658402	phase I
BRD-K33005991	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)c1ccncc1	CID:54658423	phase I
BRD-K30055322	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3nccs3)CC[C@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54658437	phase I
BRD-K29649571	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)Nc3nccs3)CC[C@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54658438	phase I
BRD-K29144516	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)Nc3nccs3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54658440	phase I
BRD-K56847293	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54658466	phase I
BRD-K71379723	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54658467	phase I
BRD-K03476588	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54658468	phase I
BRD-K34407242	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54658470	phase I
BRD-K22816026	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@H]2N(C1)C(=O)Nc1ccc(Cl)cc1	CID:54658498	phase I
BRD-K49047615	CCC(=O)N1C[C@H](O)COC[C@@H]2O[C@@H](CC(=O)NC)CC[C@@H]12	CID:54658535	phase I
BRD-K80832690	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(CC2CCOCC2)C1	CID:54658559	phase I
BRD-K83413046	CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2cccnc2)O1	CID:54658632	phase I
BRD-K66638849	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NC3Cc4ccccc4C3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54658651	phase I
BRD-K99775299	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1ccc(F)cc1	CID:54658669	phase I
BRD-K15410616	O[C@@H]1COC[C@@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54658688	phase I
BRD-K87723457	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54658692	phase I
BRD-K48668625	O[C@H]1COC[C@H]2O[C@@H](CC(=O)N3CCN(CC3)c3ccccc3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54658693	phase I
BRD-K34741779	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)c1ccccn1	CID:54658741	phase I
BRD-K07104840	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NC3CCC3)CC[C@H]2N(C1)C(=O)c1ccccn1	CID:54658744	phase I
BRD-K89204222	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(F)cc1	CID:54658765	phase I
BRD-K65600666	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccc(cc2)C(F)(F)F)C1	CID:54658771	phase I
BRD-K94498396	O[C@H]1COC[C@@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@H]2N(Cc2ccc(cc2)C(F)(F)F)C1	CID:54658772	phase I
BRD-K31441680	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658780	phase I
BRD-K45383235	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCc3cccc(F)c3)CC[C@@H]2N(Cc2ccc(Cl)cc2)C1	CID:54658782	phase I
BRD-K48116811	CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2ccc3OCOc3c2)O1	CID:54658802	phase I
BRD-K56758884	CNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2Cc2ccc(cc2)C(F)(F)F)O1	CID:54658832	phase I
BRD-K68702347	CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2S(=O)(=O)c2ccccc2Cl)O1	CID:54658844	phase I
BRD-K65315692	O[C@@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Oc4ccccc4)cc3)CC[C@H]2N(Cc2nccs2)C1	CID:54658855	phase I
BRD-K07921357	COc1ccccc1CNC(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@@H](O)CN2Cc2ccccc2)O1	CID:54658895	phase I
BRD-K26168764	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCC3CC3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54658965	phase I
BRD-K99386687	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54658969	phase I
BRD-K74566474	O[C@@H]1COC[C@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@@H]2N(Cc2ccc(cc2)C(F)(F)F)C1	CID:54658979	phase I
BRD-K41513507	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@H]2N(Cc2ccc(cc2)C(F)(F)F)C1	CID:54658980	phase I
BRD-K62876373	O[C@H]1COC[C@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@@H]2N(Cc2ccc(cc2)C(F)(F)F)C1	CID:54658983	phase I
BRD-K03464662	O[C@H]1COC[C@H]2O[C@@H](CC(=O)NCC3CCCCC3)CC[C@@H]2N(C1)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54659022	phase I
BRD-K70595525	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCCCC3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54659297	phase I
BRD-K02037345	CCCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54659308	phase I
BRD-K67276432	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54659344	phase I
BRD-K16736749	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccc(F)cc2)C1	CID:54659352	phase I
BRD-K12537676	O[C@H]1COC[C@H]2O[C@H](CC(=O)NC3CCC3)CC[C@@H]2N(C1)C(=O)Cc1ccccc1	CID:54659373	phase I
BRD-K19696793	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)N3CCOCC3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54659411	phase I
BRD-K28282859	CN1CCN(CC1)C(=O)C[C@@H]1CC[C@H]2[C@@H](COC[C@H](O)CN2Cc2ccc(Oc3ccccc3)cc2)O1	CID:54659592	phase I
BRD-K91633589	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)S(=O)(=O)c1ccccc1	CID:54659596	phase I
BRD-K41200778	CNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2C(=O)Nc2cccc(OC)c2)O1	CID:54659614	phase I
BRD-K43407019	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54659633	phase I
BRD-K64665684	O[C@H]1COC[C@@H]2O[C@@H](CC[C@H]2N(C1)C(=O)Nc1ccccc1)CC(=O)NCCc1ccncc1	CID:54659755	phase I
BRD-K04021425	COc1ccc(CN2C[C@@H](O)COC[C@H]3O[C@H](CC(=O)N4CCc5ccccc5C4)CC[C@H]23)cc1	CID:54659765	phase I
BRD-K98822179	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccncc3)CC[C@H]2N(Cc2cccc(F)c2)C1	CID:54659792	phase I
BRD-K73444552	Cc1ccc(cc1)S(=O)(=O)N1C[C@H](O)COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@H]12	CID:54659817	phase I
BRD-K30741962	O[C@H]1COC[C@@H]2O[C@@H](CC[C@H]2N(C1)Cc1cccc(C(F)(F)F)c1)CC(=O)NCc1ccncc1	CID:54659868	phase I
BRD-K39657507	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3cc(F)cc(F)c3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54659991	phase I
BRD-K52105642	CCNC(=O)C[C@H]1CC[C@@H]2[C@H](COC[C@@H](O)CN2Cc2ccc(Cl)c(Cl)c2)O1	CID:54660070	phase I
BRD-K05308647	CCCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2ccccn2)O1	CID:54660081	phase I
BRD-K60103096	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(F)cc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54660111	phase I
BRD-K67472330	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccc(Cl)c(Cl)c3)CC[C@@H]2N(C1)S(=O)(=O)c1ccc(Cl)cc1	CID:54660156	phase I
BRD-K70658964	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCCc3ccccc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54660174	phase I
BRD-K06650446	CCNC(=O)C[C@@H]1CC[C@@H]2[C@H](COC[C@H](O)CN2C(=O)c2cccnc2)O1	CID:54660187	phase I
BRD-K97699469	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCOCC3)CC[C@@H]2N(Cc2ccc(Oc3ccccc3)cc2)C1	CID:54660194	phase I
BRD-K71714567	O[C@@H]1COC[C@H]2O[C@@H](CC(=O)NCc3ccccc3)CC[C@@H]2N(C1)C(=O)c1ccccc1F	CID:54660375	phase I
BRD-K49873138	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccccc3)CC[C@H]2N(C1)C(=O)c1cccnc1	CID:54660437	phase I
BRD-K85030001	CN1C[C@@H](O)COC[C@H]2O[C@H](CC(=O)NC3CCCC3)CC[C@H]12	CID:54660558	phase I
BRD-K24383920	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1ccncc1	CID:54660614	phase I
BRD-K31435439	O[C@H]1COC[C@@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@H]2N(C1)C(=O)c1ccccc1	CID:54660617	phase I
BRD-K62122103	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccccc3)CC[C@H]2N(Cc2cccc(c2)C(F)(F)F)C1	CID:54660630	phase I
BRD-K62044515	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)N1CCCCC1)N2Cc1cocn1	CID:54660637	phase I
BRD-K83077741	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)N1CCCCC1)N2Cc1cocn1	CID:54660638	phase I
BRD-K35083768	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H](N2)[C@H]1C(=O)NCCCN1CCOCC1	CID:54660645	phase I
BRD-K85462489	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H](N2)[C@@H]1C(=O)NCCCN1CCOCC1	CID:54660646	phase I
BRD-K69790925	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N[C@H]1C(=O)NC1Cc2ccccc2C1	CID:54660647	phase I
BRD-K26511533	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N[C@@H]1C(=O)NC1Cc2ccccc2C1	CID:54660648	phase I
BRD-K48374441	COCC(=O)N1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCOCC1	CID:54660649	phase I
BRD-K74832096	COCC(=O)N1[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCOCC1	CID:54660650	phase I
BRD-K72072919	CN(C)CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2C(=O)Nc1cc(F)ccc1F	CID:54660651	phase I
BRD-K20790586	CN(C)CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2C(=O)Nc1cc(F)ccc1F	CID:54660652	phase I
BRD-K54219003	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]([C@@H]1C(O)=O)N2C(=O)c1cccnc1	CID:54660653	phase I
BRD-K13870698	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]([C@H]1C(O)=O)N2C(=O)c1cccnc1	CID:54660654	phase I
BRD-K34739003	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@H]2N1CC1CCOCC1	CID:54660655	phase I
BRD-K19938940	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@@H]2N1CC1CCOCC1	CID:54660656	phase I
BRD-K86291677	COc1ccccc1CN1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N(C)C	CID:54660657	phase I
BRD-K85790491	COc1ccccc1CN1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N(C)C	CID:54660658	phase I
BRD-K04058031	CS(=O)(=O)N1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCCCC1	CID:54660667	phase I
BRD-K04291521	CS(=O)(=O)N1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCCCC1	CID:54660668	phase I
BRD-K69344898	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]([C@@H]1C(=O)NCC1CC1)N2Cc1nccs1	CID:54660669	phase I
BRD-K25706980	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]([C@H]1C(=O)NCC1CC1)N2Cc1nccs1	CID:54660670	phase I
BRD-K92439564	Cn1cnc(CCNC(=O)[C@@H]2[C@@H](CO)[C@@H]3Cn4c(cccc4=O)[C@@H]3N2C(=O)Nc2ccccc2)c1	CID:54660671	phase I
BRD-K76028541	Cn1cnc(CCNC(=O)[C@H]2[C@H](CO)[C@H]3Cn4c(cccc4=O)[C@H]3N2C(=O)Nc2ccccc2)c1	CID:54660672	phase I
BRD-K33258928	COc1ccc(cc1)-c1ccc2[C@@H]3N[C@@H]([C@@H](CO)[C@@H]3Cn2c1=O)C(=O)N1CCOCC1	CID:54660673	phase I
BRD-K17223851	COc1ccc(cc1)-c1ccc2[C@H]3N[C@H]([C@H](CO)[C@H]3Cn2c1=O)C(=O)N1CCOCC1	CID:54660674	phase I
BRD-K28027757	COc1cccc(CNC(=O)[C@H]2[C@H](CO)[C@H]3Cn4c(ccc(-c5cncnc5)c4=O)[C@@H]2N3C(C)=O)c1	CID:54660681	phase I
BRD-K48138407	COc1cccc(CNC(=O)[C@@H]2[C@@H](CO)[C@@H]3Cn4c(ccc(-c5cncnc5)c4=O)[C@H]2N3C(C)=O)c1	CID:54660682	phase I
BRD-K64302818	CN(C)C(=O)c1cccc(c1)-c1ccc2[C@@H]3N[C@H](Cn2c1=O)[C@@H](CO)[C@@H]3C(=O)NC1CCC1	CID:54660683	phase I
BRD-K79968414	CN(C)C(=O)c1cccc(c1)-c1ccc2[C@H]3N[C@@H](Cn2c1=O)[C@H](CO)[C@H]3C(=O)NC1CCC1	CID:54660684	phase I
BRD-K22695599	OC[C@H]1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]2N[C@@H]1C(=O)NCCc1ccncc1	CID:54660685	phase I
BRD-K31290914	OC[C@@H]1[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]2N[C@H]1C(=O)NCCc1ccncc1	CID:54660686	phase I
BRD-K04687955	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCc1ccc3OCOc3c1)N2Cc1cccnc1	CID:54660687	phase I
BRD-K07923524	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCc1ccc3OCOc3c1)N2Cc1cccnc1	CID:54660688	phase I
BRD-K97103850	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(Cc2cccc(F)c2)[C@@H]1C(=O)NCC(F)(F)F	CID:54660689	phase I
BRD-K46185480	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(Cc2cccc(F)c2)[C@H]1C(=O)NCC(F)(F)F	CID:54660690	phase I
BRD-K78121324	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]2N([C@@H]1C(O)=O)C(=O)C1CCCCC1	CID:54660691	phase I
BRD-K39550135	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]2N([C@H]1C(O)=O)C(=O)C1CCCCC1	CID:54660692	phase I
BRD-K22177698	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)Nc1nccs1)N2C(=O)C1CCCC1	CID:54660693	phase I
BRD-K28049955	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)Nc1nccs1)N2C(=O)C1CCCC1	CID:54660694	phase I
BRD-K84121492	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]2N1C(=O)c1cnccn1	CID:54660695	phase I
BRD-K83744912	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]2N1C(=O)c1cnccn1	CID:54660696	phase I
BRD-K89226093	C[C@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2CCC(F)(F)F)c1ccccc1	CID:54660697	phase I
BRD-K42634310	C[C@@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2CCC(F)(F)F)c1ccccc1	CID:54660698	phase I
BRD-K05323441	C[C@@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2CCC(F)(F)F)c1ccccc1	CID:54660699	phase I
BRD-K63853782	C[C@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2CCC(F)(F)F)c1ccccc1	CID:54660700	phase I
BRD-K57393707	OC[C@H]1[C@@H]2Cn3c(=O)c(\C=C\c4ccccc4)ccc3[C@@H]2N(Cc2ccc3OCOc3c2)[C@@H]1C(O)=O	CID:54660701	phase I
BRD-K66064682	OC[C@@H]1[C@H]2Cn3c(=O)c(\C=C\c4ccccc4)ccc3[C@H]2N(Cc2ccc3OCOc3c2)[C@H]1C(O)=O	CID:54660702	phase I
BRD-K59893315	CCC(=O)N1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)OC	CID:54660709	phase I
BRD-K20428479	CCC(=O)N1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)OC	CID:54660710	phase I
BRD-K39032190	C[C@@H](NC(=O)[C@@H]1N[C@H]2[C@H](Cn3c2ccc(C2=CCCC2)c3=O)[C@H]1CO)c1ccccc1	CID:54660717	phase I
BRD-K47681666	C[C@H](NC(=O)[C@@H]1N[C@H]2[C@H](Cn3c2ccc(C2=CCCC2)c3=O)[C@H]1CO)c1ccccc1	CID:54660718	phase I
BRD-K31183432	C[C@@H](NC(=O)[C@H]1N[C@@H]2[C@@H](Cn3c2ccc(C2=CCCC2)c3=O)[C@@H]1CO)c1ccccc1	CID:54660719	phase I
BRD-K18412690	C[C@H](NC(=O)[C@H]1N[C@@H]2[C@@H](Cn3c2ccc(C2=CCCC2)c3=O)[C@@H]1CO)c1ccccc1	CID:54660720	phase I
BRD-K90073570	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]2N(CCC(F)(F)F)[C@@H]1C(=O)N1CCOCC1	CID:54660721	phase I
BRD-K15232561	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]2N(CCC(F)(F)F)[C@H]1C(=O)N1CCOCC1	CID:54660722	phase I
BRD-K32185509	CCCNC(=O)N1[C@H]2Cn3c(cccc3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCC(Cc2ccccc2)CC1	CID:54660723	phase I
BRD-K96352830	CCCNC(=O)N1[C@@H]2Cn3c(cccc3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCC(Cc2ccccc2)CC1	CID:54660724	phase I
BRD-K16048293	CC(C)NC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]12)C(=O)NC1CCC1	CID:54660725	phase I
BRD-K85126547	CC(C)NC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]12)C(=O)NC1CCC1	CID:54660726	phase I
BRD-K97173328	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N(CC2CC2)[C@@H]1C(=O)N1CCCCC1	CID:54660727	phase I
BRD-K67489890	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N(CC2CC2)[C@H]1C(=O)N1CCCCC1	CID:54660728	phase I
BRD-K20555710	OC[C@H]1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]([C@@H]1C(=O)NCc1ccccn1)N2CC1CC1	CID:54660729	phase I
BRD-K50298819	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N([C@@H]1C(=O)NCC1CCCCC1)C(=O)CC1CC1	CID:54660730	phase I
BRD-K46670060	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N([C@H]1C(=O)NCC1CCCCC1)C(=O)CC1CC1	CID:54660731	phase I
BRD-K95622068	CCCN1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCCc1cn(C)cn1	CID:54660732	phase I
BRD-K84471959	CCCN1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCCc1cn(C)cn1	CID:54660733	phase I
BRD-K75394059	CN1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCc1cc(F)cc(F)c1	CID:54660734	phase I
BRD-K09780243	CN1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCc1cc(F)cc(F)c1	CID:54660735	phase I
BRD-K39581664	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(OC)c4)c3=O)[C@H]2N1Cc1nccs1	CID:54660742	phase I
BRD-K88027520	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(OC)c4)c3=O)[C@@H]2N1Cc1nccs1	CID:54660743	phase I
BRD-K51961561	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]1N2	CID:54660744	phase I
BRD-K86758801	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]1N2	CID:54660745	phase I
BRD-K90640851	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(Cc2ccccc2Cl)[C@H]1C(=O)N1CCCCC1	CID:54660746	phase I
BRD-K34332181	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(Cc2ccccc2Cl)[C@@H]1C(=O)N1CCCCC1	CID:54660747	phase I
BRD-K16347954	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]([C@@H]1C(=O)N1CCOCC1)N2C(=O)c1ccncc1	CID:54660748	phase I
BRD-K73288268	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]([C@H]1C(=O)N1CCOCC1)N2C(=O)c1ccncc1	CID:54660749	phase I
BRD-K36725752	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]([C@@H]1C(=O)NC1CCCC1)N2CCc1ccccc1	CID:54660750	phase I
BRD-K71353154	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]([C@H]1C(=O)NC1CCCC1)N2CCc1ccccc1	CID:54660751	phase I
BRD-K67583114	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H](N2)[C@@H]1C(=O)NCc1cc(F)cc(F)c1	CID:54660752	phase I
BRD-K51951665	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H](N2)[C@H]1C(=O)NCc1cc(F)cc(F)c1	CID:54660753	phase I
BRD-K02511275	COc1ccccc1-c1ccc2[C@@H]3N[C@@H]([C@@H](CO)[C@@H]3Cn2c1=O)C(=O)NCc1ccccc1Cl	CID:54660754	phase I
BRD-K60087207	COc1ccccc1-c1ccc2[C@H]3N[C@H]([C@H](CO)[C@H]3Cn2c1=O)C(=O)NCc1ccccc1Cl	CID:54660755	phase I
BRD-K96150242	CCCNC(=O)N1[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCC	CID:54660756	phase I
BRD-K39839146	CCCNC(=O)N1[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCC	CID:54660757	phase I
BRD-K39431644	CS(=O)(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]12)C(=O)NCCc1ccncc1	CID:54660758	phase I
BRD-K51036109	CS(=O)(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]12)C(=O)NCCc1ccncc1	CID:54660759	phase I
BRD-K63090665	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H](N2)[C@H]1C(=O)NCCc1ccncc1	CID:54660760	phase I
BRD-K31290842	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H](N2)[C@@H]1C(=O)NCCc1ccncc1	CID:54660761	phase I
BRD-K11144279	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]2N1C(=O)c1cccnc1	CID:54660762	phase I
BRD-K62430643	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]2N1C(=O)c1cccnc1	CID:54660763	phase I
BRD-K92347680	CCCNC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]12)C(=O)N1CCCCC1	CID:54660764	phase I
BRD-K08520424	CCCNC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]12)C(=O)N1CCCCC1	CID:54660765	phase I
BRD-K03346718	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]1N2S(=O)(=O)c1ccccc1C	CID:54660766	phase I
BRD-K62063025	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]1N2S(=O)(=O)c1ccccc1C	CID:54660767	phase I
BRD-K16425314	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCc1ccc(F)cc1)N2C(=O)Cc1ccccn1	CID:54660774	phase I
BRD-K32183200	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCc1ccc(F)cc1)N2C(=O)Cc1ccccn1	CID:54660775	phase I
BRD-K00766524	COc1ccc(cc1)-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3C)C(=O)Nc1ccccc1	CID:54660782	phase I
BRD-K93876350	COc1ccc(cc1)-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3C)C(=O)Nc1ccccc1	CID:54660783	phase I
BRD-K46575753	COc1ccc(cc1)-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3CC1CCCC1)C(=O)N(C)C	CID:54660784	phase I
BRD-K26715911	COc1ccc(cc1)-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3CC1CCCC1)C(=O)N(C)C	CID:54660785	phase I
BRD-K93123387	C[C@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]1N2)c1ccccc1	CID:54660786	phase I
BRD-K46393778	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2Cc1nccs1	CID:54660787	phase I
BRD-K35809598	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2Cc1nccs1	CID:54660788	phase I
BRD-K31720784	CCN1[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCc1ccc(F)cc1	CID:54660789	phase I
BRD-K24746925	CCN1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCc1ccc(F)cc1	CID:54660790	phase I
BRD-K26604645	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]2N[C@H]1C(=O)NCCN1CCCCC1	CID:54660791	phase I
BRD-K04078927	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]2N[C@@H]1C(=O)NCCN1CCCCC1	CID:54660792	phase I
BRD-K04366697	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]2N([C@@H]1C(O)=O)C(=O)c1ccccn1	CID:54660793	phase I
BRD-K84381175	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]2N([C@H]1C(O)=O)C(=O)c1ccccn1	CID:54660794	phase I
BRD-K68279832	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NC1CCC1)N2Cc1cc(F)ccc1F	CID:54660795	phase I
BRD-K23703347	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NC1CCC1)N2Cc1cc(F)ccc1F	CID:54660796	phase I
BRD-K57579117	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]12)C(=O)NCCCN1CCOCC1	CID:54660797	phase I
BRD-K07609594	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]12)C(=O)NCCCN1CCOCC1	CID:54660798	phase I
BRD-K11402657	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]12)C(=O)NC1Cc2ccccc2C1	CID:54660805	phase I
BRD-K76269942	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]12)C(=O)NC1Cc2ccccc2C1	CID:54660806	phase I
BRD-K39801870	COCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]12)C(=O)Nc1ccccc1	CID:54660807	phase I
BRD-K59174142	COCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]12)C(=O)Nc1ccccc1	CID:54660808	phase I
BRD-K02734624	CN(C)CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1N2Cc1cocn1	CID:54660815	phase I
BRD-K58600416	CN(C)CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]1N2Cc1cocn1	CID:54660816	phase I
BRD-K50052949	CC(=O)N1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCc2ccccc2C1	CID:54660817	phase I
BRD-K42953652	CC(=O)N1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCc2ccccc2C1	CID:54660818	phase I
BRD-K08799867	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]1N2C(=O)NC1CCCC1	CID:54660819	phase I
BRD-K83157442	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]1N2C(=O)NC1CCCC1	CID:54660820	phase I
BRD-K00484200	COc1ccccc1CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]12)C(=O)NCCc1ccncc1	CID:54660821	phase I
BRD-K40050963	COc1ccccc1CN1[C@H]([C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]12)C(=O)NCCc1ccncc1	CID:54660822	phase I
BRD-K41527436	COc1cccc(c1)-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3Cc1ccccc1F)C(O)=O	CID:54660823	phase I
BRD-K68844146	COc1cccc(c1)-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3Cc1ccccc1F)C(O)=O	CID:54660824	phase I
BRD-K47664103	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCCN1CCCC1)N2C(=O)c1ccccc1	CID:54660825	phase I
BRD-K80666761	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCCN1CCCC1)N2C(=O)c1ccccc1	CID:54660826	phase I
BRD-K60027289	CN(C)CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1N2C(=O)CC1CC1	CID:54660830	phase I
BRD-K15679280	CN(C)CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1N2C(=O)CC1CC1	CID:54660831	phase I
BRD-K61764820	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]2N(Cc2cocn2)[C@H]1C(=O)N1CCCCC1	CID:54660832	phase I
BRD-K69464603	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]2N(Cc2cocn2)[C@@H]1C(=O)N1CCCCC1	CID:54660833	phase I
BRD-K88903268	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]2N(CC2CC2)[C@@H]1C(=O)NCc1ccncn1	CID:54660834	phase I
BRD-K81752795	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]2N(CC2CC2)[C@H]1C(=O)NCc1ccncn1	CID:54660835	phase I
BRD-K81476029	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]2N1Cc1cc(F)ccc1F	CID:54660836	phase I
BRD-K10662075	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]2N1Cc1cc(F)ccc1F	CID:54660837	phase I
BRD-K70512038	COCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]1N2C(=O)NC(C)C	CID:54660838	phase I
BRD-K81468789	COCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]1N2C(=O)NC(C)C	CID:54660839	phase I
BRD-K86124549	COc1ccccc1-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3CC1CC1)C(=O)N1CCOCC1	CID:54660840	phase I
BRD-K19882533	COc1ccccc1-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3CC1CC1)C(=O)N1CCOCC1	CID:54660841	phase I
BRD-K42516959	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N1C(=O)c1ccccc1F	CID:54660848	phase I
BRD-K50694553	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N1C(=O)c1ccccc1F	CID:54660849	phase I
BRD-K88196769	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)N1CCc3ccccc3C1)N2CC1CC1	CID:54660856	phase I
BRD-K04262969	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)N1CCc3ccccc3C1)N2CC1CC1	CID:54660857	phase I
BRD-K56975856	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]2N[C@H]1C(=O)N1CCc2ccccc2C1	CID:54660858	phase I
BRD-K54585147	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]2N[C@@H]1C(=O)N1CCc2ccccc2C1	CID:54660859	phase I
BRD-K00951345	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@@H]2N1C(=O)C1CCC1	CID:54660860	phase I
BRD-K78586486	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@H]2N1C(=O)C1CCC1	CID:54660861	phase I
BRD-K26252750	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]([C@H]1C(O)=O)N2C(=O)Cc1ccccn1	CID:54660862	phase I
BRD-K20044426	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]([C@@H]1C(O)=O)N2C(=O)Cc1ccccn1	CID:54660863	phase I
BRD-K88363359	COc1ccccc1-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3S(C)(=O)=O)C(=O)NCC1CC1	CID:54660864	phase I
BRD-K16009699	COc1ccccc1-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3S(C)(=O)=O)C(=O)NCC1CC1	CID:54660865	phase I
BRD-K58493574	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]12)C(=O)N1CCN(C)CC1	CID:54660866	phase I
BRD-K13183999	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]12)C(=O)N1CCN(C)CC1	CID:54660867	phase I
BRD-K54014179	CN1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCC(Cc2ccccc2)CC1	CID:54660868	phase I
BRD-K94715393	CN1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCC(Cc2ccccc2)CC1	CID:54660869	phase I
BRD-K56370195	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(CCc2ccccc2)[C@H]1C(=O)NC1CCC1	CID:54660870	phase I
BRD-K95047072	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(CCc2ccccc2)[C@@H]1C(=O)NC1CCC1	CID:54660871	phase I
BRD-K02315839	CC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]12)C(=O)NCc1ccccc1F	CID:54660872	phase I
BRD-K75094920	CC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]12)C(=O)NCc1ccccc1F	CID:54660873	phase I
BRD-K15990364	COc1cccc(c1)-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3C)C(=O)NCCN1CCCCC1	CID:54660880	phase I
BRD-K41761456	COc1cccc(c1)-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3C)C(=O)NCCN1CCCCC1	CID:54660881	phase I
BRD-K11415638	CN1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NC1Cc2ccccc2C1	CID:54660882	phase I
BRD-K50388099	CN1[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NC1Cc2ccccc2C1	CID:54660883	phase I
BRD-K11002182	CCCN1[C@@H]2Cn3c(ccc(-c4cccc(c4)C(=O)N(C)C)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)OC	CID:54660884	phase I
BRD-K02861439	CCCN1[C@H]2Cn3c(ccc(-c4cccc(c4)C(=O)N(C)C)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)OC	CID:54660885	phase I
BRD-K30456673	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCC(F)(F)F)N2CC1CCOCC1	CID:54660886	phase I
BRD-K56327795	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCC(F)(F)F)N2CC1CCOCC1	CID:54660887	phase I
BRD-K28841686	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N1C(=O)Cc1cccnc1	CID:54660888	phase I
BRD-K15023392	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N1C(=O)Cc1cccnc1	CID:54660889	phase I
BRD-K89399567	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)Nc1ccc(cc1)-c1ccccc1)N2Cc1ccncc1	CID:54660890	phase I
BRD-K56240483	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)Nc1ccc(cc1)-c1ccccc1)N2Cc1ccncc1	CID:54660891	phase I
BRD-K29827452	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1N2C(=O)C1CCCCC1	CID:54660892	phase I
BRD-K72798501	COc1ccc(cc1)-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3C(=O)c1cnccn1)C(=O)N(C)C	CID:54660893	phase I
BRD-K11847435	COc1ccc(cc1)-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3C(=O)c1cnccn1)C(=O)N(C)C	CID:54660894	phase I
BRD-K15457570	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]12)C(=O)Nc1nccs1	CID:54660895	phase I
BRD-K32027259	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]12)C(=O)Nc1nccs1	CID:54660896	phase I
BRD-K23781896	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]([C@H]1C(=O)N1CCCCC1)N2Cc1nccs1	CID:54660897	phase I
BRD-K25761622	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]([C@@H]1C(=O)N1CCCCC1)N2Cc1nccs1	CID:54660898	phase I
BRD-K15460493	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]([C@@H]1C(O)=O)N2CC1CCCCC1	CID:54660899	phase I
BRD-K19658687	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]([C@H]1C(O)=O)N2CC1CCCCC1	CID:54660900	phase I
BRD-K98990727	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@H]2N1C	CID:54660901	phase I
BRD-K91627479	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@@H]2N1C	CID:54660902	phase I
BRD-K82151990	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H](N2)[C@@H]1C(=O)N1CCCCC1	CID:54660903	phase I
BRD-K71087530	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H](N2)[C@H]1C(=O)N1CCCCC1	CID:54660904	phase I
BRD-K42758410	CN1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)Nc1nccs1	CID:54660905	phase I
BRD-K32910761	CN1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)Nc1nccs1	CID:54660906	phase I
BRD-K77908171	CS(=O)(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]12)C(O)=O	CID:54660907	phase I
BRD-K90381642	CS(=O)(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]12)C(O)=O	CID:54660908	phase I
BRD-K26148755	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]([C@@H]1C(O)=O)N2C(=O)C1CC1	CID:54660909	phase I
BRD-K94823396	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]([C@H]1C(O)=O)N2C(=O)C1CC1	CID:54660910	phase I
BRD-K22932079	CN1CCN(CC1)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]2N1CC1CC1	CID:54660917	phase I
BRD-K13245569	CN1CCN(CC1)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]2N1CC1CC1	CID:54660918	phase I
BRD-K69332942	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]([C@@H]1C(=O)NCc1cccc(F)c1)N2CC1CC1	CID:54660919	phase I
BRD-K88709513	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]([C@H]1C(=O)NCc1cccc(F)c1)N2CC1CC1	CID:54660920	phase I
BRD-K75906982	CN1[C@H]2Cn3c(cccc3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCC1CC1	CID:54660921	phase I
BRD-K79106006	CN1[C@@H]2Cn3c(cccc3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCC1CC1	CID:54660922	phase I
BRD-K79983157	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]([C@@H]1C(=O)NCC1CC1)N2CCC(F)(F)F	CID:54660923	phase I
BRD-K39685946	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]([C@H]1C(=O)NCC1CC1)N2CCC(F)(F)F	CID:54660924	phase I
BRD-K32128027	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]2N1Cc1ccc2OCOc2c1	CID:54660925	phase I
BRD-K31295191	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N1Cc1ccc2OCOc2c1	CID:54660926	phase I
BRD-K32759520	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H](N2)[C@H]1C(=O)NCC1CCCCC1	CID:54660933	phase I
BRD-K19358815	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H](N2)[C@@H]1C(=O)NCC1CCCCC1	CID:54660934	phase I
BRD-K73428213	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N([C@@H]1C(=O)NC1Cc2ccccc2C1)C(=O)c1cnccn1	CID:54660935	phase I
BRD-K47070211	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N([C@H]1C(=O)NC1Cc2ccccc2C1)C(=O)c1cnccn1	CID:54660936	phase I
BRD-K71182858	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]2N[C@@H]1C(=O)NC1CCCCC1	CID:54660943	phase I
BRD-K08624646	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]2N[C@H]1C(=O)NC1CCCCC1	CID:54660944	phase I
BRD-K06745755	C[C@@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]2N1C)c1ccccc1	CID:54660945	phase I
BRD-K21473123	C[C@@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]2N1C)c1ccccc1	CID:54660946	phase I
BRD-K20211345	C[C@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]2N1C)c1ccccc1	CID:54660947	phase I
BRD-K61152698	C[C@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]2N1C)c1ccccc1	CID:54660948	phase I
BRD-K14659422	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NC1Cc3ccccc3C1)N2C(=O)CC1CC1	CID:54660949	phase I
BRD-K41325905	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NC1Cc3ccccc3C1)N2C(=O)CC1CC1	CID:54660950	phase I
BRD-K93679872	CC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]12)C(=O)NCc1ccccc1Cl	CID:54660951	phase I
BRD-K59977049	CC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]12)C(=O)NCc1ccccc1Cl	CID:54660952	phase I
BRD-K83529035	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]2N1C(=O)CC1CC1	CID:54660953	phase I
BRD-K30155575	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]2N1C(=O)CC1CC1	CID:54660954	phase I
BRD-K19331234	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]1N2S(=O)(=O)c1cn(C)cn1	CID:54660955	phase I
BRD-K58745468	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1N2S(=O)(=O)c1cn(C)cn1	CID:54660956	phase I
BRD-K92210276	CCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]12)C(=O)NCc1cccc(OC)c1	CID:54660957	phase I
BRD-K75609900	CCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]12)C(=O)NCc1cccc(OC)c1	CID:54660958	phase I
BRD-K24748809	CC(C)NC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]12)C(=O)N1CCc2ccccc2C1	CID:54660959	phase I
BRD-K33341138	CC(C)NC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]12)C(=O)N1CCc2ccccc2C1	CID:54660960	phase I
BRD-K10689551	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(Cc2ccccn2)[C@@H]1C(=O)NCCN1CCCCC1	CID:54660961	phase I
BRD-K15400899	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(Cc2ccccn2)[C@H]1C(=O)NCCN1CCCCC1	CID:54660962	phase I
BRD-K95138368	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]1N2C(=O)c1ccncc1	CID:54660963	phase I
BRD-K97955841	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]1N2C(=O)c1ccncc1	CID:54660964	phase I
BRD-K30114694	C[C@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@@H]2N1S(C)(=O)=O)c1ccccc1	CID:54660971	phase I
BRD-K63435201	C[C@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@H]2N1S(C)(=O)=O)c1ccccc1	CID:54660972	phase I
BRD-K13649454	C[C@@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@@H]2N1S(C)(=O)=O)c1ccccc1	CID:54660973	phase I
BRD-K81636483	C[C@@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@H]2N1S(C)(=O)=O)c1ccccc1	CID:54660974	phase I
BRD-K02544880	CC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]12)C(=O)Nc1nccs1	CID:54660975	phase I
BRD-K29720768	CC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]12)C(=O)Nc1nccs1	CID:54660976	phase I
BRD-K50157880	CN(C)CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]2N1C(C)=O	CID:54660977	phase I
BRD-K52719892	CN(C)CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]2N1C(C)=O	CID:54660978	phase I
BRD-K46922721	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]12)C(=O)OC	CID:54660991	phase I
BRD-K42862966	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]12)C(=O)OC	CID:54660992	phase I
BRD-K98641517	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]12)C(=O)NCc1ccncn1	CID:54660993	phase I
BRD-K50381033	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]([C@@H]1C(=O)N1CCCCC1)N2CCC(F)(F)F	CID:54660994	phase I
BRD-K92313046	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]([C@H]1C(=O)N1CCCCC1)N2CCC(F)(F)F	CID:54660995	phase I
BRD-K15958865	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]([C@@H]1C(=O)NCc1ccccn1)N2Cc1cccnc1	CID:54660996	phase I
BRD-K56917655	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]([C@H]1C(=O)NCc1ccccn1)N2Cc1cccnc1	CID:54660997	phase I
BRD-K28668737	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]12)C(=O)NCCCN1CCOCC1	CID:54660998	phase I
BRD-K76276139	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]12)C(=O)NCCCN1CCOCC1	CID:54660999	phase I
BRD-K65049758	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]([C@H]1C(=O)N1CCCCC1)N2C(=O)C1CCC1	CID:54661000	phase I
BRD-K06380515	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]([C@@H]1C(=O)N1CCCCC1)N2C(=O)C1CCC1	CID:54661001	phase I
BRD-K35801103	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]2N([C@H]1C(=O)NCCc1ccncc1)C(=O)C1CC1	CID:54661002	phase I
BRD-K83477078	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]2N([C@@H]1C(=O)NCCc1ccncc1)C(=O)C1CC1	CID:54661003	phase I
BRD-K80204570	CCC(=O)N1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NC1Cc2ccccc2C1	CID:54661004	phase I
BRD-K42614769	CCC(=O)N1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NC1Cc2ccccc2C1	CID:54661005	phase I
BRD-K24175855	OC[C@H]1[C@@H]2Cn3c(=O)cccc3[C@@H]2N(Cc2ncoc2)[C@@H]1C(=O)N1CCC(CC1)Cc1ccccc1	CID:54661012	phase I
BRD-K66480544	OC[C@@H]1[C@H]2Cn3c(=O)cccc3[C@H]2N(Cc2ncoc2)[C@H]1C(=O)N1CCC(CC1)Cc1ccccc1	CID:54661013	phase I
BRD-K38187891	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]1N2Cc1ccccc1F	CID:54661014	phase I
BRD-K24626857	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N(Cc2cocn2)[C@H]1C(=O)Nc1ccccc1	CID:54661015	phase I
BRD-K32436461	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]2N(Cc2cocn2)[C@@H]1C(=O)Nc1ccccc1	CID:54661016	phase I
BRD-K19917828	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]2N(CC2CCCC2)[C@H]1C(=O)Nc1nccs1	CID:54661017	phase I
BRD-K59283736	COc1ccc(cc1)-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3C(=O)NC(C)C)C(=O)NCC1CC1	CID:54661018	phase I
BRD-K50727748	COc1ccc(cc1)-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3C(=O)NC(C)C)C(=O)NCC1CC1	CID:54661019	phase I
BRD-K69506839	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]12)C(=O)N1CCc2ccccc2C1	CID:54661020	phase I
BRD-K93906979	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]12)C(=O)N1CCc2ccccc2C1	CID:54661021	phase I
BRD-K60308664	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]2N1Cc1ccncc1	CID:54661022	phase I
BRD-K39892211	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]2N1Cc1ccncc1	CID:54661023	phase I
BRD-K04985042	COCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]12)C(=O)N1CCOCC1	CID:54661024	phase I
BRD-K45485804	COCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]12)C(=O)N1CCOCC1	CID:54661025	phase I
BRD-K52725924	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]1N2C(=O)c1ccccn1	CID:54661032	phase I
BRD-K02927581	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]1N2C(=O)c1ccccn1	CID:54661033	phase I
BRD-K93116089	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]([C@H]1C(=O)NC1CCC1)N2Cc1cocn1	CID:54661034	phase I
BRD-K27433204	OC[C@H]1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]2N(Cc2cncnc2)[C@@H]1C(=O)NC1CCC1	CID:54661037	phase I
BRD-K08477148	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N(Cc2ccccc2F)[C@@H]1C(=O)NCC1CC1	CID:54661038	phase I
BRD-K17427497	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N(Cc2ccccc2F)[C@H]1C(=O)NCC1CC1	CID:54661039	phase I
BRD-K08171986	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N([C@@H]1C(O)=O)C(=O)NC1CCCC1	CID:54661046	phase I
BRD-K23051555	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N([C@H]1C(O)=O)C(=O)NC1CCCC1	CID:54661047	phase I
BRD-K80201761	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N1C(=O)C1CC1	CID:54661048	phase I
BRD-K24680618	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N1C(=O)C1CC1	CID:54661049	phase I
BRD-K49620695	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]([C@@H]1C(=O)N1CCOCC1)N2Cc1cccnc1	CID:54661050	phase I
BRD-K01520647	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]([C@H]1C(=O)N1CCOCC1)N2Cc1cccnc1	CID:54661051	phase I
BRD-K92399508	COc1cccc(c1)-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3S(C)(=O)=O)C(=O)NCC1CC1	CID:54661052	phase I
BRD-K32503834	COc1cccc(c1)-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3S(C)(=O)=O)C(=O)NCC1CC1	CID:54661053	phase I
BRD-K82494420	CCCN1[C@@H]2Cn3c(cccc3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N(C)C	CID:54661054	phase I
BRD-K84673192	CCCN1[C@H]2Cn3c(cccc3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N(C)C	CID:54661055	phase I
BRD-K89960068	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(CC2CC2)[C@H]1C(=O)Nc1ccc(cc1)-c1ccccc1	CID:54661056	phase I
BRD-K77318689	COc1cccc(CNC(=O)[C@@H]2[C@@H](CO)[C@@H]3Cn4c(cccc4=O)[C@H]2N3C(=O)C2CCCCC2)c1	CID:54661057	phase I
BRD-K86578973	COc1cccc(CNC(=O)[C@H]2[C@H](CO)[C@H]3Cn4c(cccc4=O)[C@@H]2N3C(=O)C2CCCCC2)c1	CID:54661058	phase I
BRD-K89507938	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)N1CCOCC1)N2Cc1cccc(Cl)c1	CID:54661059	phase I
BRD-K45466167	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)N1CCOCC1)N2Cc1cccc(Cl)c1	CID:54661060	phase I
BRD-K85656047	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]2N1C(=O)C1CCCC1	CID:54661063	phase I
BRD-K83183082	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]2N1C(=O)C1CCCC1	CID:54661064	phase I
BRD-K51147043	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]2N(Cc2ccncc2)[C@H]1C(=O)NCC(F)(F)F	CID:54661065	phase I
BRD-K25736729	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]2N(Cc2ccncc2)[C@@H]1C(=O)NCC(F)(F)F	CID:54661066	phase I
BRD-K59352217	CN(C)CC(=O)N1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCN(C)CC1	CID:54661067	phase I
BRD-K22863062	CN(C)CC(=O)N1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCN(C)CC1	CID:54661068	phase I
BRD-K85568664	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]12)C(=O)NCC1CCCCC1	CID:54661069	phase I
BRD-K85072179	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]12)C(=O)NCC1CCCCC1	CID:54661070	phase I
BRD-K34007913	Cc1cccc(c1)S(=O)(=O)N1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(O)=O	CID:54661077	phase I
BRD-K86684694	Cc1cccc(c1)S(=O)(=O)N1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(O)=O	CID:54661078	phase I
BRD-K13417398	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)N1CCCCC1)N2C(=O)c1ccccn1	CID:54661079	phase I
BRD-K52379384	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)N1CCCCC1)N2C(=O)c1ccccn1	CID:54661080	phase I
BRD-K84307821	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]2N(CC2CCOCC2)[C@H]1C(=O)NCC1CC1	CID:54661081	phase I
BRD-K82332258	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]2N(CC2CCOCC2)[C@@H]1C(=O)NCC1CC1	CID:54661082	phase I
BRD-K76991985	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]2N(Cc2ccccn2)[C@@H]1C(=O)NC1CCC1	CID:54661083	phase I
BRD-K24522647	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]2N(Cc2ccccn2)[C@H]1C(=O)NC1CCC1	CID:54661084	phase I
BRD-K82150563	CN(C)C(=O)c1ccc(cc1)-c1ccc2[C@@H]3N[C@@H]([C@@H](CO)[C@@H]3Cn2c1=O)C(=O)NCCc1ccccc1	CID:54661085	phase I
BRD-K74530260	CN(C)C(=O)c1ccc(cc1)-c1ccc2[C@H]3N[C@H]([C@H](CO)[C@H]3Cn2c1=O)C(=O)NCCc1ccccc1	CID:54661086	phase I
BRD-K42365464	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCCCN1CCOCC1)N2C(=O)NC1CCCC1	CID:54661087	phase I
BRD-K56325098	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCCCN1CCOCC1)N2C(=O)NC1CCCC1	CID:54661088	phase I
BRD-K74732057	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]1N2Cc1ccccc1	CID:54661089	phase I
BRD-K15420741	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]1N2Cc1ccccc1	CID:54661090	phase I
BRD-K07591847	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]2N1Cc1ccc2OCOc2c1	CID:54661097	phase I
BRD-K05649470	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]2N1Cc1ccc2OCOc2c1	CID:54661098	phase I
BRD-K46118045	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]12)C(=O)NCC(F)(F)F	CID:54661099	phase I
BRD-K96779965	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]12)C(=O)NCC(F)(F)F	CID:54661100	phase I
BRD-K49383373	C[C@@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]1N2C)c1ccccc1	CID:54661101	phase I
BRD-K41215666	C[C@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]1N2C)c1ccccc1	CID:54661102	phase I
BRD-K46017924	C[C@@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]1N2C)c1ccccc1	CID:54661103	phase I
BRD-K19593593	C[C@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]1N2C)c1ccccc1	CID:54661104	phase I
BRD-K27237215	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]1N2C(=O)CC	CID:54661105	phase I
BRD-K41767152	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1N2C(=O)CC	CID:54661106	phase I
BRD-K22846014	COCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]1N2S(C)(=O)=O	CID:54661107	phase I
BRD-K40425733	COCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]1N2S(C)(=O)=O	CID:54661108	phase I
BRD-K47663354	COc1ccccc1-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3C)C(=O)N1CCCCC1	CID:54661109	phase I
BRD-K20954269	COc1ccccc1-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3C)C(=O)N1CCCCC1	CID:54661110	phase I
BRD-K93680063	CCCN1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCc2ccccc2C1	CID:54661111	phase I
BRD-K75990896	CCCN1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)N1CCc2ccccc2C1	CID:54661112	phase I
BRD-K14336497	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2C(=O)C1CC1	CID:54661119	phase I
BRD-K75882457	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2C(=O)C1CC1	CID:54661120	phase I
BRD-K28149578	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]([C@@H]1C(=O)NC1CCCC1)N2C(=O)CC1CC1	CID:54661133	phase I
BRD-K99786514	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]([C@H]1C(=O)NC1CCCC1)N2C(=O)CC1CC1	CID:54661134	phase I
BRD-K43407975	CN1CCN(CC1)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]1N2S(C)(=O)=O	CID:54661135	phase I
BRD-K74066682	CN1CCN(CC1)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1N2S(C)(=O)=O	CID:54661136	phase I
BRD-K97165733	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCc1cc(F)cc(F)c1)N2C(=O)c1cnccn1	CID:54661137	phase I
BRD-K25755601	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCc1cc(F)cc(F)c1)N2C(=O)c1cnccn1	CID:54661138	phase I
BRD-K99327410	CN(C)CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N1CCC(F)(F)F	CID:54661139	phase I
BRD-K58129723	CN(C)CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N1CCC(F)(F)F	CID:54661140	phase I
BRD-K88990907	COCC(=O)N1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCc1ccccn1	CID:54661141	phase I
BRD-K93406741	COCC(=O)N1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCc1ccccn1	CID:54661142	phase I
BRD-K08707982	COc1cccc(c1)-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3C(=O)C1CC1)C(=O)N(C)C	CID:54661143	phase I
BRD-K67086788	COc1cccc(c1)-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3C(=O)C1CC1)C(=O)N(C)C	CID:54661144	phase I
BRD-K65729053	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]([C@@H]1C(O)=O)N2C(=O)Nc1cc(F)ccc1F	CID:54661145	phase I
BRD-K89332300	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]([C@H]1C(O)=O)N2C(=O)Nc1cc(F)ccc1F	CID:54661146	phase I
BRD-K32106123	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]1N2C(=O)Nc1ccccc1	CID:54661147	phase I
BRD-K87688096	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]1N2C(=O)Nc1ccccc1	CID:54661148	phase I
BRD-K43036943	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCCc1ccccc1)N2Cc1ccccn1	CID:54661149	phase I
BRD-K97865175	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCCc1ccccc1)N2Cc1ccccn1	CID:54661150	phase I
BRD-K43771394	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]2N1C(=O)Cc1cccnc1	CID:54661151	phase I
BRD-K35562235	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]2N1C(=O)Cc1cccnc1	CID:54661152	phase I
BRD-K58524976	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H](N2)[C@@H]1C(=O)NC1Cc2ccccc2C1	CID:54661159	phase I
BRD-K54565270	CN(C)C(=O)c1cccc(c1)-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3C)C(=O)NCC(F)(F)F	CID:54661160	phase I
BRD-K93681700	CN(C)C(=O)c1cccc(c1)-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3C)C(=O)NCC(F)(F)F	CID:54661161	phase I
BRD-K43411248	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]2N(Cc2ccccc2F)[C@H]1C(O)=O	CID:54661168	phase I
BRD-K69493165	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]2N(Cc2ccccc2F)[C@@H]1C(O)=O	CID:54661169	phase I
BRD-K19645992	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]1N2Cc1ccccc1F	CID:54661170	phase I
BRD-K82019527	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]1N2Cc1ccccc1F	CID:54661171	phase I
BRD-K49640920	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H](N2)[C@@H]1C(=O)NCc1ccccc1	CID:54661172	phase I
BRD-K59689930	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H](N2)[C@H]1C(=O)NCc1ccccc1	CID:54661173	phase I
BRD-K19073426	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCc1ccncn1)N2CC1CC1	CID:54661174	phase I
BRD-K62902932	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCc1ccncn1)N2CC1CC1	CID:54661175	phase I
BRD-K65160163	CN(C)C(=O)[C@H]1N[C@@H]2[C@@H](Cn3c2ccc(-c2ccc(F)cc2)c3=O)[C@@H]1CO	CID:54661176	phase I
BRD-K58679476	CN(C)C(=O)[C@@H]1N[C@H]2[C@H](Cn3c2ccc(-c2ccc(F)cc2)c3=O)[C@H]1CO	CID:54661177	phase I
BRD-K04147035	CCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]12)C(=O)NCCCN(C)C	CID:54661190	phase I
BRD-K55251364	CCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]12)C(=O)NCCCN(C)C	CID:54661191	phase I
BRD-K90496835	CCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]12)C(=O)NCCc1cn(C)cn1	CID:54661192	phase I
BRD-K86654865	CCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]12)C(=O)NCCc1cn(C)cn1	CID:54661193	phase I
BRD-K62123687	CN(C)CC(=O)N1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NC1CCC1	CID:54661197	phase I
BRD-K68908437	CN(C)CC(=O)N1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NC1CCC1	CID:54661198	phase I
BRD-K20191348	OC[C@@H]1[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]([C@H]1C(=O)NCC1CC1)N2C(=O)C1CCC1	CID:54661199	phase I
BRD-K78247419	OC[C@H]1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]([C@@H]1C(=O)NCC1CC1)N2C(=O)C1CCC1	CID:54661200	phase I
BRD-K09927308	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]([C@@H]1C(=O)NC1CCCC1)N2C(=O)c1ccccc1	CID:54661201	phase I
BRD-K90562112	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]([C@H]1C(=O)NC1CCCC1)N2C(=O)c1ccccc1	CID:54661202	phase I
BRD-K79900369	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]([C@@H]1C(=O)NCCc1ccncc1)N2CC1CC1	CID:54661203	phase I
BRD-K04061325	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]([C@H]1C(=O)NCCc1ccncc1)N2CC1CC1	CID:54661204	phase I
BRD-K54022924	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]2N1C(=O)c1ccccc1F	CID:54661205	phase I
BRD-K09416407	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]2N1C(=O)c1ccccc1F	CID:54661206	phase I
BRD-K12805419	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]2N(Cc2cocn2)[C@@H]1C(=O)NCc1ccccc1	CID:54661207	phase I
BRD-K01798544	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]2N(Cc2cocn2)[C@H]1C(=O)NCc1ccccc1	CID:54661208	phase I
BRD-K50670216	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]1N2CC1CC1	CID:54661209	phase I
BRD-K16794723	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]1N2CC1CC1	CID:54661210	phase I
BRD-K23091084	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(Cc2cc(F)ccc2F)[C@H]1C(=O)N1CCOCC1	CID:54661217	phase I
BRD-K34940426	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(Cc2cc(F)ccc2F)[C@@H]1C(=O)N1CCOCC1	CID:54661218	phase I
BRD-K41326905	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]([C@H]1C(=O)NCC1CC1)N2Cc1cccnc1	CID:54661231	phase I
BRD-K88995397	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]([C@@H]1C(=O)NCC1CC1)N2Cc1cccnc1	CID:54661232	phase I
BRD-K18481678	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@@H]([C@H]1C(=O)NCC1CCCCC1)N2C(=O)c1cccnc1	CID:54661233	phase I
BRD-K05643885	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@H]([C@@H]1C(=O)NCC1CCCCC1)N2C(=O)c1cccnc1	CID:54661234	phase I
BRD-K64133040	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]1N2Cc1ccccc1	CID:54661235	phase I
BRD-K21216453	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]1N2Cc1ccccc1	CID:54661236	phase I
BRD-K66860235	CN1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NC1CCC1	CID:54661237	phase I
BRD-K09880340	CN1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NC1CCC1	CID:54661238	phase I
BRD-K09876067	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(OC)cc4)c3=O)[C@H]1N2CC1CC1	CID:54661239	phase I
BRD-K14302953	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(OC)cc4)c3=O)[C@@H]1N2CC1CC1	CID:54661240	phase I
BRD-K50570214	CCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]12)C(=O)N1CCCCC1	CID:54661241	phase I
BRD-K19054042	CCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]12)C(=O)N1CCCCC1	CID:54661242	phase I
BRD-K05717370	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(Cc2cncnc2)[C@H]1C(=O)NCC1CC1	CID:54661243	phase I
BRD-K87833465	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(Cc2cncnc2)[C@@H]1C(=O)NCC1CC1	CID:54661244	phase I
BRD-K97031447	CCCNC(=O)N1[C@@H]2Cn3c(ccc(-c4cccc(OC)c4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NC1CCC1	CID:54661245	phase I
BRD-K14356681	CCCNC(=O)N1[C@H]2Cn3c(ccc(-c4cccc(OC)c4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NC1CCC1	CID:54661246	phase I
BRD-K27113545	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(cc4)C(=O)N(C)C)c3=O)[C@H]12)C(=O)NCCOC	CID:54661247	phase I
BRD-K13094522	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(cc4)C(=O)N(C)C)c3=O)[C@@H]12)C(=O)NCCOC	CID:54661248	phase I
BRD-K85727265	CCN1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCCCN1CCOCC1	CID:54661249	phase I
BRD-K80313395	CCN1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCCCN1CCOCC1	CID:54661250	phase I
BRD-K51640940	COc1ccc(cc1)-c1ccc2[C@@H]3[C@@H]([C@@H](CO)[C@H](Cn2c1=O)N3C(=O)c1ccccc1F)C(O)=O	CID:54661251	phase I
BRD-K73517214	COc1ccc(cc1)-c1ccc2[C@H]3[C@H]([C@H](CO)[C@@H](Cn2c1=O)N3C(=O)c1ccccc1F)C(O)=O	CID:54661252	phase I
BRD-K51826244	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]2N[C@@H]1C(=O)N1CCC(Cc2ccccc2)CC1	CID:54661259	phase I
BRD-K33064169	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N[C@H]1C(=O)N1CCC(Cc2ccccc2)CC1	CID:54661260	phase I
BRD-K66602457	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]12)C(=O)N[C@H](C)c1ccccc1	CID:54661261	phase I
BRD-K08394807	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]12)C(=O)N[C@H](C)c1ccccc1	CID:54661262	phase I
BRD-K38370145	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]12)C(=O)N[C@@H](C)c1ccccc1	CID:54661263	phase I
BRD-K68303822	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]12)C(=O)N[C@@H](C)c1ccccc1	CID:54661264	phase I
BRD-K29802265	CCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(c4)C(=O)N(C)C)c3=O)[C@H]12)C(=O)N(C)C	CID:54661265	phase I
BRD-K45525014	CCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(c4)C(=O)N(C)C)c3=O)[C@@H]12)C(=O)N(C)C	CID:54661266	phase I
BRD-K90004145	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2CCc1ccccc1	CID:54661267	phase I
BRD-K71533863	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2CCc1ccccc1	CID:54661268	phase I
BRD-K43179840	COCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]2N1C(=O)C1CCCC1	CID:54661269	phase I
BRD-K15989099	COCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]2N1C(=O)C1CCCC1	CID:54661270	phase I
BRD-K21230248	CC(C)NC(=O)N1[C@@H]2Cn3c(ccc(-c4cccc(c4)C(=O)N(C)C)c3=O)[C@H]1[C@H]([C@@H]2CO)C(O)=O	CID:54661271	phase I
BRD-K31122916	CC(C)NC(=O)N1[C@H]2Cn3c(ccc(-c4cccc(c4)C(=O)N(C)C)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(O)=O	CID:54661272	phase I
BRD-K00697836	COc1ccc(cc1)-c1ccc2[C@@H]3[C@H](Cn2c1=O)[C@@H](CO)[C@@H](N3S(C)(=O)=O)C(=O)NC1CCC1	CID:54661273	phase I
BRD-K46751125	COc1ccc(cc1)-c1ccc2[C@H]3[C@@H](Cn2c1=O)[C@H](CO)[C@H](N3S(C)(=O)=O)C(=O)NC1CCC1	CID:54661274	phase I
BRD-K74835229	CCCNC(=O)N1[C@H]2Cn3c(cccc3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCC(F)(F)F	CID:54661275	phase I
BRD-K39779204	CCCNC(=O)N1[C@@H]2Cn3c(cccc3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCC(F)(F)F	CID:54661276	phase I
BRD-K41341398	CCCN1[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCC1CC1	CID:54661277	phase I
BRD-K37284732	CCCN1[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCC1CC1	CID:54661278	phase I
BRD-K62395041	CCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]12)C(=O)N(C)C	CID:54661279	phase I
BRD-K83058591	CCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]12)C(=O)N(C)C	CID:54661280	phase I
BRD-K53193280	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]2N([C@H]1C(=O)NCC1CC1)C(=O)NC1CCCC1	CID:54661281	phase I
BRD-K26199553	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]2N([C@@H]1C(=O)NCC1CC1)C(=O)NC1CCCC1	CID:54661282	phase I
BRD-K69521358	CCCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]12)C(=O)NC1CCC1	CID:54661283	phase I
BRD-K99299141	CCCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]12)C(=O)NC1CCC1	CID:54661284	phase I
BRD-K59455917	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]1N2C(C)=O	CID:54661291	phase I
BRD-K78845122	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]1N2C(C)=O	CID:54661292	phase I
BRD-K31422806	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]12)C(=O)NC1Cc2ccccc2C1	CID:54661293	phase I
BRD-K74799293	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]12)C(=O)NC1Cc2ccccc2C1	CID:54661294	phase I
BRD-K72956282	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]2N[C@H]1C(=O)NCC1CCCCC1	CID:54661295	phase I
BRD-K97258019	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H](N2)[C@H]1C(=O)N1CCc2ccccc2C1	CID:54661296	phase I
BRD-K49299173	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H](N2)[C@@H]1C(=O)N1CCc2ccccc2C1	CID:54661297	phase I
BRD-K05657439	CCCN1[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCc1ccccn1	CID:54661298	phase I
BRD-K28001738	CCCN1[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCc1ccccn1	CID:54661299	phase I
BRD-K41028488	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1N2CCC(F)(F)F	CID:54661300	phase I
BRD-K49178877	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1N2CCC(F)(F)F	CID:54661301	phase I
BRD-K58593815	CN1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCCc1ccccc1	CID:54661302	phase I
BRD-K10701104	CN1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCCc1ccccc1	CID:54661303	phase I
BRD-K12981857	CC(=O)N1[C@H]2Cn3c(cccc3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NC1CCCC1	CID:54661304	phase I
BRD-K46407773	CC(=O)N1[C@@H]2Cn3c(cccc3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NC1CCCC1	CID:54661305	phase I
BRD-K84368021	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N([C@@H]1C(=O)NCc1ccccc1Cl)C(=O)C1CCOCC1	CID:54661306	phase I
BRD-K64937432	CCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]12)C(=O)NCc1ccc(F)cc1	CID:54661313	phase I
BRD-K61161989	CCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]12)C(=O)NCc1ccc(F)cc1	CID:54661314	phase I
BRD-K87758256	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]2N1CC1CCCC1	CID:54661321	phase I
BRD-K87838848	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]2N1CC1CCCC1	CID:54661322	phase I
BRD-K20793945	CN1CCN(CC1)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2Cc1ccncc1	CID:54661323	phase I
BRD-K65761985	CN1CCN(CC1)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2Cc1ccncc1	CID:54661324	phase I
BRD-K85689251	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]1N2CC1CCCC1	CID:54661325	phase I
BRD-K88272013	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]1N2CC1CCCC1	CID:54661326	phase I
BRD-K76595742	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@H]2N1CC1CCCCC1	CID:54661327	phase I
BRD-K09817289	CCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@@H]2N1CC1CCCCC1	CID:54661328	phase I
BRD-K79025148	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]([C@@H]1C(O)=O)N2CCc1ccccc1	CID:54661329	phase I
BRD-K69425327	CCN1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)N1CCCCC1	CID:54661330	phase I
BRD-K11436949	CN(C)CC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]12)C(=O)NC1CCC1	CID:54661331	phase I
BRD-K17546203	CN(C)CC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]12)C(=O)NC1CCC1	CID:54661332	phase I
BRD-K39812368	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]2N1Cc1ccccn1	CID:54661333	phase I
BRD-K16113530	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N1Cc1ccccn1	CID:54661334	phase I
BRD-K13272610	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]12)C(=O)Nc1ccccc1	CID:54661341	phase I
BRD-K06832445	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]12)C(=O)Nc1ccccc1	CID:54661342	phase I
BRD-K29390829	CN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]12)C(=O)NCc1ccccn1	CID:54661343	phase I
BRD-K87539610	CN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]12)C(=O)NCc1ccccn1	CID:54661344	phase I
BRD-K74043769	COCC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]12)C(=O)NCc1ccccc1	CID:54661345	phase I
BRD-K13544395	COCC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]12)C(=O)NCc1ccccc1	CID:54661346	phase I
BRD-K20016217	CCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@@H]12)C(=O)NCc1ccc(F)cc1	CID:54661347	phase I
BRD-K06482871	CCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4OC)c3=O)[C@H]12)C(=O)NCc1ccc(F)cc1	CID:54661348	phase I
BRD-K55813437	OC[C@@H]1[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]([C@H]1C(=O)NCC1CC1)N2C(=O)C1CC1	CID:54661349	phase I
BRD-K93666423	OC[C@H]1[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]([C@@H]1C(=O)NCC1CC1)N2C(=O)C1CC1	CID:54661350	phase I
BRD-K16512302	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N([C@@H]1C(=O)NCC(F)(F)F)C(=O)C1CC1	CID:54661363	phase I
BRD-K65541951	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N([C@H]1C(=O)NCC(F)(F)F)C(=O)C1CC1	CID:54661364	phase I
BRD-K10600561	CN1[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCC1CCCCC1	CID:54661365	phase I
BRD-K32030161	CN1[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCC1CCCCC1	CID:54661366	phase I
BRD-K84061726	OC[C@H]1[C@@H]2Cn3c(cccc3=O)[C@@H]2N(CCC(F)(F)F)[C@@H]1C(=O)NCc1ccc(F)cc1	CID:54661379	phase I
BRD-K74152422	OC[C@@H]1[C@H]2Cn3c(cccc3=O)[C@H]2N(CCC(F)(F)F)[C@H]1C(=O)NCc1ccc(F)cc1	CID:54661380	phase I
BRD-K48257023	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@@H]2N1CC1CC1	CID:54661381	phase I
BRD-K69097792	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4F)c3=O)[C@H]2N1CC1CC1	CID:54661382	phase I
BRD-K65836281	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]1N2C(=O)C1CCC1	CID:54661383	phase I
BRD-K03515977	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]1N2C(=O)C1CCC1	CID:54661384	phase I
BRD-K14437503	OC[C@H]1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@@H]2N[C@@H]1C(=O)N1CCCCC1	CID:54661391	phase I
BRD-K24164383	CCN1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@H]12)C(=O)N1CCCCC1	CID:54661398	phase I
BRD-K74101931	CCN1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(-c4cccc(F)c4)c3=O)[C@@H]12)C(=O)N1CCCCC1	CID:54661399	phase I
BRD-K47423282	COc1cccc(c1)-c1ccc2[C@@H]3N[C@@H]([C@@H](CO)[C@@H]3Cn2c1=O)C(=O)NC1Cc2ccccc2C1	CID:54661400	phase I
BRD-K36701739	COc1cccc(c1)-c1ccc2[C@H]3N[C@H]([C@H](CO)[C@H]3Cn2c1=O)C(=O)NC1Cc2ccccc2C1	CID:54661401	phase I
BRD-K00754679	CN1CCN(CC1)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@H]2N1CC1CC1	CID:54661402	phase I
BRD-K50949213	CN1CCN(CC1)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cncnc4)c3=O)[C@@H]2N1CC1CC1	CID:54661403	phase I
BRD-K28589277	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2C(=O)c1ccc(F)cc1	CID:54661404	phase I
BRD-K62124038	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2C(=O)c1ccc(F)cc1	CID:54661405	phase I
BRD-K46120075	C[C@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]1N2C(C)=O)c1ccccc1	CID:54661406	phase I
BRD-K20827972	C[C@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1N2C(C)=O)c1ccccc1	CID:54661407	phase I
BRD-K23406211	C[C@@H](NC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]1N2C(C)=O)c1ccccc1	CID:54661408	phase I
BRD-K86530412	C[C@@H](NC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1N2C(C)=O)c1ccccc1	CID:54661409	phase I
BRD-K45466793	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]1N2C(=O)Nc1ccccc1	CID:54661410	phase I
BRD-K34553907	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1N2C(=O)Nc1ccccc1	CID:54661411	phase I
BRD-K59793998	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(=O)c(ccc3[C@H]2N1C(=O)C1CCC1)-c1ccc(F)cc1	CID:54661412	phase I
BRD-K55106539	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(=O)c(ccc3[C@@H]2N1C(=O)C1CCC1)-c1ccc(F)cc1	CID:54661413	phase I
BRD-K02602944	CN(C)CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(cccc3=O)[C@@H]1N2CC1CC1	CID:54661414	phase I
BRD-K90671064	CN(C)CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(cccc3=O)[C@H]1N2CC1CC1	CID:54661415	phase I
BRD-K52918979	OC[C@@H]1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]([C@H]1C(O)=O)N2S(=O)(=O)c1ccccc1F	CID:54661416	phase I
BRD-K78704198	OC[C@H]1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]([C@@H]1C(O)=O)N2S(=O)(=O)c1ccccc1F	CID:54661417	phase I
BRD-K89440651	CN(C)C(=O)c1cccc(c1)-c1ccc2[C@@H]3N[C@@H]([C@@H](CO)[C@@H]3Cn2c1=O)C(=O)NCC1CC1	CID:54661424	phase I
BRD-K47204106	CN(C)C(=O)c1cccc(c1)-c1ccc2[C@H]3N[C@H]([C@H](CO)[C@H]3Cn2c1=O)C(=O)NCC1CC1	CID:54661425	phase I
BRD-K60807183	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]1N2Cc1cccnc1	CID:54661432	phase I
BRD-K20736932	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]1N2Cc1cccnc1	CID:54661433	phase I
BRD-K25799352	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@@H]2N1Cc1cccc(F)c1	CID:54661434	phase I
BRD-K93736495	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4cccnc4)c3=O)[C@H]2N1Cc1cccc(F)c1	CID:54661435	phase I
BRD-K57228329	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]2N1CCC(F)(F)F	CID:54661436	phase I
BRD-K91834385	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]2N1CCC(F)(F)F	CID:54661437	phase I
BRD-K71761800	CCN1[C@@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)Nc1ccccc1	CID:54661438	phase I
BRD-K90781287	CCN1[C@H]2Cn3c(ccc(-c4ccncc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)Nc1ccccc1	CID:54661439	phase I
BRD-K32083350	CCCN1[C@@H]2Cn3c(ccc(\C=C\c4ccccc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCC	CID:54661440	phase I
BRD-K13896696	CCN1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCCOC	CID:54661441	phase I
BRD-K42379673	CCN1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCCOC	CID:54661442	phase I
BRD-K14622703	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]2N[C@@H]1C(=O)NCC1CC1	CID:54661443	phase I
BRD-K37451830	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N[C@H]1C(=O)NCC1CC1	CID:54661444	phase I
BRD-K44911253	CCCN1[C@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCCOC	CID:54661445	phase I
BRD-K52303942	CCCN1[C@@H]2Cn3c(ccc(-c4ccc(F)cc4)c3=O)[C@H]1[C@H]([C@@H]2CO)C(=O)NCCOC	CID:54661446	phase I
BRD-K81054062	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H](N2)[C@@H]1C(=O)NCc1ccc(F)cc1	CID:54661453	phase I
BRD-K62366931	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H](N2)[C@H]1C(=O)NCc1ccc(F)cc1	CID:54661454	phase I
BRD-K10837140	CN(C)C(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]1N2CC1CCOCC1	CID:54661455	phase I
BRD-K92770212	CN(C)C(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]1N2CC1CCOCC1	CID:54661456	phase I
BRD-K61519911	COC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@H]2N1Cc1ccccn1	CID:54661457	phase I
BRD-K72383170	COC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(-c4ccccc4)c3=O)[C@@H]2N1Cc1ccccn1	CID:54661458	phase I
BRD-K57476701	CC(=O)N1[C@@H]([C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]12)C(=O)Nc1ccccc1	CID:54661459	phase I
BRD-K84443834	CC(=O)N1[C@H]([C@H](CO)[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]12)C(=O)Nc1ccccc1	CID:54661460	phase I
BRD-K11345845	OC[C@H]1[C@@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@@H]2N(Cc2nccs2)[C@@H]1C(=O)N1CCOCC1	CID:54661461	phase I
BRD-K19558952	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCC4)c3=O)[C@H]2N(Cc2nccs2)[C@H]1C(=O)N1CCOCC1	CID:54661462	phase I
BRD-K13641963	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N[C@H]1C(=O)N1CCc2ccccc2C1	CID:54662042	phase I
BRD-K51878684	CCCNC(=O)[C@@H]1[C@@H](CO)[C@@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]2N1Cc1ccccc1F	CID:54662640	phase I
BRD-K87440499	CCCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N1Cc1ccccc1F	CID:54662641	phase I
BRD-K85821758	CC(=O)N1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@@H]1[C@@H]([C@H]2CO)C(=O)NCc1cc(F)cc(F)c1	CID:54662957	phase I
BRD-K43637338	CCNC(=O)[C@H]1[C@H](CO)[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N1CC1CC1	CID:54664745	phase I
BRD-K76193256	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccc2OCOc2c1)C#Cc1ccc(F)cc1	CID:54664787	phase I
BRD-K44923117	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1ccc2OCOc2c1)C#Cc1ccc(F)cc1	CID:54664788	phase I
BRD-K18840975	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccc2OCOc2c1)C#Cc1ccc(F)cc1	CID:54664789	phase I
BRD-K66621600	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1ccc2OCOc2c1)C#Cc1ccc(F)cc1	CID:54664790	phase I
BRD-K93338495	Cn1cnc(c1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C1=CCCCC1	CID:54664791	phase I
BRD-K29966477	COc1cccc(c1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@H]2CO)C#Cc1cccnc1	CID:54664792	phase I
BRD-K04388421	COc1cccc(c1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@H]2CO)C#Cc1cccnc1	CID:54664793	phase I
BRD-K92333822	COc1cccc(c1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)C#Cc1cccnc1	CID:54664794	phase I
BRD-K97114030	CN1[C@@H](CO)[C@H]2CCN[C@H]2c2cc(Br)ccc12	CID:54664795	phase I
BRD-K71138839	CN1[C@H](CO)[C@@H]2CCN[C@@H]2c2cc(Br)ccc12	CID:54664796	phase I
BRD-K01849255	COc1ccccc1CN1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)-c1ccc(cc1)C(=O)N(C)C	CID:54664797	phase I
BRD-K17120478	COc1ccccc1CN1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)-c1ccc(cc1)C(=O)N(C)C	CID:54664798	phase I
BRD-K13489056	COc1ccccc1CN1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)-c1ccc(cc1)C(=O)N(C)C	CID:54664799	phase I
BRD-K81838897	OC[C@@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)C1CCOCC1	CID:54664800	phase I
BRD-K69546841	OC[C@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)C1CCOCC1	CID:54664801	phase I
BRD-K04613932	OC[C@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)C1CCOCC1	CID:54664802	phase I
BRD-K59371957	COc1ccc(cc1)C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccccn1	CID:54664807	phase I
BRD-A18573497	CC1C=NC(=N1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@H]2CO)-c1ccccc1F	CID:54664808	phase I
BRD-A59046243	CC1C=NC(=N1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@@H]2CO)-c1ccccc1F	CID:54664809	phase I
BRD-A91404865	CC1C=NC(=N1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)-c1ccccc1F	CID:54664810	phase I
BRD-A99702332	CC1C=NC(=N1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@H]2CO)-c1ccccc1F	CID:54664811	phase I
BRD-K25804113	COc1ccc(cc1)C#Cc1ccc2N(C)[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Nc1ccc(cc1)C(F)(F)F	CID:54664812	phase I
BRD-K34992378	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cccc(F)c1)-c1ccccc1F	CID:54664813	phase I
BRD-K26654895	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cccc(F)c1)-c1ccccc1F	CID:54664814	phase I
BRD-K00900096	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1cccc(F)c1)-c1ccccc1F	CID:54664815	phase I
BRD-K23470676	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1cccc(F)c1)-c1ccccc1F	CID:54664816	phase I
BRD-K81312543	C\C=C\c1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)Cc1cccnc1	CID:54664817	phase I
BRD-K84568319	C\C=C\c1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)Cc1cccnc1	CID:54664818	phase I
BRD-K60056473	C\C=C\c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Cc1cccnc1	CID:54664819	phase I
BRD-K17347940	C\C=C\c1ccc2N(C)[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Cc1cccnc1	CID:54664820	phase I
BRD-K10526563	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C1=CCCCC1)C(=O)Nc1cc(F)ccc1F	CID:54664821	phase I
BRD-K19105325	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1ccccc1C	CID:54664822	phase I
BRD-K02032571	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccccc1C	CID:54664823	phase I
BRD-K62290501	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1ccccc1C	CID:54664824	phase I
BRD-K46999092	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccccc1C	CID:54664825	phase I
BRD-K67336565	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C#Cc1ccccc1F)C(=O)c1cnccn1	CID:54664826	phase I
BRD-K46242161	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccncc1)-c1cccc(F)c1	CID:54664827	phase I
BRD-K61890750	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1ccncc1)-c1cccc(F)c1	CID:54664828	phase I
BRD-K26667087	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccncc1)-c1cccc(F)c1	CID:54664829	phase I
BRD-K84168393	CCCC#Cc1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)CC1CC1	CID:54664830	phase I
BRD-K69869536	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccc(cc1)C#N)S(=O)(=O)c1ccc(C)cc1	CID:54664831	phase I
BRD-K36203049	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccc(cc1)C#N)S(=O)(=O)c1ccc(C)cc1	CID:54664832	phase I
BRD-K93885794	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccc(cc1)C#N)S(=O)(=O)c1ccc(C)cc1	CID:54664833	phase I
BRD-K14199536	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccc(cc1)C#N)S(=O)(=O)c1ccc(C)cc1	CID:54664834	phase I
BRD-K62999057	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)CN1CCOCC1	CID:54664835	phase I
BRD-K11913456	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)CN1CCOCC1	CID:54664836	phase I
BRD-K46384573	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)CN1CCOCC1	CID:54664837	phase I
BRD-K35100006	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)CN1CCOCC1	CID:54664838	phase I
BRD-K21113341	C\C=C\c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccc(C)cc1	CID:54664839	phase I
BRD-K41958183	C\C=C\c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1ccc(C)cc1	CID:54664840	phase I
BRD-K74475430	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccc2OCOc2c1)-c1ccc(cc1)C#N	CID:54664841	phase I
BRD-K78160230	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccc2OCOc2c1)-c1ccc(cc1)C#N	CID:54664842	phase I
BRD-K62423074	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccc2OCOc2c1)-c1ccc(cc1)C#N	CID:54664843	phase I
BRD-K59164282	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccc2OCOc2c1)-c1ccc(cc1)C#N	CID:54664844	phase I
BRD-K50748030	COc1ccc(cc1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)CN1CCOCC1	CID:54664845	phase I
BRD-K05778965	COc1ccc(cc1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)CN1CCOCC1	CID:54664846	phase I
BRD-K19232452	COc1ccc(cc1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)CN1CCOCC1	CID:54664847	phase I
BRD-K05620072	COc1ccc(cc1)-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)CN1CCOCC1	CID:54664848	phase I
BRD-K52215487	C\C=C\c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1cnccn1	CID:54664849	phase I
BRD-K38197770	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)S(=O)(=O)c1cccc(F)c1	CID:54664850	phase I
BRD-K90916892	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)S(=O)(=O)c1cccc(F)c1	CID:54664851	phase I
BRD-K91279674	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)S(=O)(=O)c1cccc(F)c1	CID:54664852	phase I
BRD-K74470016	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)S(=O)(=O)c1cccc(F)c1	CID:54664853	phase I
BRD-K29137607	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cccnc1)C1=CCCCC1	CID:54664854	phase I
BRD-K23138236	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1nccs1)C#Cc1ccccc1	CID:54664855	phase I
BRD-K24392866	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1nccs1)C#Cc1ccccc1	CID:54664856	phase I
BRD-K27188211	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2S(=O)(=O)c1ccc(F)cc1)-c1cccc(c1)C#N	CID:54664857	phase I
BRD-K33906096	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2S(=O)(=O)c1ccc(F)cc1)-c1cccc(c1)C#N	CID:54664858	phase I
BRD-K33056518	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2S(=O)(=O)c1ccc(F)cc1)-c1cccc(c1)C#N	CID:54664859	phase I
BRD-K73006286	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2S(=O)(=O)c1ccc(F)cc1)-c1cccc(c1)C#N	CID:54664860	phase I
BRD-K11385710	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C#Cc1ccc(F)cc1)S(=O)(=O)c1ccccc1C	CID:54664861	phase I
BRD-K75899251	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccc(cc1)C#N)C(=O)Nc1cccc(F)c1	CID:54664862	phase I
BRD-K72001456	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccccc1F)C(=O)Cc1ccccn1	CID:54664864	phase I
BRD-K51220638	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccccc1F)C(=O)Cc1ccccn1	CID:54664865	phase I
BRD-K33943748	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCC1)C#Cc1cccc(F)c1	CID:54664866	phase I
BRD-K07340176	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCC1)C#Cc1cccc(F)c1	CID:54664867	phase I
BRD-K62177026	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCC1)C#Cc1cccc(F)c1	CID:54664868	phase I
BRD-K51428159	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCC1)C#Cc1cccc(F)c1	CID:54664869	phase I
BRD-K05496005	COc1ccccc1-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCCCC1	CID:54664870	phase I
BRD-K63227090	COc1ccccc1-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)C1CCCCC1	CID:54664871	phase I
BRD-K81763433	COc1cccc(c1)-c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Cc1ccncc1	CID:54664872	phase I
BRD-K56953341	COCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)-c1cccc(c1)C(=O)N(C)C	CID:54664873	phase I
BRD-K79748109	COCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)-c1cccc(c1)C(=O)N(C)C	CID:54664874	phase I
BRD-K99626290	COCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)-c1cccc(c1)C(=O)N(C)C	CID:54664875	phase I
BRD-K75371115	COCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)-c1cccc(c1)C(=O)N(C)C	CID:54664876	phase I
BRD-K71947697	COc1ccc(cc1)-c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)NC1CCCCC1	CID:54664877	phase I
BRD-K68915174	COc1ccc(cc1)-c1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)NC1CCCCC1	CID:54664878	phase I
BRD-K10655148	COc1ccc(cc1)-c1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)NC1CCCCC1	CID:54664879	phase I
BRD-K92522487	COc1ccccc1C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)Cc1ccccc1	CID:54664880	phase I
BRD-K11911738	COc1ccc(cc1)-c1ccc2N[C@@H](CO)[C@H]3CCN(Cc4cncnc4)[C@H]3c2c1	CID:54664881	phase I
BRD-K95820322	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C#Cc1cccnc1)C(=O)C1CCCCC1	CID:54664882	phase I
BRD-K89354425	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C#Cc1cccnc1)C(=O)C1CCCCC1	CID:54664883	phase I
BRD-K11970601	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C#Cc1cccnc1)C(=O)C1CCCCC1	CID:54664884	phase I
BRD-K09943620	CC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)-c1ccc(F)cc1	CID:54664885	phase I
BRD-K34585937	CC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)-c1ccc(F)cc1	CID:54664886	phase I
BRD-K37958236	CC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)-c1ccc(F)cc1	CID:54664887	phase I
BRD-K44134539	COc1ccccc1C#Cc1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(C)=O	CID:54664888	phase I
BRD-K27534253	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)Nc1ccccc1F	CID:54664889	phase I
BRD-K47519681	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)Nc1ccccc1F	CID:54664890	phase I
BRD-K83726109	COc1ccccc1-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1cccc(F)c1	CID:54664891	phase I
BRD-K32272500	COc1ccccc1-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1cccc(F)c1	CID:54664892	phase I
BRD-K51102238	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)Cc1ccccn1)-c1cccc(F)c1	CID:54664893	phase I
BRD-K32657617	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)Cc1ccccn1)-c1cccc(F)c1	CID:54664894	phase I
BRD-K62590692	COc1ccccc1C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54664895	phase I
BRD-K48023456	CC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C#Cc1cccnc1	CID:54664896	phase I
BRD-K52593146	CC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1cccnc1	CID:54664897	phase I
BRD-K02445308	CC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1cccnc1	CID:54664898	phase I
BRD-K80879725	OC[C@@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2S(=O)(=O)c1ccccc1	CID:54664899	phase I
BRD-K53920100	OC[C@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2S(=O)(=O)c1ccccc1	CID:54664900	phase I
BRD-K53488338	OC[C@@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2S(=O)(=O)c1ccccc1	CID:54664901	phase I
BRD-K48150994	OC[C@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2S(=O)(=O)c1ccccc1	CID:54664902	phase I
BRD-K10362791	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)C1CCOCC1	CID:54664903	phase I
BRD-K07418207	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)C1CCOCC1	CID:54664904	phase I
BRD-K11528380	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)C1CCOCC1	CID:54664905	phase I
BRD-K12342133	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)C1CCOCC1	CID:54664906	phase I
BRD-K24469285	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C1=CCCCC1)C(=O)c1ccc2OCOc2c1	CID:54664907	phase I
BRD-K56399425	COc1cccc(c1)-c1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccccc1F	CID:54664908	phase I
BRD-K11258147	COc1cccc(c1)-c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1ccccc1F	CID:54664909	phase I
BRD-K75369250	COc1cccc(c1)-c1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccccc1F	CID:54664910	phase I
BRD-K69077316	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccc(F)cc1)C#Cc1ccccc1F	CID:54664911	phase I
BRD-K39709536	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccc(F)cc1)C#Cc1ccccc1F	CID:54664912	phase I
BRD-K79906422	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccc(F)cc1)C#Cc1ccccc1F	CID:54664913	phase I
BRD-K65677539	COc1cccc(c1)C#Cc1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccccc1F	CID:54664914	phase I
BRD-K77525326	COc1ccc(cc1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1cccc(OC)c1	CID:54664915	phase I
BRD-K21967348	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccncc1)-c1ccccc1	CID:54664916	phase I
BRD-K44363560	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccncc1)-c1ccccc1	CID:54664917	phase I
BRD-K17258761	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccncc1)-c1ccccc1	CID:54664918	phase I
BRD-K11236606	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccncc1)-c1ccccc1	CID:54664919	phase I
BRD-K53577657	OC[C@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)c1ccccc1F	CID:54664920	phase I
BRD-K47014407	OC[C@@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)c1ccccc1F	CID:54664921	phase I
BRD-K18722825	OC[C@@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)c1ccccc1F	CID:54664922	phase I
BRD-K82374143	OC[C@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)c1ccccc1F	CID:54664923	phase I
BRD-K65617968	COCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)-c1ccc(F)cc1	CID:54664924	phase I
BRD-K67943760	COCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@H]2CO)-c1ccc(F)cc1	CID:54664925	phase I
BRD-K55767217	COCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@H]2CO)-c1ccc(F)cc1	CID:54664926	phase I
BRD-K36588736	COCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@@H]2CO)-c1ccc(F)cc1	CID:54664927	phase I
BRD-K51133104	OC[C@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)Cc1ccncc1	CID:54664928	phase I
BRD-K36115238	OC[C@@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)Cc1ccncc1	CID:54664929	phase I
BRD-K51431550	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(c1)C#N)C(=O)CC1CC1	CID:54664930	phase I
BRD-K27272622	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(c1)C#N)C(=O)CC1CC1	CID:54664931	phase I
BRD-K73895377	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(c1)C#N)C(=O)CC1CC1	CID:54664932	phase I
BRD-K66253082	CCCC#Cc1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccccc1	CID:54664933	phase I
BRD-A26627799	COc1ccc(cc1)C#Cc1ccc2N(C)[C@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)C1=NC(C)C=N1	CID:54664934	phase I
BRD-A02726762	COc1ccc(cc1)C#Cc1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)C1=NC(C)C=N1	CID:54664935	phase I
BRD-K15226746	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1ccccc1F)-c1ccccc1	CID:54664936	phase I
BRD-K08594759	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1ccccc1F)-c1ccccc1	CID:54664937	phase I
BRD-K23240772	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccccc1F)-c1ccccc1	CID:54664938	phase I
BRD-K45358881	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2S(=O)(=O)c1ccccc1F)-c1ccccc1F	CID:54664939	phase I
BRD-K22935984	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2S(=O)(=O)c1ccccc1F)-c1ccccc1F	CID:54664940	phase I
BRD-K97166443	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2S(=O)(=O)c1ccccc1F)-c1ccccc1F	CID:54664941	phase I
BRD-K78207246	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2S(=O)(=O)c1ccccc1F)-c1ccccc1F	CID:54664942	phase I
BRD-K55330917	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN(Cc4nccs4)[C@H]3c2c1	CID:54664943	phase I
BRD-K91351577	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@H](CO)[C@H]3CCN(Cc4nccs4)[C@H]3c2c1	CID:54664944	phase I
BRD-K16673836	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN(Cc4nccs4)[C@@H]3c2c1	CID:54664945	phase I
BRD-K99182933	COCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccc(F)cc1	CID:54664946	phase I
BRD-K04232710	COCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccc(F)cc1	CID:54664947	phase I
BRD-K44598486	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccc(C)cc1	CID:54664948	phase I
BRD-K88504936	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1ccc(C)cc1	CID:54664949	phase I
BRD-K51395794	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1ccc(C)cc1	CID:54664950	phase I
BRD-K64741770	CN(C)C(=O)c1cccc(c1)-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1ccc(C)cc1	CID:54664951	phase I
BRD-K39244640	COc1ccc(cc1)C#Cc1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccncc1	CID:54664952	phase I
BRD-K97351331	COc1ccc(cc1)NC(=O)N1CC[C@@H]2[C@@H](CO)N(C)c3ccc(cc3[C@H]12)-c1cccc(c1)C(=O)N(C)C	CID:54664953	phase I
BRD-K82368009	COc1ccc(cc1)NC(=O)N1CC[C@H]2[C@H](CO)N(C)c3ccc(cc3[C@@H]12)-c1cccc(c1)C(=O)N(C)C	CID:54664954	phase I
BRD-K77165899	COc1ccccc1NC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)C#Cc1cccc(F)c1	CID:54664955	phase I
BRD-K89960860	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)C1CCCCC1	CID:54664956	phase I
BRD-K25031586	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)C1CCCCC1	CID:54664957	phase I
BRD-K29125789	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)C1CCCCC1	CID:54664958	phase I
BRD-K60828552	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)C1CCCCC1	CID:54664959	phase I
BRD-K80247389	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Cc1ccccc1	CID:54664960	phase I
BRD-K29150200	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)Cc1ccccc1	CID:54664961	phase I
BRD-K02823077	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Cc1ccccc1	CID:54664962	phase I
BRD-K29182094	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)Cc1ccccc1	CID:54664963	phase I
BRD-K67520049	COc1ccccc1S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)-c1ccc(cc1)C#N	CID:54664964	phase I
BRD-K22488594	COc1ccccc1S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)-c1ccc(cc1)C#N	CID:54664965	phase I
BRD-K55809413	COc1ccccc1S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)-c1ccc(cc1)C#N	CID:54664966	phase I
BRD-K49333293	COc1ccccc1S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)-c1ccc(cc1)C#N	CID:54664967	phase I
BRD-K21787157	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCCCC1)-c1ccc(cc1)C#N	CID:54664968	phase I
BRD-K52197325	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCCCC1)-c1ccc(cc1)C#N	CID:54664969	phase I
BRD-K25989885	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCCCC1)-c1ccc(cc1)C#N	CID:54664970	phase I
BRD-K72692763	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCCCC1)-c1ccc(cc1)C#N	CID:54664971	phase I
BRD-K84421421	COc1cccc(c1)C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)CC1CC1	CID:54664972	phase I
BRD-K95462612	COc1cccc(c1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C1=CCCCC1	CID:54664973	phase I
BRD-K78160105	COc1ccccc1CN1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccccc1	CID:54664974	phase I
BRD-K18260949	COc1ccccc1CN1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccccc1	CID:54664975	phase I
BRD-K99032206	COc1ccccc1CN1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccccc1	CID:54664976	phase I
BRD-K00183357	COc1ccccc1CN1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccccc1	CID:54664977	phase I
BRD-K72452617	Cc1ccccc1S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccccc1	CID:54664978	phase I
BRD-K39446093	Cc1ccccc1S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccccc1	CID:54664979	phase I
BRD-K31373683	Cc1ccccc1S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccccc1	CID:54664980	phase I
BRD-K80033497	Cc1ccccc1S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccccc1	CID:54664981	phase I
BRD-K13109628	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2Cc1ccc2OCOc2c1)-c1cccc(c1)C#N	CID:54664982	phase I
BRD-K62697007	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccc2OCOc2c1)-c1cccc(c1)C#N	CID:54664983	phase I
BRD-K83311737	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2Cc1ccc2OCOc2c1)-c1cccc(c1)C#N	CID:54664984	phase I
BRD-K68937579	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)c1cccc(F)c1	CID:54664985	phase I
BRD-K61762092	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)c1cccc(F)c1	CID:54664986	phase I
BRD-K93229898	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)c1cccc(F)c1	CID:54664987	phase I
BRD-K48853765	CC(C)NC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@H]2CO)C#Cc1ccccc1	CID:54664988	phase I
BRD-K74919500	CC(C)NC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)C#Cc1ccccc1	CID:54664989	phase I
BRD-K90219001	COc1ccc(cc1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@H]2CO)-c1ccc(F)cc1	CID:54664990	phase I
BRD-K88647644	COc1ccc(cc1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@H]2CO)-c1ccc(F)cc1	CID:54664991	phase I
BRD-K28991565	COc1ccc(cc1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)-c1ccc(F)cc1	CID:54664992	phase I
BRD-K16827616	COc1ccc(cc1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@@H]2CO)-c1ccc(F)cc1	CID:54664993	phase I
BRD-K14787141	COc1ccccc1CN1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C1=CCCCC1	CID:54664994	phase I
BRD-K45680746	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1cnccn1	CID:54664995	phase I
BRD-K11943259	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1cnccn1	CID:54664996	phase I
BRD-K70896405	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@H](CO)[C@H]3CCN(Cc4ccc5OCOc5c4)[C@H]3c2c1	CID:54664997	phase I
BRD-K22148752	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@@H](CO)[C@@H]3CCN(Cc4ccc5OCOc5c4)[C@@H]3c2c1	CID:54664998	phase I
BRD-K52721673	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@@H](CO)[C@H]3CCN(Cc4ccc5OCOc5c4)[C@H]3c2c1	CID:54664999	phase I
BRD-K19234078	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@H](CO)[C@@H]3CCN(Cc4ccc5OCOc5c4)[C@@H]3c2c1	CID:54665000	phase I
BRD-K67287181	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(c1)C#N)S(=O)(=O)c1ccccc1C	CID:54665001	phase I
BRD-K97898255	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(c1)C#N)S(=O)(=O)c1ccccc1C	CID:54665002	phase I
BRD-K17890048	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C#Cc1cccnc1)C(=O)Nc1cc(F)ccc1F	CID:54665003	phase I
BRD-K10589286	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)Cc1ccccc1)C1=CCCCC1	CID:54665004	phase I
BRD-K83448282	COc1ccc(cc1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)C#Cc1ccccc1OC	CID:54665005	phase I
BRD-K76880231	COc1ccc(cc1)C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCOCC1	CID:54665006	phase I
BRD-K03936430	COc1ccc(cc1)C#Cc1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)C1CCOCC1	CID:54665007	phase I
BRD-K17233740	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)Cc1ccccc1	CID:54665008	phase I
BRD-K14489740	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(Br)ccc12)C(=O)Cc1ccccc1	CID:54665009	phase I
BRD-K60918127	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(Br)ccc12)C(=O)Cc1ccccc1	CID:54665010	phase I
BRD-K83491689	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C1=CCCCC1)C(=O)C1CCCC1	CID:54665011	phase I
BRD-K98569658	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C1=CCCCC1)C(=O)C1CCCC1	CID:54665012	phase I
BRD-K10938308	Cc1ccc(cc1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccc(F)cc1	CID:54665013	phase I
BRD-K31678340	Cc1ccc(cc1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccc(F)cc1	CID:54665014	phase I
BRD-K19385772	Cc1ccc(cc1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccc(F)cc1	CID:54665015	phase I
BRD-K38544238	Cc1ccc(cc1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccc(F)cc1	CID:54665016	phase I
BRD-K90939315	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665017	phase I
BRD-K39267498	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665018	phase I
BRD-K39260562	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665019	phase I
BRD-K16796151	CN(C)C(=O)c1ccc(cc1)-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665020	phase I
BRD-K50822286	CCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@H]2CO)C#Cc1cccc(F)c1	CID:54665021	phase I
BRD-K69449860	CN(C)CC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)-c1ccc(cc1)C(=O)N(C)C	CID:54665022	phase I
BRD-K35101110	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccccc1F)-c1cccc(c1)C#N	CID:54665023	phase I
BRD-K20652606	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccccc1F)-c1cccc(c1)C#N	CID:54665024	phase I
BRD-K65385622	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1ccccc1F)-c1cccc(c1)C#N	CID:54665025	phase I
BRD-K96103104	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1ccccc1F)-c1cccc(c1)C#N	CID:54665026	phase I
BRD-K26586614	CCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccccc1	CID:54665027	phase I
BRD-K56832078	CCC(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N[C@H]2CO)C#Cc1ccccc1	CID:54665028	phase I
BRD-K44525591	CCC(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N[C@@H]2CO)C#Cc1ccccc1	CID:54665029	phase I
BRD-K95795676	CN(C)C(=O)c1ccc(cc1)-c1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCC1	CID:54665030	phase I
BRD-K06111933	CN(C)C(=O)c1ccc(cc1)-c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)C1CCC1	CID:54665031	phase I
BRD-K05858751	CN(C)C(=O)c1ccc(cc1)-c1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCC1	CID:54665032	phase I
BRD-K80494270	CN(C)C(=O)c1ccc(cc1)-c1ccc2N(C)[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)C1CCC1	CID:54665033	phase I
BRD-A35430844	CC1C=NC(=N1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@@H]2CO)C1=CCCCC1	CID:54665034	phase I
BRD-A53271750	CC1C=NC(=N1)S(=O)(=O)N1CC[C@H]2[C@@H]1c1cc(ccc1N(C)[C@H]2CO)C1=CCCCC1	CID:54665035	phase I
BRD-A41228941	CC1C=NC(=N1)S(=O)(=O)N1CC[C@@H]2[C@H]1c1cc(ccc1N(C)[C@@H]2CO)C1=CCCCC1	CID:54665036	phase I
BRD-K02717912	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)c1ccccc1F	CID:54665037	phase I
BRD-K01615361	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)c1ccccc1F	CID:54665038	phase I
BRD-K11221750	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)c1ccccc1F	CID:54665039	phase I
BRD-K78959251	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)c1ccccc1F	CID:54665040	phase I
BRD-K22244182	COc1ccccc1-c1ccc2N(C)[C@@H](CO)[C@H]3CCN(C(=O)CN4CCOCC4)[C@H]3c2c1	CID:54665041	phase I
BRD-K63806140	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccc(cc1)C#N)C(C)=O	CID:54665042	phase I
BRD-K34030207	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccc(cc1)C#N)C(C)=O	CID:54665043	phase I
BRD-K21642579	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccc(cc1)C#N)C(C)=O	CID:54665044	phase I
BRD-K06511061	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccc(cc1)C#N)C(C)=O	CID:54665045	phase I
BRD-K19821569	COc1ccccc1-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccc2OCOc2c1	CID:54665046	phase I
BRD-K21159035	OC[C@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)c1ccccn1	CID:54665047	phase I
BRD-K22166546	OC[C@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)c1ccccn1	CID:54665048	phase I
BRD-K74452256	OC[C@@H]1Nc2ccc(Br)cc2[C@@H]2[C@H]1CCN2C(=O)c1ccccn1	CID:54665049	phase I
BRD-K05387676	OC[C@@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)c1ccccn1	CID:54665050	phase I
BRD-K78217164	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccccc1F)S(=O)(=O)c1cccc(C)c1	CID:54665051	phase I
BRD-K15627143	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccccc1F)S(=O)(=O)c1cccc(C)c1	CID:54665052	phase I
BRD-K21448715	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1ccccc1F)S(=O)(=O)c1cccc(C)c1	CID:54665053	phase I
BRD-K92827116	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1ccccc1F)S(=O)(=O)c1cccc(C)c1	CID:54665054	phase I
BRD-K50795243	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)Cc1ccncc1)-c1ccccc1F	CID:54665055	phase I
BRD-K48183516	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)Cc1ccncc1)-c1ccccc1F	CID:54665056	phase I
BRD-K84145110	COc1cccc(c1)-c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1ccc2OCOc2c1	CID:54665057	phase I
BRD-K79998171	COc1cccc(c1)-c1ccc2N(C)[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1ccc2OCOc2c1	CID:54665058	phase I
BRD-K66626628	COc1cccc(c1)-c1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccc2OCOc2c1	CID:54665059	phase I
BRD-K55507662	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCOCC1)-c1cccc(F)c1	CID:54665060	phase I
BRD-K98225498	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCOCC1)-c1cccc(F)c1	CID:54665061	phase I
BRD-K44452237	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCOCC1)-c1cccc(F)c1	CID:54665062	phase I
BRD-K48752687	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCOCC1)-c1cccc(F)c1	CID:54665063	phase I
BRD-K65598260	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)Cc1cccnc1	CID:54665064	phase I
BRD-K08884733	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)Cc1cccnc1	CID:54665065	phase I
BRD-K92132228	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)Cc1cccnc1	CID:54665066	phase I
BRD-K51888384	CN1[C@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)-c1cccc(F)c1)C(=O)Cc1cccnc1	CID:54665067	phase I
BRD-K33385950	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cccnc1)-c1ccc(cc1)C#N	CID:54665068	phase I
BRD-K83242582	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1ccc(F)cc1	CID:54665069	phase I
BRD-K69048763	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccc(F)cc1	CID:54665070	phase I
BRD-K62774106	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1ccc(F)cc1	CID:54665071	phase I
BRD-K19268781	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1ccc(F)cc1	CID:54665072	phase I
BRD-K74327009	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)CC1CC1)-c1ccccc1	CID:54665073	phase I
BRD-K75976016	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)CC1CC1)-c1ccccc1	CID:54665074	phase I
BRD-K14567384	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)CC1CC1)-c1ccccc1	CID:54665075	phase I
BRD-K37935437	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)CC1CC1)-c1ccccc1	CID:54665076	phase I
BRD-K28107603	COc1ccc(cc1)-c1ccc2N(C)[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)Nc1ccccc1OC	CID:54665077	phase I
BRD-K16914190	COc1ccc(cc1)-c1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)Nc1ccccc1OC	CID:54665078	phase I
BRD-K80806019	CN1[C@@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C#Cc1cccnc1)S(=O)(=O)c1ccccc1F	CID:54665079	phase I
BRD-K58893765	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C#Cc1cccnc1)S(=O)(=O)c1ccccc1F	CID:54665080	phase I
BRD-K39647256	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C#Cc1cccnc1)S(=O)(=O)c1ccccc1F	CID:54665081	phase I
BRD-K42363645	COc1ccc(cc1)C#Cc1ccc2N(C)[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)CN1CCOCC1	CID:54665082	phase I
BRD-K30820123	COc1ccc(cc1)C#Cc1ccc2N(C)[C@@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)CN1CCOCC1	CID:54665083	phase I
BRD-K16063772	COc1ccc(cc1)C#Cc1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1cccc(F)c1	CID:54665084	phase I
BRD-K79998087	COc1ccc(cc1)C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)c1cccc(F)c1	CID:54665085	phase I
BRD-K96306575	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cnccn1)-c1ccccc1F	CID:54665086	phase I
BRD-K84770655	OC[C@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cnccn1)-c1ccccc1F	CID:54665087	phase I
BRD-K87026780	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1cnccn1)-c1ccccc1F	CID:54665088	phase I
BRD-K33171119	OC[C@@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1cnccn1)-c1ccccc1F	CID:54665089	phase I
BRD-K89830699	COc1ccc(NC(=O)N2CC[C@H]3[C@@H]2c2cc(Br)ccc2N(C)[C@H]3CO)cc1	CID:54665090	phase I
BRD-K03958924	COc1ccc(NC(=O)N2CC[C@@H]3[C@H]2c2cc(Br)ccc2N(C)[C@@H]3CO)cc1	CID:54665091	phase I
BRD-K63711119	COc1ccc(NC(=O)N2CC[C@@H]3[C@H]2c2cc(Br)ccc2N(C)[C@H]3CO)cc1	CID:54665092	phase I
BRD-K39187484	COc1ccc(NC(=O)N2CC[C@H]3[C@@H]2c2cc(Br)ccc2N(C)[C@@H]3CO)cc1	CID:54665093	phase I
BRD-K62767164	CC(C)NC(=O)N1CC[C@@H]2[C@H]1c1cc(Br)ccc1N(C)[C@@H]2CO	CID:54665094	phase I
BRD-K41721525	CC(C)NC(=O)N1CC[C@H]2[C@@H]1c1cc(Br)ccc1N(C)[C@@H]2CO	CID:54665095	phase I
BRD-K72947048	CC(C)NC(=O)N1CC[C@@H]2[C@H]1c1cc(Br)ccc1N(C)[C@H]2CO	CID:54665096	phase I
BRD-K12977357	CC(C)NC(=O)N1CC[C@H]2[C@@H]1c1cc(Br)ccc1N(C)[C@H]2CO	CID:54665097	phase I
BRD-K35654724	COc1cccc(c1)-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665098	phase I
BRD-K07888312	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665099	phase I
BRD-K32290015	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)S(=O)(=O)c1cn(C)cn1	CID:54665100	phase I
BRD-K74889969	CC(=O)N1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1ccccc1	CID:54666385	phase I
BRD-K70330256	CC(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1ccccc1	CID:54666386	phase I
BRD-K85174275	OC[C@H]1[C@@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666387	phase I
BRD-K27209353	OC[C@@H]1[C@@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666388	phase I
BRD-K75992528	OC[C@H]1[C@@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666389	phase I
BRD-K45615006	OC[C@H]1[C@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666390	phase I
BRD-K80913219	OC[C@H]1[C@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666391	phase I
BRD-K14478589	OC[C@@H]1[C@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666392	phase I
BRD-K61793536	OC[C@@H]1[C@@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666393	phase I
BRD-K29252735	OC[C@@H]1[C@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666394	phase I
BRD-K95790481	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666395	phase I
BRD-K27084624	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666396	phase I
BRD-K70690367	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666397	phase I
BRD-K56366698	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666398	phase I
BRD-K69197522	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666399	phase I
BRD-K22265882	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666400	phase I
BRD-K03006541	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)C#CCC(C)C	CID:54666402	phase I
BRD-K43073442	OC[C@@H]1[C@@H]([C@H]2CNCCCCN12)c1ccc(Br)cc1	CID:54666407	phase I
BRD-K58873027	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CCC(F)(F)F)C[C@@H]12	CID:54666408	phase I
BRD-K44218044	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CCC(F)(F)F)C[C@@H]12	CID:54666409	phase I
BRD-K29426933	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CCC(F)(F)F)C[C@H]12	CID:54666410	phase I
BRD-K24112840	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CCC(F)(F)F)C[C@H]12	CID:54666411	phase I
BRD-K52758732	OC[C@H]1[C@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666412	phase I
BRD-K13234528	OC[C@@H]1[C@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666413	phase I
BRD-K58791909	OC[C@H]1[C@@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666414	phase I
BRD-K27366480	OC[C@H]1[C@@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666415	phase I
BRD-K07786204	OC[C@@H]1[C@@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666416	phase I
BRD-K77608452	OC[C@@H]1[C@@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666417	phase I
BRD-K29651341	OC[C@@H]1[C@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666418	phase I
BRD-K03043432	OC[C@H]1[C@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)C#Cc1ccccc1F	CID:54666419	phase I
BRD-K20203275	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666420	phase I
BRD-K02131961	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666421	phase I
BRD-K73045999	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666422	phase I
BRD-K43947390	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666423	phase I
BRD-K02931142	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666424	phase I
BRD-K91868345	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666425	phase I
BRD-K83507699	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666426	phase I
BRD-K87720600	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)C#Cc1cccnc1	CID:54666427	phase I
BRD-K20658410	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1cccs1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666428	phase I
BRD-K20449903	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1cccs1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666429	phase I
BRD-K42919101	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1cccs1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666430	phase I
BRD-K00842536	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1cccs1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666431	phase I
BRD-K50827439	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1cccs1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666432	phase I
BRD-K85297392	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1cccs1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666433	phase I
BRD-K72814870	COc1cccc(CN2CCCCN3[C@@H](CO)[C@H]([C@H]3C2)c2ccc(cc2)-c2cccnc2)c1	CID:54666434	phase I
BRD-K41520872	COc1cccc(CN2CCCCN3[C@@H](CO)[C@@H]([C@H]3C2)c2ccc(cc2)-c2cccnc2)c1	CID:54666435	phase I
BRD-K45025380	COc1cccc(CN2CCCCN3[C@H](CO)[C@H]([C@H]3C2)c2ccc(cc2)-c2cccnc2)c1	CID:54666436	phase I
BRD-K49156662	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666437	phase I
BRD-K66123981	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666438	phase I
BRD-K66808842	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666439	phase I
BRD-K48566675	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666440	phase I
BRD-K49916352	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666441	phase I
BRD-K25642832	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666442	phase I
BRD-K84696632	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666443	phase I
BRD-K52421542	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)-c1cncnc1	CID:54666444	phase I
BRD-K63851915	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)NC1CCCC1	CID:54666445	phase I
BRD-K79149684	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)NC1CCCC1	CID:54666446	phase I
BRD-K93662714	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)NC1CCCC1	CID:54666447	phase I
BRD-K40155511	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)NC1CCCC1	CID:54666448	phase I
BRD-K44339679	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)NC1CCCC1	CID:54666449	phase I
BRD-K12067499	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)NC1CCCC1	CID:54666450	phase I
BRD-K33685212	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)NC1CCCC1	CID:54666451	phase I
BRD-K89000385	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)NC1CCCC1	CID:54666452	phase I
BRD-K61382850	OC[C@@H]1[C@H]([C@@H]2CN(Cc3ccccc3F)CCCCN12)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666453	phase I
BRD-K15419834	OC[C@H]1[C@@H]([C@H]2CN(Cc3ccccc3F)CCCCN12)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666454	phase I
BRD-K69711545	OC[C@H]1[C@H]([C@H]2CN(Cc3ccccc3F)CCCCN12)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666455	phase I
BRD-K43472599	OC[C@@H]1[C@H]([C@H]2CN(Cc3ccccc3F)CCCCN12)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666456	phase I
BRD-K77301526	OC[C@@H]1[C@@H]([C@@H]2CN(Cc3ccccc3F)CCCCN12)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666457	phase I
BRD-K85438393	CCS(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)C#Cc1ccccn1	CID:54666458	phase I
BRD-K43955935	CCS(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)C#Cc1ccccn1	CID:54666459	phase I
BRD-K38627245	CCS(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)C#Cc1ccccn1	CID:54666460	phase I
BRD-K61285042	CCS(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)C#Cc1ccccn1	CID:54666461	phase I
BRD-K62702428	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666462	phase I
BRD-K87790979	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666463	phase I
BRD-K82637111	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666464	phase I
BRD-K13064257	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666465	phase I
BRD-K81438145	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666466	phase I
BRD-K80427968	C[C@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666467	phase I
BRD-K46477974	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666468	phase I
BRD-K10422753	C[C@H](O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666469	phase I
BRD-K94274196	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666470	phase I
BRD-K21741022	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666471	phase I
BRD-K47788798	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666472	phase I
BRD-K86925364	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666473	phase I
BRD-K42618289	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc2OCOc2c1	CID:54666474	phase I
BRD-K58446572	C[C@H](O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666475	phase I
BRD-K07448100	C[C@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666476	phase I
BRD-K00868395	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc2OCOc2c1	CID:54666477	phase I
BRD-K24820372	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cc(F)ccc1F)c1ccc(cc1)C1=CCCCC1	CID:54666478	phase I
BRD-K26542939	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cc(F)ccc1F)c1ccc(cc1)C1=CCCCC1	CID:54666479	phase I
BRD-K90544854	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)Nc1cc(F)ccc1F)c1ccc(cc1)C1=CCCCC1	CID:54666480	phase I
BRD-K33907901	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CCC)C[C@H]12	CID:54666481	phase I
BRD-K21668646	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CCC)C[C@@H]12	CID:54666482	phase I
BRD-K97175782	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1cccnc1	CID:54666483	phase I
BRD-K88231082	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1cccnc1	CID:54666484	phase I
BRD-K92476250	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1cccnc1	CID:54666485	phase I
BRD-K50795058	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1cccnc1	CID:54666486	phase I
BRD-K64892842	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1cccnc1	CID:54666487	phase I
BRD-K28066515	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1cccnc1	CID:54666488	phase I
BRD-K95351169	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1cccnc1	CID:54666489	phase I
BRD-K82469533	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1cccnc1	CID:54666490	phase I
BRD-K82276260	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccccn1	CID:54666491	phase I
BRD-K63614890	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccccn1	CID:54666492	phase I
BRD-K83625314	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccccn1	CID:54666493	phase I
BRD-K74833731	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccccn1	CID:54666494	phase I
BRD-K24956360	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccccn1	CID:54666495	phase I
BRD-K04890734	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccccn1	CID:54666496	phase I
BRD-K30211346	OC[C@H]1[C@H]([C@@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666497	phase I
BRD-K65392546	OC[C@H]1[C@H]([C@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666498	phase I
BRD-K54642063	OC[C@@H]1[C@@H]([C@@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666499	phase I
BRD-K56450018	OC[C@H]1[C@@H]([C@@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666500	phase I
BRD-K42132006	OC[C@@H]1[C@H]([C@@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666501	phase I
BRD-K00568440	OC[C@H]1[C@@H]([C@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666502	phase I
BRD-K92455228	OC[C@@H]1[C@H]([C@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666503	phase I
BRD-K37127287	OC[C@@H]1[C@@H]([C@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(Br)cc1	CID:54666504	phase I
BRD-K79138145	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666505	phase I
BRD-K99311353	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666506	phase I
BRD-K10268154	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666507	phase I
BRD-K85698453	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666508	phase I
BRD-K19645792	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666509	phase I
BRD-K45038844	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666510	phase I
BRD-K90168790	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666511	phase I
BRD-K45861923	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)CN1CCOCC1)c1ccc(Br)cc1	CID:54666512	phase I
BRD-K23647039	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)Cc1ccccc1	CID:54666513	phase I
BRD-K92048968	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)Cc1ccccc1	CID:54666514	phase I
BRD-K48421284	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)Cc1ccccc1	CID:54666515	phase I
BRD-K62600822	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)Cc1ccccc1	CID:54666516	phase I
BRD-K19288011	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)Cc1ccccc1	CID:54666517	phase I
BRD-K86764949	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)Cc1ccccc1	CID:54666518	phase I
BRD-K04239420	OC[C@H]1[C@H]([C@@H]2CN(Cc3ccncc3)CCCCN12)c1ccc(cc1)C1=CCCC1	CID:54666519	phase I
BRD-K88590679	OC[C@@H]1[C@@H]([C@H]2CN(Cc3ccncc3)CCCCN12)c1ccc(cc1)C1=CCCC1	CID:54666520	phase I
BRD-K18024030	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CCC1	CID:54666521	phase I
BRD-K02223457	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CCC1	CID:54666522	phase I
BRD-K93036747	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CCC1	CID:54666523	phase I
BRD-K36773541	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CCC1	CID:54666524	phase I
BRD-K18300217	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CCC1	CID:54666525	phase I
BRD-K43168251	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CCC1	CID:54666526	phase I
BRD-K64716911	COc1ccccc1C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CCC1	CID:54666527	phase I
BRD-K14193256	COc1ccccc1C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CCC1	CID:54666528	phase I
BRD-K80779790	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1F	CID:54666529	phase I
BRD-K01966678	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1F	CID:54666530	phase I
BRD-K93081895	Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1F	CID:54666531	phase I
BRD-K68855692	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1F	CID:54666532	phase I
BRD-K26945408	Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1F	CID:54666533	phase I
BRD-K73008154	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1F	CID:54666534	phase I
BRD-K20154295	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C)C[C@@H]12	CID:54666535	phase I
BRD-K80472040	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C)C[C@@H]12	CID:54666536	phase I
BRD-K14245765	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C)C[C@H]12	CID:54666537	phase I
BRD-K87931486	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C)C[C@@H]12	CID:54666538	phase I
BRD-K46297593	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C)C[C@@H]12	CID:54666539	phase I
BRD-K68078697	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C)C[C@H]12	CID:54666540	phase I
BRD-K50176356	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C)C[C@H]12	CID:54666541	phase I
BRD-K97372925	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666542	phase I
BRD-K55569739	COc1ccc(NC(=O)N2CCCCN3[C@H](CO)[C@H]([C@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666543	phase I
BRD-K64469479	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@H]([C@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666544	phase I
BRD-K68638497	COc1ccc(NC(=O)N2CCCCN3[C@H](CO)[C@@H]([C@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666545	phase I
BRD-K92012565	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666546	phase I
BRD-K79552375	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@H]([C@@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666547	phase I
BRD-K66898048	COc1ccc(NC(=O)N2CCCCN3[C@H](CO)[C@H]([C@@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666548	phase I
BRD-K32088574	COc1ccc(NC(=O)N2CCCCN3[C@H](CO)[C@@H]([C@@H]3C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:54666549	phase I
BRD-K33312838	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666550	phase I
BRD-K46707147	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666551	phase I
BRD-K43708940	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666552	phase I
BRD-K04123911	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666553	phase I
BRD-K57565683	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666554	phase I
BRD-K36826042	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666555	phase I
BRD-K27242547	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666556	phase I
BRD-K94993557	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)c1cccc(F)c1)c1ccc(cc1)C#CC1(O)CCCC1	CID:54666557	phase I
BRD-K35842817	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54666558	phase I
BRD-K45327589	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54666559	phase I
BRD-K62409349	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54666560	phase I
BRD-K69500068	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54666561	phase I
BRD-K58490891	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54666562	phase I
BRD-K28344523	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54666563	phase I
BRD-K10743257	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54666564	phase I
BRD-K24755528	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54666565	phase I
BRD-K36826784	COc1ccccc1NC(=O)N1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666566	phase I
BRD-K43713542	COc1ccccc1NC(=O)N1CCCCN2[C@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666567	phase I
BRD-K63667213	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666568	phase I
BRD-K05639119	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666569	phase I
BRD-K74381836	COc1ccccc1NC(=O)N1CCCCN2[C@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666570	phase I
BRD-K31444894	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666571	phase I
BRD-K58860003	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666572	phase I
BRD-K11432829	COc1ccccc1NC(=O)N1CCCCN2[C@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666573	phase I
BRD-K87920770	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1cccnc1	CID:54666574	phase I
BRD-K98370047	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1cccnc1	CID:54666575	phase I
BRD-K73143149	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1cccnc1	CID:54666576	phase I
BRD-K21136828	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1cccnc1	CID:54666577	phase I
BRD-K27425684	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1cccnc1	CID:54666578	phase I
BRD-K98245706	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1cccnc1	CID:54666579	phase I
BRD-K80236176	COc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1cccnc1	CID:54666580	phase I
BRD-K18483660	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1cccnc1	CID:54666581	phase I
BRD-K30857073	CC(C)(O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(C)(=O)=O	CID:54666582	phase I
BRD-K30437434	CC(C)(O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(C)(=O)=O	CID:54666583	phase I
BRD-K31906558	CC(C)(O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(C)(=O)=O	CID:54666584	phase I
BRD-K77874118	CC(C)(O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)S(C)(=O)=O	CID:54666585	phase I
BRD-K41363665	CC(C)(O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(C)(=O)=O	CID:54666586	phase I
BRD-K45472161	CC(C)(O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)S(C)(=O)=O	CID:54666587	phase I
BRD-K76237504	CC(C)(O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(C)(=O)=O	CID:54666588	phase I
BRD-K40408048	CC(C)(O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(C)(=O)=O	CID:54666589	phase I
BRD-K22282523	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1C	CID:54666590	phase I
BRD-K05729886	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1C	CID:54666591	phase I
BRD-K84499554	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1C	CID:54666592	phase I
BRD-K73907604	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1C	CID:54666593	phase I
BRD-K33449128	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1C	CID:54666594	phase I
BRD-K58292285	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1C	CID:54666595	phase I
BRD-K73676286	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1C	CID:54666596	phase I
BRD-K67470245	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)S(=O)(=O)c1ccccc1C	CID:54666597	phase I
BRD-K72500499	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1F	CID:54666598	phase I
BRD-K65927019	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1F	CID:54666599	phase I
BRD-K25193669	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1F	CID:54666600	phase I
BRD-K68756928	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1F	CID:54666601	phase I
BRD-K44485049	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1F	CID:54666602	phase I
BRD-K62357899	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1F	CID:54666603	phase I
BRD-K10806720	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1F	CID:54666604	phase I
BRD-K10082717	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1F	CID:54666605	phase I
BRD-K53539078	CCS(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:54666606	phase I
BRD-K09620519	CCS(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:54666607	phase I
BRD-K77800502	CCS(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:54666608	phase I
BRD-K97143621	CCS(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:54666609	phase I
BRD-K20490522	CCS(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:54666610	phase I
BRD-K07129792	CCS(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C)C	CID:54666611	phase I
BRD-K05841102	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccncc1	CID:54666612	phase I
BRD-K94159777	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccncc1	CID:54666613	phase I
BRD-K74085580	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccncc1	CID:54666614	phase I
BRD-K00540336	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccncc1	CID:54666615	phase I
BRD-K49483184	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccncc1	CID:54666616	phase I
BRD-K45891353	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccncc1	CID:54666617	phase I
BRD-K73233900	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Cc1ccncc1	CID:54666618	phase I
BRD-K17854785	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)\C=C\C	CID:54666619	phase I
BRD-K47033137	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)\C=C\C	CID:54666620	phase I
BRD-K77320816	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)\C=C\C	CID:54666621	phase I
BRD-K59606716	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)\C=C\C	CID:54666622	phase I
BRD-K01409647	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)\C=C\C	CID:54666623	phase I
BRD-K57556784	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)\C=C\C	CID:54666624	phase I
BRD-K63158888	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)\C=C\C	CID:54666625	phase I
BRD-K64062072	COc1ccc(cc1)S(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)\C=C\C	CID:54666626	phase I
BRD-K43540029	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666627	phase I
BRD-K40311869	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666628	phase I
BRD-K48995011	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666629	phase I
BRD-K25866746	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666630	phase I
BRD-K51358551	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666631	phase I
BRD-K43234208	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666632	phase I
BRD-K94074846	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666633	phase I
BRD-K06816133	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)C#CC1CCCC1	CID:54666634	phase I
BRD-K23954640	OC[C@H]1[C@@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666635	phase I
BRD-K26755359	OC[C@H]1[C@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666636	phase I
BRD-K28594113	OC[C@H]1[C@@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666637	phase I
BRD-K46183911	OC[C@@H]1[C@@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666638	phase I
BRD-K26499328	OC[C@@H]1[C@@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666639	phase I
BRD-K02560333	OC[C@H]1[C@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666640	phase I
BRD-K93944867	OC[C@@H]1[C@H]([C@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666641	phase I
BRD-K07257078	OC[C@@H]1[C@H]([C@@H]2CN(Cc3cncnc3)CCCCN12)c1ccc(cc1)-c1ccccc1F	CID:54666642	phase I
BRD-K95583033	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccc(F)cc1	CID:54666643	phase I
BRD-K05502425	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccc(F)cc1	CID:54666644	phase I
BRD-K91946056	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccc(F)cc1	CID:54666645	phase I
BRD-K75514176	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccc(F)cc1	CID:54666646	phase I
BRD-K85815049	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccc(F)cc1	CID:54666647	phase I
BRD-K56215828	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccc(F)cc1	CID:54666648	phase I
BRD-K56104093	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccc(F)cc1	CID:54666649	phase I
BRD-K40910787	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccc(F)cc1	CID:54666650	phase I
BRD-K52418167	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(Cc3ccncc3)C[C@@H]12	CID:54666651	phase I
BRD-K14079892	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(Cc3ccncc3)C[C@H]12	CID:54666652	phase I
BRD-K28956095	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(Cc3ccncc3)C[C@H]12	CID:54666653	phase I
BRD-K74954602	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(Cc3ccncc3)C[C@@H]12	CID:54666654	phase I
BRD-K90194420	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(Cc3ccncc3)C[C@H]12	CID:54666655	phase I
BRD-K46943684	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666656	phase I
BRD-K14471579	OC[C@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666657	phase I
BRD-K45889441	OC[C@@H]1[C@H]([C@@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666658	phase I
BRD-K14697199	OC[C@@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666659	phase I
BRD-K07778122	OC[C@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666660	phase I
BRD-K99536165	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666661	phase I
BRD-K76764002	OC[C@@H]1[C@@H]([C@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666662	phase I
BRD-K30275524	OC[C@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)NC1CCCC1)c1ccc(cc1)-c1cccnc1	CID:54666663	phase I
BRD-K95582125	CN1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666664	phase I
BRD-K39827602	CN1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666665	phase I
BRD-K13774281	CN1CCCCN2[C@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666666	phase I
BRD-K79793579	CN1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666667	phase I
BRD-K62450654	CN1CCCCN2[C@H](CO)[C@@H]([C@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666668	phase I
BRD-K47443018	CN1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666669	phase I
BRD-K53107914	CN1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666670	phase I
BRD-K53295358	CN1CCCCN2[C@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1ccc(F)cc1	CID:54666671	phase I
BRD-K49477330	CN(C)CC(=O)N1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666672	phase I
BRD-K55767450	CN(C)CC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666673	phase I
BRD-K87125912	CN(C)CC(=O)N1CCCCN2[C@H](CO)[C@@H]([C@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666674	phase I
BRD-K97194822	CN(C)CC(=O)N1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666675	phase I
BRD-K84447616	CN(C)CC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666676	phase I
BRD-K74461819	CN(C)CC(=O)N1CCCCN2[C@H](CO)[C@H]([C@@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666677	phase I
BRD-K91663486	CN(C)CC(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(\C=C\c2ccccc2)cc1	CID:54666678	phase I
BRD-K89824424	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc(F)cc1	CID:54666679	phase I
BRD-K95695488	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc(F)cc1	CID:54666680	phase I
BRD-K90463980	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc(F)cc1	CID:54666681	phase I
BRD-K73423175	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc(F)cc1	CID:54666682	phase I
BRD-K69048063	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc(F)cc1	CID:54666683	phase I
BRD-K60172814	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)c1ccc(F)cc1	CID:54666684	phase I
BRD-K99438709	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc(F)cc1	CID:54666685	phase I
BRD-K11071576	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)c1ccc(F)cc1	CID:54666686	phase I
BRD-K63423329	OC[C@H]1[C@H]([C@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666687	phase I
BRD-K34104948	OC[C@H]1[C@@H]([C@@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666688	phase I
BRD-K05132143	OC[C@@H]1[C@@H]([C@@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666689	phase I
BRD-K07689498	OC[C@H]1[C@H]([C@@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666690	phase I
BRD-K68906258	OC[C@@H]1[C@H]([C@@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666691	phase I
BRD-K30373477	OC[C@@H]1[C@@H]([C@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666692	phase I
BRD-K41335306	OC[C@H]1[C@@H]([C@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666693	phase I
BRD-K43122204	OC[C@@H]1[C@H]([C@H]2CN(Cc3cccnc3)CCCCN12)c1ccc(\C=C\c2ccccc2)cc1	CID:54666694	phase I
BRD-K59194364	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1	CID:54666695	phase I
BRD-K83003953	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1	CID:54666696	phase I
BRD-K18241892	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1	CID:54666697	phase I
BRD-K53134312	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)Nc1ccccc1	CID:54666698	phase I
BRD-K46476822	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1	CID:54666699	phase I
BRD-K14095788	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)Nc1ccccc1	CID:54666700	phase I
BRD-K09064372	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)S(=O)(=O)c1ccccc1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54666790	phase I
BRD-K71053953	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Cc1ccccc1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:54666820	phase I
BRD-K85756431	Cc1ccccc1S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1cccnc1	CID:54666825	phase I
BRD-K77399257	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@@H]3C2)c2ccc(cc2)C#Cc2ccccn2)cc1	CID:54666869	phase I
BRD-K85943445	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(Cc3cccnc3)C[C@@H]12	CID:54666906	phase I
BRD-K23021002	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(Cc3cccnc3)C[C@H]12	CID:54666907	phase I
BRD-K69392286	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:54667012	phase I
BRD-K67575276	OC[C@H]1[C@H]([C@@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54667051	phase I
BRD-K00645031	OC[C@H]1[C@@H]([C@@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54667053	phase I
BRD-K73952419	OC[C@@H]1[C@H]([C@H]2CN(Cc3ccccn3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54667054	phase I
BRD-K79797318	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@@H]3C2)c2ccc(cc2)C#CCC(C)C)cc1	CID:54667061	phase I
BRD-K35451338	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54667072	phase I
BRD-K58611676	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54667074	phase I
BRD-K40189164	CN1CCCCN2[C@@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1cccnc1	CID:54667335	phase I
BRD-K06087483	CN1CCCCN2[C@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccnc1	CID:54667339	phase I
BRD-K62374815	OC[C@@H]1[C@@H]([C@@H]2CN(CC3CC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54667344	phase I
BRD-K93380196	OC[C@H]1[C@H]([C@H]2CN(CC3CC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54667347	phase I
BRD-K59675434	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Cc1cccnc1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54667389	phase I
BRD-K72765491	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1cccc(F)c1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54667404	phase I
BRD-K27465870	Cc1ccccc1S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(F)c1	CID:54667575	phase I
BRD-K23651361	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1	CID:54667764	phase I
BRD-K96072301	CS(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54667769	phase I
BRD-K73281599	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(F)c1	CID:54667822	phase I
BRD-K21953167	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(Cc3ccncc3)C[C@H]12	CID:54667931	phase I
BRD-K15181238	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@@H]3C2)c2ccc(\C=C\C)cc2)cc1	CID:54667998	phase I
BRD-K88081783	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)Cc1ccccn1	CID:54668348	phase I
BRD-K92412252	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1C	CID:54668530	phase I
BRD-K44791842	CCS(=O)(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54668617	phase I
BRD-K61551326	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)C#Cc1ccccc1	CID:54668627	phase I
BRD-K31441776	Cc1ccccc1S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1cncnc1	CID:54668813	phase I
BRD-K74489738	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Cc1ccncc1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54668868	phase I
BRD-K11264391	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@@H]3C2)c2ccc(cc2)-c2ccccc2C)cc1	CID:54668907	phase I
BRD-K35747889	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)S(=O)(=O)c1ccccc1C	CID:54668959	phase I
BRD-K85873301	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CCC(F)(F)F)C[C@H]12	CID:54668984	phase I
BRD-K62511324	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CCC(F)(F)F)C[C@@H]12	CID:54668986	phase I
BRD-K45185691	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CCC(F)(F)F)C[C@H]12	CID:54668988	phase I
BRD-K41008930	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CCC(F)(F)F)C[C@@H]12	CID:54668989	phase I
BRD-K35208671	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CCC(F)(F)F)C[C@@H]12	CID:54668991	phase I
BRD-K07604665	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1ccccc1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54669029	phase I
BRD-K29392278	COc1cccc(c1)S(=O)(=O)N1CCCCN2[C@H](CO)[C@H]([C@H]2C1)c1ccc(cc1)-c1cncnc1	CID:54669037	phase I
BRD-K60398284	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Cc1ccccc1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54669111	phase I
BRD-K11672960	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1cccc(C)c1	CID:54669118	phase I
BRD-K29771961	OC[C@H]1[C@@H]([C@@H]2CN(CCCCN12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(c1)C#N	CID:54669151	phase I
BRD-K51750373	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(Cc3cccnc3)C[C@@H]12	CID:54669183	phase I
BRD-K57977694	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(Cc3cccnc3)C[C@H]12	CID:54669184	phase I
BRD-K48805623	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(Cc3cccnc3)C[C@@H]12	CID:54669187	phase I
BRD-K90660470	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54669268	phase I
BRD-K63476888	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54669269	phase I
BRD-K14020943	C[C@@H](O)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54669270	phase I
BRD-K82021299	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54669271	phase I
BRD-K04013642	C[C@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54669272	phase I
BRD-K20807411	C[C@H](O)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54669275	phase I
BRD-K25699844	C[C@@H](O)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@H]12	CID:54669276	phase I
BRD-K55623459	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CC3CCOCC3)C[C@@H]12	CID:54669290	phase I
BRD-K97255584	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CC3CC3)C[C@H]12	CID:54669301	phase I
BRD-K41899231	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CC3)C[C@@H]12	CID:54669302	phase I
BRD-K93203589	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CC3CC3)C[C@H]12	CID:54669303	phase I
BRD-K58601216	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(CC3CC3)C[C@@H]12	CID:54669304	phase I
BRD-K82379643	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CC3)C[C@H]12	CID:54669305	phase I
BRD-K09989112	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(CC3CC3)C[C@H]12	CID:54669306	phase I
BRD-K01312966	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2CCCCN(CC3CC3)C[C@@H]12	CID:54669307	phase I
BRD-K25257305	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(CC3CC3)C[C@@H]12	CID:54669308	phase I
BRD-K76485827	OC[C@@H]1[C@@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669309	phase I
BRD-K07695007	OC[C@H]1[C@@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669310	phase I
BRD-K36909552	OC[C@H]1[C@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669312	phase I
BRD-K18390106	OC[C@@H]1[C@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669313	phase I
BRD-K14090520	OC[C@@H]1[C@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669314	phase I
BRD-K57879743	OC[C@H]1[C@@H]([C@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669315	phase I
BRD-K93845141	OC[C@H]1[C@H]([C@@H]2CN(CC3CCOCC3)CCCCN12)c1ccc(cc1)-c1cccnc1	CID:54669316	phase I
BRD-K05932219	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)-c1ccccc1	CID:54669335	phase I
BRD-K23807807	Cc1ccccc1S(=O)(=O)N1CCCCN2[C@@H](CO)[C@H]([C@@H]2C1)c1ccc(cc1)-c1ccccc1	CID:54669344	phase I
BRD-K99640003	OC[C@H]1[C@@H]([C@H]2CN(CCC(F)(F)F)CCCCN12)c1ccc(cc1)C1=CCCC1	CID:54669456	phase I
BRD-K58800409	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CC1	CID:54669462	phase I
BRD-K87765798	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CC1	CID:54669463	phase I
BRD-K75674991	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CC1	CID:54669467	phase I
BRD-K24663282	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CC1	CID:54669469	phase I
BRD-K24319929	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2CCCCN(C[C@H]12)C(=O)C1CCCC1	CID:54669492	phase I
BRD-K21193980	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2CCCCN(C[C@@H]12)C(=O)C1CCCC1	CID:54669493	phase I
BRD-K71154829	OC[C@@H]1[C@H]([C@H]2CN(CCCCN12)C(=O)Nc1ccccc1F)c1ccc(cc1)C1=CCCCC1	CID:54669567	phase I
BRD-K91044787	COc1ccc(NC(=O)N2CCCCN3[C@H](CO)[C@H]([C@@H]3C2)c2ccc(cc2)C2=CCCC2)cc1	CID:54669575	phase I
BRD-K24251672	COc1ccc(NC(=O)N2CCCCN3[C@@H](CO)[C@@H]([C@H]3C2)c2ccc(cc2)C2=CCCC2)cc1	CID:54669576	phase I
BRD-K05658747	Cc1nnc(o1)C(=O)NC(C)(C)c1nc(C(=O)NCc2ccc(F)cc2)c(O)c(=O)n1C	CID:54671008	phase I
BRD-K85307935	CO[C@@H]1[C@@H](OC(N)=O)[C@@H](O)[C@H](Oc2ccc3c(O)c(NC(=O)c4ccc(O)c(CC=C(C)C)c4)c(=O)oc3c2C)OC1(C)C	CID:54675769	phase I
BRD-K82236179	Oc1c(Cc2c(O)c3ccccc3oc2=O)c(=O)oc2ccccc12	CID:54676038	phase I
BRD-K03384561	CN(C(=O)c1c(O)c2ccccc2n(C)c1=O)c1ccccc1	CID:54676478	phase I
BRD-K81847782	COc1c(CC=C(C)C)c2OC(C)(C)C=Cc2c3oc(=O)c(c(O)c13)c4ccc(O)cc4	CID:54676535	phase I
BRD-A65051990	CC(=O)CC(c1ccc(cc1)[N+]([O-])=O)c1c(O)c2ccccc2oc1=O	CID:54676537	phase I
BRD-K54411430	COc1ccc(cc1)c2c(O)c3c(OC)c4C=CC(C)(C)Oc4cc3oc2=O	CID:54677407	phase I
BRD-A24514565	CC(=O)CC(c1ccccc1)c1c(O)c2ccccc2oc1=O	CID:54678486	phase I
BRD-K08109516	Oc1c(-c2cccc(Oc3ccccc3)c2)c(=O)[nH]c2cc(Cl)ccc12	CID:54682505	phase I
BRD-K07325606	Oc1cc(/C=C/c2ccc(O)c(O)c2)oc(=O)c1	CID:54685921	phase I
BRD-K94412972	COc1ccc(cc1)c2c(O)c3c(OC)c4CCC(C)(C)Oc4cc3oc2=O	CID:54686939	phase I
BRD-K10176267	Oc1c(C(=O)C2CC2)c(=O)[nH]c2cc(Cl)ccc12	CID:54687453	phase I
BRD-K25991148	CC(=O)C[C@@H](c1ccccc1)c1c(O)c2ccccc2oc1=O	CID:54688261	phase I
BRD-K30570479	Clc1cc(NC(=O)c2ccccn2)ccc1N1C(=O)[C@H]2[C@@H]3C[C@@H](C=C3)[C@H]2C1=O	CID:54752951	phase I
BRD-K26863634	COc1ccc(cc1)C(=O)Oc1ccc(CCn2c(NC(=O)c3ccc(cc3)C(F)(F)F)nc3cc(ccc23)C(O)=O)cc1	CID:56676725	phase I
BRD-K58663279	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835197	phase I
BRD-K19016650	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835198	phase I
BRD-K71287386	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835199	phase I
BRD-K11609893	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835201	phase I
BRD-K11880681	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835202	phase I
BRD-K26301430	CO[C@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO)c4ccccc4	CID:56835203	phase I
BRD-K86427056	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4ccccc4C1=O	CID:56835204	phase I
BRD-K35979672	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835205	phase I
BRD-K63686806	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835207	phase I
BRD-K76581294	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835211	phase I
BRD-K59848706	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835213	phase I
BRD-K29568987	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835214	phase I
BRD-K61076106	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:56835215	phase I
BRD-K26779385	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835216	phase I
BRD-K66633149	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835217	phase I
BRD-K32231531	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc3OCCCOc23)OCc4ccccc4-c5ccccc5C1=O	CID:56835218	phase I
BRD-K62337120	COc1ccc(OC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:56835219	phase I
BRD-K42696220	CO[C@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO)c4ccccc4	CID:56835220	phase I
BRD-K15651660	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835221	phase I
BRD-K31160185	COc1ccc(CNC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO)cc1	CID:56835222	phase I
BRD-K47811236	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:56835223	phase I
BRD-K54889769	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:56835224	phase I
BRD-K86171512	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835225	phase I
BRD-K45442578	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835226	phase I
BRD-K41652832	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)c1	CID:56835227	phase I
BRD-K79235289	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835228	phase I
BRD-K37960810	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835230	phase I
BRD-K42712649	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835231	phase I
BRD-K80174954	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO)c4ccccc4	CID:56835235	phase I
BRD-K30912278	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835236	phase I
BRD-K96612763	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:56835237	phase I
BRD-K41944296	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835238	phase I
BRD-K75614533	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835241	phase I
BRD-K17661785	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835242	phase I
BRD-K09029418	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:56835245	phase I
BRD-K85068586	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)CC2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835246	phase I
BRD-K45542432	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835247	phase I
BRD-K97925203	CC(C)OC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:56835248	phase I
BRD-K10808435	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835250	phase I
BRD-K20965564	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835251	phase I
BRD-K90528929	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835255	phase I
BRD-K33044853	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@@H](C)CO)n(C)c4ccccc34	CID:56835258	phase I
BRD-K96475865	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835259	phase I
BRD-K45745416	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835260	phase I
BRD-K97481912	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:56835263	phase I
BRD-K07462139	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(O)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835264	phase I
BRD-K83549059	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835265	phase I
BRD-K44015831	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835266	phase I
BRD-K68327489	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835268	phase I
BRD-K45714982	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:56835269	phase I
BRD-K56215045	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:56835270	phase I
BRD-K59024058	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835271	phase I
BRD-K96039110	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835272	phase I
BRD-K29368169	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835273	phase I
BRD-K56079297	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:56835274	phase I
BRD-K00954272	CC(C)[C@@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:56835275	phase I
BRD-K01222176	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835276	phase I
BRD-K88608081	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835281	phase I
BRD-K25068941	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835282	phase I
BRD-K87885716	COc1ccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:56835283	phase I
BRD-K84388104	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:56835284	phase I
BRD-K12570990	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835285	phase I
BRD-K50513128	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835286	phase I
BRD-K50737884	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835287	phase I
BRD-K64900763	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:56835288	phase I
BRD-K65778880	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835290	phase I
BRD-K97722864	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835291	phase I
BRD-K17375958	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835292	phase I
BRD-K40505314	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835295	phase I
BRD-K18552758	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835297	phase I
BRD-K60477859	CO[C@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3c(C(=O)N(C[C@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:56835298	phase I
BRD-K95718241	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835299	phase I
BRD-K22814206	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835300	phase I
BRD-K79780092	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:56835302	phase I
BRD-K19815647	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835303	phase I
BRD-K25148849	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:56835304	phase I
BRD-K65416492	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4c(C(=O)N(C[C@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c1	CID:56835305	phase I
BRD-K74318028	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835306	phase I
BRD-K22479833	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835307	phase I
BRD-K38431902	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835308	phase I
BRD-K74712058	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835312	phase I
BRD-K07400331	COc1cccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c1	CID:56835314	phase I
BRD-K21037590	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835315	phase I
BRD-K56483755	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835320	phase I
BRD-K25542589	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835321	phase I
BRD-K64341172	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835322	phase I
BRD-K70243592	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:56835324	phase I
BRD-K41017712	COc1ccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:56835325	phase I
BRD-K24465933	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:56835326	phase I
BRD-K64520484	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835328	phase I
BRD-K50078508	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835329	phase I
BRD-K75252623	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835333	phase I
BRD-K11877130	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835334	phase I
BRD-K99128867	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835336	phase I
BRD-K00391235	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:56835337	phase I
BRD-K87079453	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)CC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835339	phase I
BRD-K62839271	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835340	phase I
BRD-K51072560	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835344	phase I
BRD-K45265806	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835348	phase I
BRD-K52204603	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835349	phase I
BRD-K66199575	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835350	phase I
BRD-K39321814	CC(C)COC(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@@H](C)CO)n(C)c4ccccc34	CID:56835351	phase I
BRD-K01289045	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835353	phase I
BRD-K20500634	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835355	phase I
BRD-K00043782	COc1ccc(CNC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45)cc1	CID:56835356	phase I
BRD-K44897098	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:56835357	phase I
BRD-K39844985	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835358	phase I
BRD-K29280435	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835360	phase I
BRD-K88866336	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835362	phase I
BRD-K19294102	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccnc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835363	phase I
BRD-K08094365	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835364	phase I
BRD-K62560708	COc1ccccc1S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:56835365	phase I
BRD-K44818533	COc1ccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45)c(OC)c1	CID:56835366	phase I
BRD-K98286370	CO[C@@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:56835367	phase I
BRD-K58189273	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835368	phase I
BRD-K57659231	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@@H](C)CO)n(C)c5ccccc45	CID:56835369	phase I
BRD-K87357593	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835371	phase I
BRD-K44752364	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835380	phase I
BRD-K30226385	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835382	phase I
BRD-K55743364	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835385	phase I
BRD-K16619158	CO[C@H](C(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@H](C)CO)n(C)c4ccccc34)c5ccccc5	CID:56835386	phase I
BRD-K63837190	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835387	phase I
BRD-K43980524	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835389	phase I
BRD-K08590382	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835390	phase I
BRD-K45785972	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835391	phase I
BRD-K84079653	CC(C)COC(=O)N(C)C[C@H]1OCc2ccccc2-c3c(C(=O)N(C[C@@H]1C)[C@H](C)CO)n(C)c4ccccc34	CID:56835392	phase I
BRD-K05448102	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835394	phase I
BRD-K11901207	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835395	phase I
BRD-K67037986	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835396	phase I
BRD-K22650859	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835399	phase I
BRD-K23724349	CC(C)OC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:56835401	phase I
BRD-K99159184	CC(C)[C@@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:56835402	phase I
BRD-K78778476	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:56835404	phase I
BRD-K56931391	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835405	phase I
BRD-K31042078	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835406	phase I
BRD-K70016992	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835407	phase I
BRD-K94348552	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5c(C1=O)n(C)c6ccccc56	CID:56835410	phase I
BRD-K09276254	COc1cccc(c1)S(=O)(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45	CID:56835411	phase I
BRD-K38942541	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835412	phase I
BRD-K98168679	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835414	phase I
BRD-K10325955	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835416	phase I
BRD-K71397492	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccnc(c2)N3CCOCC3)OCc4ccccc4-c5ccccc5C1=O	CID:56835417	phase I
BRD-K83030741	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO	CID:56835418	phase I
BRD-K16561564	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:56835419	phase I
BRD-K05745800	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835420	phase I
BRD-K21787371	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835421	phase I
BRD-K98695146	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:56835422	phase I
BRD-K75749796	CC(C)[C@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@H](C)CO	CID:56835423	phase I
BRD-K14493775	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835426	phase I
BRD-K99643744	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO	CID:56835428	phase I
BRD-K99026889	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3c(C1=O)n(C)c4ccccc34	CID:56835429	phase I
BRD-K77434972	CO[C@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO)c4ccccc4	CID:56835430	phase I
BRD-K15530151	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835431	phase I
BRD-K81392055	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCC(F)(F)F)OCc2ccccc2-c3ccccc3C1=O	CID:56835432	phase I
BRD-K74556269	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835433	phase I
BRD-K32864614	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835434	phase I
BRD-K28862107	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)CCN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835435	phase I
BRD-K26835110	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:56835436	phase I
BRD-K04847305	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835438	phase I
BRD-K39114105	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835439	phase I
BRD-K01146969	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835440	phase I
BRD-K09929560	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835441	phase I
BRD-K25564095	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)c2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835442	phase I
BRD-K20914452	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO)c4ccccc4	CID:56835443	phase I
BRD-K91416922	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835444	phase I
BRD-K25560306	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:56835445	phase I
BRD-K06096379	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835446	phase I
BRD-K99718824	COc1cccc(NC(=O)N(C)C[C@H]2OCc3ccccc3-c4c(C(=O)N(C[C@@H]2C)[C@H](C)CO)n(C)c5ccccc45)c1	CID:56835451	phase I
BRD-K94988014	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835452	phase I
BRD-K07479774	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)N[C@H](C)c2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835453	phase I
BRD-K97805274	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO	CID:56835457	phase I
BRD-K40907206	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:56835458	phase I
BRD-K42048463	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:56835459	phase I
BRD-K71859938	COc1ccc(CNC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:56835460	phase I
BRD-K49877948	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835461	phase I
BRD-K04086909	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835462	phase I
BRD-K05442673	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835465	phase I
BRD-K97185232	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)C2CC2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835466	phase I
BRD-K19597888	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835468	phase I
BRD-K66357706	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835469	phase I
BRD-K53467073	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(Cl)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835470	phase I
BRD-K61342953	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(F)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835473	phase I
BRD-K02944060	CC(C)[C@@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:56835474	phase I
BRD-K36109933	COc1ccc(OC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:56835475	phase I
BRD-K80195617	COc1ccccc1NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:56835476	phase I
BRD-K09426613	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835478	phase I
BRD-K76103468	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)CC2CC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835479	phase I
BRD-K12415987	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835480	phase I
BRD-K51832753	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2c(C)noc2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835481	phase I
BRD-K77579348	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835482	phase I
BRD-K44681861	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835483	phase I
BRD-K02581961	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835484	phase I
BRD-K70756309	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835485	phase I
BRD-K86219348	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835489	phase I
BRD-K75745425	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835492	phase I
BRD-K70657810	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835493	phase I
BRD-K79003015	CC(C)OC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:56835494	phase I
BRD-K25354424	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:56835495	phase I
BRD-K01787550	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:56835496	phase I
BRD-K87878159	CC(C)[C@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:56835497	phase I
BRD-K40483165	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835499	phase I
BRD-K44480417	COc1ccccc1S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:56835500	phase I
BRD-K05051567	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccs2)OCc3ccccc3-c4ccccc4C1=O	CID:56835501	phase I
BRD-K98676361	CC(C)COC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO	CID:56835503	phase I
BRD-K29136476	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccsc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835504	phase I
BRD-K59893964	COc1cccc(c1)S(=O)(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO	CID:56835505	phase I
BRD-K06199632	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:56835506	phase I
BRD-K43874853	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:56835507	phase I
BRD-K34829873	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H]2CCCN2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835508	phase I
BRD-K92953840	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2cccc(C#N)c2)OCc3ccccc3-c4ccccc4C1=O	CID:56835509	phase I
BRD-K27363274	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835510	phase I
BRD-K96522480	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835511	phase I
BRD-K81415316	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)[C@H]2CCCN2C)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835514	phase I
BRD-K16229712	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2c(C)noc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835515	phase I
BRD-K63164901	COc1ccc(OC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO)cc1	CID:56835516	phase I
BRD-K58194762	COc1cccc(NC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@H](C)CO)c1	CID:56835517	phase I
BRD-K50733069	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835518	phase I
BRD-K69692345	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3OCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:56835519	phase I
BRD-K23603287	COc1cccc(CN(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO)c1	CID:56835520	phase I
BRD-K84733605	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835521	phase I
BRD-K08246588	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835522	phase I
BRD-K87133350	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835525	phase I
BRD-K49723782	COc1ccc(CNC(=O)N(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@H]2C)[C@@H](C)CO)cc1	CID:56835526	phase I
BRD-K59039774	CO[C@@H](C(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@H]1C)[C@@H](C)CO)c4ccccc4	CID:56835528	phase I
BRD-K78228015	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835529	phase I
BRD-K54876931	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835530	phase I
BRD-K28812281	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)C(=O)Cc2ccccc2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:56835531	phase I
BRD-K44098776	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2cccc(c2)C(F)(F)F)OCc3ccccc3-c4ccccc4C1=O	CID:56835532	phase I
BRD-K22825029	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)N[C@@H](C)c2ccccc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835533	phase I
BRD-K87913872	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)S(=O)(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835536	phase I
BRD-K60065591	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835539	phase I
BRD-K75961033	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:56835541	phase I
BRD-K70036333	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2F)OCc3ccccc3-c4ccccc4C1=O	CID:56835544	phase I
BRD-K06688693	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2cn(C)cn2)OCc3ccccc3-c4ccccc4C1=O	CID:56835545	phase I
BRD-K55295918	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2ccc3N(C)CCOc3c2)OCc4ccccc4-c5ccccc5C1=O	CID:56835547	phase I
BRD-K25878320	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835548	phase I
BRD-K62595167	CC(C)[C@H](C)NC(=O)N(C)C[C@@H]1OCc2ccccc2-c3ccccc3C(=O)N(C[C@@H]1C)[C@@H](C)CO	CID:56835550	phase I
BRD-K38717348	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(c2)C(=O)O)OCc3ccccc3-c4ccccc4C1=O	CID:56835552	phase I
BRD-K28663733	COc1ccccc1CN(C)C[C@@H]2OCc3ccccc3-c4ccccc4C(=O)N(C[C@@H]2C)[C@@H](C)CO	CID:56835554	phase I
BRD-K39156670	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)Nc2ccc(F)cc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835555	phase I
BRD-K70358157	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C#N)OCc3ccccc3-c4ccccc4C1=O	CID:56835556	phase I
BRD-K08482401	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)S(=O)(=O)c2ccccc2C)OCc3ccccc3-c4ccccc4C1=O	CID:56835557	phase I
BRD-K83837862	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C(=O)NC2CCCCC2)OCc3ccccc3-c4ccccc4C1=O	CID:56835558	phase I
BRD-K19114437	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)c2ccncc2)OCc3ccccc3-c4ccccc4C1=O	CID:56835559	phase I
BRD-K20848134	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:56835560	phase I
BRD-K19826330	C[C@@H](CO)N1C[C@H](C)[C@H](CN(C)C)OCc2ccccc2-c3ccccc3C1=O	CID:56835561	phase I
BRD-K13000360	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)[C@@H](Cc2ccccc2)N(C)C)OCc3ccccc3-c4ccccc4C1=O	CID:56835564	phase I
BRD-K92523103	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@@H]1CCO)c3cccc(C#CCC4CCCC4)c3)C(=O)NCCCN5CCOCC5	CID:56835565	phase I
BRD-K35691352	COc1cccc(c1)c2cccc(c2)c3nc(cc4CN([C@H](CCO)c43)S(=O)C(C)(C)C)C(=O)O	CID:56835566	phase I
BRD-K54051742	CN(C)CC#Cc1cccc(c1)c2nc(cc3CN([C@H](CCO)c32)S(=O)C(C)(C)C)C(=O)N4CCN(C)CC4	CID:56835567	phase I
BRD-K62189562	COCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)c3cccc(c3)c4cccc(OC)c4)S(=O)C(C)(C)C	CID:56835568	phase I
BRD-K75012089	CCOC(=O)c1cc2CN([C@H](CCO)c2c(n1)c3cccc(C#CCN(C)C)c3)S(=O)C(C)(C)C	CID:56835569	phase I
BRD-K88176535	COc1cccc(c1)c2cccc(c2)c3nc(cc4CN([C@@H](CCO)c43)S(=O)C(C)(C)C)C(=O)O	CID:56835570	phase I
BRD-K22674439	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@H]1CCO)c3cccc(C#CC(C)(C)O)c3)C(=O)N4CCN(Cc5ccccc5)CC4	CID:56835571	phase I
BRD-K42001678	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@@H]1CCO)c3cccc(C#CC(C)(C)O)c3)C(=O)O	CID:56835572	phase I
BRD-K31449336	COc1cccc(c1)c2cccc(c2)c3nc(cc4CN([C@H](CCO)c43)S(=O)C(C)(C)C)C(=O)NCCCN5CCOCC5	CID:56835573	phase I
BRD-K58999044	COc1cccc(c1)c2cccc(c2)c3nc(cc4CN([C@H](CCO)c43)S(=O)C(C)(C)C)C(=O)N5CCN(C)CC5	CID:56835574	phase I
BRD-K84586204	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@H]1CCO)c3cccc(c3)c4cccc(F)c4)C(=O)NCCCN5CCOCC5	CID:56835575	phase I
BRD-K01490356	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@@H]1CCO)c3cccc(c3)c4cc5ccccc5o4)C(=O)O	CID:56835576	phase I
BRD-K72014243	CN1CCN(CC1)C(=O)c2cc3CN([C@@H](CCO)c3c(n2)c4cccc(c4)c5cccc(F)c5)S(=O)C(C)(C)C	CID:56835577	phase I
BRD-K27865298	CN1CCN(CC1)C(=O)c2cc3CN([C@H](CCO)c3c(n2)c4cccc(c4)c5cccc(F)c5)S(=O)C(C)(C)C	CID:56835578	phase I
BRD-K18449990	COc1ccc(C#Cc2cccc(c2)c3nc(cc4CN([C@H](CCO)c43)S(=O)C(C)(C)C)C(=O)NCCCN5CCOCC5)cc1OC	CID:56835579	phase I
BRD-K48719132	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@@H]1CCO)c3cccc(c3)c4cccc(F)c4)C(=O)NCCCN5CCOCC5	CID:56835580	phase I
BRD-K44521151	COc1ccc(C#Cc2cccc(c2)c3nc(cc4CN([C@@H](CCO)c43)S(=O)C(C)(C)C)C(=O)O)cc1OC	CID:56835582	phase I
BRD-K61079130	CN(C)CC#Cc1cccc(c1)c2nc(cc3CN([C@@H](CCO)c32)S(=O)C(C)(C)C)C(=O)NCc4ccc5OCOc5c4	CID:56835583	phase I
BRD-K65873444	CN(C)CC#Cc1cccc(c1)c2nc(cc3CN([C@H](CCO)c32)S(=O)C(C)(C)C)C(=O)NCc4ccc5OCOc5c4	CID:56835584	phase I
BRD-K06956443	COc1ccc(C#Cc2cccc(c2)c3nc(cc4CN([C@H](CCO)c43)S(=O)C(C)(C)C)C(=O)O)cc1OC	CID:56835585	phase I
BRD-K96742509	CCOC(=O)c1cc2CN([C@H](CCO)c2c(n1)c3cccc(c3)c4cccc(OC)c4)S(=O)C(C)(C)C	CID:56835586	phase I
BRD-K98466889	CN(C)CC#Cc1cccc(c1)c2nc(cc3CN([C@@H](CCO)c32)S(=O)C(C)(C)C)C(=O)N4CCN(C)CC4	CID:56835587	phase I
BRD-K32173944	CN(C)CC#Cc1cccc(c1)c2nc(cc3CN([C@@H](CCO)c32)S(=O)C(C)(C)C)C(=O)NCCCN4CCOCC4	CID:56835588	phase I
BRD-K00472408	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@H]1CCO)c3cccc(C#CC(C)(C)O)c3)C(=O)NCCCN4CCOCC4	CID:56835589	phase I
BRD-K87621813	CN1CCN(CC1)C(=O)c2cc3CN([C@H](CCO)c3c(n2)c4cccc(C#CCC5CCCC5)c4)S(=O)C(C)(C)C	CID:56835590	phase I
BRD-K47071092	CCOC(=O)c1cc2CN([C@@H](CCO)c2c(n1)c3cccc(c3)c4cccc(OC)c4)S(=O)C(C)(C)C	CID:56835591	phase I
BRD-K85123694	CN(C)CC#Cc1cccc(c1)c2nc(cc3CN([C@@H](CCO)c32)S(=O)C(C)(C)C)C(=O)O	CID:56835592	phase I
BRD-K00347903	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@H]1CCO)c3cccc(c3)c4cccc(F)c4)C(=O)O	CID:56835593	phase I
BRD-K55569103	COCCNC(=O)c1cc2CN([C@H](CCO)c2c(n1)c3cccc(c3)c4cccc(F)c4)S(=O)C(C)(C)C	CID:56835594	phase I
BRD-K69947829	CN1CCN(CC1)C(=O)c2cc3CN([C@@H](CCO)c3c(n2)c4cccc(C#CCC5CCCC5)c4)S(=O)C(C)(C)C	CID:56835595	phase I
BRD-K30695296	COCCNC(=O)c1cc2CN([C@@H](CCO)c2c(n1)c3cccc(c3)c4cccc(F)c4)S(=O)C(C)(C)C	CID:56835597	phase I
BRD-K98948170	OC(=O)[C@H]1CCCC[C@H]1C(=O)N1CCc2ccccc2[C@H]1CN1C(=O)c2ccccc2C1=O	CID:56840728	phase I
BRD-K81925854	C[C@@H]1C[C@@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]2(C)[C@H]1C(=O)COC(=O)C(C)(C)C	CID:56840865	phase I
BRD-K16604218	O=C(NC1=C(N2CCN(CC2)c2ccccc2)C(=O)c2ccccc2C1=O)c1ccccc1	CID:56928031	phase I
BRD-K24859147	COCCNCCCn1c(C(=O)CF)c(-c2ccc(C)cc2)c2c(N)ncnc12	CID:56965963	phase I
BRD-A22740840	CN(C)[C@H]1[C@@H]2[C@@H](O)[C@H]3C(C(=O)c4c(O)cccc4[C@@]3(C)O)C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O	CID:57004235	phase I
BRD-A31374339	Nc1nc(F)nc2n(cnc12)[C@@H]1O[C@H](CO)C(O)C1O	CID:57007282	phase I
BRD-K96390176	C[C@H](C=C[C@@H](O)C1CC1)[C@H]1CC[C@H]2C(CCC[C@]12C)=CC=C1C[C@@H](O)C[C@H](O)C1=C	CID:57118766	phase I
BRD-A74767450	OC[C@H]1O[C@H](C(O)C1O)n1cnc2c(Nc3ccc(cc3)S(O)(=O)=O)ncnc12	CID:57241630	phase I
BRD-K83972459	CCN1CCN(Cc2ccc(Nc3ncc4N(C)C(=O)c5ccccc5N(C)c4n3)cc2C(F)(F)F)CC1	CID:57340671	phase I
BRD-K61860715	CN(C)C\C=C\C(=O)Nc1ccc(cc1)C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1	CID:57340680	phase I
BRD-K56994829	N[C@H](Cc1ccc(O)cc1O)C(O)=O	CID:57367711	phase I
BRD-K61341215	CC(=O)O[C@H]1[C@H](C[C@@H]2[C@H]3CC[C@@H]4C[C@H](OC(C)=O)[C@H](C[C@@]4(C)[C@@H]3CC[C@@]12C)N1CCCCC1)[N+]1(C)CCCCC1	CID:57369718	phase I
BRD-K86940322	CCC[C@H](N[C@@H](C)C(=O)N1[C@H]2CCCC[C@@H]2C[C@H]1C(O)=O)C(=O)OCC	CID:58153637	phase I
BRD-K19220233	N#Cc1cc(cc(c1)-c1ccnc(Nc2ccc(cc2)-n2cnc(n2)-c2cccnc2)n1)N1CCOCC1	CID:59588070	phase I
BRD-K91449330	COC(=O)N1N(C(=O)OC)[C@](C(C)C)(C1=O)c1ccc(Cl)cc1	CID:60138064	phase I
BRD-K20914082	COC(=O)N1N(C(=O)OC)[C@](C(C)C)(C1=O)c1ccsc1	CID:60138134	phase I
BRD-K60219430	C(Cc1c[nH]c2ccccc12)Nc1cccc(Nc2ccncc2)c1	CID:60167550	phase I
BRD-K50012739	CC(C)CC#Cc1cnc2O[C@H](CN(C)C(=O)CC3CC3)[C@H](C)CN([C@@H](C)CO)C(=O)c2c1	CID:60182493	phase I
BRD-K34810022	OC[C@H]1N[C@H](CNC(=O)C2CCCC2)[C@H]1c1ccc(cc1)-c1cncnc1	CID:60182592	phase I
BRD-K27096101	CCCNC(=O)N1[C@H](CO)[C@@H]([C@H]1CNC(C)C)c1ccc(cc1)C1=CCCCC1	CID:60182621	phase I
BRD-K38465286	CCNC[C@H]1[C@H]([C@@H](CO)N1C(=O)C1CCCC1)c1ccc(cc1)\C=C\C	CID:60182633	phase I
BRD-K63662683	CCCNC(=O)N1[C@H](CO)[C@@H]([C@@H]1CNC(C)C)c1ccc(cc1)C1=CCCCC1	CID:60182656	phase I
BRD-K99398689	CC(C)N(C[C@@H]1[C@H]([C@@H](CO)N1CC1CC1)c1ccc(cc1)C1=CCCC1)C(C)=O	CID:60182667	phase I
BRD-K94719962	OC[C@H]1N[C@H](CNC(=O)C2CCC2)[C@H]1c1ccc(cc1)-c1cccc(c1)C#N	CID:60182680	phase I
BRD-K31800869	CN(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)-c1cccnc1)C(=O)NC1CCCC1	CID:60182741	phase I
BRD-K70923866	CCC(=O)N1[C@H](CO)[C@@H]([C@H]1CNCC1CCC1)c1ccc(cc1)C1=CCCCC1	CID:60182794	phase I
BRD-K02448874	CC(C)N(C[C@H]1N[C@H](CO)[C@@H]1c1ccc(cc1)C1=CCCCC1)C(=O)CN(C)C	CID:60182807	phase I
BRD-K78235165	OC[C@H]1N[C@H](CNC(=O)C2CCCCC2)[C@H]1c1ccc(cc1)-c1cncnc1	CID:60182852	phase I
BRD-K51916742	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CCc1ccccc1	CID:60182932	phase I
BRD-K07276035	COC(=O)c1ccc(CN2C[C@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60182960	phase I
BRD-K07508147	COC(=O)c1ccc(CN2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60182962	phase I
BRD-K82750814	COC(=O)c1ccc(CN2C[C@@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60182963	phase I
BRD-K73224765	COC(=O)c1ccc(CN2C[C@@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60182993	phase I
BRD-K31931684	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)C#CCC1CCCC1	CID:60183177	phase I
BRD-K76528265	CN(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60183353	phase I
BRD-K48105325	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)c1cccc(F)c1)C#Cc1ccccc1	CID:60183407	phase I
BRD-K75725875	COc1ccccc1-c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)C1CCCC1	CID:60183411	phase I
BRD-K38632726	OC[C@H]1[C@@H]([C@@H](C#N)N1C(=O)NC1CCCC1)c1ccc(cc1)C1=CCCCC1	CID:60183420	phase I
BRD-K14023656	OC[C@H]1[C@@H]([C@H](C#N)N1c1nc(cs1)-c1ccccc1)c1ccc(cc1)C1=CCCC1	CID:60183443	phase I
BRD-K87268239	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCCC1)-c1ccc(cc1)C#N	CID:60183492	phase I
BRD-K37268490	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C1=CCCCC1)C(=O)C1CCC1	CID:60183604	phase I
BRD-K96903816	CC(C)(C)S(=O)N1Cc2cc(nc(c2[C@@H]1CCO)c3cccc(C#CC(C)(C)O)c3)C(=O)N[C@@H]4CCN(Cc5ccccc5)C4	CID:60183843	phase I
BRD-K26119753	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2cc(F)ccc2F)CC1)C(=O)Nc1ccc(F)cc1	CID:60184001	phase I
BRD-K52497027	CCC(=O)N1CC[C@@]2(CC1)CN(Cc1cc(F)ccc1F)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60184075	phase I
BRD-K59196958	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccncc1)C[C@]31CN(CC2CCOCC2)C1	CID:60184097	phase I
BRD-K92302554	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccccc1)C(=O)c1cccc(F)c1	CID:60184116	phase I
BRD-K37185609	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4Cl)C[C@]33CN(C3)C(=O)CC3CC3)n(C)c2c1	CID:60184146	phase I
BRD-K13175698	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4Cl)C[C@]33CN(C3)C(=O)CC3CC3)n(C)c2c1	CID:60184147	phase I
BRD-K41342615	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccc1F)C(=O)Nc1ccccc1F	CID:60184150	phase I
BRD-K70880645	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CCN(CC1)C(=O)C1CCC1	CID:60184192	phase I
BRD-K64551861	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CCN(CC3)C(=O)c3ccc4OCOc4c3)n(C)c2c1	CID:60184193	phase I
BRD-K41908462	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CCN(CC1)C(=O)C1CCC1	CID:60184231	phase I
BRD-K51237366	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)Nc1ccccc1)C(=O)Nc1ccc(F)cc1	CID:60184300	phase I
BRD-K29309835	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)S(=O)(=O)c3ccc(C)cc3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60184372	phase I
BRD-K46674611	C[C@@H](CO)N1C[C@@H](C)[C@H](CN(C)Cc2cccc(F)c2)OCc3ccccc3-c4c(C1=O)n(C)c5ccccc45	CID:60184577	phase I
BRD-K71838325	COc1cccc(c1)S(=O)(=O)N1C[C@]2(CCN(C)CC2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60184814	phase I
BRD-K17116894	CCCNC(=O)N1C[C@]2(CCN(CC2)C(=O)c2cccc(F)c2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60184815	phase I
BRD-K84678141	CCCNC(=O)N1C[C@]2(CCN(CC2)C(=O)c2cccc(F)c2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60184816	phase I
BRD-K64416059	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1F)C[C@]31CN(CC2CC2)C1	CID:60184817	phase I
BRD-K02098145	COc1ccc2c3c([C@H](CO)N(Cc4cccnc4)C[C@]33CN(C3)C(=O)c3cccnc3)n(C)c2c1	CID:60184818	phase I
BRD-K51288770	COc1ccc2c3c([C@@H](CO)N(Cc4cccnc4)C[C@]33CN(C3)C(=O)c3cccnc3)n(C)c2c1	CID:60184819	phase I
BRD-K07291429	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1cccnc1)S(C)(=O)=O	CID:60184820	phase I
BRD-K21299908	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)c1cccnc1)S(C)(=O)=O	CID:60184821	phase I
BRD-K73722380	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(CC1CC1)C[C@]31CCN(CC1)C(=O)Nc1cccc(F)c1	CID:60184822	phase I
BRD-K74794453	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(CC1CC1)C[C@]31CCN(CC1)C(=O)Nc1cccc(F)c1	CID:60184823	phase I
BRD-K28121452	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccc(Cl)cc1)C[C@]31CCN(Cc2nccs2)CC1	CID:60184824	phase I
BRD-K60850838	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1cccs1)C(=O)c1ccc(F)cc1	CID:60184842	phase I
BRD-K20601561	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)CC1CC1)C(=O)CC1CC1	CID:60184843	phase I
BRD-K87733826	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)CC1CC1)C(=O)CC1CC1	CID:60184844	phase I
BRD-K16126971	COc1ccc2c3c([C@H](CO)N(Cc4cccc(F)c4)C[C@]33CCN(CC3)C(=O)Cc3ccccc3)n(C)c2c1	CID:60184845	phase I
BRD-K70416046	COc1ccc2c3c([C@@H](CO)N(Cc4cccc(F)c4)C[C@]33CCN(CC3)C(=O)Cc3ccccc3)n(C)c2c1	CID:60184846	phase I
BRD-K86297549	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)c3ccc4OCOc4c3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60184847	phase I
BRD-K62058497	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)c3ccc4OCOc4c3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60184848	phase I
BRD-K64589075	COCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Nc1ccccc1F	CID:60184865	phase I
BRD-K90830878	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CCN(CC1)C(=O)CN(C)C	CID:60184866	phase I
BRD-K00550058	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CCN(CC1)C(=O)CN(C)C	CID:60184867	phase I
BRD-K27671514	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(Cc4ccc(cc4)-c4ccccn4)C3)n(C)c2c1	CID:60184868	phase I
BRD-K27711805	COc1ccc2c3c([C@H](CO)NC[C@]33CN(Cc4ccc(cc4)-c4ccccn4)C3)n(C)c2c1	CID:60184869	phase I
BRD-K29654204	CCCN1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)CN1CCOCC1	CID:60184870	phase I
BRD-K96408604	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4Cl)C[C@]33CN(C3)C(=O)CN(C)C)n(C)c2c1	CID:60184871	phase I
BRD-K94934810	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CN(C1)S(=O)(=O)c1cccc(C)c1	CID:60184872	phase I
BRD-K36953952	COc1ccc2c3c([C@H](CO)N(CC4CCOCC4)C[C@]33CCN(CC3)C(=O)CN(C)C)n(C)c2c1	CID:60184873	phase I
BRD-K78105568	COc1ccc(CN2C[C@]3(CN(C3)C(=O)c3ccccc3)c3c([nH]c4cc(OC)ccc34)[C@H]2CO)cc1	CID:60184885	phase I
BRD-K45217009	COc1ccc(CN2C[C@]3(CN(C3)C(=O)c3ccccc3)c3c([nH]c4cc(OC)ccc34)[C@@H]2CO)cc1	CID:60184886	phase I
BRD-K05994859	COc1ccc2c3c([C@@H](CO)N(Cc4ccncc4)C[C@]33CN(C3)C(=O)Nc3cccc(F)c3)n(C)c2c1	CID:60184887	phase I
BRD-K96692572	COc1ccc2c3c([C@H](CO)N(Cc4ccncc4)C[C@]33CN(C3)C(=O)Nc3cccc(F)c3)n(C)c2c1	CID:60184888	phase I
BRD-K22486133	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)C(=O)Nc3ccc4OCOc4c3)n(C)c2c1	CID:60184889	phase I
BRD-K73533033	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC3)C(=O)Nc3ccc4OCOc4c3)n(C)c2c1	CID:60184890	phase I
BRD-K61484309	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)C3CCCC3)S(C)(=O)=O)n(C)c2c1	CID:60184891	phase I
BRD-K80676896	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)C3CCCC3)S(C)(=O)=O)n(C)c2c1	CID:60184892	phase I
BRD-K03048862	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CN(Cc2cc(F)ccc2F)C1	CID:60184895	phase I
BRD-K50728502	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccc2OCOc2c1)C[C@]31CCN(CC1)C(=O)Nc1c(C)noc1C	CID:60184896	phase I
BRD-K20345035	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Cc1ccccn1	CID:60184897	phase I
BRD-K77295570	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Cc1ccccn1	CID:60184898	phase I
BRD-K81701287	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC2CCCCC2)CC1)S(=O)(=O)c1cn(C)cn1	CID:60184899	phase I
BRD-K70109596	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC2CCCCC2)CC1)S(=O)(=O)c1cn(C)cn1	CID:60184900	phase I
BRD-K90928795	COc1ccc2c3c([C@@H](CO)N(CC4CCOCC4)C[C@]33CN(Cc4nccs4)C3)n(C)c2c1	CID:60184901	phase I
BRD-K78032863	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4nccs4)CC3)C(=O)NC(C)C)n(C)c2c1	CID:60184902	phase I
BRD-K43638827	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)c3ccc4OCOc4c3)n(C)c2c1	CID:60184903	phase I
BRD-K79460683	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)c3ccc4OCOc4c3)n(C)c2c1	CID:60184904	phase I
BRD-K95605061	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccc2OCOc2c1)C(C)=O	CID:60184905	phase I
BRD-K57512343	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccc2OCOc2c1)C(C)=O	CID:60184906	phase I
BRD-K16144417	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4F)C[C@]33CCN(CC3)C(=O)C3CCOCC3)n(C)c2c1	CID:60184907	phase I
BRD-K17706493	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccc(Cl)cc1)C[C@]31CCN(Cc2nccs2)CC1	CID:60184915	phase I
BRD-K24625151	CCC(=O)N1C[C@]2(CN(C2)C(C)=O)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60184916	phase I
BRD-K08008963	CCC(=O)N1C[C@]2(CN(C2)C(C)=O)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60184917	phase I
BRD-K92300676	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C)C3)C(=O)Cc3ccccc3)n(C)c2c1	CID:60184918	phase I
BRD-K33380066	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C)C3)C(=O)Cc3ccccc3)n(C)c2c1	CID:60184919	phase I
BRD-K75313893	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(C)CC1)C(=O)C1CCCCC1	CID:60184920	phase I
BRD-K66340791	COCC(=O)N1CC[C@@]2(CC1)CN(Cc1cc(F)ccc1F)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60184921	phase I
BRD-K02427049	CCS(=O)(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1cccc(F)c1	CID:60184922	phase I
BRD-K62433344	CCS(=O)(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1cccc(F)c1	CID:60184923	phase I
BRD-K18823018	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1cn(C)cn1)C(=O)Nc1ccc(F)cc1	CID:60184924	phase I
BRD-K81031294	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1cn(C)cn1)C(=O)Nc1ccc(F)cc1	CID:60184925	phase I
BRD-K41280229	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CN(C3)S(=O)(=O)c3cccs3)n(C)c2c1	CID:60184926	phase I
BRD-K93596678	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1cc(F)ccc1F)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60184927	phase I
BRD-K91701366	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1cc(F)ccc1F)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60184928	phase I
BRD-K21576808	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)c1cnccn1)C(=O)NC(C)C	CID:60184929	phase I
BRD-K79962460	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4F)C[C@]33CCN(CC3)C(=O)C3CCOCC3)n(C)c2c1	CID:60184930	phase I
BRD-K59255802	CCCNC(=O)N1CC[C@@]2(CC1)CN(Cc1ccccn1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60184931	phase I
BRD-K20315727	CCCNC(=O)N1CC[C@@]2(CC1)CN(Cc1ccccn1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60184932	phase I
BRD-K38586507	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(OC)cc(OC)c1)C[C@]31CCN(CC1)C(=O)c1cccnc1	CID:60184938	phase I
BRD-K74144406	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)S(C)(=O)=O)C(=O)CN(C)C)n(C)c2c1	CID:60184939	phase I
BRD-K61540796	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)S(C)(=O)=O)C(=O)CN(C)C)n(C)c2c1	CID:60184940	phase I
BRD-K78816294	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)Cc1cccnc1)S(=O)(=O)c1ccc(C)cc1	CID:60184941	phase I
BRD-K94114461	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)Cc3ccncc3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60184942	phase I
BRD-K74176341	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CN(C3)S(=O)(=O)c3cccs3)n(C)c2c1	CID:60184943	phase I
BRD-K51368944	COc1ccc2c3c([C@H](CO)NC[C@]33CN(C3)C(=O)CC3CC3)n(C)c2c1	CID:60184944	phase I
BRD-K56153762	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)C(=O)CC3CC3)n(C)c2c1	CID:60184945	phase I
BRD-K38024502	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(C)=O)C(=O)c3ccncc3)n(C)c2c1	CID:60184946	phase I
BRD-K45392462	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(C)=O)C(=O)c3ccncc3)n(C)c2c1	CID:60184947	phase I
BRD-K41908552	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1cnccn1)C(=O)NC(C)C	CID:60184951	phase I
BRD-K33475837	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2cc(on2)-c2ccccc2)C1)C(=O)Nc1ccc(F)cc1	CID:60184952	phase I
BRD-K32253397	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2cc(on2)-c2ccccc2)C1)C(=O)Nc1ccc(F)cc1	CID:60184953	phase I
BRD-K16897811	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(CC1CC1)C[C@]31CN(C1)C(=O)c1ccc(F)cc1	CID:60184954	phase I
BRD-K77687238	COc1cccc(CN2C[C@@]3(C2)CN([C@H](CO)c2[nH]c4cc(OC)ccc4c32)S(C)(=O)=O)c1	CID:60184965	phase I
BRD-K78636275	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)S(=O)(=O)c1ccccc1)C(=O)c1cnccn1	CID:60184966	phase I
BRD-K09922076	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cc(OC)cc(OC)c1)C[C@]31CN(C1)S(=O)(=O)c1cccc(F)c1	CID:60184967	phase I
BRD-K51134784	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(Cc4ccncc4)C3)C(=O)CC3CC3)n(C)c2c1	CID:60184968	phase I
BRD-K26798591	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)Cc3ccncc3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60184969	phase I
BRD-K36289669	CCS(=O)(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)Nc1c(C)noc1C	CID:60184970	phase I
BRD-K50131804	CCS(=O)(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)Nc1c(C)noc1C	CID:60184971	phase I
BRD-K73329392	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(C)CC3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60184972	phase I
BRD-K65257892	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(C)CC3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60184973	phase I
BRD-K65946722	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2ccc(F)cc2)C1)C(=O)NC(C)C	CID:60184991	phase I
BRD-K33493537	CCCNC(=O)N1C[C@]2(CCN(CC2)S(=O)(=O)c2ccccc2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60184992	phase I
BRD-K01566563	CCCNC(=O)N1C[C@]2(CCN(CC2)S(=O)(=O)c2ccccc2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60184993	phase I
BRD-K47549778	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccc(F)cc1F)C(C)=O	CID:60184994	phase I
BRD-K07378992	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccc(F)cc1F)C(C)=O	CID:60184995	phase I
BRD-K36754063	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC4CCCC4)CC3)C(=O)C3CCC3)n(C)c2c1	CID:60184996	phase I
BRD-K12985993	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccn1)C(=O)C1CCC1	CID:60185015	phase I
BRD-K20146413	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccn1)C(=O)C1CCC1	CID:60185016	phase I
BRD-K02372107	CCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1cnccn1	CID:60185017	phase I
BRD-K18026907	CCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1cnccn1	CID:60185018	phase I
BRD-K99306975	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccncc1)C[C@]31CCN(CC2CCOCC2)CC1	CID:60185019	phase I
BRD-K96521176	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccncc1)C[C@]31CCN(CC2CCOCC2)CC1	CID:60185020	phase I
BRD-K23674074	COc1ccc2c3c([C@H](CO)N(Cc4cc(OC)cc(OC)c4)C[C@]33CCN(CC3)S(=O)(=O)c3cn(C)cn3)n(C)c2c1	CID:60185021	phase I
BRD-K96400713	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)S(C)(=O)=O	CID:60185031	phase I
BRD-K50037482	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)S(C)(=O)=O	CID:60185032	phase I
BRD-K95047050	COCC(=O)N1C[C@]2(CCN(Cc3cccnc3)CC2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60185033	phase I
BRD-K21340447	COCC(=O)N1C[C@]2(CCN(Cc3cccnc3)CC2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60185034	phase I
BRD-K46998548	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccc1F)C(=O)Nc1ccc(F)cc1	CID:60185035	phase I
BRD-K66046647	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccc1F)C(=O)Nc1ccc(F)cc1	CID:60185036	phase I
BRD-K42251804	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C)C[C@]31CCN(CC1)S(=O)(=O)c1ccc(C)cc1	CID:60185037	phase I
BRD-K78822312	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C)C[C@]31CCN(CC1)S(=O)(=O)c1ccc(C)cc1	CID:60185038	phase I
BRD-K05671267	COc1ccc2c3c([C@H](CO)N(Cc4ccccn4)C[C@]33CN(Cc4ccccn4)C3)n(C)c2c1	CID:60185039	phase I
BRD-K15245489	CCCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1ccc(C)cc1	CID:60185043	phase I
BRD-K90761527	CCCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1ccc(C)cc1	CID:60185044	phase I
BRD-K75323473	COc1ccc2c3c([C@H](CO)N(Cc4ccncc4)C[C@]33CN(C3)C(=O)C3CCCCC3)n(C)c2c1	CID:60185045	phase I
BRD-K51285422	COc1ccc2c3c([C@@H](CO)N(Cc4ccncc4)C[C@]33CN(C3)C(=O)C3CCCCC3)n(C)c2c1	CID:60185046	phase I
BRD-K73825454	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4cc(on4)-c4ccccc4)CC3)n(C)c2c1	CID:60185047	phase I
BRD-K70125131	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(Cc4cc(on4)-c4ccccc4)CC3)n(C)c2c1	CID:60185048	phase I
BRD-K17663482	COc1ccc2c3c([C@@H](CO)N(Cc4cc(OC)cc(OC)c4)C[C@]33CCN(CC3)S(=O)(=O)c3cn(C)cn3)n(C)c2c1	CID:60185049	phase I
BRD-K37273423	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)c3ccccc3F)C(=O)Nc3ccccc3F)n(C)c2c1	CID:60185050	phase I
BRD-K21095834	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(Cc4ccccc4OC)C3)C(=O)C3CC3)n(C)c2c1	CID:60185051	phase I
BRD-K18512301	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(Cc4ccccc4OC)C3)C(=O)C3CC3)n(C)c2c1	CID:60185052	phase I
BRD-K38620156	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)Cc1ccncc1)C(=O)Nc1ccc(F)cc1	CID:60185053	phase I
BRD-K62932832	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccncc1)C[C@]31CN(C1)C(=O)CN(C)C	CID:60185059	phase I
BRD-K85371697	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccncc1)C[C@]31CN(C1)C(=O)CN(C)C	CID:60185060	phase I
BRD-K03319520	COCC(=O)N1C[C@]2(CN(Cc3ccc(Cl)cc3)C2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60185061	phase I
BRD-K12654187	COCC(=O)N1C[C@]2(CN(Cc3ccc(Cl)cc3)C2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60185062	phase I
BRD-K18972207	CCS(=O)(=O)N1CC[C@@]2(CC1)CN[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185063	phase I
BRD-K09551497	CCS(=O)(=O)N1CC[C@@]2(CC1)CN[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185064	phase I
BRD-K97095445	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1OC)C[C@]31CN(C1)C(C)=O	CID:60185065	phase I
BRD-K45333259	CCCNC(=O)N1C[C@]2(CN(C2)C(=O)CN(C)C)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60185066	phase I
BRD-K16318272	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC2CCOCC2)CC1)C(=O)Nc1ccc(F)cc1	CID:60185067	phase I
BRD-K70260503	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)CN(C)C)C(=O)c1cccnc1	CID:60185068	phase I
BRD-K76060215	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)CN(C)C)C(=O)c1cccnc1	CID:60185069	phase I
BRD-K76811126	COc1ccc2c3c([C@@H](CO)N(Cc4cccc(Cl)c4)C[C@]33CCN(CC3)C(=O)C3CC3)n(C)c2c1	CID:60185070	phase I
BRD-K19004531	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)Cc1cccnc1	CID:60185071	phase I
BRD-K10417524	CCCNC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)CN1CCOCC1	CID:60185072	phase I
BRD-K44352336	CCCNC(=O)N1C[C@]2(CN(Cc3cccnc3)C2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60185073	phase I
BRD-K70053541	CCCNC(=O)N1C[C@]2(CN(Cc3cccnc3)C2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60185074	phase I
BRD-K23062161	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1nccs1)C[C@]31CCN(CC1)C(=O)C1CCCCC1	CID:60185075	phase I
BRD-K22101161	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2cncnc2)CC1)C(=O)CN(C)C	CID:60185076	phase I
BRD-K01037390	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2cncnc2)CC1)C(=O)CN(C)C	CID:60185077	phase I
BRD-K70539465	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C)C[C@]31CCN(CC1)C(=O)c1ccccc1F	CID:60185078	phase I
BRD-K87508191	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC4CCCC4)CC3)C(=O)C3CCC3)n(C)c2c1	CID:60185083	phase I
BRD-K87073769	COc1ccc2c3c([C@H](CO)NC[C@]33CN(C3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60185084	phase I
BRD-K07385663	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60185085	phase I
BRD-K25298364	CCS(=O)(=O)N1CC[C@@]2(CC1)CN[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185086	phase I
BRD-K00715257	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC2CCCC2)CC1)C(=O)CN1CCOCC1	CID:60185087	phase I
BRD-K11932360	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC2CCCC2)CC1)C(=O)CN1CCOCC1	CID:60185088	phase I
BRD-K39049859	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CCN(CC3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60185089	phase I
BRD-K41302766	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CCN(CC3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60185090	phase I
BRD-K44242139	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4cccc(F)c4)CC3)C(=O)C3CC3)n(C)c2c1	CID:60185091	phase I
BRD-K20109053	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4cccc(F)c4)CC3)C(=O)C3CC3)n(C)c2c1	CID:60185092	phase I
BRD-K00199388	COCC(=O)N1C[C@]2(CCN(CC2)C(=O)c2ccccn2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60185093	phase I
BRD-K80579043	COCC(=O)N1C[C@]2(CCN(CC2)C(=O)c2ccccn2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60185094	phase I
BRD-K97626184	COc1cccc(CN2C[C@]3(CN(C)C3)c3c([nH]c4cc(OC)ccc34)[C@H]2CO)c1	CID:60185095	phase I
BRD-K08502366	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1nccs1)C[C@]31CCN(CC1)C(=O)C1CCCCC1	CID:60185098	phase I
BRD-K42790191	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(CC4CCCCC4)C3)C(=O)Cc3ccccn3)n(C)c2c1	CID:60185099	phase I
BRD-K29514489	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4cncnc4)CC3)S(C)(=O)=O)n(C)c2c1	CID:60185100	phase I
BRD-K59768094	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)C(=O)Nc3ccc(F)cc3F)n(C)c2c1	CID:60185101	phase I
BRD-K37606648	COCC(=O)N1C[C@@]2(C1)CN(Cc1nccs1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185111	phase I
BRD-K75852825	COCC(=O)N1C[C@@]2(C1)CN(Cc1nccs1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185112	phase I
BRD-K05835710	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2nccs2)CC1)S(=O)(=O)c1ccc(C)cc1	CID:60185113	phase I
BRD-K81335986	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2nccs2)CC1)S(=O)(=O)c1ccc(C)cc1	CID:60185114	phase I
BRD-K22031742	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)NC(C)C)C(=O)C1CCOCC1	CID:60185115	phase I
BRD-K48254300	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)NC(C)C)C(=O)C1CCOCC1	CID:60185116	phase I
BRD-K26893932	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CN(CC4CC4)C3)n(C)c2c1	CID:60185117	phase I
BRD-K66187495	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CN(CC4CC4)C3)n(C)c2c1	CID:60185118	phase I
BRD-K12695722	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)S(=O)(=O)c1ccccc1	CID:60185119	phase I
BRD-K87640646	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CN(Cc4ccc(F)cc4)C3)n(C)c2c1	CID:60185120	phase I
BRD-K36984542	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CN(Cc4ccc(F)cc4)C3)n(C)c2c1	CID:60185121	phase I
BRD-K88994971	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(CC1CCCCC1)C[C@]31CN(C1)C(=O)C1CCOCC1	CID:60185122	phase I
BRD-K90544334	COc1ccc2c3c([C@H](CO)NC[C@]33CN(Cc4ccccc4Cl)C3)n(C)c2c1	CID:60185123	phase I
BRD-K30282337	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)S(=O)(=O)c1ccccc1	CID:60185140	phase I
BRD-K78130859	COc1ccc2c3c([C@H](CO)N(CC4CCCC4)C[C@]33CN(C3)C(=O)Nc3ccccc3)n(C)c2c1	CID:60185141	phase I
BRD-K81408913	COc1ccc2c3c([C@@H](CO)N(CC4CCCC4)C[C@]33CN(C3)C(=O)Nc3ccccc3)n(C)c2c1	CID:60185142	phase I
BRD-K61520982	CCCNC(=O)N1C[C@@]2(C1)CN(Cc1ccc(F)cc1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185143	phase I
BRD-K00596555	CCCNC(=O)N1C[C@@]2(C1)CN(Cc1ccc(F)cc1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185144	phase I
BRD-K16481946	CCCNC(=O)N1C[C@]2(CN(C2)C(=O)Cc2cccnc2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60185145	phase I
BRD-K50257410	CCCNC(=O)N1C[C@]2(CN(C2)C(=O)Cc2cccnc2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60185146	phase I
BRD-K24404115	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC3)C(=O)Nc3ccc(F)cc3F)n(C)c2c1	CID:60185159	phase I
BRD-K64279463	COc1cccc(CN2C[C@]3(CN(C)C3)c3c([C@@H]2CO)n(C)c2cc(OC)ccc32)c1	CID:60185160	phase I
BRD-K51030799	COc1cccc(CN2C[C@]3(CN(C)C3)c3c([C@H]2CO)n(C)c2cc(OC)ccc32)c1	CID:60185161	phase I
BRD-K48180773	CCCC(=O)N1C[C@]2(CN(Cc3nccs3)C2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60185162	phase I
BRD-K93411257	CCCC(=O)N1C[C@]2(CN(Cc3nccs3)C2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60185163	phase I
BRD-K25776214	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C)C1)C(=O)c1ccncc1	CID:60185164	phase I
BRD-K20369357	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C)C1)C(=O)c1ccncc1	CID:60185165	phase I
BRD-K09708845	CCCNC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)S(C)(=O)=O	CID:60185166	phase I
BRD-K53717189	CCCNC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)S(C)(=O)=O	CID:60185167	phase I
BRD-K82248240	COc1cccc(CN2C[C@]3(CN(C)C3)c3c([nH]c4cc(OC)ccc34)[C@@H]2CO)c1	CID:60185177	phase I
BRD-K93946290	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC4CCOCC4)CC3)C(=O)NC(C)C)n(C)c2c1	CID:60185178	phase I
BRD-K28746839	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CCN(CC3)C(=O)NC3CCCC3)n(C)c2c1	CID:60185179	phase I
BRD-K85885948	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CCN(CC3)C(=O)NC3CCCC3)n(C)c2c1	CID:60185180	phase I
BRD-K27133763	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2cc(on2)-c2ccccc2)CC1)C(C)=O	CID:60185181	phase I
BRD-K44874209	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2cc(on2)-c2ccccc2)CC1)C(C)=O	CID:60185182	phase I
BRD-K13559434	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cccc(F)c1)C[C@]31CCN(CC1)C(C)=O	CID:60185183	phase I
BRD-K98710661	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cccc(F)c1)C[C@]31CCN(CC1)C(C)=O	CID:60185184	phase I
BRD-K31129604	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)CC1CC1)C(=O)c1cccc(F)c1	CID:60185185	phase I
BRD-K67737641	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)Nc1cccc(F)c1)C(=O)c1cccnc1	CID:60185186	phase I
BRD-K03992415	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)Nc1cccc(F)c1)C(=O)c1cccnc1	CID:60185187	phase I
BRD-K23020884	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)c3ccccn3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60185188	phase I
BRD-K77502932	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)c3ccccn3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60185189	phase I
BRD-K23769006	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CCN(CC3)S(=O)(=O)c3cccc(F)c3)n(C)c2c1	CID:60185190	phase I
BRD-K29662826	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CCN(CC3)S(=O)(=O)c3cccc(F)c3)n(C)c2c1	CID:60185191	phase I
BRD-K20609812	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CN(C1)C(=O)Nc1ccc2OCOc2c1	CID:60185192	phase I
BRD-K75436517	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CN(C1)C(=O)Nc1ccc2OCOc2c1	CID:60185193	phase I
BRD-K31411295	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccccc1)S(C)(=O)=O	CID:60185194	phase I
BRD-K11615943	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(C)(=O)=O)C(=O)NC1CCCC1	CID:60185195	phase I
BRD-K65801064	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1cccc(C)c1)C(=O)Nc1cccc(F)c1	CID:60185196	phase I
BRD-K17446297	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(CC4CCOCC4)C3)C(=O)c3ccc(F)cc3)n(C)c2c1	CID:60185197	phase I
BRD-K65738831	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(CC4CCOCC4)C3)C(=O)c3ccc(F)cc3)n(C)c2c1	CID:60185198	phase I
BRD-K15380586	COc1cccc(CN2C[C@]3(CCN(Cc4ccccn4)CC3)c3c([nH]c4cc(OC)ccc34)[C@H]2CO)c1	CID:60185199	phase I
BRD-K14783598	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(Cc4ccccc4Cl)C3)n(C)c2c1	CID:60185207	phase I
BRD-K75145803	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccc(F)cc1)C[C@]31CCN(C)CC1	CID:60185208	phase I
BRD-K46512534	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccc(F)cc1)C[C@]31CCN(C)CC1	CID:60185209	phase I
BRD-K18929270	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(Cc4nccs4)C3)C(=O)Nc3cccc(F)c3)n(C)c2c1	CID:60185210	phase I
BRD-K85411199	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(Cc4nccs4)C3)C(=O)Nc3cccc(F)c3)n(C)c2c1	CID:60185211	phase I
BRD-K30229575	COc1ccc2c3c([C@H](CO)N(Cc4cc(OC)cc(OC)c4)C[C@]33CN(C3)C(=O)CN3CCOCC3)n(C)c2c1	CID:60185212	phase I
BRD-K43433419	COc1ccc2c3c([C@@H](CO)N(Cc4cc(OC)cc(OC)c4)C[C@]33CN(C3)C(=O)CN3CCOCC3)n(C)c2c1	CID:60185213	phase I
BRD-K78018080	CCCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)c1ccc(F)cc1	CID:60185214	phase I
BRD-K02004525	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)CC1CC1)C(=O)c1cccc(F)c1	CID:60185215	phase I
BRD-K21400518	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(CC4CCOCC4)C3)S(C)(=O)=O)n(C)c2c1	CID:60185216	phase I
BRD-K94250811	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)NC(C)C)C(=O)c1ccc(F)cc1	CID:60185217	phase I
BRD-K22204517	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)NC(C)C)C(=O)c1ccc(F)cc1	CID:60185218	phase I
BRD-K56301236	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C)C1)C(=O)Cc1ccccc1	CID:60185219	phase I
BRD-K89207838	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C)C1)C(=O)Cc1ccccc1	CID:60185220	phase I
BRD-K29029059	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2ccccc2Cl)C1)C(C)=O	CID:60185221	phase I
BRD-K02242562	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2ccccc2Cl)C1)C(C)=O	CID:60185222	phase I
BRD-K75686993	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)C(=O)Nc1c(C)noc1C	CID:60185223	phase I
BRD-K65983169	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)C(=O)Nc1c(C)noc1C	CID:60185224	phase I
BRD-K65126127	COCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)NC1CCCC1	CID:60185225	phase I
BRD-K86566782	COc1cccc(CN2C[C@]3(CCN(Cc4ccccn4)CC3)c3c([nH]c4cc(OC)ccc34)[C@@H]2CO)c1	CID:60185226	phase I
BRD-K17611527	CCC(=O)N1C[C@]2(CCN(Cc3ccc(Cl)cc3)CC2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60185227	phase I
BRD-K82195532	CCCC(=O)N1C[C@]2(CN(C2)C(=O)C2CC2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60185232	phase I
BRD-K59765229	CCCC(=O)N1C[C@]2(CN(C2)C(=O)C2CC2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60185233	phase I
BRD-K20032161	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3cccc(F)c3)S(C)(=O)=O)n(C)c2c1	CID:60185234	phase I
BRD-K66295388	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3cccc(F)c3)S(C)(=O)=O)n(C)c2c1	CID:60185235	phase I
BRD-K33486590	CCCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)c1ccc(F)cc1	CID:60185236	phase I
BRD-K72624437	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CCN(Cc2ccc(F)cc2)CC1	CID:60185237	phase I
BRD-K29642604	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)S(=O)(=O)c3cccc(C)c3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60185238	phase I
BRD-K68287477	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)S(=O)(=O)c3cccc(C)c3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60185239	phase I
BRD-K59134391	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)S(=O)(=O)c1ccc(C)cc1)C(=O)Nc1ccc(F)cc1	CID:60185240	phase I
BRD-K54173022	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)S(=O)(=O)c1ccc(C)cc1)C(=O)Nc1ccc(F)cc1	CID:60185241	phase I
BRD-K18032654	COCC(=O)N1CC[C@@]2(CC1)CN[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185242	phase I
BRD-K44802037	COCC(=O)N1CC[C@@]2(CC1)CN[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185243	phase I
BRD-K03641022	CCCNC(=O)N1C[C@]2(CCN(CC2)C(=O)C2CCOCC2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60185244	phase I
BRD-K82414981	CCCNC(=O)N1C[C@]2(CCN(CC2)C(=O)C2CCOCC2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60185245	phase I
BRD-K84797952	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)Nc1c(C)noc1C)C(=O)Nc1ccc(F)cc1	CID:60185246	phase I
BRD-K81860076	COCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)NC1CCCC1	CID:60185247	phase I
BRD-K46044238	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CCN(CC3)C(=O)NC(C)C)n(C)c2c1	CID:60185257	phase I
BRD-K21690323	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CCN(CC3)C(=O)NC(C)C)n(C)c2c1	CID:60185258	phase I
BRD-K16930585	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CCN(CC1)C(=O)Nc1ccccc1F	CID:60185259	phase I
BRD-K53549200	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)Nc1ccccc1F	CID:60185260	phase I
BRD-K98328967	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1)C[C@]31CCN(CC1)C(=O)NC(C)C	CID:60185261	phase I
BRD-K12126940	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4ccccn4)CC3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60185262	phase I
BRD-K29582182	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4ccccn4)CC3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60185263	phase I
BRD-K81227048	COCC(=O)N1CC[C@@]2(CC1)CN(Cc1ccccc1Cl)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185264	phase I
BRD-K13624944	COCC(=O)N1CC[C@@]2(CC1)CN(Cc1ccccc1Cl)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185265	phase I
BRD-K49831518	CCCC(=O)N1CC[C@@]2(CC1)CN(Cc1ccc(Cl)cc1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185266	phase I
BRD-K37174007	CCCC(=O)N1CC[C@@]2(CC1)CN(Cc1ccc(Cl)cc1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60185267	phase I
BRD-K78486523	CCS(=O)(=O)N1C[C@@]2(C1)CN(CC1CCOCC1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185268	phase I
BRD-K00818202	CCS(=O)(=O)N1C[C@@]2(C1)CN(CC1CCOCC1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60185269	phase I
BRD-K41814765	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4cc(F)ccc4F)CC3)n(C)c2c1	CID:60185270	phase I
BRD-K46746428	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(Cc4cc(F)ccc4F)CC3)n(C)c2c1	CID:60185271	phase I
BRD-K71590271	CCC(=O)N1C[C@]2(CCN(Cc3ccc(Cl)cc3)CC2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60185284	phase I
BRD-K32631210	COc1cccc(c1)S(=O)(=O)N1C[C@]2(CCN(C)CC2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60185285	phase I
BRD-K25464116	COc1cccc(CN2C[C@]3(CN(Cc4ccccn4)C3)c3c([nH]c4cc(OC)ccc34)[C@@H]2CO)c1	CID:60185339	phase I
BRD-K28890604	COCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Nc1ccccc1F	CID:60185356	phase I
BRD-K76073136	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccn1)C[C@]31CN(C1)C(=O)CC1CC1	CID:60185358	phase I
BRD-K55204560	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1cccc(C)c1)C(=O)Nc1cccc(F)c1	CID:60185359	phase I
BRD-K68205606	C[C@@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:60185638	phase I
BRD-K41633701	C[C@H](CO)N1C[C@H](C)[C@H](CN(C)Cc2cccc(F)c2)Oc3ncc(C#CCN(C)C)cc3C1=O	CID:60185673	phase I
BRD-K43814749	OC[C@@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)C1CCC1	CID:60186110	phase I
BRD-K96285502	COc1ccc(NC(=O)N2C[C@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCC2)cc1	CID:60186146	phase I
BRD-K03194608	COc1ccc(NC(=O)N2C[C@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCC2)cc1	CID:60186147	phase I
BRD-K23543378	COc1ccc(NC(=O)N2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCC2)cc1	CID:60186184	phase I
BRD-K43498025	COc1ccc(NC(=O)N2C[C@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCC2)cc1	CID:60186224	phase I
BRD-K45845536	COCC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60186644	phase I
BRD-K48475203	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CCN(Cc4ccc(F)cc4)CC3)n(C)c2c1	CID:60186697	phase I
BRD-K40446801	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccn1)C(=O)Nc1ccc(F)cc1	CID:60186762	phase I
BRD-K67526586	COCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(Cl)c1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60186793	phase I
BRD-K61880255	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2nccs2)C1)C(=O)Nc1ccc(F)cc1	CID:60186794	phase I
BRD-K25284112	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)C(=O)Nc1ccc(F)cc1	CID:60186824	phase I
BRD-K72736188	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)Nc1ccc2OCOc2c1)C(=O)Nc1ccc(F)cc1	CID:60186845	phase I
BRD-K21368140	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)C(=O)Nc1cccc(F)c1	CID:60186945	phase I
BRD-K57008746	CCCNC(=O)N1C[C@@]2(C1)CN(Cc1cccc(OC)c1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60186973	phase I
BRD-K27797475	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CCOCC2)C1)C(=O)CN(C)C	CID:60186978	phase I
BRD-K08146255	CCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(OC)c1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60186994	phase I
BRD-K46883633	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccccc1)C(=O)CC1CC1	CID:60187003	phase I
BRD-K10846668	CCC(=O)N1CC[C@@]2(CC1)CN(Cc1ccc(Cl)cc1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60187119	phase I
BRD-K33528640	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1F)C[C@]31CCN(CC2CC2)CC1	CID:60187154	phase I
BRD-K60218284	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(Cc4ccccn4)C3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60187163	phase I
BRD-K72345505	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)S(=O)(=O)c3ccccc3)n(C)c2c1	CID:60187247	phase I
BRD-K42951169	COc1ccc(cc1)S(=O)(=O)N1CC[C@@]2(CC1)CN(Cc1ccncc1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60187272	phase I
BRD-K48199580	COc1ccc(cc1)S(=O)(=O)N1CC[C@@]2(CC1)CN(Cc1ccncc1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60187274	phase I
BRD-K50160200	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1Cl)C[C@]31CN(C1)C(C)=O	CID:60187279	phase I
BRD-K86048057	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CN(C3)S(=O)(=O)c3cn(C)cn3)n(C)c2c1	CID:60187282	phase I
BRD-K55260239	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CN(C3)S(=O)(=O)c3cn(C)cn3)n(C)c2c1	CID:60187283	phase I
BRD-K10937407	CCCNC(=O)N1C[C@]2(CCN(Cc3nccs3)CC2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60187284	phase I
BRD-K99469128	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)c3ccccc3)n(C)c2c1	CID:60187317	phase I
BRD-K22836524	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4)C[C@]33CCN(CC4CC4)CC3)n(C)c2c1	CID:60187335	phase I
BRD-K56647759	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)C(=O)Nc3ccc(F)cc3F)n(C)c2c1	CID:60187371	phase I
BRD-K38851002	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60187403	phase I
BRD-K12968907	CCCC(=O)N1C[C@@]2(C1)CN(Cc1ccccc1F)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60187466	phase I
BRD-K77433548	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1nccs1)C[C@]31CN(Cc2ccncc2)C1	CID:60187467	phase I
BRD-K28924448	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1nccs1)C[C@]31CN(Cc2ccncc2)C1	CID:60187469	phase I
BRD-K46504268	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2cccnc2)C1)C(=O)CC1CC1	CID:60187471	phase I
BRD-K73028742	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2cccnc2)C1)C(=O)CC1CC1	CID:60187472	phase I
BRD-K77758624	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1F)C[C@]31CCN(CC1)C(=O)C1CC1	CID:60187473	phase I
BRD-K45235808	CCC(=O)N1C[C@]2(CCN(CC2)C(=O)Nc2c(C)noc2C)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60187474	phase I
BRD-K08039986	COc1ccc2c3c([C@H](CO)N(Cc4ccc(Cl)cc4)C[C@]33CN(CC4CC4)C3)n(C)c2c1	CID:60187499	phase I
BRD-K87972615	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccccc1)S(C)(=O)=O	CID:60187506	phase I
BRD-K99750636	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccn1)C[C@]31CCN(CC1)C(C)=O	CID:60187511	phase I
BRD-K34665338	CCC(=O)N1C[C@]2(CCN(CC2)C(=O)Nc2c(C)noc2C)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60187512	phase I
BRD-K24893212	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CCN(CC3)C(=O)CN3CCOCC3)n(C)c2c1	CID:60187513	phase I
BRD-K15524596	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CCN(CC3)C(=O)c3ccccc3F)n(C)c2c1	CID:60187514	phase I
BRD-K00409771	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1)C[C@]31CCN(Cc2cncnc2)CC1	CID:60187515	phase I
BRD-K62768824	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(CC1CC1)C[C@]31CCN(CC1)S(=O)(=O)c1cccc(F)c1	CID:60187516	phase I
BRD-K88537788	COCC(=O)N1C[C@@]2(C1)CN(Cc1ccc3OCOc3c1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60187518	phase I
BRD-K67498554	COCC(=O)N1C[C@@]2(C1)CN(Cc1ccc3OCOc3c1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60187519	phase I
BRD-K55290744	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)C(=O)Nc3ccccc3F)n(C)c2c1	CID:60187600	phase I
BRD-K39683987	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)Nc1ccc2OCOc2c1	CID:60187611	phase I
BRD-K63261117	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(Cc4ccc(cc4)-c4ccccn4)CC3)n(C)c2c1	CID:60187613	phase I
BRD-K81249055	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4ccc(cc4)-c4ccccn4)CC3)n(C)c2c1	CID:60187614	phase I
BRD-K81119027	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cccc(Cl)c1)C[C@]31CN(C)C1	CID:60187720	phase I
BRD-K63874400	COc1ccc2c3c([C@H](CO)NC[C@]33CN(Cc4cc(on4)-c4ccccc4)C3)n(C)c2c1	CID:60187750	phase I
BRD-K00412766	CN1[C@H](CO)[C@@H]2CCN([C@@H]2c2cc(ccc12)C1=CCCCC1)C(=O)NC1CCCC1	CID:60187786	phase I
BRD-K67794838	COc1cccc(c1)-c1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCCCC1	CID:60187817	phase I
BRD-K31695944	OC[C@@H]1Nc2ccc(Br)cc2[C@H]2[C@@H]1CCN2C(=O)C1CCCC1	CID:60187853	phase I
BRD-K99842945	CN1[C@@H](CO)[C@H]2CCN([C@H]2c2cc(ccc12)C1=CCCCC1)C(=O)NC1CCCC1	CID:60187856	phase I
BRD-K40397365	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)c1cccc(F)c1)-c1ccccc1	CID:60187910	phase I
BRD-K47170156	OC[C@H]1Nc2ccc(cc2[C@@H]2[C@H]1CCN2C(=O)C1CCC1)-c1ccc(cc1)C#N	CID:60187952	phase I
BRD-K16128171	OC[C@H]1[C@H]([C@@H](C#N)N1C(=O)NC1CCCCC1)c1ccccc1C1=CCCCC1	CID:60187989	phase I
BRD-K91501298	COc1ccc(cc1)C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCCC1	CID:60188007	phase I
BRD-K44401329	COc1ccc(cc1)C#Cc1ccc2N[C@H](CO)[C@@H]3CCN([C@@H]3c2c1)C(=O)C1CCC1	CID:60188036	phase I
BRD-K13369161	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60188067	phase I
BRD-K66254772	O=C1C=CCCN1S(=O)(=O)\C=C\c1ccccc1	CID:60188101	phase I
BRD-K10799838	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(Cc1ccccc1)CC2=O	CID:60188399	phase I
BRD-K42136113	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(Cc1ccccc1)CC2=O	CID:60188411	phase I
BRD-K45534781	OC[C@@H]1Nc2ccc(cc2[C@H]2[C@@H]1CCN2C(=O)C1CCCC1)C1=CCCCC1	CID:60188647	phase I
BRD-K53582057	OC[C@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCCC1	CID:60188667	phase I
BRD-K10542638	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CC1)c1ccc(cc1)C1=CCCCC1	CID:60188674	phase I
BRD-K05378136	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60188698	phase I
BRD-K55341184	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60188702	phase I
BRD-K62865272	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCC1	CID:60188733	phase I
BRD-K87634799	OC[C@@H]1[C@H]([C@@H](C#N)N1C(=O)NC1CCCC1)c1ccc(cc1)C1=CCCCC1	CID:60188849	phase I
BRD-K14628187	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCCC1	CID:60189055	phase I
BRD-K84963986	OC[C@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCCC1	CID:60189083	phase I
BRD-K17808354	OC[C@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCCC1	CID:60189084	phase I
BRD-K00505809	OC[C@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCCC1	CID:60189085	phase I
BRD-K46268437	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCCC1	CID:60189086	phase I
BRD-K10302728	COc1ccc(NC(=O)N2C[C@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189159	phase I
BRD-K75620843	COc1ccc(NC(=O)N2C[C@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189160	phase I
BRD-K67561376	COc1ccc(NC(=O)N2C[C@@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189161	phase I
BRD-K22145792	COc1ccc(NC(=O)N2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189162	phase I
BRD-K83098569	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189163	phase I
BRD-K14055576	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189164	phase I
BRD-K21990111	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189165	phase I
BRD-K06425073	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189166	phase I
BRD-K42307233	COc1ccccc1NC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(C)c1	CID:60189167	phase I
BRD-K70673311	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(C)c1	CID:60189168	phase I
BRD-K20065789	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(C)c1	CID:60189169	phase I
BRD-K01125214	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189170	phase I
BRD-K86831676	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189171	phase I
BRD-K82735282	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189172	phase I
BRD-K96522482	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189173	phase I
BRD-K00502422	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189174	phase I
BRD-K59294904	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189175	phase I
BRD-K72794452	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189176	phase I
BRD-K62263376	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189177	phase I
BRD-K52929685	COc1ccc(NC(=O)N2C[C@@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189196	phase I
BRD-K49434474	COc1ccc(NC(=O)N2C[C@@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189197	phase I
BRD-K33078666	COc1ccc(NC(=O)N2C[C@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189198	phase I
BRD-K93993903	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189199	phase I
BRD-K76537832	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189200	phase I
BRD-K15029638	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189201	phase I
BRD-K59777289	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189202	phase I
BRD-K23091373	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189203	phase I
BRD-K40628462	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(C)c1	CID:60189204	phase I
BRD-K43050752	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccncc1)c1ccc(Br)cc1	CID:60189205	phase I
BRD-K56870772	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccncc1)c1ccc(Br)cc1	CID:60189206	phase I
BRD-K66551929	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccncc1)c1ccc(Br)cc1	CID:60189207	phase I
BRD-K35861449	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)NC1CCCCC1)c1ccc(cc1)-c1ccncc1	CID:60189208	phase I
BRD-K94011376	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)NC1CCCCC1)c1ccc(cc1)-c1ccncc1	CID:60189209	phase I
BRD-K37529519	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)NC1CCCCC1)c1ccc(cc1)-c1ccncc1	CID:60189210	phase I
BRD-K34985200	CN(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CN(C)C	CID:60189211	phase I
BRD-K58576935	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189212	phase I
BRD-K75984692	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189239	phase I
BRD-K03213425	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189240	phase I
BRD-K87324885	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CCc1ccccc1	CID:60189241	phase I
BRD-K16663346	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CNCC2=O	CID:60189242	phase I
BRD-K51919154	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CNCC2=O	CID:60189243	phase I
BRD-K06373645	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CNCC2=O	CID:60189244	phase I
BRD-K69100231	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CNCC2=O	CID:60189245	phase I
BRD-K52688277	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60189246	phase I
BRD-K22597651	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60189247	phase I
BRD-K64119425	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60189248	phase I
BRD-K58407898	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1cc(F)ccc1F)c1ccc(\C=C\c2ccccc2)cc1	CID:60189269	phase I
BRD-K16227029	O[C@H]1COC[C@@H]2O[C@@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(CC2CCCC2)C1	CID:60189280	phase I
BRD-K11880555	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189286	phase I
BRD-K22314621	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189287	phase I
BRD-K07591425	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189288	phase I
BRD-K73202406	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189289	phase I
BRD-K13673853	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189290	phase I
BRD-K85865817	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60189291	phase I
BRD-K89107430	C\C=C\c1ccc2N[C@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)C1CCCC1	CID:60189295	phase I
BRD-K48744855	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1cc(F)ccc1F)c1ccc(\C=C\c2ccccc2)cc1	CID:60189302	phase I
BRD-K75143842	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1cc(F)ccc1F)c1ccc(\C=C\c2ccccc2)cc1	CID:60189303	phase I
BRD-K95147502	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1cc(F)ccc1F)c1ccc(\C=C\c2ccccc2)cc1	CID:60189304	phase I
BRD-K90397906	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189305	phase I
BRD-K61565464	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189306	phase I
BRD-K70407915	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189307	phase I
BRD-K34825242	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189308	phase I
BRD-K35827873	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189309	phase I
BRD-K32240435	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C#Cc1cccnc1	CID:60189310	phase I
BRD-K93527821	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccn1	CID:60189311	phase I
BRD-K96393402	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccn1	CID:60189312	phase I
BRD-K91007808	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccn1	CID:60189313	phase I
BRD-K02929561	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccn1	CID:60189314	phase I
BRD-K30842998	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccccn1)c1ccc(cc1)C1=CCCC1	CID:60189315	phase I
BRD-K58781576	OC[C@@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189316	phase I
BRD-K54647312	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189317	phase I
BRD-K18255961	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189318	phase I
BRD-K54877231	OC[C@@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189319	phase I
BRD-K78298277	OC[C@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189320	phase I
BRD-K86300178	OC[C@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189321	phase I
BRD-K24243182	OC[C@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189322	phase I
BRD-K12951693	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccccc1)c1ccc(cc1)-c1ccccc1	CID:60189345	phase I
BRD-K35176035	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189346	phase I
BRD-K59078549	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189347	phase I
BRD-K45807461	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189348	phase I
BRD-K77643021	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189349	phase I
BRD-K46774516	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189350	phase I
BRD-K11923178	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189351	phase I
BRD-K37470774	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)C#CC1CC1	CID:60189352	phase I
BRD-K48710089	COC(=O)c1ccc(CN2C[C@@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)-c2cccnc2)cc1	CID:60189353	phase I
BRD-K54092557	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccn1	CID:60189354	phase I
BRD-K27401646	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccn1	CID:60189355	phase I
BRD-K25337138	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:60189356	phase I
BRD-K91738126	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:60189357	phase I
BRD-K10483446	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:60189358	phase I
BRD-K04192660	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:60189359	phase I
BRD-K50655333	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:60189360	phase I
BRD-K39394160	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)-c1cccc(F)c1	CID:60189361	phase I
BRD-K62415056	OC[C@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C1=CCCC1	CID:60189362	phase I
BRD-K35970781	CCN1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189363	phase I
BRD-K00504156	CCN1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189364	phase I
BRD-K10701803	CCN1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189365	phase I
BRD-K36473494	CCN1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189366	phase I
BRD-K72128077	CCN1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189367	phase I
BRD-K62157654	CCN1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189368	phase I
BRD-K94288726	OC[C@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C#CC1CCCCC1	CID:60189389	phase I
BRD-K52276780	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C#CC1CCCCC1	CID:60189390	phase I
BRD-K18076490	OC[C@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C#CC1CCCCC1	CID:60189391	phase I
BRD-K23903329	OC[C@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C#CC1CCCCC1	CID:60189392	phase I
BRD-K97994060	OC[C@@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C#CC1CCCCC1	CID:60189393	phase I
BRD-K39548949	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C#CC1CCCCC1	CID:60189394	phase I
BRD-K13752834	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189395	phase I
BRD-K60175505	COC(=O)c1ccc(CN2C[C@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)-c2cccnc2)cc1	CID:60189396	phase I
BRD-K46842958	COC(=O)c1ccc(CN2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)-c2cccnc2)cc1	CID:60189397	phase I
BRD-K77058876	COC(=O)c1ccc(CN2C[C@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)-c2cccnc2)cc1	CID:60189398	phase I
BRD-K16698502	COC(=O)c1ccc(CN2C[C@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)-c2cccnc2)cc1	CID:60189399	phase I
BRD-K25902674	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189400	phase I
BRD-K30025108	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189401	phase I
BRD-K38381720	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189402	phase I
BRD-K90819764	CCN1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189403	phase I
BRD-K24639784	CCN1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60189404	phase I
BRD-K96343378	O[C@H]1COC[C@@H]2O[C@H](CC(=O)NCc3ccc(Cl)cc3)CC[C@H]2N(CC2CCCC2)C1	CID:60189405	phase I
BRD-K40704255	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189421	phase I
BRD-K02485640	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189422	phase I
BRD-K57572982	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189423	phase I
BRD-K79287095	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189424	phase I
BRD-K10196668	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189425	phase I
BRD-K23674935	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189426	phase I
BRD-K76718418	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60189427	phase I
BRD-K12148366	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1cccnc1	CID:60189428	phase I
BRD-K85567359	COc1cccc(c1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1cccnc1	CID:60189429	phase I
BRD-K08982647	COc1cccc(c1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1cccnc1	CID:60189430	phase I
BRD-K11219023	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189431	phase I
BRD-K53636670	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189445	phase I
BRD-K19651468	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189446	phase I
BRD-K47686040	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189455	phase I
BRD-K68731612	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189456	phase I
BRD-K12034365	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189457	phase I
BRD-K98711518	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189458	phase I
BRD-K38810814	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189459	phase I
BRD-K38997615	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189460	phase I
BRD-K10954923	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189461	phase I
BRD-K92022308	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccccc1F	CID:60189462	phase I
BRD-K45145114	COc1cccc(NC(=O)N2C[C@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCCC2)c1	CID:60189463	phase I
BRD-K29655991	COc1cccc(NC(=O)N2C[C@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCCC2)c1	CID:60189464	phase I
BRD-K05248013	COc1cccc(NC(=O)N2C[C@@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCCC2)c1	CID:60189465	phase I
BRD-K91269812	COc1cccc(NC(=O)N2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C2=CCCCC2)c1	CID:60189466	phase I
BRD-K65170870	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189487	phase I
BRD-K93791165	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)S(=O)(=O)Cc1ccccc1)c1ccc(cc1)C#Cc1ccccc1	CID:60189488	phase I
BRD-K41169041	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189489	phase I
BRD-K71132173	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189490	phase I
BRD-K70543679	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189491	phase I
BRD-K23243038	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189492	phase I
BRD-K88955481	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189493	phase I
BRD-K68013677	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189494	phase I
BRD-K77990919	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189495	phase I
BRD-K54639145	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189496	phase I
BRD-K03770502	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189497	phase I
BRD-K31883641	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189498	phase I
BRD-K22691925	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189499	phase I
BRD-K93716900	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189500	phase I
BRD-K00119817	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189501	phase I
BRD-K62717630	COc1cccc(c1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1cccnc1	CID:60189524	phase I
BRD-K33967077	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189525	phase I
BRD-K08722369	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189526	phase I
BRD-K83754856	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189527	phase I
BRD-K20962057	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189528	phase I
BRD-K62794454	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189529	phase I
BRD-K90787403	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189530	phase I
BRD-K01715539	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(Cc1ccc(F)cc1)CC2=O	CID:60189531	phase I
BRD-K69607079	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189532	phase I
BRD-K36221157	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60189533	phase I
BRD-K58577862	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(C)(=O)=O	CID:60189534	phase I
BRD-K65109005	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(C)(=O)=O	CID:60189535	phase I
BRD-K16254782	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(C)(=O)=O	CID:60189536	phase I
BRD-K00846914	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(C)(=O)=O	CID:60189537	phase I
BRD-K06111088	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(C)(=O)=O	CID:60189538	phase I
BRD-K71944937	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1C	CID:60189539	phase I
BRD-K82933801	CCS(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C1=CCCCC1	CID:60189566	phase I
BRD-K41035516	CCCNC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189567	phase I
BRD-K31844452	CCCNC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189568	phase I
BRD-K54254994	CCCNC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189569	phase I
BRD-K21075720	CCCNC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189570	phase I
BRD-K74236049	CCCNC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189571	phase I
BRD-K23496480	CCCNC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189572	phase I
BRD-K63145939	CCCNC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189573	phase I
BRD-K55692246	CCCNC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60189574	phase I
BRD-K79157816	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189575	phase I
BRD-K02689622	COc1ccc(NC(=O)N2C[C@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(Br)cc2)cc1	CID:60189599	phase I
BRD-K82483257	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189600	phase I
BRD-K27838482	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189601	phase I
BRD-K02749944	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189602	phase I
BRD-K35073835	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189603	phase I
BRD-K79032360	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189616	phase I
BRD-K97226655	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189617	phase I
BRD-K46298622	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(cc1)C#Cc1cccc(F)c1	CID:60189618	phase I
BRD-K89469595	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189619	phase I
BRD-K20505830	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189620	phase I
BRD-K88700643	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189621	phase I
BRD-K14428604	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccccc1F	CID:60189622	phase I
BRD-K63211577	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189623	phase I
BRD-K75889393	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189624	phase I
BRD-K14842933	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60189625	phase I
BRD-K00348196	COCC(=O)N1C[C@]2(CN(Cc3ccccc3)C2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60189639	phase I
BRD-K96697180	COc1ccc(CN2C[C@]3(CCN(CC3)C(=O)Cc3ccncc3)c3c([nH]c4cc(OC)ccc34)[C@@H]2CO)cc1	CID:60189640	phase I
BRD-K04512584	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)S(C)(=O)=O)C(=O)C1CCC1	CID:60189641	phase I
BRD-K88819433	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cccc(Cl)c1)C[C@]31CCN(C)CC1	CID:60189643	phase I
BRD-K19888970	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4OC)C[C@]33CN(C)C3)n(C)c2c1	CID:60189645	phase I
BRD-K55277887	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(CC3CCOCC3)C2)N1Cc1cncnc1	CID:60189646	phase I
BRD-K44012584	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3cccnc3)C2)N1C(=O)CC1CC1	CID:60189647	phase I
BRD-K55706946	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N(CC2CC2)C11CN(C1)S(C)(=O)=O	CID:60189648	phase I
BRD-K94397824	COc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N(CC2CC2)C11CN(C1)S(C)(=O)=O	CID:60189649	phase I
BRD-K04445149	COc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N(CC2CC2)C11CN(C1)S(C)(=O)=O	CID:60189650	phase I
BRD-K07493822	CCC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccc2OCOc2c1	CID:60189651	phase I
BRD-K69698931	CCC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccc2OCOc2c1	CID:60189652	phase I
BRD-K31969867	CCC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)c1ccc2OCOc2c1	CID:60189653	phase I
BRD-K08150827	OC[C@@H]1[C@H](c2ccccc2)C2(CN(CCC(F)(F)F)C2)N1Cc1cccnc1	CID:60189654	phase I
BRD-K42540297	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(CCC(F)(F)F)C2)N1Cc1cccnc1	CID:60189655	phase I
BRD-K02914492	CC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)CC1CC1)c1ccc(cc1)-c1ccccc1C	CID:60189656	phase I
BRD-K48350747	CC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)CC1CC1)c1ccc(cc1)-c1ccccc1C	CID:60189657	phase I
BRD-K64579699	CC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)CC1CC1)c1ccc(cc1)-c1ccccc1C	CID:60189658	phase I
BRD-K51390731	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N(C(=O)C2CC2)C11CN(C1)C(C)=O	CID:60189659	phase I
BRD-K74823182	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(=O)C2CC2)C11CN(C1)C(C)=O	CID:60189660	phase I
BRD-K72901512	CCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)CC)c1ccc(cc1)-c1ccc(F)cc1	CID:60189662	phase I
BRD-K09057839	CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccc1	CID:60189663	phase I
BRD-K76050206	COc1ccc2c3c([C@@H](CO)N(Cc4ccc(F)cc4)C[C@]33CCN(C)CC3)n(C)c2c1	CID:60189664	phase I
BRD-K76397886	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccncc1)C[C@]31CCN(Cc2ccc(cc2)-c2ccccn2)CC1	CID:60189666	phase I
BRD-K17138170	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccncc1)C[C@]31CCN(Cc2ccc(cc2)-c2ccccn2)CC1	CID:60189667	phase I
BRD-K54553362	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)NC(C)C)C(=O)CC3CC3)n(C)c2c1	CID:60189669	phase I
BRD-K99049289	CCCNC(=O)N1C[C@]2(CN(CC3CCCCC3)C2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60189670	phase I
BRD-K38965191	CCCNC(=O)N1C[C@]2(CN(CC3CCCCC3)C2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60189671	phase I
BRD-K36194373	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1cccc(Cl)c1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60189672	phase I
BRD-K51797651	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1cccc(Cl)c1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60189673	phase I
BRD-K70727050	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccc(Cl)cc1)C[C@]31CN(C1)S(C)(=O)=O	CID:60189677	phase I
BRD-K27882424	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccc(Cl)cc1)C[C@]31CN(C1)S(C)(=O)=O	CID:60189679	phase I
BRD-K37569719	COc1ccc(NC(=O)N2CC[C@@]3(CC2)CN([C@@H](CO)c2[nH]c4cc(OC)ccc4c32)C(=O)CN2CCOCC2)cc1	CID:60189680	phase I
BRD-K25255972	COc1ccc(NC(=O)N2CC[C@@]3(CC2)CN([C@H](CO)c2[nH]c4cc(OC)ccc4c32)C(=O)CN2CCOCC2)cc1	CID:60189681	phase I
BRD-K94740841	COc1ccc(NC(=O)N2CC[C@@]3(CC2)CN([C@@H](CO)c2c3c3ccc(OC)cc3n2C)C(=O)C2CCC2)cc1	CID:60189682	phase I
BRD-K42863614	COc1ccc(NC(=O)N2CC[C@@]3(CC2)CN([C@H](CO)c2c3c3ccc(OC)cc3n2C)C(=O)C2CCC2)cc1	CID:60189683	phase I
BRD-K59722298	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)Nc1cccc(F)c1)C(=O)NC1CCCC1	CID:60189685	phase I
BRD-K99633760	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)c3cccnc3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60189687	phase I
BRD-K89840812	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)c3cccnc3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60189688	phase I
BRD-K66658536	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4OC)C[C@]33CN(C)C3)n(C)c2c1	CID:60189690	phase I
BRD-K70697816	CCCNC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Nc1ccc(F)cc1	CID:60189691	phase I
BRD-K60528884	CCCNC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Nc1ccc(F)cc1	CID:60189692	phase I
BRD-K86249754	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC2CCCC2)CC1)S(C)(=O)=O	CID:60189693	phase I
BRD-K87829407	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC2CCCC2)CC1)S(C)(=O)=O	CID:60189694	phase I
BRD-K47967838	COc1ccc2c3c([C@@H](CO)N(Cc4ccccn4)C[C@]33CN(C3)C(=O)NC(C)C)n(C)c2c1	CID:60189695	phase I
BRD-K44937047	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2ccccc2)C1)S(=O)(=O)c1ccc(C)cc1	CID:60189696	phase I
BRD-K03223506	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2ccccc2)C1)S(=O)(=O)c1ccc(C)cc1	CID:60189698	phase I
BRD-K58985955	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1CCC(F)(F)F	CID:60189699	phase I
BRD-K95935167	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1CCC(F)(F)F	CID:60189701	phase I
BRD-K68589684	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1CCC(F)(F)F	CID:60189702	phase I
BRD-K98546418	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N(C11CN(C1)C(=O)C1CCCC1)S(=O)(=O)Cc1ccccc1	CID:60189703	phase I
BRD-K71214345	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)C2CCOCC2)C11CN(C1)C(=O)NC(C)C	CID:60189704	phase I
BRD-K92979098	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(=O)C2CCOCC2)C11CN(C1)C(=O)NC(C)C	CID:60189705	phase I
BRD-K13089870	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3cccc(Cl)c3)C2)N1C(=O)C1CCOCC1	CID:60189707	phase I
BRD-K40043058	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)C2CC2)C11CN(C1)C(C)=O	CID:60189708	phase I
BRD-K73032790	COCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)NC1CCCC1)c1ccccc1	CID:60189710	phase I
BRD-K75880427	COCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)NC1CCCC1)c1ccccc1	CID:60189712	phase I
BRD-K12743465	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C)C[C@]31CN(C1)C(=O)C1CC1	CID:60189713	phase I
BRD-K23162766	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C)C[C@]31CN(C1)C(=O)C1CC1	CID:60189714	phase I
BRD-K48549412	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)Cc3ccccc3)C(=O)c3ccccn3)n(C)c2c1	CID:60189715	phase I
BRD-K36627189	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)Cc3ccccc3)C(=O)c3ccccn3)n(C)c2c1	CID:60189716	phase I
BRD-K41705395	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)NC3CCCC3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60189717	phase I
BRD-K56704970	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)NC3CCCC3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60189718	phase I
BRD-K62384871	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccn1)C[C@]31CCN(CC1)C(=O)c1ccccn1	CID:60189719	phase I
BRD-K58043445	COc1ccc2c3c([C@@H](CO)N(Cc4cccnc4)C[C@]33CCN(CC3)C(=O)NC(C)C)n(C)c2c1	CID:60189720	phase I
BRD-K83871946	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CC2)C1)C(=O)Nc1cccc(F)c1	CID:60189721	phase I
BRD-K11628545	CCCC(=O)N1C[C@@]2(C1)CN(Cc1cccnc1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189722	phase I
BRD-K79094264	CCCC(=O)N1C[C@@]2(C1)CN(Cc1cccnc1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189723	phase I
BRD-K04418684	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3c(C)noc3C)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60189724	phase I
BRD-K98988824	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3c(C)noc3C)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60189725	phase I
BRD-K43263266	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4ccccc4OC)CC3)C(C)=O)n(C)c2c1	CID:60189726	phase I
BRD-K85236313	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4ccccc4OC)CC3)C(C)=O)n(C)c2c1	CID:60189727	phase I
BRD-K58607374	CCC(=O)N1C[C@]2(CCN(Cc3ccccc3Cl)CC2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60189729	phase I
BRD-K88899793	CCC(=O)N1C[C@]2(CCN(Cc3ccccc3Cl)CC2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60189730	phase I
BRD-K67215204	COCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)S(C)(=O)=O	CID:60189731	phase I
BRD-K51410836	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)c1ccc(F)cc1	CID:60189732	phase I
BRD-K16769902	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)c1ccc(F)cc1	CID:60189733	phase I
BRD-K21483310	CCCNC(=O)N1C[C@]2(CN(C2)S(C)(=O)=O)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60189734	phase I
BRD-K76656279	CCCNC(=O)N1C[C@]2(CN(C2)S(C)(=O)=O)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60189735	phase I
BRD-K96178772	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CN(C)C1	CID:60189736	phase I
BRD-K67301423	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CN(C)C1	CID:60189737	phase I
BRD-K63565086	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1cccc(OC)c1	CID:60189738	phase I
BRD-K40951733	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1cccc(OC)c1	CID:60189739	phase I
BRD-K65393151	COc1ccc2c3c([C@H](CO)N(Cc4ccncc4)C[C@]33CCN(CC3)C(=O)Cc3ccncc3)n(C)c2c1	CID:60189741	phase I
BRD-K93253774	OC[C@H]1[C@@H](c2ccccc2)C2(CN(Cc3cccc(Cl)c3)C2)N1C(=O)C1CCOCC1	CID:60189742	phase I
BRD-K82528406	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CN2CCOCC2)N1Cc1ccc(F)cc1	CID:60189744	phase I
BRD-K18220124	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)CN2CCOCC2)N1Cc1ccc(F)cc1	CID:60189745	phase I
BRD-K90365097	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)NC(C)C)c1ccccc1	CID:60189746	phase I
BRD-K87471235	CCCNC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)C1CCCCC1	CID:60189747	phase I
BRD-K16074065	CCCNC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)C1CCCCC1	CID:60189748	phase I
BRD-K07184814	CCCNC(=O)N1[C@@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)C1CCCCC1	CID:60189749	phase I
BRD-K90198040	CCCNC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)C1CCCCC1	CID:60189751	phase I
BRD-K11957915	CCC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)CN1CCOCC1	CID:60189752	phase I
BRD-K13059702	CCC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)CN1CCOCC1	CID:60189753	phase I
BRD-K32197572	CCCNC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)c1ccccc1	CID:60189754	phase I
BRD-K40115967	CCCNC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)c1ccccc1	CID:60189755	phase I
BRD-K85981997	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CN(C1)C(=O)C1CCC1	CID:60189756	phase I
BRD-K03515135	CCCC(=O)N1C[C@]2(CN(C2)C(=O)NC(C)C)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60189757	phase I
BRD-K62536321	CCCC(=O)N1C[C@]2(CN(C2)C(=O)NC(C)C)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60189759	phase I
BRD-K29243968	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC4CC4)CC3)C(=O)c3ccncc3)n(C)c2c1	CID:60189760	phase I
BRD-K20170530	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC4CC4)CC3)C(=O)c3ccncc3)n(C)c2c1	CID:60189761	phase I
BRD-K76373654	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)c3cnccn3)C(C)=O)n(C)c2c1	CID:60189762	phase I
BRD-K96797558	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)c3cnccn3)C(C)=O)n(C)c2c1	CID:60189764	phase I
BRD-K50790730	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2ccccc2)C1)C(=O)c1cccnc1	CID:60189766	phase I
BRD-K57420195	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2ccccc2)C1)C(=O)c1cccnc1	CID:60189768	phase I
BRD-K14200107	COCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)S(C)(=O)=O	CID:60189769	phase I
BRD-K48424967	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(C)CC3)C(=O)NC3CCCCC3)n(C)c2c1	CID:60189771	phase I
BRD-K19402218	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(C)CC3)C(=O)NC3CCCCC3)n(C)c2c1	CID:60189772	phase I
BRD-K31633278	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1nccs1)C[C@]31CCN(Cc2cccnc2)CC1	CID:60189773	phase I
BRD-K99310510	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1nccs1)C[C@]31CCN(Cc2cccnc2)CC1	CID:60189774	phase I
BRD-K99354840	COc1ccc2c3c([C@H](CO)N(Cc4nccs4)C[C@]33CCN(CC3)C(=O)CN(C)C)n(C)c2c1	CID:60189775	phase I
BRD-K44715408	COc1ccc2c3c([C@@H](CO)N(Cc4nccs4)C[C@]33CCN(CC3)C(=O)CN(C)C)n(C)c2c1	CID:60189776	phase I
BRD-K61148205	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)CC3CC3)C(=O)C3CCCC3)n(C)c2c1	CID:60189777	phase I
BRD-K95052025	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)CC3CC3)C(=O)C3CCCC3)n(C)c2c1	CID:60189778	phase I
BRD-K59253994	COc1ccc2c3c([C@@H](CO)N(Cc4ccncc4)C[C@]33CCN(CC3)C(=O)Cc3ccncc3)n(C)c2c1	CID:60189779	phase I
BRD-K26359746	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)C3CCOCC3)C(C)=O)n(C)c2c1	CID:60189781	phase I
BRD-K69557760	COCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)NC1CCCC1)c1ccccc1	CID:60189782	phase I
BRD-K83365102	CN(C)CC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(Cc2cc(F)ccc2F)C1	CID:60189784	phase I
BRD-K43566466	CC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccc1	CID:60189785	phase I
BRD-K74338856	CC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccc1	CID:60189787	phase I
BRD-K73548235	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2ccccc2F)CC1)S(=O)(=O)c1cn(C)cn1	CID:60189788	phase I
BRD-K26441788	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2ccccc2F)CC1)S(=O)(=O)c1cn(C)cn1	CID:60189790	phase I
BRD-K86413298	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4cccnc4)CC3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60189792	phase I
BRD-K56040567	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4cccnc4)CC3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60189793	phase I
BRD-K54492529	CCCNC(=O)N1CC[C@@]2(CC1)CN(Cc1cccc(OC)c1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189794	phase I
BRD-K87959840	CCCNC(=O)N1CC[C@@]2(CC1)CN(Cc1cccc(OC)c1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189795	phase I
BRD-K67887361	CCCNC(=O)N1C[C@]2(CN(C2)C(=O)c2cnccn2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60189796	phase I
BRD-K16483711	CCCNC(=O)N1C[C@]2(CN(C2)C(=O)c2cnccn2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60189798	phase I
BRD-K79356120	CCCNC(=O)N1C[C@]2(CCN(Cc3cccc(OC)c3)CC2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60189799	phase I
BRD-K60944301	CCCNC(=O)N1C[C@]2(CCN(Cc3cccc(OC)c3)CC2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60189800	phase I
BRD-K95964003	COc1ccc2c3c([C@H](CO)N(Cc4cc(F)ccc4F)C[C@]33CN(C3)C(=O)C3CC3)n(C)c2c1	CID:60189802	phase I
BRD-K06555318	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CN2CCOCC2)N1Cc1ccc(F)cc1	CID:60189803	phase I
BRD-K66694259	CC(=O)N1[C@H](CO)[C@@H](c2ccc(cc2)-c2ccc(cc2)C#N)C11CN(C1)C(=O)C1CC1	CID:60189804	phase I
BRD-K62982188	CN(C)CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(Cc2cc(F)ccc2F)C1	CID:60189805	phase I
BRD-K54360306	COc1cccc(CN2CC3(C2)[C@@H]([C@H](CO)N3C(=O)Cc2ccccc2)c2ccccc2)c1	CID:60189806	phase I
BRD-K54791528	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2cccc(F)c2)N1C(=O)C1CCCCC1	CID:60189807	phase I
BRD-K81550430	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2cccc(F)c2)N1C(=O)C1CCCCC1	CID:60189809	phase I
BRD-K87634307	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2cccc(F)c2)N1C(=O)C1CCCCC1	CID:60189810	phase I
BRD-K21200579	CCCNC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(CCC(F)(F)F)C1	CID:60189811	phase I
BRD-K33693037	CCCNC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(CCC(F)(F)F)C1	CID:60189812	phase I
BRD-K68937877	OC[C@@H]1N(C(=O)C2CCCC2)C2(CN(Cc3ccc(F)cc3)C2)[C@@H]1c1ccccc1	CID:60189813	phase I
BRD-K34639069	CS(=O)(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CCC(F)(F)F)c1ccccc1	CID:60189814	phase I
BRD-K17983173	CS(=O)(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CCC(F)(F)F)c1ccccc1	CID:60189815	phase I
BRD-K43026564	CS(=O)(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CCC(F)(F)F)c1ccccc1	CID:60189816	phase I
BRD-K72700227	CS(=O)(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)C1CCC1)c1ccccc1	CID:60189817	phase I
BRD-K17367351	CS(=O)(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)C1CCC1)c1ccccc1	CID:60189818	phase I
BRD-K34451734	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3ccccn3)C2)N1Cc1cncnc1	CID:60189819	phase I
BRD-K15706160	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cc(F)ccc1F)C[C@]31CN(C1)C(=O)C1CCC1	CID:60189820	phase I
BRD-K74704013	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4)C[C@]33CN(C3)C(=O)c3ccccc3F)n(C)c2c1	CID:60189821	phase I
BRD-K75872636	CCCC(=O)N1C[C@]2(CN(C2)S(C)(=O)=O)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60189822	phase I
BRD-K12916986	CCCC(=O)N1C[C@]2(CN(C2)S(C)(=O)=O)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60189823	phase I
BRD-K91473136	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(CC4CC4)C3)C(=O)Nc3c(C)noc3C)n(C)c2c1	CID:60189824	phase I
BRD-K08412560	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(CC4CC4)C3)C(=O)Nc3c(C)noc3C)n(C)c2c1	CID:60189826	phase I
BRD-K86457545	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccncc1)S(C)(=O)=O	CID:60189828	phase I
BRD-K80907598	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccncc1)S(C)(=O)=O	CID:60189829	phase I
BRD-K22264435	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CN(C1)C(=O)Nc1ccc(F)cc1F	CID:60189830	phase I
BRD-K31635696	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4ccncc4)CC3)C(=O)CN3CCOCC3)n(C)c2c1	CID:60189832	phase I
BRD-K97924280	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccccn1)C(=O)Nc1ccc(F)cc1	CID:60189833	phase I
BRD-K69572618	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccccn1)C(=O)Nc1ccc(F)cc1	CID:60189834	phase I
BRD-K38908436	CC(=O)N1[C@H](CO)[C@H](c2ccc(cc2)-c2ccc(cc2)C#N)C11CN(C1)C(=O)C1CC1	CID:60189838	phase I
BRD-K30021624	CC(=O)N1[C@@H](CO)[C@@H](c2ccc(cc2)-c2ccc(cc2)C#N)C11CN(C1)C(=O)C1CC1	CID:60189839	phase I
BRD-K15240833	CC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)S(=O)(=O)c1ccccc1	CID:60189840	phase I
BRD-K90721481	CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)S(=O)(=O)c1ccccc1	CID:60189841	phase I
BRD-K93413915	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(C)=O)c1ccc(cc1)-c1ccccc1OC	CID:60189843	phase I
BRD-K74709515	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(C)=O)c1ccc(cc1)-c1ccccc1OC	CID:60189844	phase I
BRD-K86715767	CCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(C)=O)c1ccc(cc1)-c1ccccc1OC	CID:60189845	phase I
BRD-K47662318	CC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CC1CC1)c1ccc(cc1)-c1ccc(F)cc1	CID:60189846	phase I
BRD-K61242280	CC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2Cc1ccccc1F)c1ccccc1	CID:60189847	phase I
BRD-K74972903	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)Cc2cccnc2)N1C(=O)C1CCOCC1	CID:60189849	phase I
BRD-K04729818	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)Cc2cccnc2)N1C(=O)C1CCOCC1	CID:60189850	phase I
BRD-K36841620	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)Cc2cccnc2)N1C(=O)C1CCOCC1	CID:60189851	phase I
BRD-K56395592	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1Cc1nccs1	CID:60189852	phase I
BRD-K31285743	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1Cc1nccs1	CID:60189853	phase I
BRD-K96270963	OC[C@H]1[C@@H](c2ccccc2)C2(CN(Cc3ccccn3)C2)N1Cc1cncnc1	CID:60189854	phase I
BRD-K17800788	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1C(=O)CC1CC1	CID:60189855	phase I
BRD-K13383838	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1C(=O)CC1CC1	CID:60189856	phase I
BRD-K06715209	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1C(=O)CC1CC1	CID:60189857	phase I
BRD-K35304243	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(C)=O)C11CN(C1)C(=O)NC1CCCCC1	CID:60189858	phase I
BRD-K85410924	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(C)=O)C11CN(C1)C(=O)NC1CCCCC1	CID:60189859	phase I
BRD-K04802065	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1Cc1cccc(F)c1	CID:60189861	phase I
BRD-K85573444	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1Cc1cccc(F)c1	CID:60189862	phase I
BRD-K18721752	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1Cc1cccc(F)c1	CID:60189863	phase I
BRD-K40522524	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4)C[C@]33CN(C3)C(=O)c3ccccc3F)n(C)c2c1	CID:60189864	phase I
BRD-K92967637	COCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)S(C)(=O)=O	CID:60189865	phase I
BRD-K37650321	COCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)S(C)(=O)=O	CID:60189866	phase I
BRD-K42943439	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1)C[C@]31CN(C1)C(=O)Nc1cccc(F)c1	CID:60189867	phase I
BRD-K16621373	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1)C[C@]31CN(C1)C(=O)Nc1cccc(F)c1	CID:60189868	phase I
BRD-K27559321	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccccc1F)C(=O)Cc1ccccc1	CID:60189869	phase I
BRD-K29625564	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccccc1F)C(=O)Cc1ccccc1	CID:60189870	phase I
BRD-K48930263	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CCN(CC3)C(=O)c3cccnc3)n(C)c2c1	CID:60189871	phase I
BRD-K99660708	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CN(C3)C(=O)C3CCC3)n(C)c2c1	CID:60189872	phase I
BRD-K15858225	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(CC1CC1)C[C@]31CN(C1)C(=O)NC1CCCC1	CID:60189873	phase I
BRD-K09014535	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(CC1CC1)C[C@]31CN(C1)C(=O)NC1CCCC1	CID:60189874	phase I
BRD-K01193369	CCCNC(=O)N1C[C@]2(CN(Cc3cccc(F)c3)C2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60189875	phase I
BRD-K48193278	CCCNC(=O)N1C[C@]2(CN(Cc3cccc(F)c3)C2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60189876	phase I
BRD-K79734497	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)c1ccccc1	CID:60189878	phase I
BRD-K47512679	COc1ccc2c3c([C@@H](CO)N(Cc4cc(F)ccc4F)C[C@]33CN(C3)C(=O)C3CC3)n(C)c2c1	CID:60189879	phase I
BRD-K30298702	CCS(=O)(=O)N1C[C@@]2(C1)CN(C)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60189881	phase I
BRD-K52721778	CCS(=O)(=O)N1C[C@@]2(C1)CN(C)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60189882	phase I
BRD-K80749795	COc1ccc2c3c([C@@H](CO)N(Cc4ccc(Cl)cc4)C[C@]33CCN(CC4CC4)CC3)n(C)c2c1	CID:60189883	phase I
BRD-K71424167	CC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CCC(F)(F)F)c1ccc(cc1)-c1cccc(c1)C#N	CID:60189886	phase I
BRD-K08436070	CC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CCC(F)(F)F)c1ccc(cc1)-c1cccc(c1)C#N	CID:60189887	phase I
BRD-K94734308	CC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CCC(F)(F)F)c1ccc(cc1)-c1cccc(c1)C#N	CID:60189888	phase I
BRD-K81976047	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(CCC(F)(F)F)C2)N1S(=O)(=O)Cc1ccccc1	CID:60189889	phase I
BRD-K26150272	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)c2cnccn2)C11CN(C1)C(C)=O	CID:60189890	phase I
BRD-K46815185	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)c2cnccn2)C11CN(C1)C(C)=O	CID:60189891	phase I
BRD-K38274933	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(=O)c2cnccn2)C11CN(C1)C(C)=O	CID:60189892	phase I
BRD-K29328696	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2cccnc2)N1Cc1ccc(Cl)cc1	CID:60189893	phase I
BRD-K58609008	CC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CC1CC1)c1ccc(cc1)-c1ccc(F)cc1	CID:60189894	phase I
BRD-K53224568	CC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CC1CC1)c1ccc(cc1)-c1ccc(F)cc1	CID:60189895	phase I
BRD-K83395537	CCC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(Cc2ccccc2Cl)C1	CID:60189896	phase I
BRD-K56068611	COc1cccc(CN2[C@H](CO)[C@H](c3ccccc3)C22CN(C2)C(=O)C2CCCCC2)c1	CID:60189897	phase I
BRD-K14217854	COc1cccc(CN2[C@H](CO)[C@@H](c3ccccc3)C22CN(C2)C(=O)C2CCCCC2)c1	CID:60189898	phase I
BRD-K78869873	COc1cccc(CN2[C@@H](CO)[C@H](c3ccccc3)C22CN(C2)C(=O)C2CCCCC2)c1	CID:60189899	phase I
BRD-K17619118	COc1cccc(CN2[C@@H](CO)[C@@H](c3ccccc3)C22CN(C2)C(=O)C2CCCCC2)c1	CID:60189900	phase I
BRD-K59465228	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1Cc1nccs1	CID:60189901	phase I
BRD-K04750859	CCC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1cnccn1	CID:60189902	phase I
BRD-K83705009	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(C)=O)C11CN(C1)C(=O)c1ccc(F)cc1	CID:60189903	phase I
BRD-K91565112	COCC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccccc1	CID:60189905	phase I
BRD-K39062398	COCC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)c1ccccc1	CID:60189906	phase I
BRD-K84831408	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CCN(CC3)C(=O)c3cccnc3)n(C)c2c1	CID:60189907	phase I
BRD-K81739235	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1ccccc1)C(C)=O	CID:60189909	phase I
BRD-K60159779	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1ccccc1)C(C)=O	CID:60189910	phase I
BRD-K55426263	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(CC4CCOCC4)C3)n(C)c2c1	CID:60189911	phase I
BRD-K00518397	COc1ccc2c3c([C@H](CO)NC[C@]33CN(CC4CCOCC4)C3)n(C)c2c1	CID:60189912	phase I
BRD-K31928320	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccc2OCOc2c1)C(=O)Nc1ccc(F)cc1	CID:60189913	phase I
BRD-K31593641	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccc2OCOc2c1)C(=O)Nc1ccc(F)cc1	CID:60189914	phase I
BRD-K58340898	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CCN(CC1)C(=O)c1ccccc1	CID:60189915	phase I
BRD-K16157799	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C)C[C@]31CCN(CC1)S(=O)(=O)c1cn(C)cn1	CID:60189916	phase I
BRD-K89951364	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(C)CC1)C(=O)c1ccccc1	CID:60189917	phase I
BRD-K15697250	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(C)CC1)C(=O)c1ccccc1	CID:60189918	phase I
BRD-K38832878	COc1ccc2c3c([C@H](CO)N(Cc4ccc(Cl)cc4)C[C@]33CCN(CC4CC4)CC3)n(C)c2c1	CID:60189920	phase I
BRD-K29943481	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccncc1)C(=O)CN(C)C	CID:60189922	phase I
BRD-K20862010	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)c1ccncc1)C(=O)CN(C)C	CID:60189924	phase I
BRD-K74782274	COc1ccc2c(c1)n(C)c1[C@@H](CO)N(C[C@]3(CCN(C)CC3)c21)C(=O)c1ccc(F)cc1	CID:60189925	phase I
BRD-K38451408	COc1ccc2c(c1)n(C)c1[C@H](CO)N(C[C@]3(CCN(C)CC3)c21)C(=O)c1ccc(F)cc1	CID:60189927	phase I
BRD-K94200504	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1ccc(F)cc1	CID:60189928	phase I
BRD-K60751982	COc1ccc(C#Cc2cnc3O[C@@H](CN(C)CC4CC4)[C@@H](C)CN([C@@H](C)CO)C(=O)c3c2)cc1	CID:60189929	phase I
BRD-K93195783	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2cccnc2)N1Cc1ccc(Cl)cc1	CID:60189930	phase I
BRD-K39896319	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2cccnc2)N1Cc1ccc(Cl)cc1	CID:60189931	phase I
BRD-K90146477	CC(C)NC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(C)=O)c1ccc(cc1)C1=CCCC1	CID:60189932	phase I
BRD-K32066855	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(C)=O)c1ccc(cc1)C1=CCCC1	CID:60189933	phase I
BRD-K07476637	CCC(=O)N1CC2(C1)[C@H]([C@H](CO)N2S(=O)(=O)CC)c1ccc(cc1)-c1ccc(C)cc1	CID:60189934	phase I
BRD-K00232157	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2S(=O)(=O)CC)c1ccc(cc1)-c1ccc(C)cc1	CID:60189935	phase I
BRD-K19398444	CC(=O)N1[C@H](CO)[C@@H](c2ccc(cc2)-c2ccccc2F)C11CN(CC2CCOCC2)C1	CID:60189936	phase I
BRD-K97748657	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)NC2CCCCC2)N1CC1CCCC1	CID:60189937	phase I
BRD-K00303543	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)Nc2ccccc2F)N1C(=O)CC1CC1	CID:60189938	phase I
BRD-K65266817	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)Nc2ccccc2F)N1C(=O)CC1CC1	CID:60189939	phase I
BRD-K33230547	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)Nc2ccccc2F)N1C(=O)CC1CC1	CID:60189940	phase I
BRD-K92129795	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2ccccc2)C1)C(=O)CN1CCOCC1	CID:60189941	phase I
BRD-K35945912	CCCNC(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)COC	CID:60189942	phase I
BRD-K70842558	CCCNC(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)COC	CID:60189943	phase I
BRD-K62473389	COc1ccc(CN2C[C@]3(CN(C3)C(C)=O)c3c([C@@H]2CO)n(C)c2cc(OC)ccc32)cc1	CID:60189944	phase I
BRD-K97239800	COc1ccc(CN2C[C@]3(CN(C3)C(C)=O)c3c([C@H]2CO)n(C)c2cc(OC)ccc32)cc1	CID:60189945	phase I
BRD-K68223173	COc1ccc2c3c([C@H](CO)NC[C@]33CN(Cc4ccc(F)cc4)C3)n(C)c2c1	CID:60189946	phase I
BRD-K43212439	CCCC(=O)N1C[C@@]2(C1)CN(CC1CC1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189947	phase I
BRD-K50890172	CCCC(=O)N1C[C@]2(CCN(CC2)S(=O)(=O)CC)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60189949	phase I
BRD-K35046689	CCCC(=O)N1C[C@]2(CCN(CC2)S(=O)(=O)CC)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60189950	phase I
BRD-K69237309	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1ccc(F)cc1	CID:60189952	phase I
BRD-K90417358	CCC(=O)N1C[C@]2(CN(Cc3ccc(F)cc3)C2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60189953	phase I
BRD-K48332988	CCC(=O)N1C[C@]2(CN(Cc3ccc(F)cc3)C2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60189954	phase I
BRD-K76263948	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC3)C(=O)c3ccc(F)cc3)n(C)c2c1	CID:60189955	phase I
BRD-K06209369	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)C(=O)c3ccc(F)cc3)n(C)c2c1	CID:60189956	phase I
BRD-K36991730	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(C)(=O)=O)C(=O)c1cnccn1	CID:60189957	phase I
BRD-K14951088	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)S(C)(=O)=O)C(=O)c1cnccn1	CID:60189959	phase I
BRD-K99450499	COCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(F)c1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60189960	phase I
BRD-K63684048	COCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(F)c1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60189961	phase I
BRD-K97281677	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)NC2CCCCC2)N1CC1CCCC1	CID:60189962	phase I
BRD-K65426421	CS(=O)(=O)N1CC2(C1)[C@H]([C@@H](CO)N2Cc1ccccn1)c1ccccc1	CID:60189964	phase I
BRD-K04087697	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(C(C)=O)C11CN(C1)C(=O)c1ccc(F)cc1	CID:60189965	phase I
BRD-K53682606	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(C)=O)C11CN(C1)C(=O)c1ccc(F)cc1	CID:60189966	phase I
BRD-K18287297	COCC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccccc1	CID:60189967	phase I
BRD-K64320360	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)NC(C)C)c1ccccc1	CID:60189968	phase I
BRD-K83443720	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C)C[C@]31CCN(CC1)S(=O)(=O)c1cn(C)cn1	CID:60189969	phase I
BRD-K36820092	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)C1CCC1)C(=O)c1ccncc1	CID:60189970	phase I
BRD-K64404931	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(C)CC3)S(=O)(=O)c3cn(C)cn3)n(C)c2c1	CID:60189971	phase I
BRD-K50953983	COc1cccc(CN2C[C@]3(CCN(CC3)S(C)(=O)=O)c3c([C@@H]2CO)n(C)c2cc(OC)ccc32)c1	CID:60189973	phase I
BRD-K82078087	COc1cccc(CN2C[C@]3(CCN(CC3)S(C)(=O)=O)c3c([C@H]2CO)n(C)c2cc(OC)ccc32)c1	CID:60189975	phase I
BRD-K21537090	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1Cl)C[C@]31CN(C1)C(=O)C1CC1	CID:60189976	phase I
BRD-K27398156	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1Cl)C[C@]31CN(C1)C(=O)C1CC1	CID:60189977	phase I
BRD-K39507536	COCC(=O)N1C[C@@]2(C1)CN(Cc1ccccc1F)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189981	phase I
BRD-K49534870	COCC(=O)N1C[C@@]2(C1)CN(Cc1ccccc1F)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60189982	phase I
BRD-K07935321	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2nccs2)CC1)C(=O)C1CCOCC1	CID:60189984	phase I
BRD-K22389219	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4nccs4)CC3)S(C)(=O)=O)n(C)c2c1	CID:60189985	phase I
BRD-K09977695	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(Cc2cncnc2)C11CN(C1)C(=O)CC1CC1	CID:60189986	phase I
BRD-K64601990	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(Cc2cncnc2)C11CN(C1)C(=O)CC1CC1	CID:60189987	phase I
BRD-K03610256	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)c2ccccn2)C11CN(CCC(F)(F)F)C1	CID:60189988	phase I
BRD-K90045406	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)c2ccccn2)C11CN(CCC(F)(F)F)C1	CID:60189989	phase I
BRD-K90526552	OC[C@@H]1N(Cc2ccccn2)C2(CN(C2)C(=O)c2cccc(F)c2)[C@@H]1c1ccccc1	CID:60189990	phase I
BRD-K70273200	OC[C@@H]1N(Cc2ccccn2)C2(CN(C2)C(=O)c2cccc(F)c2)[C@H]1c1ccccc1	CID:60189991	phase I
BRD-K85935038	OC[C@H]1N(Cc2ccccn2)C2(CN(C2)C(=O)c2cccc(F)c2)[C@@H]1c1ccccc1	CID:60189992	phase I
BRD-K32893176	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)C1CCC1)C(=O)c1ccncc1	CID:60189993	phase I
BRD-K14989056	COc1ccc2c3c([C@H](CO)NC[C@]33CN(C3)C(=O)Nc3ccccc3F)n(C)c2c1	CID:60189994	phase I
BRD-K38294141	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)C(=O)Nc3ccccc3F)n(C)c2c1	CID:60189995	phase I
BRD-K89808696	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccc(F)cc1)C[C@]31CN(Cc2ccccn2)C1	CID:60189997	phase I
BRD-K04340915	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccc(F)cc1)C[C@]31CN(Cc2ccccn2)C1	CID:60189998	phase I
BRD-K87748349	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)Nc3ccc(F)cc3F)n(C)c2c1	CID:60189999	phase I
BRD-K33841609	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)Nc3ccc(F)cc3F)n(C)c2c1	CID:60190000	phase I
BRD-K78957196	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3ccccc3F)C(C)=O)n(C)c2c1	CID:60190001	phase I
BRD-K55345749	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1C(=O)c1ccccc1	CID:60190005	phase I
BRD-K91035379	OC[C@@H]1[C@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1C(=O)c1ccccc1	CID:60190006	phase I
BRD-K18309252	OC[C@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1C(=O)c1ccccc1	CID:60190007	phase I
BRD-K83518844	OC[C@H]1N(C(=O)c2cccnc2)C2(CN(C(=O)Cc3ccccn3)C2)[C@@H]1c1ccccc1	CID:60190008	phase I
BRD-K62625902	OC[C@H]1N(C(=O)c2cccnc2)C2(CN(C(=O)Cc3ccccn3)C2)[C@H]1c1ccccc1	CID:60190009	phase I
BRD-K03673270	COCC(=O)N1CC2(C1)N(CCC(F)(F)F)[C@H](CO)[C@@H]2c1ccc(\C=C\C)cc1	CID:60190010	phase I
BRD-K98367403	COCC(=O)N1CC2(C1)N(CCC(F)(F)F)[C@@H](CO)[C@H]2c1ccc(\C=C\C)cc1	CID:60190011	phase I
BRD-K03925537	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1C(=O)c1ccccn1	CID:60190012	phase I
BRD-K34161817	OC[C@H]1N(Cc2ccccn2)C2(CN(C2)C(=O)c2cccc(F)c2)[C@H]1c1ccccc1	CID:60190013	phase I
BRD-K71994465	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2S(C)(=O)=O)c1ccc(cc1)\C=C\C	CID:60190014	phase I
BRD-K80108679	CCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2S(C)(=O)=O)c1ccc(cc1)\C=C\C	CID:60190015	phase I
BRD-K83045795	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2S(C)(=O)=O)c1ccc(cc1)\C=C\C	CID:60190017	phase I
BRD-K77663706	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)S(=O)(=O)c2ccccc2)N1CC1CCCC1	CID:60190019	phase I
BRD-K35522276	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)S(=O)(=O)c2ccccc2)N1CC1CCCC1	CID:60190020	phase I
BRD-K84276102	CCC(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1ccccc1	CID:60190023	phase I
BRD-K79600112	CCC(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1ccccc1	CID:60190024	phase I
BRD-K09335206	CCCNC(=O)N1C[C@]2(CCN(CC2)S(=O)(=O)CC)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60190025	phase I
BRD-K67485291	CCCNC(=O)N1C[C@]2(CCN(CC2)S(=O)(=O)CC)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60190026	phase I
BRD-K54588025	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C)C3)C(=O)C3CCOCC3)n(C)c2c1	CID:60190027	phase I
BRD-K55093794	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(C)(=O)=O)C(=O)C1CCOCC1	CID:60190028	phase I
BRD-K32014638	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)S(C)(=O)=O)C(=O)C1CCOCC1	CID:60190029	phase I
BRD-K27925875	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3cccc(F)c3)C(=O)CN3CCOCC3)n(C)c2c1	CID:60190030	phase I
BRD-K86149906	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4Cl)C[C@]33CCN(CC3)C(=O)CC3CC3)n(C)c2c1	CID:60190031	phase I
BRD-K43345858	CCCC(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Cc1ccccn1	CID:60190032	phase I
BRD-K88701555	CCCC(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Cc1ccccn1	CID:60190034	phase I
BRD-K45986013	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Nc1c(C)noc1C	CID:60190035	phase I
BRD-K87458009	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)Nc1c(C)noc1C	CID:60190036	phase I
BRD-K82110567	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(OC)cc(OC)c1)C[C@]31CN(C1)C(=O)Nc1c(C)noc1C	CID:60190037	phase I
BRD-K17407318	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(Cc4nccs4)CC3)S(C)(=O)=O)n(C)c2c1	CID:60190038	phase I
BRD-K07040635	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccc1)C(=O)CC1CC1	CID:60190039	phase I
BRD-K25828886	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)c1ccccc1)C(=O)CC1CC1	CID:60190041	phase I
BRD-K95437400	CCS(=O)(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1ccc(C)cc1	CID:60190043	phase I
BRD-K67985577	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2Cc1cccc(F)c1)c1ccc(\C=C\C)cc1	CID:60190046	phase I
BRD-K02037850	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3ccc4OCOc4c3)C2)N1Cc1ccccc1	CID:60190047	phase I
BRD-K74133758	CC(C)NC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(Cc2cc(F)cc(F)c2)C1	CID:60190048	phase I
BRD-K78989575	CS(=O)(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)c1ccccc1F	CID:60190049	phase I
BRD-K17466145	CS(=O)(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccccc1F	CID:60190050	phase I
BRD-K82869745	CS(=O)(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccccc1F	CID:60190052	phase I
BRD-K61553906	COc1ccccc1CN1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccc1	CID:60190053	phase I
BRD-K95152807	COc1ccccc1CN1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccc1	CID:60190054	phase I
BRD-K19237705	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1C(=O)c1ccccn1	CID:60190055	phase I
BRD-K68698887	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1C(=O)c1ccccn1	CID:60190056	phase I
BRD-K87807408	OC[C@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1C(=O)c1ccccn1	CID:60190057	phase I
BRD-K60823407	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2Cc1cncnc1)c1ccccc1	CID:60190058	phase I
BRD-K26130452	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(CC2CC2)C11CN(C1)C(=O)c1ccc2OCOc2c1	CID:60190059	phase I
BRD-K33284065	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(CC2CC2)C11CN(C1)C(=O)c1ccc2OCOc2c1	CID:60190060	phase I
BRD-K57170492	CCCNC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2Cc1cccc(Cl)c1)c1ccccc1	CID:60190062	phase I
BRD-K17712828	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)S(=O)(=O)c2ccccc2)N1CC1CCCC1	CID:60190063	phase I
BRD-K28096758	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1S(=O)(=O)Cc1ccccc1	CID:60190064	phase I
BRD-K61891887	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1S(=O)(=O)Cc1ccccc1	CID:60190065	phase I
BRD-K62919978	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)S(=O)(=O)c3ccccc3)C(C)=O)n(C)c2c1	CID:60190071	phase I
BRD-K70210716	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1)C[C@]31CN(C1)S(=O)(=O)c1ccc(C)cc1	CID:60190072	phase I
BRD-K57580310	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccc1)C[C@]31CN(C1)S(=O)(=O)c1ccc(C)cc1	CID:60190073	phase I
BRD-K94915559	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1cn(C)cn1	CID:60190074	phase I
BRD-K78124775	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1cn(C)cn1	CID:60190076	phase I
BRD-K30760376	COc1ccc2c3c([C@H](CO)N(Cc4cc(OC)cc(OC)c4)C[C@]33CCN(CC3)C(=O)Nc3c(C)noc3C)n(C)c2c1	CID:60190077	phase I
BRD-K76243153	COc1ccc2c3c([C@@H](CO)N(Cc4cc(OC)cc(OC)c4)C[C@]33CCN(CC3)C(=O)Nc3c(C)noc3C)n(C)c2c1	CID:60190078	phase I
BRD-K16643204	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3cccc(F)c3)C(=O)CN3CCOCC3)n(C)c2c1	CID:60190079	phase I
BRD-K79579182	COc1cccc(CN2C[C@@]3(C2)CN([C@H](CO)c2[nH]c4cc(OC)ccc4c32)C(=O)C2CC2)c1	CID:60190081	phase I
BRD-K81953058	COc1cccc(CN2C[C@@]3(C2)CN([C@@H](CO)c2[nH]c4cc(OC)ccc4c32)C(=O)C2CC2)c1	CID:60190082	phase I
BRD-K47950966	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CCN(CC1)C(=O)C1CCOCC1	CID:60190083	phase I
BRD-K30007764	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)C1CCOCC1	CID:60190084	phase I
BRD-K23217353	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)Nc3ccc(F)cc3)C(=O)c3ccc(F)cc3)n(C)c2c1	CID:60190085	phase I
BRD-K27682288	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)Nc3ccc(F)cc3)C(=O)c3ccc(F)cc3)n(C)c2c1	CID:60190086	phase I
BRD-K20120164	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cc(OC)cc(OC)c1)C[C@]31CN(C1)C(=O)Nc1c(C)noc1C	CID:60190087	phase I
BRD-K99102143	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)CN(C)C)C(=O)C3CC3)n(C)c2c1	CID:60190088	phase I
BRD-K35522326	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2nccs2)CC1)C(=O)C1CCOCC1	CID:60190089	phase I
BRD-K26522558	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CCN(CC3)C(=O)c3ccc4OCOc4c3)n(C)c2c1	CID:60190091	phase I
BRD-K53927732	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CCN(CC3)C(=O)c3ccc4OCOc4c3)n(C)c2c1	CID:60190093	phase I
BRD-K61753121	CCS(=O)(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)S(=O)(=O)c1ccc(C)cc1	CID:60190094	phase I
BRD-K22571527	CCC(=O)N1C[C@]2(CCN(CC2)C(=O)Cc2ccccc2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60190095	phase I
BRD-K68108628	CCC(=O)N1C[C@]2(CCN(CC2)C(=O)Cc2ccccc2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:60190097	phase I
BRD-K98386238	CCCC(=O)N1CC[C@@]2(CC1)CN[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190099	phase I
BRD-K64716493	CCCC(=O)N1CC[C@@]2(CC1)CN[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190100	phase I
BRD-K45319408	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(C)=O)C(C)=O	CID:60190102	phase I
BRD-K96782963	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(C)=O)C(C)=O	CID:60190103	phase I
BRD-K90341035	COCC(=O)N1CC2(C1)[C@H]([C@H](CO)N2C(=O)COC)c1ccc(cc1)-c1cccc(F)c1	CID:60190104	phase I
BRD-K36617229	COCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)COC)c1ccc(cc1)-c1cccc(F)c1	CID:60190105	phase I
BRD-K02162441	COCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)COC)c1ccc(cc1)-c1cccc(F)c1	CID:60190106	phase I
BRD-K41595225	CCCNC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)c1ccncc1)c1ccccc1	CID:60190107	phase I
BRD-K65561930	CCCNC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)c1ccncc1)c1ccccc1	CID:60190108	phase I
BRD-K22941245	CCCNC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)c1ccncc1)c1ccccc1	CID:60190109	phase I
BRD-K54048734	CCCNC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2Cc1cccc(Cl)c1)c1ccccc1	CID:60190110	phase I
BRD-K46664882	CCCNC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2Cc1cccc(Cl)c1)c1ccccc1	CID:60190112	phase I
BRD-K35080107	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2ccncc2)N1CC1CCOCC1	CID:60190113	phase I
BRD-K24184187	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(Cc4nccs4)C3)C(=O)CN(C)C)n(C)c2c1	CID:60190114	phase I
BRD-K81614512	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(Cc4nccs4)C3)C(=O)CN(C)C)n(C)c2c1	CID:60190115	phase I
BRD-K71673735	COc1ccc(NC(=O)N2C[C@@]3(C2)CN([C@H](CO)c2[nH]c4cc(OC)ccc4c32)C(C)=O)cc1	CID:60190116	phase I
BRD-K18471876	COc1ccc(NC(=O)N2C[C@@]3(C2)CN([C@@H](CO)c2[nH]c4cc(OC)ccc4c32)C(C)=O)cc1	CID:60190118	phase I
BRD-K49367140	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(CC2CC2)C1)C(=O)CN(C)C	CID:60190119	phase I
BRD-K86694468	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(CC2CC2)C1)C(=O)CN(C)C	CID:60190120	phase I
BRD-K02274189	COc1ccc2c3c([C@H](CO)N(Cc4nccs4)C[C@]33CCN(CC4CCCC4)CC3)n(C)c2c1	CID:60190121	phase I
BRD-K28138218	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2cc(F)ccc2F)C1)C(=O)Nc1ccc(F)cc1	CID:60190122	phase I
BRD-K17996849	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(Cc2cc(F)ccc2F)C1)C(=O)Nc1ccc(F)cc1	CID:60190124	phase I
BRD-K32857328	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C)C[C@]31CCN(CC1)C(=O)CN(C)C	CID:60190126	phase I
BRD-K05344363	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CN(C3)S(=O)(=O)c3cccc(C)c3)n(C)c2c1	CID:60190127	phase I
BRD-K54335715	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CN(C3)S(=O)(=O)c3cccc(C)c3)n(C)c2c1	CID:60190129	phase I
BRD-K41115759	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CN(C1)S(=O)(=O)c1cccs1	CID:60190131	phase I
BRD-K45153357	COc1ccc2c3c([nH]c2c1)[C@@H](CO)NC[C@]31CN(C1)S(=O)(=O)c1cccs1	CID:60190132	phase I
BRD-K33821902	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4)C[C@]33CN(CC4CC4)C3)n(C)c2c1	CID:60190133	phase I
BRD-K40013467	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(Cc4ccc(Cl)cc4)C3)C(C)=O)n(C)c2c1	CID:60190135	phase I
BRD-K31770065	CCCNC(=O)N1C[C@]2(CCN(CC2)C(=O)Nc2cccc(F)c2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60190136	phase I
BRD-K84431964	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)c3ccccc3F)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60190137	phase I
BRD-K67795523	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)c3ccccc3F)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60190138	phase I
BRD-K93207153	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cccnc1)C[C@]31CCN(CC1)C(=O)CN(C)C	CID:60190139	phase I
BRD-K82886296	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1cccnc1)C[C@]31CCN(CC1)C(=O)CN(C)C	CID:60190140	phase I
BRD-K75579936	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)CN1CCOCC1)C(C)=O	CID:60190141	phase I
BRD-K04139743	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)CN1CCOCC1)C(C)=O	CID:60190142	phase I
BRD-K37820137	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)c3cccc(F)c3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60190143	phase I
BRD-K39766484	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)c3cccc(F)c3)C(=O)c3cccc(F)c3)n(C)c2c1	CID:60190144	phase I
BRD-K66710853	COc1cccc(NC(=O)N2CC3(C2)[C@H]([C@@H](CO)N3C(C)=O)c2ccccc2)c1	CID:60190145	phase I
BRD-K66499109	COc1cccc(NC(=O)N2CC3(C2)[C@@H]([C@H](CO)N3C(C)=O)c2ccccc2)c1	CID:60190146	phase I
BRD-K54521353	COc1cccc(NC(=O)N2CC3(C2)[C@@H]([C@@H](CO)N3C(C)=O)c2ccccc2)c1	CID:60190147	phase I
BRD-K67507121	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1S(=O)(=O)Cc1ccccc1	CID:60190149	phase I
BRD-K79838525	CCS(=O)(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)c1ccccc1)c1ccccc1	CID:60190151	phase I
BRD-K63596086	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(CC1CCCC1)C[C@]31CN(C)C1	CID:60190152	phase I
BRD-K13982317	CCCC(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(C)=O	CID:60190153	phase I
BRD-K51930253	CCCC(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(C)=O	CID:60190154	phase I
BRD-K70165913	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)CN(C)C)C(=O)C3CC3)n(C)c2c1	CID:60190155	phase I
BRD-K11145711	CCCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)C1CCCC1	CID:60190156	phase I
BRD-K83954980	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC4CCCCC4)CC3)S(C)(=O)=O)n(C)c2c1	CID:60190159	phase I
BRD-K49508167	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC4CCCCC4)CC3)S(C)(=O)=O)n(C)c2c1	CID:60190160	phase I
BRD-K49258689	COCC(=O)N1C[C@]2(CCN(Cc3ccccc3)CC2)c2c([nH]c3cc(OC)ccc23)[C@@H]1CO	CID:60190162	phase I
BRD-K44732214	COCC(=O)N1C[C@]2(CCN(Cc3ccccc3)CC2)c2c([nH]c3cc(OC)ccc23)[C@H]1CO	CID:60190163	phase I
BRD-K20537503	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccc3OCOc3c1)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60190164	phase I
BRD-K96703103	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccc3OCOc3c1)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60190166	phase I
BRD-K66757073	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)Nc1cccc(F)c1)C(=O)NC1CCCC1	CID:60190167	phase I
BRD-K27586181	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)S(C)(=O)=O)C(=O)C1CCC1	CID:60190169	phase I
BRD-K07444373	CCS(=O)(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)c1ccccc1)c1ccccc1	CID:60190171	phase I
BRD-K93620106	CCS(=O)(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)c1ccccc1)c1ccccc1	CID:60190173	phase I
BRD-K25624315	CN(C)CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(CC2CCOCC2)C1	CID:60190174	phase I
BRD-K06851272	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccn2)N1Cc1ccccc1	CID:60190176	phase I
BRD-K89562272	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)COC)c1ccc(cc1)C1=CCCC1	CID:60190177	phase I
BRD-K84121706	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)CN(C)C)C11CN(C1)C(=O)C1CCC1	CID:60190178	phase I
BRD-K36128472	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(=O)CN(C)C)C11CN(C1)C(=O)C1CCC1	CID:60190179	phase I
BRD-K17087588	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccccc1F)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190180	phase I
BRD-K49955466	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccccc1F)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190181	phase I
BRD-K41034329	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)C(=O)C1CCCC1)C(=O)NC(C)C	CID:60190182	phase I
BRD-K18340348	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)C1CCCC1)C(=O)NC(C)C	CID:60190183	phase I
BRD-K91773518	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)CC2CCCC2)Oc3cc(C#CCN(C)C)ccc3S1(=O)=O	CID:60190184	phase I
BRD-K24925721	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)C(=O)c1cccnc1)C(=O)NC(C)C	CID:60190185	phase I
BRD-K72010491	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)c1cccnc1)C(=O)NC(C)C	CID:60190186	phase I
BRD-K18981886	CCCN1CC[C@@]2(CC1)CN(Cc1ccc3OCOc3c1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190187	phase I
BRD-K65920478	COc1cccc(CN2C[C@]3(CN(CC4CCOCC4)C3)c3c([nH]c4cc(OC)ccc34)[C@H]2CO)c1	CID:60190188	phase I
BRD-K99749622	COc1cccc(NC(=O)N2CC3(C2)[C@H]([C@H](CO)N3C(C)=O)c2ccccc2)c1	CID:60190189	phase I
BRD-K66857089	CCC(=O)N1[C@H](CO)[C@@H](c2ccc(\C=C\c3ccccc3)cc2)C11CN(C1)S(C)(=O)=O	CID:60190191	phase I
BRD-K76202646	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccncc2)N1CC1CCOCC1	CID:60190192	phase I
BRD-K19911709	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1S(=O)(=O)c1ccccc1	CID:60190194	phase I
BRD-K02635441	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1S(=O)(=O)c1ccccc1	CID:60190195	phase I
BRD-K68935991	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1S(=O)(=O)c1ccccc1	CID:60190197	phase I
BRD-K77877235	CCS(=O)(=O)N1CC2(C1)[C@@H]([C@H](CO)N2Cc1ccc(F)cc1)c1ccccc1	CID:60190198	phase I
BRD-K38227596	CCS(=O)(=O)N1CC2(C1)[C@H]([C@H](CO)N2Cc1ccc(F)cc1)c1ccccc1	CID:60190199	phase I
BRD-K18237196	CCS(=O)(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2Cc1ccc(F)cc1)c1ccccc1	CID:60190200	phase I
BRD-K60331845	CCS(=O)(=O)N1CC2(C1)[C@H]([C@@H](CO)N2Cc1ccc(F)cc1)c1ccccc1	CID:60190202	phase I
BRD-K52515416	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)CN(C)C)C11CN(C1)C(=O)C1CCC1	CID:60190203	phase I
BRD-K28436871	OC[C@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1CC1CCOCC1	CID:60190204	phase I
BRD-K25979847	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1CC1CCOCC1	CID:60190205	phase I
BRD-K90205161	OC[C@@H]1[C@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1CC1CCOCC1	CID:60190207	phase I
BRD-K58149752	COc1cccc(CN2[C@H](CO)[C@@H](c3ccccc3)C22CN(Cc3ccccc3OC)C2)c1	CID:60190208	phase I
BRD-K24962261	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)S(=O)(=O)Cc2ccccc2)N1CC1CCOCC1	CID:60190210	phase I
BRD-K95995661	CCC(=O)N1CC2(C1)[C@H]([C@H](CO)N2C(=O)CC)c1ccc(cc1)-c1ccc(F)cc1	CID:60190211	phase I
BRD-K48089931	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)CC)c1ccc(cc1)-c1ccc(F)cc1	CID:60190212	phase I
BRD-K58826761	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)CC)c1ccc(cc1)-c1ccc(F)cc1	CID:60190213	phase I
BRD-K16106362	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(Cc4ccncc4)CC3)n(C)c2c1	CID:60190214	phase I
BRD-K44828732	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4ccncc4)CC3)n(C)c2c1	CID:60190216	phase I
BRD-K25298922	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C)C[C@]31CCN(CC1)C(=O)CN(C)C	CID:60190217	phase I
BRD-K26066252	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)CC3CC3)n(C)c2c1	CID:60190218	phase I
BRD-K78327149	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CN(C3)C(=O)CC3CC3)n(C)c2c1	CID:60190219	phase I
BRD-K91461129	CCCC(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)Nc1cccc(F)c1	CID:60190220	phase I
BRD-K59744203	CCCC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)Nc1cccc(F)c1	CID:60190221	phase I
BRD-K09651570	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)S(C)(=O)=O)C(=O)c1ccccn1	CID:60190222	phase I
BRD-K55697606	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CN(C1)S(C)(=O)=O)C(=O)c1ccccn1	CID:60190223	phase I
BRD-K62176618	COCC(=O)N1C[C@]2(CN(C2)S(C)(=O)=O)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60190224	phase I
BRD-K87864638	COc1cccc(CN2C[C@]3(CN(CC4CCOCC4)C3)c3c([nH]c4cc(OC)ccc34)[C@@H]2CO)c1	CID:60190226	phase I
BRD-K93185112	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(C)CC3)C(=O)Cc3ccccn3)n(C)c2c1	CID:60190228	phase I
BRD-K71101608	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4cncnc4)CC3)C(=O)CN(C)C)n(C)c2c1	CID:60190230	phase I
BRD-K81052803	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)CN3CCOCC3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60190231	phase I
BRD-K21683465	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)C(=O)CN3CCOCC3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:60190232	phase I
BRD-K96396151	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC3)S(=O)(=O)c3cccc(C)c3)n(C)c2c1	CID:60190233	phase I
BRD-K21626096	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(CC3)S(=O)(=O)c3cccc(C)c3)n(C)c2c1	CID:60190234	phase I
BRD-K01886140	COCC(=O)N1C[C@]2(CN(Cc3ccccc3)C2)c2c([C@@H]1CO)n(C)c1cc(OC)ccc21	CID:60190235	phase I
BRD-K30883461	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)S(=O)(=O)c3cccc(C)c3)n(C)c2c1	CID:60190244	phase I
BRD-K10731645	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4ccccc4Cl)CC3)n(C)c2c1	CID:60190271	phase I
BRD-K59733592	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(Cc4ccccc4Cl)CC3)n(C)c2c1	CID:60190301	phase I
BRD-K81524996	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(Cc4ccccc4F)CC3)n(C)c2c1	CID:60190306	phase I
BRD-K60631585	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4ccccc4F)CC3)n(C)c2c1	CID:60190307	phase I
BRD-K28782753	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:60190310	phase I
BRD-K42678365	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(Cc4ccc(Cl)cc4)C3)n(C)c2c1	CID:60190319	phase I
BRD-K62346407	CCCC(=O)N1CC[C@@]2(CC1)CN[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60190336	phase I
BRD-K78014537	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(Cc4cc(F)ccc4F)C3)n(C)c2c1	CID:60190368	phase I
BRD-K75065443	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC3)C(=O)c3ccccc3)n(C)c2c1	CID:60190385	phase I
BRD-K45307260	COc1ccc2c3c([C@H](CO)NC[C@]33CN(Cc4ccccc4F)C3)n(C)c2c1	CID:60190446	phase I
BRD-K66732164	COc1ccc2c3c([C@H](CO)NC[C@]33CCN(Cc4ccc(Cl)cc4)CC3)n(C)c2c1	CID:60190448	phase I
BRD-K57698173	CCC(=O)N1C[C@@]2(C1)CN(Cc1ccccc1Cl)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190509	phase I
BRD-K69236395	COc1ccc(cc1)S(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccccc1OC)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60190515	phase I
BRD-K88058149	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(Cc2ccccc2)CC1	CID:60190539	phase I
BRD-K58969952	CCCN1CC[C@@]2(CC1)CN(Cc1ccccc1OC)[C@H](CO)c1c2c2ccc(OC)cc2n1C	CID:60190540	phase I
BRD-K46532981	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CCN(CC3)C(=O)Nc3ccc(F)cc3F)n(C)c2c1	CID:60190552	phase I
BRD-K56014252	CS(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1ccc(F)cc1	CID:60190939	phase I
BRD-K27296582	CS(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1ccc(F)cc1	CID:60190940	phase I
BRD-K25775504	CS(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1ccc(F)cc1	CID:60190941	phase I
BRD-K74248891	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190942	phase I
BRD-K93062774	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190943	phase I
BRD-K79181721	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190944	phase I
BRD-K31387465	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190945	phase I
BRD-K15594502	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190946	phase I
BRD-K65343560	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190947	phase I
BRD-K05487130	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCC1	CID:60190948	phase I
BRD-K34545522	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60190949	phase I
BRD-K12862164	COc1cccc(NC(=O)N2C[C@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60190950	phase I
BRD-K78088483	COc1ccccc1NC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190951	phase I
BRD-K29543879	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190952	phase I
BRD-K66783461	COc1ccccc1NC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190953	phase I
BRD-K30563791	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190954	phase I
BRD-K36675307	COc1ccccc1NC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190955	phase I
BRD-K41954709	COc1ccccc1NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190956	phase I
BRD-K95361366	CS(=O)(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1ccc(F)cc1	CID:60190959	phase I
BRD-K12912249	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190960	phase I
BRD-K99536035	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190961	phase I
BRD-K14631382	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190962	phase I
BRD-K84129690	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190963	phase I
BRD-K95270854	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190964	phase I
BRD-K18407079	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190965	phase I
BRD-K86571219	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60190966	phase I
BRD-K85685363	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)S(=O)(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60190967	phase I
BRD-K05246899	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)S(=O)(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60190968	phase I
BRD-K00859238	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)S(=O)(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCC1	CID:60190969	phase I
BRD-K76836103	CCCNC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60190970	phase I
BRD-K56473018	CCCNC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60190971	phase I
BRD-K34580085	CCCNC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60190972	phase I
BRD-K93685415	COc1ccccc1NC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190973	phase I
BRD-K70669970	COc1ccccc1NC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC(C)C	CID:60190974	phase I
BRD-K21498052	COCC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60190975	phase I
BRD-K73397518	COCC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60190976	phase I
BRD-K72343629	COCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60190977	phase I
BRD-K20766305	Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1cccc(F)c1	CID:60190979	phase I
BRD-K55155550	CCCNC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60190986	phase I
BRD-K07303702	CCCNC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60190987	phase I
BRD-K33912919	CCCNC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60190988	phase I
BRD-K64988800	CCCNC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60190989	phase I
BRD-K75155876	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190990	phase I
BRD-K51349050	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(cc1)-c1cccc(F)c1	CID:60190991	phase I
BRD-K21453918	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60190992	phase I
BRD-K86591768	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60190993	phase I
BRD-K58043213	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60190994	phase I
BRD-K93800099	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60190995	phase I
BRD-K36226647	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60190996	phase I
BRD-K20462402	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60190997	phase I
BRD-K68211814	CCCNC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60190998	phase I
BRD-K76915833	CCCNC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60190999	phase I
BRD-K38509760	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191000	phase I
BRD-K36787562	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191001	phase I
BRD-K49330073	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191002	phase I
BRD-K67087659	COCC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60191003	phase I
BRD-K61615367	COCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60191004	phase I
BRD-K19147748	CCC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191005	phase I
BRD-K70900504	CCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191006	phase I
BRD-K99827928	CCC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191007	phase I
BRD-K76264608	CCC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191008	phase I
BRD-K42957595	CCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191009	phase I
BRD-K17519289	CCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191010	phase I
BRD-K47555438	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191013	phase I
BRD-K11310449	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191014	phase I
BRD-K39981110	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191015	phase I
BRD-K10849007	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191016	phase I
BRD-K41310594	CCCNC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60191017	phase I
BRD-K23017938	CCCNC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60191018	phase I
BRD-K52643239	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191019	phase I
BRD-K29258781	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191020	phase I
BRD-K12696543	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191021	phase I
BRD-K48583488	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191022	phase I
BRD-K63061929	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191023	phase I
BRD-K28395853	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60191024	phase I
BRD-K46593635	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccccn1)c1ccc(cc1)C#CCC1CCCC1	CID:60191025	phase I
BRD-K16195716	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191026	phase I
BRD-K74495399	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191027	phase I
BRD-K69291665	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191028	phase I
BRD-K94014921	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191029	phase I
BRD-K33390612	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191030	phase I
BRD-K10804522	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C1=CCCC1	CID:60191031	phase I
BRD-K71452159	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C1=CCCC1	CID:60191032	phase I
BRD-K88307115	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C1=CCCC1	CID:60191033	phase I
BRD-K42624823	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C1=CCCC1	CID:60191034	phase I
BRD-K24632043	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)C1=CCCC1	CID:60191035	phase I
BRD-K98252401	CCC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191036	phase I
BRD-K79625260	CCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccnc1	CID:60191037	phase I
BRD-K12302379	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191038	phase I
BRD-K81202141	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191039	phase I
BRD-K87988402	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191040	phase I
BRD-K83845832	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191041	phase I
BRD-K36062164	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191042	phase I
BRD-K29834132	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191043	phase I
BRD-K83785854	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191044	phase I
BRD-K61423234	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191053	phase I
BRD-K65813884	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191054	phase I
BRD-K84099887	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191055	phase I
BRD-K56222361	Cc1ccc(CN2C[C@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:60191056	phase I
BRD-K85069227	Cc1ccc(CN2C[C@@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:60191057	phase I
BRD-K49866472	Cc1ccc(CN2C[C@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:60191058	phase I
BRD-K04429417	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191059	phase I
BRD-K06846146	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1F)c1ccc(cc1)-c1cccnc1	CID:60191060	phase I
BRD-K79610347	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191061	phase I
BRD-K55442031	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191062	phase I
BRD-K08846320	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191063	phase I
BRD-K77795481	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191064	phase I
BRD-K21081985	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191065	phase I
BRD-K69191922	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191066	phase I
BRD-K06911479	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191067	phase I
BRD-K95553255	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)CN1CCOCC1	CID:60191068	phase I
BRD-K95063618	CCCNC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60191069	phase I
BRD-K81019664	CCCNC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60191070	phase I
BRD-K95810330	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191071	phase I
BRD-K89122409	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191072	phase I
BRD-K95074209	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191073	phase I
BRD-K76411754	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191074	phase I
BRD-K67889001	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191075	phase I
BRD-K55340188	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191076	phase I
BRD-K92993117	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191077	phase I
BRD-K68948289	CC(C)NC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191078	phase I
BRD-K24351638	CC(C)NC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191079	phase I
BRD-K66177994	CC(C)NC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191080	phase I
BRD-K09324015	CC(C)NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191081	phase I
BRD-K73543260	CC(C)NC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191082	phase I
BRD-K67622458	CC(C)NC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191083	phase I
BRD-K34844610	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191084	phase I
BRD-K25807578	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191085	phase I
BRD-K24536757	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191086	phase I
BRD-K63923428	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Nc1ccc(F)cc1)c1ccc(cc1)-c1cccc(F)c1	CID:60191087	phase I
BRD-K12124649	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)C#CC1CCCCC1	CID:60191088	phase I
BRD-K09388706	Cc1ccc(CN2C[C@@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:60191091	phase I
BRD-K11093795	Cc1ccc(CN2C[C@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:60191092	phase I
BRD-K75772012	Cc1ccc(CN2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)-c2ccccc2F)cc1	CID:60191093	phase I
BRD-K47716724	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191094	phase I
BRD-K17771527	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191095	phase I
BRD-K40960913	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191096	phase I
BRD-K67035256	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191097	phase I
BRD-K91104058	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191098	phase I
BRD-K59308946	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191099	phase I
BRD-K51753035	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60191100	phase I
BRD-K67454499	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191101	phase I
BRD-K92439079	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191102	phase I
BRD-K64751731	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191103	phase I
BRD-K21751020	CCCNC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1cccc(OC)c1	CID:60191104	phase I
BRD-K45627302	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191105	phase I
BRD-K99578584	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191106	phase I
BRD-K88683417	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191107	phase I
BRD-K10593696	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191108	phase I
BRD-K70276339	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191109	phase I
BRD-K85515417	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191110	phase I
BRD-K35202752	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191111	phase I
BRD-K38842489	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191112	phase I
BRD-K10279202	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191113	phase I
BRD-K58051960	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191114	phase I
BRD-K81079621	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccccc1)c1ccc(cc1)-c1ccc(F)cc1	CID:60191115	phase I
BRD-K23578923	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1ccccc1)c1ccc(cc1)-c1ccc(F)cc1	CID:60191116	phase I
BRD-K28698886	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1ccccc1)c1ccc(cc1)-c1ccc(F)cc1	CID:60191117	phase I
BRD-K09325707	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60191118	phase I
BRD-K11742792	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60191119	phase I
BRD-K06953509	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60191120	phase I
BRD-K50388960	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191121	phase I
BRD-K87744519	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191122	phase I
BRD-K63900355	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191123	phase I
BRD-K06992369	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191124	phase I
BRD-K51475868	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191125	phase I
BRD-K21217422	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191126	phase I
BRD-K92904177	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCCCC1	CID:60191127	phase I
BRD-K45322187	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(Cc1ccccc1)CC2=O	CID:60191128	phase I
BRD-K37399041	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(Cc1ccccc1)CC2=O	CID:60191129	phase I
BRD-K41651095	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191130	phase I
BRD-K54294645	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191131	phase I
BRD-K79001525	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191132	phase I
BRD-K22361536	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191133	phase I
BRD-K36938987	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191134	phase I
BRD-K78987935	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cccnc1)c1ccc(cc1)-c1ccccc1F	CID:60191135	phase I
BRD-K35613686	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191136	phase I
BRD-K71153796	CCCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191137	phase I
BRD-K30715463	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60191139	phase I
BRD-K68208040	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(Cc1ccccc1)CC2=O	CID:60191149	phase I
BRD-K55693448	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(Cc1ccccc1)CC2=O	CID:60191150	phase I
BRD-K42100231	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(Cc1ccccc1)CC2=O	CID:60191151	phase I
BRD-K94585132	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(Cc1ccccc1)CC2=O	CID:60191152	phase I
BRD-K85799948	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CN1CCOCC1)c1ccc(cc1)C1=CCCCC1	CID:60191153	phase I
BRD-K84039354	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCCC1	CID:60191154	phase I
BRD-K12655851	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCCC1	CID:60191155	phase I
BRD-K45853100	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCCC1	CID:60191156	phase I
BRD-K03373364	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191157	phase I
BRD-K79684588	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191158	phase I
BRD-K05832178	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191159	phase I
BRD-K47505626	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191160	phase I
BRD-K65139432	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccc(F)c1	CID:60191161	phase I
BRD-K22353999	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccccc1F)c1ccc(cc1)C#Cc1ccccc1	CID:60191178	phase I
BRD-K48463604	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191179	phase I
BRD-K34886590	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191180	phase I
BRD-K57186295	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191181	phase I
BRD-K42605282	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60191183	phase I
BRD-K74227932	COc1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60191184	phase I
BRD-K15593941	COc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1cccnc1	CID:60191185	phase I
BRD-K16383683	CCS(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(F)c1	CID:60191186	phase I
BRD-K53475565	CCS(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(F)c1	CID:60191187	phase I
BRD-K85132040	CCS(=O)(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1cccc(F)c1	CID:60191188	phase I
BRD-K78574388	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C#Cc1cccnc1	CID:60191189	phase I
BRD-K42609935	OC[C@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C#Cc1cccnc1	CID:60191190	phase I
BRD-K61776649	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCCC1	CID:60191191	phase I
BRD-K95570609	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCCC1	CID:60191192	phase I
BRD-K37184875	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60191193	phase I
BRD-K69261014	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)S(=O)(=O)c1ccccc1	CID:60191194	phase I
BRD-K20075074	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191195	phase I
BRD-K76950673	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191196	phase I
BRD-K06163572	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191197	phase I
BRD-K95716640	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191198	phase I
BRD-K55878534	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191199	phase I
BRD-K64398524	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191200	phase I
BRD-K31558029	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cnccn1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191201	phase I
BRD-K31621670	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191218	phase I
BRD-K56244705	CC(C)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191219	phase I
BRD-K11914584	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191220	phase I
BRD-K25866212	CC(C)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191221	phase I
BRD-K69259014	CC(C)C#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Cc1ccccc1	CID:60191222	phase I
BRD-K94139496	CCS(=O)(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CCCCC1	CID:60191223	phase I
BRD-K19436903	OC[C@@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)C#Cc1cccnc1	CID:60191224	phase I
BRD-K64609558	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)C#Cc1cccnc1	CID:60191225	phase I
BRD-K02593152	OC[C@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191226	phase I
BRD-K54801580	OC[C@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191227	phase I
BRD-K62726279	OC[C@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191228	phase I
BRD-K85118298	OC[C@@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191229	phase I
BRD-K28772322	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191230	phase I
BRD-K45907733	OC[C@@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191231	phase I
BRD-K77349332	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191232	phase I
BRD-K32367664	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191233	phase I
BRD-K18533094	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191234	phase I
BRD-K73096789	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191235	phase I
BRD-K60863614	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191236	phase I
BRD-K39900129	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191237	phase I
BRD-K68718973	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191238	phase I
BRD-K84705102	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191239	phase I
BRD-K45956042	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191240	phase I
BRD-K54945117	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)NC1CCCC1)c1ccc(cc1)C1=CCCCC1	CID:60191241	phase I
BRD-K24193032	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191242	phase I
BRD-K91053205	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191243	phase I
BRD-K27493325	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191244	phase I
BRD-K85667327	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191245	phase I
BRD-K86992593	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191246	phase I
BRD-K65655554	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191247	phase I
BRD-K67653084	CS(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191248	phase I
BRD-K16552772	CS(=O)(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191249	phase I
BRD-K50330857	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60191252	phase I
BRD-K32712332	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60191253	phase I
BRD-K98667932	COc1ccc(cc1)C#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60191254	phase I
BRD-K05645536	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60191255	phase I
BRD-K25638721	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc(F)cc1	CID:60191256	phase I
BRD-K92242945	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191257	phase I
BRD-K02133388	Cc1ccccc1-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191258	phase I
BRD-K63892915	CCS(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CCCCC1	CID:60191259	phase I
BRD-K81363924	CCS(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CCCCC1	CID:60191260	phase I
BRD-K55648964	CCS(=O)(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CCCCC1	CID:60191261	phase I
BRD-K55196996	CCS(=O)(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CCCCC1	CID:60191262	phase I
BRD-K95850342	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191263	phase I
BRD-K66061243	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191264	phase I
BRD-K28431799	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191265	phase I
BRD-K55055560	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191266	phase I
BRD-K19014823	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191267	phase I
BRD-K76477096	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)CC1CC1)c1ccc(\C=C\c2ccccc2)cc1	CID:60191268	phase I
BRD-K97873029	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191269	phase I
BRD-K60796852	OC[C@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(Br)cc1	CID:60191270	phase I
BRD-K77444669	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)Cc1cccnc1)c1ccc(cc1)C1=CCCCC1	CID:60191271	phase I
BRD-K12961950	CCCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191272	phase I
BRD-K88197986	CCCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191273	phase I
BRD-K71636675	CCCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191274	phase I
BRD-K33842318	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccc(F)cc1	CID:60191275	phase I
BRD-K75688794	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccc(F)cc1	CID:60191276	phase I
BRD-K84521734	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccc(F)cc1	CID:60191277	phase I
BRD-K55191691	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccc(F)cc1	CID:60191278	phase I
BRD-K43966520	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1ccc(F)cc1	CID:60191279	phase I
BRD-K37290968	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1ccc(F)cc1	CID:60191280	phase I
BRD-K29094514	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:60191281	phase I
BRD-K42589221	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1cccc(F)c1)c1ccc(cc1)C1=CCCCC1	CID:60191282	phase I
BRD-K93157782	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191283	phase I
BRD-K40230514	COCC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191284	phase I
BRD-K48918097	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191285	phase I
BRD-K34834946	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191286	phase I
BRD-K10006632	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191287	phase I
BRD-K57691575	COCC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191288	phase I
BRD-K98192020	CS(=O)(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191289	phase I
BRD-K53443165	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191290	phase I
BRD-K79379353	Cc1ccccc1-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cccc(F)c1	CID:60191291	phase I
BRD-K45200389	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191292	phase I
BRD-K60257691	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191293	phase I
BRD-K65898110	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191294	phase I
BRD-K90702747	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191295	phase I
BRD-K70648728	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191296	phase I
BRD-K58290803	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191297	phase I
BRD-K23647045	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CC1CC1	CID:60191298	phase I
BRD-K27481961	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CC1CC1	CID:60191299	phase I
BRD-K94253269	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)CC1CC1	CID:60191300	phase I
BRD-K03651051	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)CC1CC1	CID:60191301	phase I
BRD-K88376874	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)CC1CC1	CID:60191302	phase I
BRD-K29503610	CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)CC1CC1	CID:60191303	phase I
BRD-K41138144	COCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccncc1	CID:60191304	phase I
BRD-K25556383	COCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccncc1	CID:60191305	phase I
BRD-K14169964	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191306	phase I
BRD-K13307254	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191307	phase I
BRD-K01497006	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191308	phase I
BRD-K86112430	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191309	phase I
BRD-K85769686	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191310	phase I
BRD-K95683812	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191311	phase I
BRD-K77007746	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191312	phase I
BRD-K78826848	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)Nc1cc(F)ccc1F	CID:60191313	phase I
BRD-K43703882	COCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccncc1	CID:60191319	phase I
BRD-K29892351	COCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccncc1	CID:60191320	phase I
BRD-K74634175	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191321	phase I
BRD-K45532244	OC[C@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191322	phase I
BRD-K12562048	OC[C@@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191323	phase I
BRD-K43782840	OC[C@@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191324	phase I
BRD-K36080978	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191325	phase I
BRD-K51329831	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CC1	CID:60191326	phase I
BRD-K82911380	CS(=O)(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191327	phase I
BRD-K00141503	CS(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191328	phase I
BRD-K27293696	CS(=O)(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191329	phase I
BRD-K72663966	CS(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(Br)cc1	CID:60191330	phase I
BRD-K37455698	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191341	phase I
BRD-K28478559	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191342	phase I
BRD-K36232729	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191343	phase I
BRD-K20810283	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191344	phase I
BRD-K40769424	CC(C)NC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(C)cc1	CID:60191346	phase I
BRD-K06303559	COCC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191347	phase I
BRD-K11141556	COCC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191348	phase I
BRD-K59341874	COCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191349	phase I
BRD-K22149853	COCC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191350	phase I
BRD-K66761585	COCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191351	phase I
BRD-K02258558	COCC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191352	phase I
BRD-K64984926	COCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191353	phase I
BRD-K16172814	OC[C@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191354	phase I
BRD-K96552587	OC[C@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191355	phase I
BRD-K34607017	COCC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191356	phase I
BRD-K61122325	COCC#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191357	phase I
BRD-K37991590	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCCC1	CID:60191358	phase I
BRD-K44475992	CCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191359	phase I
BRD-K34231896	CCC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191360	phase I
BRD-K28190569	CCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191361	phase I
BRD-K75512942	CCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191362	phase I
BRD-K57822472	CCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191363	phase I
BRD-K69694842	CCC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191364	phase I
BRD-K35939150	CCC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191365	phase I
BRD-K98010525	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccncc1	CID:60191373	phase I
BRD-K31757099	CCC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191374	phase I
BRD-K52006320	CCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191375	phase I
BRD-K29227213	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191376	phase I
BRD-K83466397	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191377	phase I
BRD-K58245095	CC(C)CC#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191378	phase I
BRD-K57286317	CC(C)CC#Cc1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccccn1	CID:60191379	phase I
BRD-K83494171	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCC1	CID:60191380	phase I
BRD-K82781769	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CCC1	CID:60191381	phase I
BRD-K00057967	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCC1	CID:60191382	phase I
BRD-K60584379	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCC1	CID:60191383	phase I
BRD-K50068201	COCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CC1CC1	CID:60191384	phase I
BRD-K08468228	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191385	phase I
BRD-K36446940	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191386	phase I
BRD-K67662618	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191387	phase I
BRD-K05418735	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191388	phase I
BRD-K18447917	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191389	phase I
BRD-K97508452	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191390	phase I
BRD-K37290471	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191391	phase I
BRD-K18647673	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CC1	CID:60191392	phase I
BRD-K46562045	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CC1	CID:60191393	phase I
BRD-K09023525	COc1ccc(cc1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CC1	CID:60191394	phase I
BRD-K17579844	C\C=C\c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC1CCCCC1	CID:60191395	phase I
BRD-K86430746	Cc1cccc(c1)-c1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60191396	phase I
BRD-K97306770	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60191397	phase I
BRD-K96609736	Cc1cccc(c1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)c1ccc2OCOc2c1	CID:60191398	phase I
BRD-K46544760	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191399	phase I
BRD-K40963620	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191400	phase I
BRD-K23488072	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191401	phase I
BRD-K98326205	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191402	phase I
BRD-K59559352	CCC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC(C)C	CID:60191403	phase I
BRD-K25899698	CS(=O)(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191404	phase I
BRD-K74790646	CS(=O)(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191405	phase I
BRD-K52183630	CS(=O)(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191406	phase I
BRD-K54288605	CS(=O)(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191407	phase I
BRD-K42245756	CS(=O)(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191408	phase I
BRD-K27181648	CS(=O)(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191409	phase I
BRD-K40161407	CS(=O)(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191410	phase I
BRD-K65526065	CS(=O)(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#CCC1CCCC1	CID:60191411	phase I
BRD-K53092731	COCC(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60191412	phase I
BRD-K45043387	CCC(=O)N1C[C@@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191416	phase I
BRD-K55864253	CCC(=O)N1C[C@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191417	phase I
BRD-K39422601	CCC(=O)N1C[C@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191418	phase I
BRD-K23393992	CCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191419	phase I
BRD-K73062881	CCC(=O)N1C[C@@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191420	phase I
BRD-K20994897	CCC(=O)N1C[C@@H]2[C@@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191421	phase I
BRD-K88195243	OC[C@@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191422	phase I
BRD-K55069932	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191423	phase I
BRD-K75981692	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)C1CCC1	CID:60191424	phase I
BRD-K21246672	CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)[C@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CCC1	CID:60191425	phase I
BRD-K64417176	OC[C@@H]1[C@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccccc1F	CID:60191426	phase I
BRD-K88539660	OC[C@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccccc1F	CID:60191427	phase I
BRD-K82024598	OC[C@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccccc1F	CID:60191428	phase I
BRD-K61925563	OC[C@@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccccc1F	CID:60191429	phase I
BRD-K44026015	OC[C@@H]1[C@@H]([C@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccccc1F	CID:60191430	phase I
BRD-K45734366	OC[C@@H]1[C@@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccccc1F	CID:60191431	phase I
BRD-K46416377	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCC1)c1ccc(Br)cc1	CID:60191433	phase I
BRD-K12729417	CS(=O)(=O)N1C[C@@H]2[C@@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)C#Cc1ccc(F)cc1	CID:60191434	phase I
BRD-K07329815	OC[C@H]1[C@H]([C@@H]2CNCC(=O)N12)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60191435	phase I
BRD-K54168930	COc1ccc(cc1)-c1ccc(cc1)[C@@H]1[C@H](CO)N2[C@@H]1CN(CC2=O)C(=O)C1CC1	CID:60191436	phase I
BRD-K27459043	COc1cccc(NC(=O)N2C[C@@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191437	phase I
BRD-K20732958	COc1cccc(NC(=O)N2C[C@@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191438	phase I
BRD-K27395235	COc1cccc(NC(=O)N2C[C@@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191439	phase I
BRD-K03608142	COc1cccc(NC(=O)N2C[C@@H]3[C@@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191440	phase I
BRD-K74436011	COc1cccc(NC(=O)N2C[C@H]3[C@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191441	phase I
BRD-K80104673	COc1cccc(NC(=O)N2C[C@H]3[C@H]([C@@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191442	phase I
BRD-K88078052	COc1cccc(NC(=O)N2C[C@H]3[C@@H]([C@H](CO)N3C(=O)C2)c2ccc(cc2)C#CCC2CCCC2)c1	CID:60191443	phase I
BRD-K47588363	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191444	phase I
BRD-K17951468	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191445	phase I
BRD-K09527783	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191446	phase I
BRD-K46592487	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)c1ccc(F)cc1)c1ccc(cc1)C#CCC1CCCC1	CID:60191447	phase I
BRD-K19868817	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191448	phase I
BRD-K63628486	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@H](CO)N2[C@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191449	phase I
BRD-K18747403	COc1ccc(cc1)C#Cc1ccc(cc1)[C@H]1[C@@H](CO)N2[C@@H]1CN(CC2=O)C(=O)NC(C)C	CID:60191450	phase I
BRD-K33318635	COCC(=O)N1C[C@H]2[C@H]([C@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccccc1F	CID:60191451	phase I
BRD-K34009110	OC[C@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191452	phase I
BRD-K46811723	OC[C@@H]1[C@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191453	phase I
BRD-K56343202	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191454	phase I
BRD-K44641066	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191455	phase I
BRD-K13542161	OC[C@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191456	phase I
BRD-K75205131	OC[C@@H]1[C@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCOCC1)c1ccc(cc1)-c1cccnc1	CID:60191457	phase I
BRD-K63853589	OC[C@H]1[C@@H]([C@H]2CN(CC(=O)N12)C(=O)Nc1ccccc1)c1ccc(cc1)C#CC1CCCCC1	CID:60191458	phase I
BRD-K89122173	CCCNC(=O)N1C[C@H]2[C@H]([C@@H](CO)N2C(=O)C1)c1ccc(cc1)-c1ccc(F)cc1	CID:60191459	phase I
BRD-K07546004	CC(C)NC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1cccnc1	CID:60191512	phase I
BRD-K70075321	CN(C)CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccc(F)cc1	CID:60191560	phase I
BRD-K90046234	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CCC(F)(F)F)c1ccccc1	CID:60191561	phase I
BRD-K41430692	CCCNC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1cccnc1	CID:60191562	phase I
BRD-K51556457	CCCNC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1cccnc1	CID:60191563	phase I
BRD-K69611470	CCCNC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)c1cccnc1	CID:60191564	phase I
BRD-K56348092	COCC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(Cc2ccccc2)C1	CID:60191565	phase I
BRD-K21453542	CC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccccn1	CID:60191566	phase I
BRD-K89263606	CC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)c1ccccn1	CID:60191567	phase I
BRD-K97781791	CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1ccccn1	CID:60191569	phase I
BRD-K78477072	OC[C@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1Cc1ccccc1F	CID:60191570	phase I
BRD-K90008192	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1Cc1ccccc1F	CID:60191571	phase I
BRD-K61160172	CC(C)NC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CCC(F)(F)F)c1ccccc1	CID:60191597	phase I
BRD-K27376241	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CCC(F)(F)F)c1ccccc1	CID:60191598	phase I
BRD-K05601431	COc1ccccc1CN1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)c1cnccn1	CID:60191599	phase I
BRD-K77888593	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(CCC(F)(F)F)C2)N1C(=O)C1CCC1	CID:60191600	phase I
BRD-K63250790	OC[C@H]1[C@@H](c2ccccc2)C2(CN(CCC(F)(F)F)C2)N1C(=O)C1CCC1	CID:60191601	phase I
BRD-K14307099	COCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(C)=O)c1ccc(cc1)-c1ccc(C)cc1	CID:60191603	phase I
BRD-K84738609	COCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(C)=O)c1ccc(cc1)-c1ccc(C)cc1	CID:60191604	phase I
BRD-K01523435	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3ccccc3F)C2)N1C(=O)CC1CC1	CID:60191605	phase I
BRD-K72738889	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1Cc1ccccc1F	CID:60191606	phase I
BRD-K48383713	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCOCC2)N1Cc1ccccc1F	CID:60191607	phase I
BRD-K60238549	COCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CC1CCOCC1)c1ccc(cc1)\C=C\C	CID:60191608	phase I
BRD-K95321016	COCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)C1CC1)c1ccc(cc1)-c1cccc(C)c1	CID:60191609	phase I
BRD-K12025316	COCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)C1CC1)c1ccc(cc1)-c1cccc(C)c1	CID:60191610	phase I
BRD-K68950762	COCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)C1CC1)c1ccc(cc1)-c1cccc(C)c1	CID:60191611	phase I
BRD-K75900905	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1C(=O)c1cnccn1	CID:60191613	phase I
BRD-K30659453	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1C(=O)c1cnccn1	CID:60191614	phase I
BRD-K89555807	CCCNC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2Cc1ccccn1)c1ccccc1	CID:60191650	phase I
BRD-K31194232	CCCNC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2Cc1ccccn1)c1ccccc1	CID:60191651	phase I
BRD-K97460860	CCCNC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2Cc1ccccn1)c1ccccc1	CID:60191652	phase I
BRD-K60600704	OC[C@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCCCC2)N1C(=O)c1cccnc1	CID:60191653	phase I
BRD-K31812476	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCCCC2)N1C(=O)c1cccnc1	CID:60191654	phase I
BRD-K03384615	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCCCC2)N1C(=O)c1cccnc1	CID:60191655	phase I
BRD-K62714403	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCCCC2)N1C(=O)c1cccnc1	CID:60191656	phase I
BRD-K52157979	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1C(=O)c1cnccn1	CID:60191657	phase I
BRD-K76494382	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1C(=O)NC1CCCC1	CID:60191659	phase I
BRD-K76987587	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1C(=O)NC1CCCC1	CID:60191660	phase I
BRD-K08443710	CCC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)NC1CCCC1	CID:60191661	phase I
BRD-K43955991	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)C1CCCC1)c1ccccc1	CID:60191692	phase I
BRD-K97209864	CC(C)NC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)C1CCCC1)c1ccccc1	CID:60191693	phase I
BRD-K34629721	CN(C)CC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2S(C)(=O)=O)c1ccccc1	CID:60191694	phase I
BRD-K23933733	CN(C)CC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2S(C)(=O)=O)c1ccccc1	CID:60191788	phase I
BRD-K98283674	CN(C)CC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2S(C)(=O)=O)c1ccccc1	CID:60191789	phase I
BRD-K66947316	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)C2CCCCC2)C11CN(C1)C(=O)NC(C)C	CID:60191849	phase I
BRD-K08378202	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)NC2CCCCC2)N1S(=O)(=O)Cc1ccccc1	CID:60191852	phase I
BRD-K63303938	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)NC2CCCCC2)N1S(=O)(=O)Cc1ccccc1	CID:60191853	phase I
BRD-K86089324	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)NC2CCCCC2)N1S(=O)(=O)Cc1ccccc1	CID:60191855	phase I
BRD-K82425094	C\C=C\c1ccc(cc1)[C@@H]1[C@@H](CO)N(C(=O)CC2CC2)C11CN(C1)S(C)(=O)=O	CID:60191856	phase I
BRD-K34086616	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(C(=O)CC2CC2)C11CN(C1)S(C)(=O)=O	CID:60191857	phase I
BRD-K54673054	C\C=C\c1ccc(cc1)[C@@H]1[C@H](CO)N(C(=O)CC2CC2)C11CN(C1)S(C)(=O)=O	CID:60191858	phase I
BRD-K22750348	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1Cc1ccc(Cl)cc1	CID:60191859	phase I
BRD-K28000085	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CC2)N1Cc1ccc(Cl)cc1	CID:60191860	phase I
BRD-K83998477	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CC1CC1)c1ccc(cc1)-c1cccc(F)c1	CID:60191921	phase I
BRD-K59389251	CCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CC1CC1)c1ccc(cc1)-c1cccc(F)c1	CID:60191922	phase I
BRD-K67118623	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CC1CC1)c1ccc(cc1)-c1cccc(F)c1	CID:60191923	phase I
BRD-K40627098	CCC(=O)N1[C@H](CO)[C@H](c2ccc(\C=C\C)cc2)C11CN(C1)C(=O)c1ccccc1	CID:60191924	phase I
BRD-K76150628	CCC(=O)N1[C@@H](CO)[C@@H](c2ccc(\C=C\C)cc2)C11CN(C1)C(=O)c1ccccc1	CID:60191925	phase I
BRD-K64597663	CCCNC(=O)N1CC2(C1)[C@H]([C@H](CO)N2C(=O)CC1CC1)c1ccccc1	CID:60191926	phase I
BRD-K56638701	CCCNC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)CC1CC1)c1ccccc1	CID:60191928	phase I
BRD-K69372544	OC[C@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)CC2CC2)N1CC1CCOCC1	CID:60191933	phase I
BRD-K57350811	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(CC3CC3)C2)N1Cc1ccc(F)cc1	CID:60191972	phase I
BRD-K81036566	OC[C@@H]1[C@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1CCC(F)(F)F	CID:60191973	phase I
BRD-K27240704	OC[C@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1CCC(F)(F)F	CID:60191974	phase I
BRD-K76909981	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1CCC(F)(F)F	CID:60191975	phase I
BRD-K95642310	CCC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CC1CCCC1)c1ccc(cc1)\C=C\C	CID:60191976	phase I
BRD-K13868095	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CC1CCCC1)c1ccc(cc1)\C=C\C	CID:60191977	phase I
BRD-K44712456	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1Cc1cccnc1	CID:60191978	phase I
BRD-K48717457	CCCNC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)CC1CC1)c1ccccc1	CID:60191979	phase I
BRD-K93373675	COCC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccn1	CID:60191981	phase I
BRD-K88311084	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCC2)N1Cc1cccnc1	CID:60192010	phase I
BRD-K00398667	COCC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccn1	CID:60192049	phase I
BRD-K61629734	CS(=O)(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(Cc2ccccn2)C1	CID:60192051	phase I
BRD-K04361415	CCS(=O)(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CC1CCCC1)c1ccccc1	CID:60192075	phase I
BRD-K24690085	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccc2)N1Cc1cc(F)ccc1F	CID:60192109	phase I
BRD-K08446420	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccc2)N1Cc1cc(F)ccc1F	CID:60192110	phase I
BRD-K14487440	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1Cc1cccnc1	CID:60192111	phase I
BRD-K60297013	OC[C@@H]1[C@H](c2ccccc2)C2(CN(Cc3nccs3)C2)N1Cc1cccnc1	CID:60192112	phase I
BRD-K14483137	CN(C)CC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(CCC(F)(F)F)C1	CID:60192113	phase I
BRD-K82870050	CN(C)CC(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(CCC(F)(F)F)C1	CID:60192115	phase I
BRD-K64687628	CN(C)CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(CCC(F)(F)F)C1	CID:60192116	phase I
BRD-K79435297	CCC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2S(C)(=O)=O)c1ccc(cc1)-c1cccc(C)c1	CID:60192117	phase I
BRD-K77456132	CCC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2S(C)(=O)=O)c1ccc(cc1)-c1cccc(C)c1	CID:60192119	phase I
BRD-K96183125	CCC(=O)N1CC2(C1)[C@H]([C@H](CO)N2S(C)(=O)=O)c1ccc(cc1)-c1cccc(C)c1	CID:60192120	phase I
BRD-K43721143	OC[C@H]1[C@H](c2ccccc2)C2(CN(Cc3ccncc3)C2)N1Cc1ccncc1	CID:60192174	phase I
BRD-K55883155	CS(=O)(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(Cc2cc(F)ccc2F)C1	CID:60192176	phase I
BRD-K05889827	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccncc2)N1C(=O)CC1CC1	CID:60192177	phase I
BRD-K39337865	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2ccncc2)N1C(=O)CC1CC1	CID:60192178	phase I
BRD-K00692337	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccncc2)N1C(=O)CC1CC1	CID:60192179	phase I
BRD-K25423005	OC[C@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2ccncc2)N1C(=O)CC1CC1	CID:60192180	phase I
BRD-K84574164	OC[C@@H]1N(Cc2ccccn2)C2(CN(C(=O)CC3CC3)C2)[C@@H]1c1ccccc1	CID:60192181	phase I
BRD-K39029679	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2C(=O)c1ccccn1)c1ccccc1	CID:60192182	phase I
BRD-K75100604	CC(C)NC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2C(=O)c1ccccn1)c1ccccc1	CID:60192183	phase I
BRD-K70685076	CC(C)NC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)c1ccccn1)c1ccccc1	CID:60192184	phase I
BRD-K34913101	CCS(=O)(=O)N1[C@@H](CO)[C@@H](c2ccc(cc2)\C=C\C)C11CN(C1)C(C)=O	CID:60192185	phase I
BRD-K25539387	OC[C@H]1[C@@H](c2ccccc2)C2(CN(Cc3cncnc3)C2)N1C(=O)C1CC1	CID:60192186	phase I
BRD-K17351089	CCS(=O)(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)C1CCCCC1	CID:60192187	phase I
BRD-K09552525	CCS(=O)(=O)N1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)C1CCCCC1	CID:60192188	phase I
BRD-K71499021	CCC(=O)N1[C@@H](CO)[C@@H](c2ccc(cc2)\C=C\C)C11CN(CCC(F)(F)F)C1	CID:60192190	phase I
BRD-K08938154	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCCC2)N1CC1CC1	CID:60192192	phase I
BRD-K01091374	OC[C@H]1N(Cc2ccccn2)C2(CN(C(=O)CC3CC3)C2)[C@@H]1c1ccccc1	CID:60192238	phase I
BRD-K26727724	CCCNC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2CC1CCOCC1)c1ccccc1	CID:60192240	phase I
BRD-K94017308	CCCNC(=O)N1CC2(C1)[C@@H]([C@H](CO)N2CC1CCOCC1)c1ccccc1	CID:60192241	phase I
BRD-K41842760	CCCNC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2CC1CCOCC1)c1ccccc1	CID:60192242	phase I
BRD-K92636280	OC[C@@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccc2F)N1CC1CC1	CID:60192243	phase I
BRD-K74198494	OC[C@H]1[C@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccc2F)N1CC1CC1	CID:60192245	phase I
BRD-K58253880	OC[C@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccc2F)N1CC1CC1	CID:60192246	phase I
BRD-K23208702	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)C2CCCC2)N1CC1CC1	CID:60192247	phase I
BRD-K39908587	CC(C)NC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1cccnc1	CID:60192249	phase I
BRD-K04983929	CC(C)NC(=O)N1[C@H](CO)[C@H](c2ccccc2)C11CN(C1)C(=O)Cc1cccnc1	CID:60192250	phase I
BRD-K15143651	OC[C@@H]1[C@@H](c2ccccc2)C2(CN(C2)C(=O)c2ccccc2F)N1CC1CC1	CID:60192284	phase I
BRD-K03073795	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(C1)C(=O)Cc1ccccc1)C(=O)Nc1ccc(F)cc1	CID:60192328	phase I
BRD-K37317589	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)C(C)=O)n(C)c2c1	CID:60192386	phase I
BRD-K94171232	COCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(OC)c1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60192484	phase I
BRD-K37728465	CN(C)CC(=O)N[C@@H]1C[C@@H]2O[C@H](CO)CC[C@@H]2O[C@@H]1CCc1ccc(cc1)C1=CCCCC1	CID:60192494	phase I
BRD-K93291593	C[C@H](CO)N1C[C@@H](C)[C@H](CN(C)C(=O)Nc2ccccc2)OCCCC[C@@H](C)Oc3ccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)cc3C1=O	CID:60192504	phase I
BRD-K26214610	OC[C@@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60192675	phase I
BRD-K74923162	OC[C@H]1[C@@H]([C@@H]2CN(CC(=O)N12)C(=O)C1CCCCC1)c1ccc(cc1)-c1ccc(cc1)C#N	CID:60192676	phase I
BRD-K08198779	OC[C@H]1[C@H]([C@H]2CN(Cc3ccc(F)cc3)CC(=O)N12)c1ccc(cc1)-c1ccccc1	CID:60192679	phase I
BRD-K26457096	OC[C@@H]1[C@@H]([C@@H]2CN(Cc3ccc(F)cc3)CC(=O)N12)c1ccc(cc1)-c1ccccc1	CID:60192682	phase I
BRD-K81261525	C\C=C\c1ccc2N[C@@H](CO)[C@H]3CCN([C@H]3c2c1)C(=O)c1ccc(F)cc1	CID:60192688	phase I
BRD-K40655550	C\C=C\c1ccc(cc1)[C@H]1[C@@H](CO)N(CC2CCCC2)[C@@H]1CNC(=O)NC(C)C	CID:60192704	phase I
BRD-K21325303	CCCNC(=O)N(C[C@H]1N[C@H](CO)[C@@H]1c1ccccc1)Cc1cccnc1	CID:60192910	phase I
BRD-K68971353	OC[C@H]1N[C@H](CNC(=O)C2CCC2)[C@H]1c1ccc(cc1)C1=CCCC1	CID:60192959	phase I
BRD-K53739837	OC[C@H]1N[C@H](CNC(=O)Cc2ccccc2)[C@H]1c1ccc(cc1)C1=CCCC1	CID:60193306	phase I
BRD-K53669914	CCCNC[C@H]1[C@H]([C@@H](CO)N1C(=O)C1CCC1)c1ccc(cc1)C1=CCCCC1	CID:60193374	phase I
BRD-K73788182	CCCN1[C@H](CO)[C@@H]([C@H]1CN(CC)C(=O)c1ccccn1)c1ccc(\C=C\C)cc1	CID:60193408	phase I
BRD-K04856990	COc1ccccc1NC(=O)N1CCCCN2[C@@H](CO)[C@@H]([C@@H]2C1)c1ccc(cc1)C#CC1CC1	CID:60193560	phase I
BRD-K82544341	OC[C@@H]1[C@H]2Cn3c(ccc(C4=CCCCC4)c3=O)[C@H]2N(CC2CC2)[C@H]1C(=O)NC1Cc2ccccc2C1	CID:60193563	phase I
BRD-K85751793	COc1ccc(cc1)S(=O)(=O)N1CC[C@@]2(CC1)CN(Cc1ccccc1OC)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:60193582	phase I
BRD-K57127959	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1nccs1)C[C@]31CCN(CC1)C(=O)C1CCCC1	CID:60193632	phase I
BRD-K83191645	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)C1CCC1	CID:60193939	phase I
BRD-K39001644	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC4CCCC4)CC3)n(C)c2c1	CID:60194036	phase I
BRD-K09854848	COc1cc(cc(OC)c1OC)\C=C\C(=O)N1CCCC=CC1=O	CID:60194076	phase I
BRD-K79877282	Cc1cc(CS(=O)(=O)c2ccccc2)cc(OCc2ccc(CN3CCC[C@@H]3CO)cc2)c1	CID:66577038	phase I
BRD-K70555272	CC[C@H]1CC[C@H]2O[C@@]3(CC[C@@H](C)[C@@H](C[C@H](C)O)O3)[C@H](C)[C@@H](OC(=O)\C=C\[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@](C)(O)[C@H](O)[C@@H](C)C\C=C\C=C\1)[C@H]2C	CID:66649023	phase I
BRD-K05350981	CC[C@H]1CC[C@H]2O[C@@]3(CC[C@@H](C)[C@@H](C[C@H](C)O)O3)[C@H](C)[C@@H](OC(=O)\C=C\[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@@H](C)C\C=C\C=C\1)[C@H]2C	CID:66690779	phase I
BRD-K46056750	NC(=O)Nc1cc(sc1C(=O)N[C@@H]1CCCNC1)-c1cccc(F)c1	CID:67077825	phase I
BRD-K79070828	Cc1cncc2cccc(c12)S(=O)(=O)N3CC[C@@H](N)C3	CID:67243342	phase I
BRD-K86274953	O=C(Nc1n[nH]c2cc(ccc12)-c1cccc(c1)C(=O)NC1CC1)C1CC1	CID:68234129	phase I
BRD-A57152259	CCNC(=O)[C@H]1O[C@H](C(O)C1O)n1cnc2c(N)nc(NCCc3ccc(CCC(O)=O)cc3)nc12	CID:68337842	phase I
BRD-A73680854	NC(CCC(O)=O)C(=O)N1CCC[C@H]1B(O)O	CID:68508601	phase I
BRD-A78236793	COc1cc2C(CN(C)CCc2cc1Br)c1ccc(N)cc1	CID:68735707	phase I
BRD-K89912164	C[C@@H]1O[C@@H](C[C@H]1O)n1cnc2c(N)ncnc12	CID:69621407	phase I
BRD-K57282030	COc1cc(OC)cc(c1)-c1ccc2ncc3ccc(=O)n(-c4ccc(N5CCNCC5)c(c4)C(F)(F)F)c3c2c1	CID:69923936	phase I
BRD-K37417543	C[C@H]1[C@H](OC(=O)CC\C=C\C[C@@H](CC(=O)NCc2ccc(Cl)cc2)C(=O)N1C)c1ccccc1	CID:70680396	phase I
BRD-K58547375	Clc1ccc(CN2C\C=C\CCC(=O)N[C@@H](COC2=O)c2ccccc2)cc1	CID:70680397	phase I
BRD-K11306851	Clc1ccc(CNC(=O)C[C@@H]2C\C=C\CCC(=O)N[C@@H](COC2=O)c2ccc(Cl)cc2)cc1	CID:70680398	phase I
BRD-K25444257	Clc1ccc(CNC(=O)C[C@@H]2C\C=C\CCC(=O)N3CCC[C@@H]3COC2=O)cc1	CID:70680399	phase I
BRD-K91338578	CC(=O)N[C@@H]1C\C=C\CCC(=O)N[C@@H](COC1=O)c1ccc(F)cc1	CID:70680400	phase I
BRD-K19326298	CC(=O)N[C@@H]1C\C=C\CCCOC(=O)[C@@H]2CCCN2C1=O	CID:70680401	phase I
BRD-K16582605	C[C@@H]1C\C=C\CCC(=O)N[C@@H](CC(=O)O1)c1ccccc1	CID:70680403	phase I
BRD-K90370028	CC(=O)N[C@@H]1C\C=C\CCC(=O)N[C@@H](COC1=O)c1ccccc1	CID:70680404	phase I
BRD-K14700434	C[C@H]1C\C=C\C[C@@H](CC(=O)NCc2ccc(Cl)cc2)C(=O)N2CCC[C@H]2CNC1=O	CID:70680405	phase I
BRD-K92084213	Clc1ccc(CNC(=O)C[C@@H]2C\C=C\CCC(=O)OC[C@H]3CCCN3C2=O)cc1	CID:70680406	phase I
BRD-K45028728	C[C@@H]1C\C=C\CCNC(=O)[C@@H](COC1=O)c1ccccc1	CID:70680407	phase I
BRD-K55896799	C[C@H]1C\C=C\CCCN[C@@H](COC1=O)c1ccccc1	CID:70680408	phase I
BRD-K73183319	Clc1ccc(CNC(=O)C[C@@H]2C\C=C\CCC(=O)N[C@H]3[C@H](Cc4ccccc34)OC2=O)cc1	CID:70680410	phase I
BRD-K58044374	CN1C[C@H](NC(=O)CC\C=C\C[C@@H](CC(=O)NCc2ccc(Cl)cc2)C1=O)c1ccccc1	CID:70680411	phase I
BRD-K23628492	CCOC(=O)N1c2ccccc2Sc2ccc(Cl)cc12	CID:71125363	phase I
BRD-K54168243	COc1ccc2[nH]cc(\C=C3/C(=O)N(CCCN(C)C)c4ccc(F)cc34)c2c1	CID:71311634	phase I
BRD-K07103434	CN(C)c1ccc2[n+](C)c(CCc3cc(C)n(c3C)-c3ccccc3)ccc2c1	CID:71311933	phase I
BRD-A43331270	CCCN1C(C)=C(C(c2cccc(c2)[N+]([O-])=O)C(C(=O)ON2CCC(CC2)(c2ccccc2)c2ccccc2)=C1C)C(=O)OC	CID:71317558	phase I
BRD-K83068825	C[N+](C)(C)CCc1c[nH]cn1	CID:71351736	phase I
BRD-K12482929	Cc1c(O)c(O)cc(O)c1CCN	CID:71371555	phase I
BRD-K52160314	CC1(C)C(=O)NN=C1c1ccc(Cl)cc1	CID:71576756	phase I
BRD-K83493571	C[C@@H]1CC(=O)NN=C1c1ccc(I)cc1	CID:71576757	phase I
BRD-K55533488	C[C@@H]1CC(=O)NN=C1c1ccc(cc1)N1CCOCC1	CID:71576758	phase I
BRD-K22587354	CC1(C)C(=O)NN=C1c1ccc(cc1)N1CCOCC1	CID:71576776	phase I
BRD-K00972013	CC(=O)N1CC2(C1)[C@@H]([C@@H](CO)N2Cc1ccccc1F)c1ccccc1	CID:71627358	phase I
BRD-K07466598	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccc3OCOc3c1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:71729870	phase I
BRD-K99252563	Cn1cc(cn1)-c1ccc2ncc3ccc(=O)n(-c4ccc5CCN(C(=O)C=C)c5c4)c3c2c1	CID:71748056	phase I
BRD-K94154731	CCCNC(=O)N1C[C@@]2(C1)CN([C@H](CO)c1[nH]c3cc(OC)ccc3c21)C(=O)CN1CCOCC1	CID:71758843	phase I
BRD-K06521224	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)c3ccncc3)C(=O)C3CCOCC3)n(C)c2c1	CID:71758896	phase I
BRD-K93000597	CC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(Cc2ccc(Cl)cc2)C1	CID:71758950	phase I
BRD-K23319301	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2cccc(F)c2)CC1)C(=O)C1CCOCC1	CID:71758969	phase I
BRD-K00317040	COc1ccc2c3c([C@@H](CO)NC[C@]33CCN(CC4CCCCC4)CC3)n(C)c2c1	CID:71758993	phase I
BRD-K65309966	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)c3ccccc3F)C(=O)Nc3ccccc3F)n(C)c2c1	CID:71758998	phase I
BRD-K11689127	COc1ccc2c3c([C@H](CO)N(Cc4cccnc4)C[C@]33CCN(CC3)C(=O)NC(C)C)n(C)c2c1	CID:71759003	phase I
BRD-K21728898	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4OC)C[C@]33CCN(CC4CC4)CC3)n(C)c2c1	CID:71759006	phase I
BRD-K28451547	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4OC)C[C@]33CCN(CC4CC4)CC3)n(C)c2c1	CID:71759010	phase I
BRD-K78268279	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1OC)C[C@]31CN(C1)C(C)=O	CID:71759014	phase I
BRD-K17731272	COc1ccc2c3c([C@H](CO)N(Cc4ccc(Cl)cc4)C[C@]33CN(C3)C(=O)NC(C)C)n(C)c2c1	CID:71759015	phase I
BRD-K89550909	OC[C@H]1N(Cc2ccccn2)C2(CN(C(=O)CC3CC3)C2)[C@H]1c1ccccc1	CID:71759019	phase I
BRD-K34428383	COc1ccc2c3c([C@@H](CO)N(Cc4ccc(Cl)cc4)C[C@]33CN(C3)C(=O)NC(C)C)n(C)c2c1	CID:71759045	phase I
BRD-K25585643	CCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(Cl)c1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:71759117	phase I
BRD-K54260596	COc1ccc2c3c([C@H](CO)N(CC4CC4)C[C@]33CCN(CC3)S(=O)(=O)c3cccs3)n(C)c2c1	CID:71759122	phase I
BRD-K44968554	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)Cc1cccnc1)S(=O)(=O)c1ccc(C)cc1	CID:71759150	phase I
BRD-K60004464	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(Cc2cccnc2)CC1)C(=O)c1ccc(F)cc1	CID:71759195	phase I
BRD-K39017054	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(C3)S(=O)(=O)c3cn(C)cn3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:71759260	phase I
BRD-K46815273	COc1ccc2c3c([C@@H](CO)N(Cc4nccs4)C[C@]33CCN(CC4CCCC4)CC3)n(C)c2c1	CID:71759329	phase I
BRD-K68190084	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4)C[C@]33CN(C3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:71759354	phase I
BRD-K64256554	COc1ccc2c3c([C@H](CO)NC[C@]33CN(Cc4cc(F)ccc4F)C3)n(C)c2c1	CID:71759415	phase I
BRD-K17350012	COc1ccc2c3c([C@H](CO)N(C)C[C@]33CN(C3)C(=O)C3CCC3)n(C)c2c1	CID:71759440	phase I
BRD-K47463456	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(C[C@]31CCN(CC1)C(=O)Nc1ccccc1)S(C)(=O)=O	CID:71759441	phase I
BRD-K91880445	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(CC1)S(=O)(=O)c1cccs1)C(=O)c1ccc(F)cc1	CID:71759446	phase I
BRD-K43524201	COc1ccc2c3c([C@@H](CO)N(C)C[C@]33CCN(CC3)C(=O)CN3CCOCC3)n(C)c2c1	CID:71759448	phase I
BRD-K22862802	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)NC(C)C	CID:71759459	phase I
BRD-K59683426	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)C(=O)Nc3cccc(F)c3)C(=O)C3CCOCC3)n(C)c2c1	CID:71759534	phase I
BRD-K60760984	CC(=O)N1CC2(C1)[C@H]([C@@H](CO)N2Cc1ccccc1F)c1ccccc1	CID:71759563	phase I
BRD-K96694631	COc1ccc2c3c([C@@H](CO)N(CC4CC4)C[C@]33CCN(CC3)S(=O)(=O)c3cccs3)n(C)c2c1	CID:71759582	phase I
BRD-K60839087	CCS(=O)(=O)N1C[C@@]2(C1)CN(Cc1ccc3OCOc3c1)[C@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:71759618	phase I
BRD-K84617556	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(Cc4ccc(Cl)cc4)C3)C(C)=O)n(C)c2c1	CID:71759654	phase I
BRD-K28934562	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2cccc(F)c2)CC1)C(=O)C1CCOCC1	CID:71759739	phase I
BRD-K93419974	COc1ccc2c3c([C@H](CO)N(Cc4ccccc4)C[C@]33CN(C3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:71759741	phase I
BRD-K61657561	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1ccccc1F)C[C@]31CN(CC2CC2)C1	CID:71759759	phase I
BRD-K77191339	CC(C)NC[C@@H]1[C@H]([C@@H](CO)N1C(=O)CC1CC1)c1ccc(cc1)C1=CCCCC1	CID:71759789	phase I
BRD-K13150695	CCC(=O)N1C[C@@]2(C1)CN(Cc1cccc(Cl)c1)[C@@H](CO)c1[nH]c3cc(OC)ccc3c21	CID:71759866	phase I
BRD-K05484452	COc1ccc2c3c([nH]c2c1)[C@H](CO)NC[C@]31CCN(CC1)C(=O)Nc1ccc(F)cc1	CID:71759907	phase I
BRD-K03228956	CCCNC(=O)N1C[C@]2(CN(C2)C(=O)CN(C)C)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:71759937	phase I
BRD-K55981249	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4Cl)C[C@]33CCN(CC3)C(=O)CC3CC3)n(C)c2c1	CID:71759949	phase I
BRD-K26545157	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4ccncc4)CC3)C(=O)CN3CCOCC3)n(C)c2c1	CID:71760052	phase I
BRD-K81029835	COc1ccc2c3c([C@H](CO)N(C[C@]33CN(Cc4ccncc4)C3)C(=O)CC3CC3)n(C)c2c1	CID:71760106	phase I
BRD-K31142225	CCCNC(=O)N1CC[C@@]2(CC1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)CC1CC1	CID:71760121	phase I
BRD-K00668050	COc1ccc2c3c([C@H](CO)NC[C@]33CN(C3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:71760147	phase I
BRD-K59854189	COCC(=O)N1C[C@]2(CN(C2)S(C)(=O)=O)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:71760199	phase I
BRD-K36115176	CCC(=O)N1[C@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)CN1CCOCC1	CID:71760221	phase I
BRD-K15768839	CCS(=O)(=O)N1CC2(C1)[C@@H]([C@H](CO)N2C(=O)C1CCCC1)c1ccc(cc1)\C=C\C	CID:71760243	phase I
BRD-K16097209	COc1ccc2c3c([C@H](CO)N(C[C@]33CCN(CC3)C(=O)Nc3ccccc3F)C(C)=O)n(C)c2c1	CID:71760344	phase I
BRD-K89915215	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CCN(Cc2cccnc2)CC1)C(=O)c1ccc(F)cc1	CID:71760361	phase I
BRD-K26772093	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(CC1CC1)C[C@]31CN(Cc2cc(F)ccc2F)C1	CID:71760370	phase I
BRD-K55792644	COc1ccc2c3c([C@@H](CO)N(C[C@]33CN(C3)S(=O)(=O)c3cn(C)cn3)C(=O)Nc3ccc(F)cc3)n(C)c2c1	CID:71760419	phase I
BRD-K64607642	COc1ccc2c3c([C@@H](CO)N(Cc4ccccc4)C[C@]33CN(CC4CC4)C3)n(C)c2c1	CID:71760478	phase I
BRD-K86574497	COc1ccc2c3c([C@@H](CO)NC[C@]33CN(C3)S(=O)(=O)c3ccc(C)cc3)n(C)c2c1	CID:71760509	phase I
BRD-K19031214	COc1ccccc1CN1[C@@H](CO)[C@@H](c2ccccc2)C11CN(C1)C(=O)Cc1ccccc1	CID:71760513	phase I
BRD-K44266302	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(Cc4nccs4)CC3)C(=O)NC(C)C)n(C)c2c1	CID:71760516	phase I
BRD-K11989341	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(C)CC3)S(=O)(=O)c3cn(C)cn3)n(C)c2c1	CID:71760552	phase I
BRD-K93210315	COc1ccc2c3c([C@H](CO)N(CC4CCOCC4)C[C@]33CN(Cc4nccs4)C3)n(C)c2c1	CID:71760614	phase I
BRD-K57181059	COc1ccc(cc1)S(=O)(=O)N1C[C@@]2(C1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)c1cccnc1	CID:71760625	phase I
BRD-K59230034	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C)C[C@]31CN(C1)S(C)(=O)=O	CID:71760649	phase I
BRD-K29540359	COc1ccc2c3c([nH]c2c1)[C@H](CO)N(Cc1cc(OC)cc(OC)c1)C[C@]31CN(C1)S(=O)(=O)c1cccc(F)c1	CID:71760691	phase I
BRD-K40906026	COc1ccc2c3c([C@@H](CO)N(C[C@]33CCN(CC3)C(=O)c3ccncc3)C(=O)C3CCOCC3)n(C)c2c1	CID:71760750	phase I
BRD-K73937887	CCCNC(=O)N1C[C@]2(CCN(CC2)C(=O)Nc2cccc(F)c2)c2c([C@H]1CO)n(C)c1cc(OC)ccc21	CID:71760777	phase I
BRD-K82423177	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(C[C@]31CN(Cc2ccc(F)cc2)C1)C(=O)NC(C)C	CID:71760799	phase I
BRD-K81500599	CCCNC(=O)N1CC[C@@]2(CC1)CN([C@@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)CC1CC1	CID:71760812	phase I
BRD-K19898724	COCC(=O)N1CC[C@@]2(CC1)CN(Cc1cc(F)ccc1F)[C@@H](CO)c1c2c2ccc(OC)cc2n1C	CID:71760854	phase I
BRD-K52959179	COc1ccc2c3c([nH]c2c1)[C@@H](CO)N(Cc1ccccn1)C[C@]31CN(C1)C(=O)CC1CC1	CID:71760866	phase I
BRD-K86529788	CCS(=O)(=O)N1C[C@@]2(C1)CN([C@H](CO)c1c2c2ccc(OC)cc2n1C)C(=O)NC(C)C	CID:71760876	phase I
BRD-K08589866	CC1(C)CC(C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12	CID:71760892	phase I
BRD-K72264770	COC(=O)c1ccc2n(CCCc3ccccc3)c(NC(=O)c4ccccc4)nc2c1	CID:72193870	phase I
BRD-K89708791	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c4nc5cc(C)ccn5c4c(NC(=O)\C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c(O)c2c(O)c3C	CID:72698618	phase I
BRD-K29313308	CC(=O)Nc1ccc(cc1)C(=O)Nc1ccc(F)cc1N	CID:72734382	phase I
BRD-K74797618	COc1cc(\C=C\C(=O)N2CCC=C(C#Cc3ccccc3F)C2=O)cc(OC)c1OC	CID:72947407	phase I
BRD-K86472598	COc1cc(cc(OC)c1OC)\C=C\C(=O)N1CCC=C(C#CC2CC2)C1=O	CID:72947410	phase I
BRD-A43155244	COc1cc(\C=C\C(=O)N2C(CC=CC2=O)c2cccs2)cc(OC)c1OC	CID:72947591	phase I
BRD-K64024097	CC(=O)Nc1ccc(cc1)C(=O)Nc2ccc(C)cc2N	CID:73055061	phase I
BRD-K05870596	COc1cc(ccc1Nc1nc(N)c(s1)C(=O)c1c(Cl)cccc1Cl)N1CCN(C)CC1	CID:73265211	phase I
BRD-K24515980	Cc1ccc(cc1NC(=O)c1ccno1)C(=O)Nc1cc(NC(=O)C=C)cc(c1)C(F)(F)F	CID:73265214	phase I
BRD-K66847579	CCN(CC)CCCCNc1ncc2CN(C(=O)N(C)c2n1)c1c(Cl)c(OC)cc(OC)c1Cl	CID:73265276	phase I
BRD-K88969189	C[C@]12CC[C@H]3[C@@H](CCc4cc(O)ccc34)[C@H]1CC[C@@]2(O)C#C	CID:73265347	phase I
BRD-K39096267	Oc1ccc(C[C@H]2N3[C@@H](CN(Cc4cccc5ccccc45)C2=O)N(CCC3=O)C(=O)NCc2ccccc2)cc1	CID:73357429	phase I
BRD-A50287119	CO[C@@H]1C[C@H](CC(C)[C@@H]2CC(=O)[C@H](C)\C=C(C)\[C@@H](O)[C@@H](OC)C(=O)[C@H](C)C[C@H](C)\C=C\C=C\C=C(C)\[C@H](C[C@@H]3CC[C@@H](C)[C@@](O)(O3)C(=O)C(=O)N3CCCC[C@H]3C(=O)O2)OC)CC[C@H]1O	CID:73438890	phase I
BRD-A72666989	C[C@H]1[C@H]2[C@H](C[C@H]3[C@@H]4CC[C@@H]5C[C@H](CC[C@]5(C)[C@H]4CC[C@]23C)O[C@@H]2O[C@H](CO)[C@H](O)[C@H](O)[C@H]2O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)O[C@]11CCC(C)OC1	CID:73438891	phase I
BRD-A72024019	CC(C)C\C=C/C(=O)NC1C(OC2OC(C)C(O)C(O)C2NC(C)=O)OC(CC(O)C2OC(C(O)C2O)n2ccc(=O)[nH]c2=O)C(O)C1O	CID:73438893	phase I
BRD-A42994615	Nc1ncnc2n([C@H]3O[C@H]4COP(O)(=O)O[C@@H]4[C@@H]3O)c(Sc3ccc(Cl)cc3)nc12	CID:73438897	phase I
BRD-K76894938	Cc1c[nH]c(n1)-c1cnc(NCCNc2ccc(cc2)C#N)nc1-c1ccc(Cl)cc1Cl	CID:73438898	phase I
BRD-K87066636	CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)NCC(=O)N[C@@H](CS)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(O)=O	CID:73438899	phase I
BRD-K82681249	CCOC(=O)N1CCN(CC1)[N+](\[O-])=N\Oc1cc(ccc1[N+]([O-])=O)[N+]([O-])=O	CID:73438900	phase I
BRD-A65140285	NC1Cc2ccc(O)cc2NC1=O	CID:73554815	phase I
BRD-A94810754	CCC[C@@H](C)C[C@H](C)C[C@H](C)C(=O)CC(=O)[C@H](C)C[C@H](C)C\C=C\[C@@H](C)[C@@H](O)[C@@H](C)[C@@H](O)C[C@@H]1CC[C@](C)(O1)C1CC[C@](C)(O1)[C@@H](C)O	CID:73652146	phase I
BRD-K84803513	OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO	CID:73707341	phase I
BRD-K98634983	OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)CCCCC(=O)NO	CID:73707342	phase I
BRD-K62768020	ONC(=O)CCCCCC(=O)N/N=C/c1ccc(o1)S(=O)(=O)O	CID:73707344	phase I
BRD-A37828317	CC(=O)O[C@@H]1C[C@@]2(C)[C@@H](C[C@H]3O[C@]32[C@@]4(C)C1[C@@]5(C)C=CC(=O)C(C)(C)C5C(=O)C4=O)c6ccoc6	CID:73707348	phase I
BRD-K08372451	ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)c2ccccc2	CID:73707349	phase I
BRD-K31041191	COc1ccc(Br)c(/C=N/NC(=O)CCCCCCC(=O)NO)c1	CID:73707350	phase I
BRD-K75081836	ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1[N+](=O)[O-]	CID:73707351	phase I
BRD-A14985772	CCCCCCCCCCCCCCCC(=O)OCC(O)[C@H]1OC(=O)C(=O)C1O	CID:73707359	phase I
BRD-K82857306	CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]2OC(=O)[C@@H](Cc3ccccc3)C\C=C\C[C@H](Cc3ccccc3)C(=O)O[C@@H]12	CID:73707364	phase I
BRD-A24396574	CC1C(=O)C(=O)C=C2C1=CC=C3[C@@]2(C)CCC4(C)[C@@H]5C[C@@](C)(CC[C@]5(C)CC[C@]34C)C(=O)O	CID:73707365	phase I
BRD-K90610876	COc1ccc(cc1)C(COCCN2CCC[C@@H](C2)C(=O)O)(c3ccc(OC)cc3)c4ccc(OC)cc4	CID:73707366	phase I
BRD-K40949493	C[C@H](CO)N1C[C@H](C)[C@@H](CN(C)Cc2ccc(Cl)c(Cl)c2)Oc3ccc(NC(=O)CCCCCC(=O)Nc4ccccc4N)cc3C1=O	CID:73707367	phase I
BRD-K96640811	O=C(N1CCCNCC1)c2cccc3cnccc23	CID:73707370	phase I
BRD-K09907482	Brc1ccc(OCc2ccccc2Br)c(/C=C\3/SC(=S)NC3=O)c1	CID:73707371	phase I
BRD-K30677119	CC(C)n1nc(-c2cccc(c2)C(=O)NC2=NCCC2)c2c(N)ncnc12	CID:73707372	phase I
BRD-K18190982	NC(=C)c1cc2c(cnc(N)c2s1)-c1cccc(c1)-c1ccccc1	CID:73707373	phase I
BRD-A23770159	CO[C@@H]1CC(CC(C)[C@@H]2CC(=O)[C@H](C)\C=C(C)\[C@@H](O)[C@@H](OC)C(=O)[C@@H](C)C[C@H](C)\C=C\C=C\C=C(C)/[C@H](C[C@@H]3CC[C@@H](C)[C@@](O)(O3)C(=O)C(=O)N3CCCC[C@H]3C(=O)O2)OC)CC[C@H]1O	CID:73707374	phase I
BRD-K79382620	CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1CCC[C@@H]1C(=O)Nc1cccc2ncccc12	CID:73707375	phase I
BRD-K79983625	COC(OC)[C@]12O[C@@H]3[C@H](O1)[C@@](O)(Oc1c3c(C)cc3c(OC)c4[C@@H](O)C[C@H](O)C(=O)c4c(O)c13)[C@@]21CO1	CID:73707376	phase I
BRD-K84924563	N[C@@H](CCC(=O)C[N+]#N)C(O)=O	CID:73707377	phase I
BRD-K80527266	CCC\C=C\C\C=C\C=C\C=N\N[NH2+][O-]	CID:73707378	phase I
BRD-A63646118	CCCC[C@@H](C)[C@@H](OC(=O)C[C@@H](CC(O)=O)C(O)=O)[C@H](CC(C)C[C@H](O)CCCC[C@@H](O)C[C@H](O)[C@H](C)N)OC(=O)C[C@@H](CC(O)=O)C(O)=O	CID:73707380	phase I
BRD-K41087962	COC(OC)[C@]12O[C@@H]3[C@H](O1)[C@@](O)(Oc1c3c(C)cc3c(OC)c4CCCC(=O)c4c(O)c13)[C@@]21CO1	CID:73707381	phase I
BRD-A76279427	CCCCCCC(=O)CCCCCC\C=C\C[C@H](O)[C@@H](O)C(N)(CO)C(O)=O	CID:73707382	phase I
BRD-A06304526	COC1CC(C)CC2=C(NCCN(C)C)C(=O)C=C(NC(=O)\C(C)=C\C=C\C(OC)C(OC(N)=O)\C(C)=C\C(C)C1O)C2=O	CID:73707383	phase I
BRD-A61304759	COC1CC(C)CC2=C(NCC=C)C(=O)C=C(NC(=O)\C(C)=C\C=C\C(OC)C(OC(N)=O)\C(C)=C\C(C)C1O)C2=O	CID:73707384	phase I
BRD-K29830875	COC(=O)[C@@H]1[C@H](C(O)=O)[C@]2([C@H](N1C)c1ccccc1)C(=O)N(C(=O)NCc1ccccc1)c1ccc(cc21)C#Cc1ccc(OC)cc1	CID:73707385	phase I
BRD-K49456190	COC[C@]1(CO)[N@@]2CC[C@@H](CC2)C1=O	CID:73707386	phase I
BRD-K55301415	C[C@]12CC[C@@H]3[C@@H](CC=C4C[C@@H](O)CC[C@@]34C)[C@@H]1CC=C2c1cccnc1	CID:73707387	phase I
BRD-K42125900	CC(=O)O[C@]12CO[C@@H]1C[C@H](O)[C@]1(C)[C@@H]2[C@H](OC(=O)c2ccccc2)[C@]2(O)C[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c3ccccc3)C(C)=C([C@@H](O)C1=O)C2(C)C	CID:73707388	phase I
BRD-K35687265	COc1cc(OC)c(\C=C\S(=O)(=O)Cc2ccc(OC)c(NCC=O)c2)c(OC)c1	CID:73707390	phase I
BRD-A41250203	COc1cc(\C=C\C(=O)N2C(CC=CC2=O)c2cccnc2)cc(OC)c1OC	CID:73707393	phase I
BRD-A63583287	COc1cc(\C=C\C(=O)N2C(CC=CC2=O)C2CCCCC2)cc(OC)c1OC	CID:73707394	phase I
BRD-A17016119	COC(=O)[C@H](Cc1ccccc1)NC(=O)C(\c1ccccc1)=C1/OC(=O)C(C1=O)c1ccccc1	CID:73707395	phase I
BRD-A47829399	C[C@@H]1CC[C@H]2[C@@H](C)C(OC(=O)CCC(O)=O)OC3O[C@]4(C)CC[C@@H]1[C@@]23OO4	CID:73707396	phase I
BRD-K83336168	COc1cc(\C=C\C(=O)N2CCC=CC2=O)cc(OC)c1OCCN(C)CCOc1c(OC)cc(\C=C\C(=O)N2CCC=CC2=O)cc1OC	CID:73707398	phase I
BRD-K14229306	O[C@H]1COC[C@H]2O[C@H](CC(=O)Nc3ccc(cc3)-c3ccccc3)CC[C@@H]2N(C1)C(=O)c1cccnc1	CID:73707399	phase I
BRD-K72996713	O[C@H]1COC[C@H]2O[C@H](CC(=O)N3CCc4ccccc4C3)CC[C@@H]2N(Cc2ccccc2F)C1	CID:73707400	phase I
BRD-A28105619	CC(C)(O)\C=C\C(=O)[C@](C)(O)C1[C@H](O)C[C@@]2(C)C3CC=C4C(CC(=O)C(=O)C4(C)C)[C@]3(C)C(=O)C[C@]12C	CID:73707401	phase I
BRD-A69951442	C[C@@H]1CC2C3CCC4=CC(=O)C=CC4(C)[C@]3(F)[C@@H](O)CC2(C)[C@]1(O)C(=O)CO	CID:73707402	phase I
BRD-A81936046	CO[C@H]1C2OP(O)(=O)OC[C@H]2O[C@H]1n1c(Sc2ccc(Cl)cc2)nc2c(N)ncnc12	CID:73707403	phase I
BRD-A77216878	CCCC[C@@H](C)\C=C(C)\C=C(/C)C(=O)NC1=C[C@@](O)(\C=C\C=C\C=C\C(=O)NC2C(=O)CCC2=O)[C@@H]2OC2C1=O	CID:73707404	phase I
BRD-K02822062	COc1cc(cc(OC)c1OCCN1CCOCC1)\C=C\C(=O)N1CCCCC1=O	CID:73707405	phase I
BRD-K50691590	CC(C)C[C@@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)C1=CNC=CN1)B(O)O	CID:73707406	phase I
BRD-K14550461	CC(C)[C@@H](C)\C=C\[C@@H](C)[C@@H]1CC[C@H]2[C@@]1(C)CCC\C2=C/C=C1/C[C@@H](O)C[C@H](O)C1=C	CID:73707407	phase I
BRD-K12002134	CC(=O)O[C@]1(CC[C@@H]2[C@H]3C=C(C)C4=CC(=O)CC[C@@]4(C)[C@@H]3CC[C@@]12C)C(C)=O	CID:73707408	phase I
BRD-K10916986	CCC1=C[C@@H]2C[N@](C1)Cc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C)[C@@H]1[C@]22CCN3CC=C[C@@](CC)([C@@H]23)[C@@H](OC(C)=O)[C@]1(O)C(=O)OC	CID:73707409	phase I
BRD-K64935403	CC[C@@H](C)[C@@H](O)[C@H](C)C(=O)[C@H](C)\C=C(/C)C[C@H](C)[C@H]1OC(=O)[C@H]1CC	CID:73707410	phase I
BRD-A67438293	CCCCC[C@H](O)CC[C@H]1[C@H](O)CC2Cc3c(C)cccc3CC12	CID:73707411	phase I
BRD-K14791739	CCC(=O)O[C@]1([C@H](C)C[C@@H]2[C@H]3C[C@H](F)C4=CC(=O)C=C[C@@]4(C)[C@]3(F)[C@@H](O)C[C@@]12C)C(=O)SCF	CID:73707412	phase I
BRD-K46503544	COc1cc(cc(OC)c1O)[C@H]1[C@H]2[C@@H](COC2=O)[C@H](O[C@@H]2O[C@@H]3CO[C@@H](C)O[C@H]3[C@H](O)[C@H]2O)c2cc3OCOc3cc12	CID:73707413	phase I
BRD-K60460488	Cc1c(O)cccc1C(=O)N[C@@H](CSc1ccccc1)[C@H](O)CN1C[C@@H]2CCCC[C@@H]2C[C@H]1C(=O)NC(C)(C)C	CID:73707414	phase I
BRD-K90543092	CC[C@@]12CC[C@@H]3[C@H](CCC4=CC(=O)CC[C@@H]34)[C@H]1CC[C@@]2(O)C#C	CID:73707415	phase I
BRD-A36707673	CC(C)[C@H](O)CCC(C)C1CCC2C3CC=C4C[C@@H](O)CC[C@@]4(C)C3CC[C@@]12C	CID:73707416	phase I
BRD-A52193669	CC([C@H]1CC[C@@H]2[C@H]3C[C@H]4O[C@@]44[C@@H](O)C=CC(=O)[C@@]4(C)C3CC[C@@]12C)[C@@H]1CC(C)=C(CO)C(=O)O1	CID:73707417	phase I
BRD-A80960055	CC1C(=O)C(=O)C=C2C1=CC=C1[C@]2(C)CC[C@]2(C)[C@H]3C[C@](C)(CC[C@@]3(C)CC[C@@]12C)C(O)=O	CID:73707418	phase I
BRD-A11702965	CO[C@@H]([C@H]1Cc2cc3cc(OC4CC(OC5CC(O)C(OC)C(C)O5)C(OC(C)=O)C(C)O4)c(C)c(O)c3c(O)c2C(=O)[C@H]1OC1CC(OC2CC(OC3CC(C)(O)C(C)C(C)O3)C(O)C(C)O2)C(O)C(C)O1)C(=O)[C@@H](O)[C@@H](C)O	CID:73707419	phase I
BRD-K32710582	O[C@H](c1ccc2ccccc2c1)P(O)(O)=O	CID:73707420	phase I
BRD-A79237180	CCCCCCCCCCCCCCCC(=O)OC[C@H](O)[C@@H]1OC(=O)C(=O)C1O	CID:73707421	phase I
BRD-A59808129	C\C=C1/C(=O)CC2C3CCC4=CC(=O)CC[C@@]4(C)C3CC[C@@]12C	CID:73707425	phase I
BRD-K93433262	CC(C)CCC[C@@H](C)[C@@H]1CC[C@H]2[C@@]1(C)CCC\C2=C/C=C1/C[C@@H](O)C[C@H](O)C1=C	CID:73707426	phase I
BRD-A84327315	CC(CCCC(C)(C)O)C1CCC2\C(CCC[C@@]12C)=C/C=C1/CC(O)C[C@H](O)C1=C	CID:73707427	phase I
BRD-A32161980	CCC(C)[C@H]1NC(=O)[C@H](Cc2ccc(OC)cc2)NC(=O)CCCSC[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](CCC(N)=O)NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(N)=O)C(C)(C)C	CID:73707428	phase I
BRD-A94793051	CC[C@]1(O)CCC2[C@@H]3CCC4=CC(=O)CCC4=C3C=C[C@@]12CC	CID:73707430	phase I
BRD-A43805296	CCC(C)C(NC(=O)C(C)NC)C(=O)N1CCCC1C(=O)NC1CCCc2ccccc12	CID:73707433	phase I
BRD-K03339442	COC(Cc1cccc2ccccc12)=C(C#N)C#N	CID:73707434	phase I
BRD-K77876724	CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)CCNC(C)=O)C(C)C)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]2CCCN2C(=O)[C@H](CCSC)NC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(N)=O	CID:73707435	phase I
BRD-K32737443	CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)CCNC(C)=O)C(C)C)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCSC)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(N)=O	CID:73707436	phase I
BRD-K45878950	CCCC[C@@H]1NC(=O)[C@@](C)(CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)CCNC(C)=O)C(C)C)[C@@H](C)CC	CID:73707437	phase I
BRD-K58306044	CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CCNC(C)=O)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCSC)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O	CID:73707438	phase I
BRD-K71199328	CCCC[C@@H]1NC(=O)[C@@](C)(CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CCNC(C)=O)[C@@H](C)CC	CID:73707439	phase I
BRD-K20514654	CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CCNC(C)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(O)=O)NC1=O)C(=O)N[C@@H](CCCNC(N)=N)C(N)=O	CID:73707440	phase I
BRD-K22507586	CCCC[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CCNC(C)=O)[C@@H](C)CC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(O)=O)NC1=O)C(=O)N[C@@H](CCCNC(N)=N)C(N)=O	CID:73707441	phase I
BRD-K55473186	CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(O)=O)NC(=O)CCNC(C)=O)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CS)NC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(N)=O	CID:73707442	phase I
BRD-K83932973	CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCNC(C)=O)C(=O)N[C@]1(C)CCC\C=C/CCC[C@@](C)(NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CS)NC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(N)=O	CID:73707443	phase I
BRD-K79873567	CC(C)[C@H]1c2ccc(F)cc2CC[C@@]1(CCN(C)CCCc1nc2ccccc2[nH]1)OC(=O)CCCC#C	CID:73707444	phase I
BRD-A63445921	COC(=O)C1=C(C)N=C(C)C(C1c1cccc(c1)[N+]([O-])=O)C(=O)OCCN(C)Cc1ccccc1	CID:73707445	phase I
BRD-A34462049	CN(C)[C@H]1[C@@H]2C[C@@H]3Cc4c(cc(NC(=O)CNC(C)(C)C)c(O)c4C(=O)C3C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O)N(C)C	CID:73707446	phase I
BRD-K36760124	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O[C@H]1C[C@H](O)[C@H](O[C@H]2C[C@H](OC(C)=O)[C@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[C@@H](C)O2)[C@@H](C)O1)O[C@H]1CC[C@@]2(C)[C@@H](CC[C@H]3[C@@H]2C[C@@H](O)[C@]2(C)[C@H](CC[C@]32O)C2=CC(=O)OC2)C1	CID:73707447	phase I
BRD-K04497194	C[C@H](CCC(O)=O)[C@@H]1CC[C@H]2[C@@H]3CC[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]12C	CID:73707448	phase I
BRD-K13688115	C[C@H]1C[C@H]2[C@H]3CC[C@H](C(C)=O)[C@@]3(C)C[C@H](O)[C@H]2[C@@]2(C)CCC(=O)C=C12	CID:73707449	phase I
BRD-A56470328	CC(=O)OCC(=O)[C@@]1(O)CC[C@H]2[C@H]3CCC4=CC(=O)CC[C@]4(C)C3(F)[C@@H](O)C[C@]12C	CID:73707451	phase I
BRD-K80110068	C[C@]12CC(=O)[C@@H]3[C@H](CCC4=CC(=O)CC[C@]34C)[C@@H]1CC[C@]2(O)C(=O)CO	CID:73707452	phase I
BRD-A51294525	CC(=O)O[C@@]1(CC[C@@H]2[C@@H]3C=C(Cl)C4=CC(=O)C5CC5[C@]4(C)[C@@H]3CC[C@]12C)C(C)=O	CID:73707455	phase I
BRD-A68650781	C[C@]12CC[C@@H]3[C@@H](CC[C@@H]4CC5SC5C[C@]34C)[C@@H]1CC[C@@H]2O	CID:73707456	phase I
BRD-K55113501	C[C@@]12[C@H](CC[C@]1(O)[C@H]1CC[C@H]3C[C@@H](O)CC[C@]3(C)[C@H]1C[C@H]2O)C1=CC(=O)OC1	CID:73707458	phase I
BRD-A15597386	CC(=C)[C@H]1[C@H]2OC(=O)C1[C@]1(O)CC3O[C@]33C(=O)O[C@@H]2[C@]13C	CID:73707459	phase I
BRD-A60052764	Cc1onc(c1C(=O)N[C@H]1[C@@H]2SC(C)(C)C(N2C1=O)C(O)=O)-c1c(F)cccc1Cl	CID:73707461	phase I
BRD-K08727137	CC(=O)OCC(=O)[C@H]1CC[C@H]2[C@H]3CC[C@H]4C[C@H](O)CC[C@]4(C)[C@@H]3C(=O)C[C@]12C	CID:73707462	phase I
BRD-A76229785	CN(C)[C@H]1[C@@H]2C[C@@H]3C(C(=O)c4c(O)cccc4[C@@]3(C)O)C(=O)[C@]2(O)C(=O)C(C(=O)NCNC(CCCCN)C(O)=O)C1=O	CID:73707463	phase I
BRD-K87210992	CC(=O)O[C@H]1[C@H](C[C@H]2[C@H]3CC[C@H]4C[C@H](OC(C)=O)[C@H](C[C@]4(C)[C@@H]3CC[C@]12C)[N+]1(C)CCCCC1)[N+]1(C)CCCCC1	CID:73707464	phase I
BRD-K92923799	C[C@]12CC[C@H]3[C@H](CC[C@H]4C[C@@H](O)CC[C@]34C)[C@@]1(O)CC[C@@H]2C1=CC(=O)OC1	CID:73707465	phase I
BRD-K40476324	C[C@H]1O[C@H](C[C@H](O)[C@@H]1O)O[C@H]1[C@@H](O)C[C@H](O[C@H]2[C@@H](O)C[C@H](O[C@H]3CC[C@@]4(C)[C@@H](CC[C@H]5[C@@H]4C[C@@H](O)[C@]4(C)[C@H](CC[C@]54O)C4=CC(=O)OC4)C3)O[C@@H]2C)O[C@@H]1C	CID:73707466	phase I
BRD-K28026280	CCC(C)(C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@H]12	CID:73707467	phase I
BRD-K74615293	C[C@@H](O)[C@H]1[C@H]2[C@@H](C)C(S[C@@H]3CN[C@@H](C3)C(=O)N(C)C)=C(N2C1=O)C(O)=O	CID:73707470	phase I
BRD-K53342282	CC(=O)OCC(=O)[C@@]1(O)CC[C@@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3[C@@H](O)C[C@]12C	CID:73707472	phase I
BRD-A58837096	NC[C@H]1O[C@H](OC2[C@@H](N)C[C@@H](N)[C@H](O)[C@@H]2O[C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)[C@H](N)[C@@H](O)[C@@H]1O	CID:73707473	phase I
BRD-K72853990	CC(C)C[C@@H]1N2C(=O)[C@](NC(=O)[C@H]3CN(C)[C@H]4Cc5c(Br)[nH]c6cccc(C4=C3)c56)(O[C@@]2(O)[C@H]2CCCN2C1=O)C(C)C	CID:73707474	phase I
BRD-A33070992	CCOC(=O)OC(C)OC(=O)[C@@H]1N2[C@@H](SC1(C)C)[C@H](NC(=O)[C@H](N)c1ccccc1)C2=O	CID:73707475	phase I
BRD-K69260336	CC(C)(C)C(=O)OCOC(=O)[C@@H]1N2[C@@H](SC1(C)C)[C@H](NC(=O)[C@H](N)c1ccccc1)C2=O	CID:73707476	phase I
BRD-K54978501	CC(C)(C)C(=O)OCOC(=O)[C@@H]1N2[C@@H](SC1(C)C)[C@H](N=CN1CCCCCC1)C2=O	CID:73707477	phase I
BRD-K95391106	CCOC(=O)O[C@@]1(CC[C@@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@]12C)C(=O)COC(=O)CC	CID:73707478	phase I
BRD-K27218697	CCC(=O)[C@@]1(C)[C@H](C)C[C@@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@]12C	CID:73707479	phase I
BRD-K57943804	C[C@]12CC[C@@H]3C(=CCc4cc(O)ccc34)[C@H]1CCC2=O	CID:73707480	phase I
BRD-A20794617	CN[C@H](CC(C)C)C(=O)N[C@@H]1[C@H](O)c2ccc(Oc3cc4cc(Oc5ccc(cc5Cl)[C@@H](O)[C@H]5NC(=O)[C@@H](NC(=O)[C@@H]4NC(=O)[C@H](CC(N)=O)NC1=O)c1ccc(O)c(c1)-c1c(O)cc(O)cc1[C@H](NC5=O)C(O)=O)c3O[C@@H]1OC(CO)[C@@H](O)[C@H](O)[C@H]1O[C@H]1C[C@](C)(N)[C@H](O)[C@H](C)O1)c(Cl)c2	CID:73707482	phase I
BRD-K45770447	C[C@@H]1CC[C@@H]2[C@@H](C)C(=O)O[C@H]3O[C@@]4(C)CC[C@@H]1[C@@]23OO4	CID:73707483	phase I
BRD-A10606614	CC1(C)S[C@H]2[C@H](NC(=O)[C@H](N)c3ccccc3)C(=O)N2[C@H]1C(=O)OC1OC(=O)c2ccccc12	CID:73707484	phase I
BRD-A51233382	CCOC1O[C@@H]([C@@H](COCc2ccccc2)OCc2ccccc2)[C@H](OCc2ccccc2)[C@H]1O	CID:73707485	phase I
BRD-K62997315	C[C@H](CCC(O)=O)[C@@H]1CC[C@H]2[C@H]3[C@@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@@H]3CC[C@]12C	CID:73707486	phase I
BRD-A39671870	CN1[C@H]2CC[C@H]1C[C@H](C2)OC(=O)C(O)c1ccccc1	CID:73707487	phase I
BRD-A58753560	CCCC1O[C@@H]2C[C@H]3[C@H]4CCC5=CC(=O)C=C[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:73707488	phase I
BRD-K43544024	C[C@]1(O)CC[C@@H]2[C@@H]3CC[C@H]4CC(=O)OC[C@]4(C)[C@@H]3CC[C@]12C	CID:73707489	phase I
BRD-K59850506	CC[C@]12C=CC3=C4CCC(=O)C=C4CC[C@H]3[C@H]1CC[C@@]2(O)C#C	CID:73707492	phase I
BRD-K30618791	CC(=O)O[C@@]12CO[C@H]1C[C@H](O)[C@]1(C)[C@H]2[C@H](OC(=O)c2ccccc2)[C@@]2(O)C[C@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c3ccccc3)C(C)=C([C@@H](O)C1=O)C2(C)C	CID:73707494	phase I
BRD-K11700078	CN(C)CCCO[C@H]1[C@@H](O[C@@H]2OC(C)(C)O[C@@H]12)[C@H](O)CO	CID:73707495	phase I
BRD-K93923542	C[C@]12CC[C@@H]3[C@@H](CC(=C)C4=CC(=O)C=C[C@]34C)[C@H]1CCC2=O	CID:73707497	phase I
BRD-A52997285	CN(C)[C@H]1[C@@H]2C[C@@H]3C(C(=O)c4c(O)cccc4[C@@]3(C)O)C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O	CID:73707498	phase I
BRD-A99314711	NC[C@@H]1O[C@H](O[C@@H]2[C@@H](CO)O[C@@H](O[C@@H]3[C@@H](O)[C@H](N)C[C@H](N)[C@@H]3OC3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3N)[C@@H]2O)[C@H](N)[C@@H](O)[C@@H]1O	CID:73707499	phase I
BRD-A42153648	C[C@]12CC[C@@H]3[C@@H](CCC4C(=O)C(=O)CC[C@]34C)[C@H]1CCC2=O	CID:73707500	phase I
BRD-A17828570	C[C@]12CC[C@H]3[C@@H]([C@H]1CC[C@@H]2O)[C@H](CCCCCCCCCS(=O)CCCC(F)(F)C(F)(F)F)Cc1cc(O)ccc31	CID:73707501	phase I
BRD-K86858124	CC(=O)O[C@@H]1C2=C(C)[C@H](C[C@@](O)([C@@H](OC(=O)c3ccccc3)[C@H]3[C@@]4(CO[C@H]4C[C@H](O)[C@@]3(C)C1=O)OC(C)=O)C2(C)C)OC(=O)[C@H](O)[C@@H](NC(=O)c1ccccc1)c1ccccc1	CID:73707502	phase I
BRD-A28019035	C[C@]12CCC3[C@@H](CC[C@@H]4C[C@H](O)CC[C@]34C)[C@H]1CCC2=O	CID:73707504	phase I
BRD-A14652656	CCCC(=O)Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2OP(O)(=O)OC[C@@H]2[C@H]1OC(=O)CCC	CID:73707507	phase I
BRD-K79224779	C[C@]12CC[C@H]3[C@@H](CCC4=CCCC[C@H]34)[C@H]1CC[C@@]2(O)C#C	CID:73707508	phase I
BRD-K58746048	CC1(C)O[C@@H]2C[C@H]3[C@H]4C[C@H](F)C5=CC(=O)CC[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO	CID:73707509	phase I
BRD-A63934767	CCC(=O)OCC(=O)C1(OC(=O)CC)[C@H](C)C[C@H]2[C@H]3[C@H](Cl)CC4=CC(=O)C=C[C@]4(C)[C@@H]3[C@@H](O)C[C@]12C	CID:73707510	phase I
BRD-K96006502	CC(=O)OCC(=O)[C@@]12N=C(C)O[C@@H]1C[C@H]1[C@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@]21C	CID:73707512	phase I
BRD-K59946044	CC(C)CC(=O)O[C@H]1[C@@H](O[C@@H]2C[C@H]([C@@H]3CC[C@@]45C[C@H](CC[C@@H]4[C@]3(C)C2)C(=C)[C@@H]5O)C(O)=O)O[C@H](CO)[C@@H](OS(O)(=O)=O)[C@@H]1OS(O)(=O)=O	CID:73707514	phase I
BRD-A72130500	CN(C)[C@H]1[C@@H]2C[C@H]3[C@H](O)c4c(Cl)ccc(O)c4C(=O)C3C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O	CID:73707518	phase I
BRD-A39210489	CN(C)[C@H]1[C@@H]2C[C@@H]3C(C(=O)c4c(O)ccc(Cl)c4[C@@]3(C)O)C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O	CID:73707519	phase I
BRD-K11451237	C[C@@H]1O[C@@H](O[C@H]2CC[C@]3(C)[C@H]4CC[C@]5(C)[C@H](CC[C@]5(O)[C@H]4CCC3=C2)c2ccc(=O)oc2)[C@H](O)[C@H](O)[C@H]1O	CID:73707522	phase I
BRD-K91511962	C[C@]12CC[C@@H]3[C@H](CCC4=CC(=O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)CO	CID:73707523	phase I
BRD-K79199004	C[C@]1(O)CC[C@@H]2[C@@H]3CC[C@H]4Cc5[nH]ncc5C[C@]4(C)[C@@H]3CC[C@]12C	CID:73707524	phase I
BRD-A59431241	NC(=O)C1C(=O)C[C@@H]2C[C@@H]3Cc4cccc(O)c4C(=O)C3C(=O)[C@]2(O)C1=O	CID:73707525	phase I
BRD-K59873006	C[C@H]1O[C@@H](C[C@H](O)[C@@H]1O)O[C@H]1[C@@H](O)C[C@@H](O[C@H]2[C@@H](O)C[C@@H](O[C@H]3CC[C@@]4(C)[C@H](CC[C@@H]5[C@@H]4CC[C@]4(C)[C@H](CC[C@]54O)C4=CC(=O)OC4)C3)O[C@@H]2C)O[C@@H]1C	CID:73707526	phase I
BRD-A88765664	C[C@@]12CC[C@@H]3[C@@]4(C)C=CC(=O)C(C)(C)C4C(=O)C(=O)[C@@]3(C)[C@]11O[C@@H]1C[C@H]2c1ccoc1	CID:73707527	phase I
BRD-A16998493	CCC1C=CC=C2C1=NC1=C2CCOC1(CC)CC(O)=O	CID:73707528	phase I
BRD-K29385665	COc1ccc(N(C(=O)Oc2cc(ccc2C)C(=O)Nc2cccc(c2)C(F)(F)F)c2ccnc(Nc3ccc(cc3)N3CCN(C)CC3)n2)c(OC)c1	CID:73707529	phase I
BRD-K72636697	Cc1ccc(cc1NC(=O)C=C)-n1c2c(ccc1=O)cnc1ccc(cc21)-c1cn[nH]c1	CID:73707530	phase I
BRD-K43568579	COc1cc(OC)c(Cl)c(NC(=O)N(Cc2ccc(NC(=O)C=C)cc2)c2cc(Nc3ccc(cc3)N3CCN(C)CC3)ncn2)c1Cl	CID:73707531	phase I
BRD-K52721289	COc1cc(ccc1Nc1nc(N)c(s1)C(=O)c1ccc(NC(=O)C=C)cc1)N1CCN(C)CC1	CID:73707532	phase I
BRD-K38113518	CN(C)C\C=C\C(=O)Nc1cccc(Nc2ncc3N(C)C(=O)c4ccccc4N(C)c3n2)c1	CID:73707533	phase I
BRD-K29358067	Clc1ccccc1OCCc1nn2c(COc3ccccc3)nnc2s1	CID:73707534	phase I
BRD-K41179159	ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1ccccn1	CID:73707535	phase I
BRD-K65031973	Cc1ccccc1-c1ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc1	CID:73707536	phase I
BRD-A54024781	CN1c2ccccc2C(NCCCCCCC(=O)NO)c2ccc(Cl)cc2S1(=O)=O	CID:73707537	phase I
BRD-K78689929	CC(=O)Nc1ccc(cc1)C(=O)Nc1cc(ccc1O)-c1cccs1	CID:73707538	phase I
BRD-K08135697	Nc1ccccc1NC(=O)c1cnc(Nc2ccccc2)nc1	CID:73707542	phase I
BRD-K46918889	ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1ccncc1	CID:73707543	phase I
BRD-K97869369	ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1cncnc1	CID:73707544	phase I
BRD-K85732814	ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1cccs1	CID:73707545	phase I
BRD-A47268303	CC(=C)[C@@H](CC=C(C)C)C[C@]12C[C@H](CC=C(C)C)C(C)(C)[C@](CC=C(C)C)(C(=O)C(C(=O)c3ccc(O)c(O)c3)C1=O)C2=O	CID:73707546	phase I
BRD-K66198023	CCCCc1nc(Cl)c(CO)n1Cc1ccc(cc1)-c1ccccc1C1=NNNN1	CID:73707547	phase I
BRD-K55914420	CN(C(C)=O)c1ccc(cc1)C(=O)Nc1ccccc1N	CID:73707548	phase I
BRD-A73972952	CN1c2ccccc2C(NCCCCCCC(=O)Nc2ccccc2N)c2ccc(Cl)cc2S1(=O)=O	CID:73707549	phase I
BRD-K51966546	ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1cccnc1	CID:73707550	phase I
BRD-K39172790	NCCc1cc(O)c(O)c(SC[C@@H](N)C(O)=O)c1	CID:73707552	phase I
BRD-K54472228	N[C@@H](CSc1cc(CCOO)cc(O)c1O)C(O)=O	CID:73707553	phase I
BRD-A92334183	NC(Cc1ccc(O)c(O)c1)C(=O)NCCCC(O)=O	CID:73707554	phase I
BRD-A86146706	NC(Cc1cc(O)c(O)c(Cl)c1)C(O)=O	CID:73707555	phase I
BRD-K47535255	CCOC(=O)NCCc1ccc(OC(=O)OCC)c(OC(=O)OCC)c1	CID:73707556	phase I
BRD-A09053961	NC(Cc1cc(O)c(O)cc1Cl)C(O)=O	CID:73707557	phase I
BRD-A29342309	NC(COO)c1cc(O)cc(O)c1	CID:73707559	phase I
BRD-K53888148	CN(C)Cc1ccccc1Sc1ccc(cc1N)[N+]#[C-]	CID:73707560	phase I
BRD-K63835783	CNCc1ccccc1Sc1ccc(cc1N)[N+]#[C-]	CID:73707561	phase I
BRD-K03608458	Oc1ccccc1C[C@H]([C@H]1OCCNC1)c1ccccc1	CID:73707562	phase I
BRD-A40163033	CCC(C)(N)CCS(C)(=N)=O	CID:73707563	phase I
BRD-K34722304	C[C@@]12N[C@@H](Cc3ccccc13)c1ccc(I)cc21	CID:73707574	phase I
BRD-K29064493	C[C@@]12N[C@@H](Cc3ccccc13)c1ccc(cc21)[Si](C)(C)C	CID:73707575	phase I
BRD-A39986918	C[C@]12NC(Cc3ccccc13)c1ccc(I)cc21	CID:73707576	phase I
BRD-K65213718	C[C@]12N[C@H](Cc3ccccc13)c1ccc(cc21)[Si](C)(C)C	CID:73707577	phase I
BRD-A69454249	COc1cc(CC(C)(N)C(O)=O)ccc1OS(O)(=O)=O	CID:73707579	phase I
BRD-K10939925	CCCC(=O)Sc1ccc(cc1)[C@@H]1CN2CCC[C@@H]2c2ccccc12	CID:73707580	phase I
BRD-K82326223	CCCN(CC#C)[C@H]1CCc2cccc(O)c2C1	CID:73707582	phase I
BRD-A92148199	CCOC(=O)C(CC(C)C)NC(=O)C(CC(C)(C)C)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C1CCCN1C(=O)C(CCCCN)NC(=O)C(N)CCCCN	CID:73707583	phase I
BRD-K43631199	OONc1ccc2nc(ccc2c1I)N1CCNCC1	CID:73707584	phase I
BRD-K33943862	Nc1ccc(CCNC(=O)[C@@H]2[C@@H](O)CC[C@@H]3CN4CCc5c([nH]c6ccccc56)[C@@H]4C[C@H]23)cc1	CID:73707585	phase I
BRD-K63124331	CCCc1c[nH]c2ccc(CS(O)(=O)=O)cc12	CID:73707586	phase I
BRD-K52436943	Cc1ccc(Cn2nc(cc2-c2ccc(Cl)c(C)c2)C(=O)N[C@H]2[C@]3(C)CC[C@H](C3)C2(C)C)cc1	CID:73707587	phase I
BRD-A12881497	NCCc1c[nH]c2ccc(OC3O[C@@H]([C@@H](O)[C@H](O)[C@H]3O)C(O)=O)cc12	CID:73707588	phase I
BRD-A75769921	COc1cc(N=[N+]=[N-])c(I)cc1C(=O)NC1CCN(Cc2ccccc2)C1C	CID:73707590	phase I
BRD-A11009626	CN1CCc2cc(Br)c(O)cc2C(C1)c1ccc(cc1)N(CCCl)CCCl	CID:73707591	phase I
BRD-A50984182	CCC(C)C(NCC(Cc1ccc(O)cc1)NC(=O)C1CCCN1C(=O)C(CCCNC(N)=N)NC(=O)C(CCCNC(N)=N)NC(=O)OC(C)(C)C)C(=O)NC(CC(C)C)C(O)=O	CID:73707593	phase I
BRD-K15181602	CN(C)CCOc1ccc(CCN)cc1OCCN(C)C	CID:73707594	phase I
BRD-A15100685	CC1O[C@@H](OCC2O[C@@H](O[C@H]3CC[C@@]4(C)C(CC[C@]5(C)C4CC=C4C6CC(C)(C)[C@H](C[C@@]6([C@H](O)C[C@@]54C)C(=O)O[C@@H]4OC(CO)[C@@H](O)[C@@H](O)[C@@H]4O[C@@H]4OC(C)[C@H](O[C@@H]5O[C@@H](CO)[C@H](O)[C@@H]5O)[C@@H](O[C@@H]5OC(CO)[C@@H](O)[C@@H](O)[C@@H]5O)[C@@H]4O)OC(=O)C(\CO)=C\CC[C@](C)(O[C@@H]4OC(C)[C@@H](OC(=O)C(\CO)=C\CCC(C)(O)C=C)[C@@H](O)[C@@H]4O)C=C)C3(C)C)[C@@H](NC(C)=O)[C@H](O)[C@@H]2O)[C@@H](O[C@@H]2OC[C@@H](O)[C@@H](O)[C@@H]2O)[C@H](O)[C@H]1O	CID:73707595	phase I
BRD-K59915259	CN(C)CCCN(c1ccccc1)c1cccc(Cl)c1	CID:73707596	phase I
BRD-K31344914	C[C@H](N)C(=O)N[C@@H](C)C(=O)NCCc1cc(O)c(O)cc1O	CID:73707597	phase I
BRD-K79052598	C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C(=O)NCCc1cc(O)c(O)cc1O	CID:73707598	phase I
BRD-A68802837	CS(=O)(=O)OC1C(O)[C@@H](CO)O[C@H]1n1cnc2c(N)nc(Cl)nc12	CID:73707599	phase I
BRD-A72322024	CCNC(=O)C1OC([C@@H](O)[C@H]1O)n1cnc2c(N)nc(NCCc3ccc(CCC(=O)NCCN)cc3)nc12	CID:73707600	phase I
BRD-K78787248	CN(C)c1ccccc1Sc1ccc(I)cc1N	CID:73707601	phase I
BRD-A02579693	COc1cc(cc(OC)c1O)C1C2C(COC2=O)C(OC2OC3COC(C)OC3C(O)C2O)C2C1=CC1=C2OCO1	CID:73707602	phase I
BRD-A93291428	CC1(O)CCC2C3CCC4CC(=O)C(CC4(C)C3CCC12C)C=O	CID:73707603	phase I
BRD-A33746814	CC1O[C@@H](OCC2O[C@@H](O[C@H]3CC[C@@]4(C)C(CC[C@]5(C)C4CC=C4C6CC(C)(C)[C@H](C[C@@]6([C@H](O)C[C@@]54C)C(=O)O[C@@H]4OC(CO)[C@@H](O)[C@@H](O)[C@@H]4O[C@@H]4OC(C)[C@H](O[C@@H]5O[C@@H](CO)[C@H](O)[C@@H]5O)[C@@H](O[C@@H]5OC(CO)[C@@H](O)[C@@H](O)[C@@H]5O)[C@@H]4O)OC(=O)C(\CO)=C\CC[C@](C)(O[C@@H]4OC(C)[C@@H](OC(=O)C(\C)=C\CCC(C)(O)C=C)[C@@H](O)[C@@H]4O)C=C)C3(C)C)[C@@H](NC(C)=O)[C@H](O)[C@@H]2O)[C@@H](O[C@@H]2OC[C@@H](O)[C@@H](O)[C@@H]2O)[C@H](O)[C@H]1O	CID:73707604	phase I
BRD-A70150975	CC1O[C@@H](OCC2O[C@@H](O[C@H]3CC[C@@]4(C)C(CC[C@]5(C)C4[C@H](O)C=C4C6CC(C)(C)[C@H](C[C@@]6([C@H](O)C[C@@]54C)C(=O)O[C@@H]4OC(CO)[C@@H](O)[C@@H](O)[C@@H]4O[C@@H]4OC(C)[C@H](O[C@@H]5O[C@@H](CO)[C@H](O)[C@@H]5O)[C@@H](O[C@@H]5OC(CO)[C@@H](O)[C@@H](O)[C@@H]5O)[C@@H]4O)OC(=O)C(\CO)=C\CC[C@](C)(O[C@@H]4OC(C)[C@@H](OC(=O)C(\CO)=C\CCC(C)(O)C=C)[C@@H](O)[C@@H]4O)C=C)C3(C)C)[C@@H](NC(C)=O)[C@H](O)[C@@H]2O)[C@@H](O[C@@H]2OC[C@@H](O)[C@@H](O)[C@@H]2O)[C@H](O)[C@H]1O	CID:73707605	phase I
BRD-A69592287	CC1O[C@@H](OCC2O[C@@H](O[C@H]3CC[C@@]4(C)C(CC[C@]5(C)C4CC=C4C6CC(C)(C)[C@H](C[C@@]6([C@H](O)C[C@@]54C)C(=O)O[C@@H]4OC(CO)[C@@H](O)[C@@H](O)[C@@H]4O[C@@H]4OC(C)[C@H](O[C@@H]5O[C@@H](CO)[C@H](O)[C@@H]5O)[C@@H](O[C@@H]5OC(CO)[C@@H](O)[C@@H](O)[C@@H]5O)[C@@H]4O)OC(=O)C(\CO)=C\CC[C@](C)(O[C@@H]4OC(C)[C@@H](OC(=O)C5COC5CCC(C)(O)C=C)[C@@H](O)[C@@H]4O)C=C)C3(C)C)[C@@H](NC(C)=O)[C@H](O)[C@@H]2O)[C@@H](O[C@@H]2OC[C@@H](O)[C@@H](O)[C@@H]2O)[C@H](O)[C@H]1O	CID:73707606	phase I
BRD-K61691971	CC1(C)[C@@H]2C[C@]34CCCN3C(=O)[C@]2(NC4=O)C=C2c3cc4nccnc4cc3[N+]([O-])=C12	CID:73707607	phase I
BRD-K42573370	CC1(C)[C@@H]2C[C@]34CCCN3C(=O)[C@]2(NC4=O)C=C2c3ccc(cc3[N+]([O-])=C12)-c1ccccc1	CID:73707608	phase I
BRD-K39569857	CC1(C)[C@@H]2C[C@]34CCCN3C(=O)[C@]2(NC4=O)C=C2c3cc4OCOc4cc3[N+]([O-])=C12	CID:73707609	phase I
BRD-A70731303	CC1(C)Oc2cc3c(cc2C=C1)C1=CC24NC(=O)C5(CCCN5C2=O)CC4C(C)(C)C1=[N+]3[O-]	CID:73707610	phase I
BRD-K50324045	CC1(C)Oc2cc3c(cc2C=C1)C1=C[C@@]2(CC(C)(C)C1=[N+]3[O-])NC(=O)[C@@H]1CCCN1C2=O	CID:73707611	phase I
BRD-A17390249	CC(=O)Nc1ccc(cc1)C(=O)NC1CCCCC1N	CID:73707612	phase I
BRD-K49327517	CN(C)C\C=C\C(=O)Nc1cccc(c1)C(=O)Nc1cccc(Nc2nccc(n2)-c2cccnc2)c1	CID:73707613	phase I
BRD-A51696495	COc1ccc(CNC2CC2c2ccc(Br)cc2)c(Cl)c1OC	CID:73707614	phase I
BRD-K56060837	[2H]C([2H])([2H])C(=O)NC([2H])([2H])C([2H])([2H])c1c[nH]c2ccc(O)cc12	CID:73707615	phase I
BRD-K71451869	CC1(C)O[C@@H]2C[C@H]3[C@H]4CCC5=CC(=O)CC[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CCl	CID:73707616	phase I
BRD-K85903480	N[C@H](CCC(=O)NCCc1ccc(O)c(O)c1)C(O)=O	CID:73707617	phase I
BRD-K91614993	COc1cc(OCc2ccccc2)cc(OCc2ccccc2)c1CC(O)=O	CID:73707618	phase I
BRD-A87384553	O=C(NC(Cc1ccccc1)Cn1cc(CN2C(COCC2=O)c2ccccc2)nn1)Nc1ccccc1	CID:74169187	phase I
BRD-A68721828	CN/1C(C=C(C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CO)cc4)C5CC5	CID:74180475	phase I
BRD-A12560204	CCOC(=O)C1C(C(=C(C)N=C1C)C(=O)OC)c2cccc(c2)[N+](=O)[O-]	CID:78428958	phase I
BRD-A24891640	COCCOC(=O)C1C(C(=C(C)N=C1C)C(=O)OC(C)C)c2cccc(c2)[N+](=O)[O-]	CID:78435479	phase I
BRD-A27489425	CN(C)[C@H]1C2CC3C(C(=O)c4c(O)cccc4[C@@]3(C)O)C(=O)[C@]2(O)C(=O)C(C(=O)NCN5CCCC5)C1=O	CID:90843500	phase I
BRD-A41555725	CN(C)[C@H]1[C@@H]2CC3C(C(=O)c4c(O)ccc(Cl)c4[C@@]3(C)O)C(=O)[C@]2(O)C(=O)C(C(N)=O)C1=O	CID:91192474	phase I
BRD-A35519318	COC(=O)C1[C@H](C(=C(C)N=C1C)C(=O)O[C@@H]2CCCN(Cc3ccccc3)C2)c4cccc(c4)[N+](=O)[O-]	CID:91522200	phase I
BRD-K30545681	O=C1CCCC(=O)C1C(C#Cc2ccccc2)C3C(=O)CCCC3=O	CID:91896203	phase I
BRD-A52282606	CCOC(=O)C1C(C(=C(C)N=C1C)C(=O)OCC)c2ccccc2/C=C/C(=O)OC(C)(C)C	CID:124202151	phase I
BRD-K58662656	CON=C(C(=O)N[C@@H]1[C@H]2SCC(C[N+]3(C)CCCC3)=C(N2C1=O)C(O)=O)c1csc(N)n1	CID:124929724	phase I
BRD-K54283240	Nc1nc(cs1)C(=NOCC(O)=O)C(=O)N[C@@H]1[C@H]2SCC(C=C)=C(N2C1=O)C(O)=O	CID:124930437	phase I
BRD-K37187815	CON=C(C(=O)N[C@@H]1[C@H]2SCC(COC(N)=O)=C(N2C1=O)C(O)=O)c1ccco1	CID:125136590	phase I
BRD-K24576554	O=C(NC1CC1)Nc1c[nH]nc1-c1nc2cc(CN3CCOCC3)ccc2[nH]1	CID:135398495	phase I
BRD-K01253243	CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccc2c(CC\C2=N\O)c1)-c1ccncc1	CID:135398506	phase I
BRD-K08206212	Nc1nc(=O)c2ncn([C@H]3C[C@H](O)[C@@H](CO)C3=C)c2[nH]1	CID:135398508	phase I
BRD-K85402309	CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O	CID:135398510	phase I
BRD-K32318651	Nc1nc2n(COCCO)cnc2c(=O)[nH]1	CID:135398513	phase I
BRD-K48692744	Cc1nc2c(O)cccc2c(=O)[nH]1	CID:135398517	phase I
BRD-K81647657	Cn1cnc(=N)c2nc[nH]c12	CID:135398661	phase I
BRD-K01507359	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c(O)c(\C=N\N4CCN(C)CC4)c(NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c(O)c2c(O)c3C	CID:135398735	phase I
BRD-K37289225	CN1CCN(CC1)C1=Nc2cc(Cl)ccc2Nc2ccccc12	CID:135398737	phase I
BRD-K99063460	OC[C@@H]1CC[C@@H](O1)n1cnc2c(O)ncnc12	CID:135398739	phase I
BRD-K22662435	Nc1nc2n(COC(CO)CO)cnc2c(=O)[nH]1	CID:135398740	phase I
BRD-K46435977	CC(C)[C@H](N)C(=O)OCCOCn1cnc2c1nc(N)[nH]c2=O	CID:135398742	phase I
BRD-K50128260	CCCc1nn(C)c2c1[nH]c(nc2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(C)CC1	CID:135398744	phase I
BRD-K18895904	CN1CCN(CC1)C1=Nc2ccccc2Nc2sc(C)cc12	CID:135398745	phase I
BRD-K47780086	Nc1nc(O)c2ncn(CCC(CO)CO)c2n1	CID:135398748	phase I
BRD-K12516989	CCCOc1ccccc1c2nc3nn[nH]c3c(=O)[nH]2	CID:135399235	phase I
BRD-K58547240	COc1ccc2nc(Nc3nc(C)c(CCC(C)C)c(=O)[nH]3)nc(C)c2c1	CID:135399523	phase I
BRD-K89839824	CN(Cc1ccc2[nH]c(C)nc(=O)c2c1)c1ccc(s1)C(=O)N[C@@H](CCC(O)=O)C(O)=O	CID:135400182	phase I
BRD-K13926615	CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CC)CC1	CID:135400189	phase I
BRD-A54927599	COc1ccc(C2CC(=NCCS2)c2c(O)cc(C)oc2=O)c(OC)c1	CID:135400439	phase I
BRD-K78373679	O=C1N=C(NCc2cccs2)S\C1=C/c1ccc2ncccc2c1	CID:135400873	phase I
BRD-K69885235	COc1cc(\C=C2/SC(Nc3ccccc3Cl)=NC2=O)ccc1O	CID:135401109	phase I
BRD-K86307448	O=c1[nH]cnc2[nH]ncc12	CID:135401907	phase I
BRD-A75919782	Nc1nc(=O)c2N(C=O)C(CNc3ccc(cc3)C(=O)N[C@@H](CCC(O)=O)C(O)=O)CNc2[nH]1	CID:135403648	phase I
BRD-K21350491	Nc1nc(N)c(nc1Cl)C(=O)NC(=N)Nc2ccccc2	CID:135403792	phase I
BRD-A06726973	CCCC(=O)Nc1nc2n(cnc2c(=O)[nH]1)C3O[C@H]4COP(=O)(O)O[C@@H]4[C@@H]3OC(=O)CCC	CID:135403793	phase I
BRD-K77317635	COC(=O)NN=Cc1c[n+]([O-])c2ccccc2[n+]1[O-]	CID:135403805	phase I
BRD-K28346421	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c(O)c(\C=N\N4CCN(CC4)C4CCCC4)c(NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c(O)c2c(O)c3C	CID:135403821	phase I
BRD-K39208132	CCSc1nc(O)cc(n1)c2ccccc2	CID:135406353	phase I
BRD-K62200014	Clc1ccc2N=C3NC(=O)CN3Cc2c1Cl	CID:135409400	phase I
BRD-K21806131	CCCCC\N=C(/N)N\N=C\c1c[nH]c2ccc(OC)cc12	CID:135409453	phase I
BRD-K10042277	Clc1ccc2Nc3ccccc3C(=Nc2c1)N1CCNCC1	CID:135409468	phase I
BRD-K76425766	Oc1nc(SCc2ccc(Cl)cc2)nc3CCCc31	CID:135412054	phase I
BRD-K21971034	COc1cc(\C=N\NC(=O)c2sc(N)nc2C)ccc1O	CID:135412158	phase I
BRD-K52827117	C[C@@H](O[C@H]1OCCN(Cc2nc(=O)[nH][nH]2)[C@H]1c1ccc(F)cc1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F	CID:135413536	phase I
BRD-K41160163	CN1CC(=O)N=C1NC(=O)Nc1cccc(Cl)c1	CID:135413554	phase I
BRD-K12762134	Oc1nc(nc2CCSCc12)-c1ccc(cc1)C(F)(F)F	CID:135418940	phase I
BRD-K35035132	CC(=O)Nc1ccc(/C=C/c2noc(n2)c3ccccc3O)cc1	CID:135419176	phase I
BRD-K59469039	CC(C)(C)c1cc(cc(c1O)C(C)(C)C)\C=C(/C#N)C(N)=S	CID:135419190	phase I
BRD-K87403606	CNC1=Nc2ccc(Cl)cc2C(=NC1)c1ccc[nH]1	CID:135422895	phase I
BRD-K36977165	O=c1[nH]c(nc2ccccc12)N3CCCC3	CID:135423697	phase I
BRD-K48115423	COc1ccc(CSc2nc(C)cc(O)n2)cc1	CID:135438809	phase I
BRD-K30849099	COc1cc(/C=C\2/SC(=NC2=O)Nc3ccc(O)cc3)ccc1O	CID:135440086	phase I
BRD-K34581968	Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2cccc(Cl)c2)cc[nH]c1=O)N1CCOCC1	CID:135440466	phase I
BRD-K70161581	Oc1cccc(/C=N/NC(=O)c2ccccc2O)c1O	CID:135444127	phase I
BRD-K99912150	CO[C@H]1C=CO[C@@]2(C)Oc3c(C2=O)c4c(O)c(C=NN5CCN(C)CC5)c(NC(=O)C(=CC=C[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(=O)C)[C@@H]1C)C)c(O)c4c(O)c3C	CID:135449527	phase I
BRD-K33297438	Oc1nc(nc2ccccc12)c3ccc(o3)c4cccc(Cl)c4	CID:135452687	phase I
BRD-K71746704	CCOC(=O)CCc1cnccc1c2cccc(OC)c2O	CID:135453978	phase I
BRD-K82837433	Oc1ccccc1C(=O)N/N=C/c2cc(Cl)cc(Cl)c2O	CID:135455583	phase I
BRD-K72615639	Oc1ccccc1C(=O)N/N=C/c2cc(Br)cc(Br)c2O	CID:135455584	phase I
BRD-K66359319	CCc1ccc2nc(Nc3nc(=O)c4ccccc4[nH]3)nc(C)c2c1	CID:135455921	phase I
BRD-K70918941	Oc1ccccc1/C=C/c2noc(n2)c3ccccc3O	CID:135460532	phase I
BRD-K19300944	COc1cc(\C=N\n2c(S)nnc2-c2ccccc2)ccc1O	CID:135470813	phase I
BRD-K83780283	Cc1nc(O)c([N+](=O)[O-])c(Nc2ccc(Br)cc2Br)n1	CID:135476231	phase I
BRD-K78930611	Oc1ccc(/C=C\2/SC(=NC2=O)NCc3ccccc3)cc1	CID:135486338	phase I
BRD-K14704318	Clc1cc(NC(=O)CSc2nc3ccccc3c(=O)[nH]2)ccc1Br	CID:135499031	phase I
BRD-K03552198	CCCCSc1nc2CCCc2c(O)n1	CID:135504848	phase I
BRD-A29437505	Nc1nc2n(C3OC(CO)C(O)C3O)c(=O)n(CC=C)c2c(=O)[nH]1	CID:135516428	phase I
BRD-A73594579	CC(C)CC1C(=C(C)Nc2nc(SCc3cccc(C)c3)nn12)C(=O)Nc4ccccc4	CID:135522119	phase I
BRD-K94920105	Cc1nc(=O)c2CSCCc2[nH]1	CID:135522417	phase I
BRD-A98777808	Nc1nc(=O)c2nc(Br)n(C3OC4COP(=O)(O)OC4C3O)c2[nH]1	CID:135526720	phase I
BRD-K41859756	CCNC(=O)c1noc(c1-c1ccc(CN2CCOCC2)cc1)-c1cc(C(C)C)c(O)cc1O	CID:135539077	phase I
BRD-K99750259	COC(=O)c1ccc(CSc2nc3CCCc3c(O)n2)cc1	CID:135546884	phase I
BRD-K38340366	COc1ccccc1NC2=NC(=O)/C(=C/c3ccc(O)c(OC)c3)/S2	CID:135547290	phase I
BRD-K70891562	Clc1ccc(OCC(=O)N\N=C\c2ccc[nH]2)c(Cl)c1	CID:135549936	phase I
BRD-K17306061	C[C@@H](O[C@@H]1OCCN(Cc2nc(=O)[nH][nH]2)[C@@H]1c1ccc(F)cc1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F	CID:135554441	phase I
BRD-K01712134	Cc1ccccc1NCC(=O)N\N=C\c1ccc[nH]1	CID:135560153	phase I
BRD-K55395145	Nc1nc2[nH]cc(CCc3ccc(cc3)C(=O)N[C@H](CCC(O)=O)C(O)=O)c2c(=O)[nH]1	CID:135565230	phase I
BRD-K03063480	Cn1cc(cn1)-c1[nH]c2cc(NC(=O)[C@H](N)C3CCCCC3)cc3c2c1cn[nH]c3=O	CID:135565545	phase I
BRD-K87112191	CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12	CID:135565635	phase I
BRD-K53472085	COc1cc(cc(Br)c1O)\C=N\n1c(S)nnc1C1CCCCC1	CID:135656310	phase I
BRD-A67788537	CC(C(=O)Nc1cccc(c1)\N=C\c1c(O)ccc2ccccc12)c1ccccc1	CID:135659046	phase I
BRD-K36258877	[O-][N+](=O)c1cc(C(=O)NCC=C)c2nc(Nc3ccc(Cl)c(Cl)c3)[nH]c(=O)c2c1	CID:135665263	phase I
BRD-K33720404	Cc1cc(Cl)ccc1OCC(=O)N\N=C\c1ccc[nH]1	CID:135688221	phase I
BRD-K30463976	Oc1nc(SCCc2ccccc2)nc2CCCc12	CID:135714026	phase I
BRD-K81601344	CO[C@H]1C=CO[C@@]2(C)Oc3c(C2=O)c4c(O)c(C=NN5CCN(CC5)C6CCCC6)c(NC(=O)C(=CC=C[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(=O)C)[C@@H]1C)C)c(O)c4c(O)c3C	CID:135749824	phase I
BRD-K93443135	Cc1noc(C)c1c2ccc3ncnc(O)c3c2	CID:135755223	phase I
BRD-K52904470	OC(=O)c1ccc(cc1)c2ccc(/C=C\3/SC(=NC3=O)Nc4cccc(c4)C(=O)O)o2	CID:135787362	phase I
BRD-K27799527	COC(=O)CCCCCCC(=O)N/N=C/c1c(OC)cc(O)cc1OC	CID:135787369	phase I
BRD-A73605923	CCC(C(=O)NC/C=C\C=C(\C)/C(OC)C(C)C1OC(\C=C/C=C\C=C(\C)/C(=O)c2c(O)cc[nH]c2=O)C(O)C1O)C3(O)OC(\C=C/C=C\C)C(C)(C)C(O)C3O	CID:135849857	phase I
BRD-K08878345	Oc1c(N=Nc2ccccc2O)c3ccccc3n1CC=C	CID:135857069	phase I
BRD-K67118123	CCCCn1c(O)c(N=Nc2ccccc2O)c3ccccc13	CID:135857071	phase I
BRD-K18970629	OC(=O)c1ccc(CSc2nc3CCCc3c(O)n2)cc1	CID:135857080	phase I
BRD-K72307842	Oc1nc(SCc2ccc(OC(F)(F)F)cc2)nc2CCCc12	CID:135859876	phase I
BRD-K14171663	C(N(Cc1ccccc1)Cc2ccccc2)c3nnc(s3)c4cc5ccccc5[nH]4	CID:135874057	phase I
BRD-K66588514	COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCC(=O)NO	CID:135882970	phase I
BRD-K76926998	COc1cc(/C=C/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)ccc1O	CID:135882987	phase I
BRD-K58972465	COc1ccc(/C=N/NC(=O)c2ccccn2)c(O)c1	CID:135882996	phase I
BRD-K79619196	Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(F)ccc2O	CID:135883071	phase I
BRD-K35004659	Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2c(O)ccc3ccccc23	CID:135883109	phase I
BRD-K60303132	COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCCCC(=O)NO	CID:135883127	phase I
BRD-K27332342	Oc1c(\C=N\NC(=O)c2cc(n[nH]2)-c2cccc(c2)[N+]([O-])=O)ccc2ccccc12	CID:135886610	phase I
BRD-K35798075	OOCc1cc(ccc1O)\N=N\c1ccc(cc1)-c1ccc(cc1)\N=N\c1ccc(O)c(c1)C(O)=O	CID:135886611	phase I
BRD-K41887956	Cc1cccc2c1[nH]c1nc(N\N=C\c3ccc(O)c(O)c3)nnc21	CID:135886612	phase I
BRD-K51704689	COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCCC(=O)NO	CID:135886613	phase I
BRD-K56956679	COC(=O)CCCCC(=O)N\N=C\c1c(OC)cc(O)cc1OC	CID:135886614	phase I
BRD-K66909449	Oc1cc2ccccc2cc1-c1nnc(SCC#CCOC(=O)c2ccc(F)cc2)o1	CID:135921706	phase I
BRD-K76935234	Fc1ccc(cc1)C(=O)OCC#CCSc1nnc(o1)-c1c[nH]c2ccccc12	CID:135921707	phase I
BRD-K15885023	Oc1ccc(-c2nn[nH]n2)c2cccnc12	CID:135921708	phase I
BRD-K87573634	CCCc1cn(nc1-c1ccc(O)cc1)-c1ccc(O)cc1	CID:135925692	phase I
BRD-K92817986	Clc1ccc(Cl)c(SCC(=O)N\N=C\c2ccc[nH]2)c1	CID:135976680	phase I
BRD-K76772814	CNC1=NC(=O)\C(S1)=C/c1cc(C)n(c1C)-c1ccccc1F	CID:135999135	phase I
BRD-K01121114	Clc1cc(Cl)c(OCC(=O)N\N=C\c2ccc[nH]2)c(Cl)c1	CID:135999136	phase I
BRD-K46625679	COc1cc(\C=C2/SC(Nc3ccccn3)=NC2=O)ccc1O	CID:136015351	phase I
BRD-K55889443	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c(O)c(\C=N\N4CCN(CC4)C4CCCC4)c(NC(=O)\C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c(O)c2c(O)c3C	CID:136073066	phase I
BRD-A67605442	CC(O)[C@H](O)C1CNc2nc(N)[nH]c(=O)c2N1	CID:136188272	phase I
BRD-A01317026	CC(O)[C@H](O)C1=Nc2c(NC1)nc(N)[nH]c2=O	CID:136235688	phase I
BRD-K83778500	Clc1cc(Cl)c(OCC(=O)NN=Cc2ccc[nH]2)c(Cl)c1	CID:137139966	phase I
BRD-K30563334	CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c(c(O)c3C)c(O)c(NC(=O)\C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c1=NC3(CCN(CC(C)C)CC3)N=c21	CID:137247591	phase I
BRD-A23689620	CC[C@H](C)[C@H]1O[C@@]2(C[C@@H]3C[C@@H](CC=C(C)C(O[C@H]4C[C@H](OC)C(O[C@H]5C[C@H](OC)[C@@H](O)[C@H](C)O5)[C@H](C)O4)[C@@H](C)C=CC=C4CO[C@H]5[C@H](O)C(C)=C[C@H](C(=O)O3)[C@]45O)O2)C=C[C@@H]1C	CID:139032007	phase I
BRD-K04949373	CC1=CCC[C@@]2(C)O[C@H]2[C@@H]2OC(=O)C(=C)[C@@H]2CC1	CID:139032026	phase I
BRD-K14036801	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(O)C[C@@H](C)C(=NOCOCCOC)[C@H](C)[C@@H](O)[C@]1(C)O	CID:139032028	phase I
BRD-K30600766	C[C@H]1O[C@@H](O[C@@H]2C[C@H]3O[C@@](O)(C[C@H](O)[C@H]3C(O)=O)C[C@@H](O)C[C@@H](O)[C@H](O)CC[C@@H](O)C[C@@H](O)CC(=O)O[C@@H](C)[C@H](C)[C@H](O)[C@@H](C)C=CC=CC=CC=CC=CC=CC=C2)[C@@H](O)[C@@H](N)[C@@H]1O	CID:139032029	phase I
BRD-M64432851	CCN(CC)CCNC(=O)c1c(C)[nH]c(C=C2/C(=O)Nc3ccc(F)cc23)c1C	CID:73707432	phase I
BRD-M47793593	CC(=C)[C@@H]1[C@H]2OC(=O)[C@@H]1[C@]3(O)C[C@H]4O[C@]45C(=O)O[C@H]2[C@@]53C.CC(C)(O)[C@@H]1[C@H]2OC(=O)[C@@H]1[C@]3(O)C[C@H]4O[C@]45C(=O)O[C@H]2[C@@]53C	CID:6473767	phase I
BRD-M45038741	COCCc1ccc(OCC(O)CNC(C)C)cc1.COCCc1ccc(OCC(O)CNC(C)C)cc1	CID:21997268	phase I
BRD-M10279501	CN[C@H](C)[C@@H]1CC[C@@H](N)[C@@H](O[C@@H]2[C@@H](N)C[C@@H](N)[C@H](O[C@H]3OC[C@](C)(O)[C@H](NC)[C@H]3O)[C@H]2O)O1.CN[C@@H]1[C@@H](O)[C@@H](O[C@H]2[C@H](N)C[C@H](N)[C@@H](O[C@H]3O[C@H](CN)CC[C@H]3N)[C@@H]2O)OC[C@]1(C)O.CN[C@@H]1[C@@H](O)[C@@H](O[C@H]2[C@H](N)C[C@H](N)[C@@H](O[C@H]3O[C@@H](CC[C@H]3N)[C@@H](C)N)[C@@H]2O)OC[C@]1(C)O	CID:6713924	phase I
BRD-M58473998	CC(CN(C)C)CN1c2ccccc2Sc3ccccc13.CC(CN(C)C)CN1c2ccccc2Sc3ccccc13	CID:73707352	phase I
BRD-M62162320	C1CC1C(NC2=NCCO2)C3CC3	CID:73707355	phase I
BRD-M19787235	CN1C[C@@H](CC2[C@@H]1Cc1c[nH]c3cccc2c13)C(=O)N[C@]1(C)O[C@@]2(O)[C@@H]3CCCN3C(=O)[C@H](Cc3ccccc3)N2C1=O.CN1C[C@@H](C[C@H]2[C@@H]1Cc1c[nH]c3cccc2c13)C(=O)N[C@]1(C)O[C@@]2(O)[C@@H]3CCCN3C(=O)[C@H](Cc3ccccc3)N2C1=O	CID:73707468	phase I
BRD-M30251550	CC(C)(C)NCC(O)COc1ccccc1C2CCCC2.CC(C)(C)NCC(O)COc1ccccc1C2CCCC2	CID:73707345	phase I
BRD-M98649031	Cn1c2nc(Cl)[nH]c2c(=O)n(C)c1=O.CN(C)CCOC(c1ccccc1)c1ccccc1	CID:10660	phase I
BRD-M73371355	CN1CCc2cccc-3c2[C@@H]1Cc1ccc(O)c(O)c-31.CN1CCc2cccc-3c2[C@@H]1Cc1ccc(O)c(O)c-31	CID:73707506	phase I
BRD-M07438658	CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1	CID:73707431	phase I
BRD-M35773784	CN1[C@@H]2CC[C@@H]1C[C@H](C2)OC(=O)C(CO)c1ccccc1.CN1[C@@H]2CC[C@@H]1C[C@H](C2)OC(=O)C(CO)c1ccccc1	CID:73707493	phase I
BRD-M02190957	CC(C)NCC(O)c1cc(O)cc(O)c1.CC(C)NCC(O)c1cc(O)cc(O)c1	CID:69049742	phase I
BRD-M86331534	CN(C)c1ccc2[n+](C)c(CCc3cc(C)n(c3C)-c3ccccc3)ccc2c1	CID:73707397	phase I
BRD-M41783010	CC(=O)NCCCS(O)(=O)=O	CID:73707392	phase I
BRD-M56587789	CCCCCCCN(CC)CCCC(O)c1ccc(NS(C)(=O)=O)cc1.CCCCCCCN(CC)CCCC(O)c1ccc(NS(C)(=O)=O)cc1	CID:73707513	phase I
BRD-M90449146	COC(N)(CO)CO.CCCCC[C@H](O)C=C[C@H]1[C@H](O)C[C@H](O)[C@@H]1CC=CCCCC(O)=O	CID:73707481	phase I
BRD-M16762496	CN(N=Cc1cnc2ccc(Br)cn12)S(=O)(=O)c1cc(ccc1C)[N+]([O-])=O	CID:73707389	phase I
BRD-M53001068	Cn1c(=O)n(C)c2nc[nH]c2c1=O.Cn1c(=O)n(C)c2nc[nH]c2c1=O	CID:18680317	phase I
BRD-M79902621	CC(C)(C)NCC(O)c1cc(O)cc(O)c1.CC(C)(C)NCC(O)c1cc(O)cc(O)c1	CID:73707356	phase I
BRD-M94527406	N[C@]12C[C@H]3C[C@H](C[C@@H](C3)C1)C2.N[C@]12C[C@H]3C[C@H](C[C@@H](C3)C1)C2	CID:21249869	phase I
BRD-M00539986	COc1ccc(C[C@H](C)NC[C@@H](O)c2ccc(O)c(NC=O)c2)cc1	CID:44483332	phase I
BRD-M61872305	CNC(C)(C)Cc1ccccc1.CNC(C)(C)Cc1ccccc1	CID:73707340	phase I
BRD-M61246020	CC(C(=O)O)c1cccc(Oc2ccccc2)c1.CC(C(=O)O)c1cccc(Oc2ccccc2)c1	CID:19905833	phase I
BRD-M08470251	CN(C)c1ccc2[n+](C)c(C=Cc3cc(C)n(c3C)-c3ccccc3)ccc2c1.CN(C)c1ccc2[n+](C)c(C=Cc3cc(C)n(c3C)-c3ccccc3)ccc2c1	CID:73707346	phase I
BRD-K44408410	COc1cc2[C@H]3CC[C@]4(C)[C@@H](O)CC[C@H]4[C@@H]3CCc2cc1O	CID:66414	phase II
BRD-K49055432	Cc1nc(NC(=O)N2CCC[C@H]2C(N)=O)sc1-c1csc(n1)C(C)(C)C	CID:42636535	phase II
BRD-K74363950	OC(C(=O)O[C@H]1C[N+]2(CCCOc3ccccc3)CCC1CC2)(c1cccs1)c1cccs1	CID:11434515	phase II
BRD-K82928847	ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N(c1ccccc1)c1ccccc1	CID:53340666	phase II
BRD-K00152668	OC(=O)\C=C\c1ccc(cc1)-c1ccc(O)c(c1)C12CC3CC(CC(C3)C1)C2	CID:9864378	phase II
BRD-K01577834	Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	CID:60961	phase II
BRD-K40718343	CCN1CCN(Cc2ccc(cc2)-c2cc3c(N[C@H](C)c4ccccc4)ncnc3[nH]2)CC1	CID:10297043	phase II
BRD-K54997624	Cc1nc(NC(=O)N2CCC[C@H]2C(N)=O)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F	CID:56649450	phase II
BRD-K42948882	NCCCCN(Cc1nc2ccccc2[nH]1)[C@H]1CCCc2cccnc12	CID:11256587	phase II
BRD-K32285926	COc1ccc2c(OCc3nnc4ccc(nn34)-c3ccccc3)ccnc2c1	CID:24864821	phase II
BRD-K64925568	CC(C)[C@@H](CS(=O)(=O)C(C)C)N1[C@@H]([C@H](C[C@](C)(CC(O)=O)C1=O)c1cccc(Cl)c1)c1ccc(Cl)cc1	CID:58573469	phase II
BRD-K45924332	Nc1cc(c[nH]c1=O)-c1ccncc1	CID:3698	phase II
BRD-K56032964	COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)N1CCC(CC1)N(C)C	CID:57390074	phase II
BRD-K10859802	CC(C)OC(=O)N1CCC(CC1)Oc1ncnc2n(ncc12)-c1ccc(cc1F)S(C)(=O)=O	CID:11705608	phase II
BRD-K67121414	COc1ccc(cc1)-n1nc(C(N)=O)c2CCN(C(=O)c12)c1ccc(cc1)N1CCCCC1=O	CID:10182969	phase II
BRD-K58435339	CC(C)c1cc(C(=O)N2Cc3ccc(CN4CCN(C)CC4)cc3C2)c(O)cc1O	CID:11955716	phase II
BRD-K87782578	COCCOc1ccc(Nc2ncc(F)c(Nc3cccc(NC(=O)C=C)c3)n2)cc1	CID:59174488	phase II
BRD-K42436189	C[C@@H]1COCCN1c1cc(nc(n1)-c1cccc2[nH]ccc12)C1(CC1)S(C)(=O)=O	CID:46244454	phase II
BRD-K99113996	CNC(=O)c1cccc(c1)-c1ccc2c(nc(nc2n1)N1CCOC[C@@H]1C)N1CCOC[C@@H]1C	CID:25262792	phase II
BRD-K28392481	COc1cc(CCc2cc(NC(=O)c3ccc(cc3)N3C[C@H](C)N[C@H](C)C3)n[nH]2)cc(OC)c1	CID:51039095	phase II
BRD-K99023089	NC1(CCN(CC1)c1ncnc2[nH]ccc12)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1	CID:25227436	phase II
BRD-K86525559	NC(=O)Nc1cc(sc1C(=O)N[C@H]1CCCNC1)-c1cccc(F)c1	CID:11152667	phase II
BRD-K98572433	CNC(=O)CN1CCC(CC1)Oc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC	CID:11488320	phase II
BRD-K31928526	CCN(CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1)CCOP(O)(O)=O	CID:11497983	phase II
BRD-K90195324	Cc1c(-c2ccc(O)cc2)n(Cc2ccc(OCCN3CCCCCC3)cc2)c2ccc(O)cc12	CID:154257	phase II
BRD-K45275534	COc1ccc(NC(=O)c2ccc(cc2)C(=N)N(C)C)c(c1)C(=O)Nc1ccc(Cl)cn1	CID:10275777	phase II
BRD-K92441787	Cc1cc2c(cc1C(=C)c1ccc(cc1)C(O)=O)C(C)(C)CCC2(C)C	CID:82146	phase II
BRD-K71221037	CC[C@H](NC(=O)[C@H](C)NC)C(=O)N1C[C@@H](O)C[C@H]1Cc1c([nH]c2cc(F)ccc12)-c1[nH]c2cc(F)ccc2c1C[C@@H]1C[C@H](O)CN1C(=O)[C@H](CC)NC(=O)[C@H](C)NC	CID:49836020	phase II
BRD-K07106112	Cc1c(NC(=O)OC[C@@H]2COCCN2)cn2ncnc(Nc3ccc4n(Cc5cccc(F)c5)ncc4c3)c12	CID:10437018	phase II
BRD-A07563059	Cc1cc2c(OCC(CNC(C)(C)C)OC(=O)c3ccccc3)cccc2[nH]1	CID:44112	phase II
BRD-K96936751	CC(C)(C)OC(=O)c1ncn-2c1[C@@H]1CCCN1C(=O)c1c(Br)cccc-21	CID:107926	phase II
BRD-K31313613	CC(C)c1cnn2c(NCc3ccccc3)cc(NCCCCCCN)nc12	CID:49867929	phase II
BRD-K28965160	CC(C)Nc1cc(-c2c[nH]c(c2)C(=O)N[C@H](CO)c2cccc(Cl)c2)c(Cl)cn1	CID:11719003	phase II
BRD-K51544265	COc1cc2nccc(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3)c2cc1OC	CID:25102847	phase II
BRD-K15179879	CC(C)C[C@H](NC(=O)[C@H](CCc1ccccc1)NC(=O)CN1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)[C@@]1(C)CO1	CID:11556711	phase II
BRD-K20722021	COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)c2cc1OC	CID:56846693	phase II
BRD-K97746869	CCCNC(=O)NS(=O)(=O)c1ccc(Cl)cc1	CID:2727	phase II
BRD-K22861715	Oc1cc(O)c2c(c1)oc(cc2=O)-c1ccccc1	CID:5281607	phase II
BRD-K35245662	CC(C)C(=O)OCC(=O)[C@@]12O[C@@H](O[C@@H]1C[C@H]1[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@]21C)C1CCCCC1	CID:6918155	phase II
BRD-K03390685	OC1(CN(C1)C(=O)c1ccc(F)c(F)c1Nc1ccc(I)cc1F)[C@@H]1CCCCN1	CID:16222096	phase II
BRD-K53508936	ONC(=O)C1(CS(=O)(=O)c2ccc(Oc3ccc(Cl)cc3)cc2)CCOCC1	CID:3342298	phase II
BRD-K81458380	OC(=O)c1ccc2c(c1)nc(Nc1cccc(Cl)c1)c1ccncc21	CID:24748573	phase II
BRD-K71822263	N[C@H](CO)C(O)=O	CID:71077	phase II
BRD-K57169635	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)\C=C\CN1CCCCC1	CID:11511120	phase II
BRD-K22482860	Nc1ccncc1	CID:1727	phase II
BRD-K44309363	COC(=O)C1=C(C)NC(C)=C([C@@H]1c1cccc(c1)[N+]([O-])=O)C(=O)OCCCN1CCC(CC1)(c1ccccc1)c1ccccc1	CID:6918097	phase II
BRD-K13662825	CCc1cnn2c(NCc3ccc[n+]([O-])c3)cc(nc12)N1CCCC[C@H]1CCO	CID:46926350	phase II
BRD-K71075609	CCN[C@@H]1C[C@H](C)S(=O)(=O)c2sc(cc12)S(N)(=O)=O	CID:6604453	phase II
BRD-K88807631	COc1cc2CCN(CCc3ccc(NC(=O)c4cccc5c4[nH]c4c(OC)cccc4c5=O)cc3)Cc2cc1OC	CID:119373	phase II
BRD-K35007173	CCCn1c2nc[nH]c2c(=O)[nH]c1=O	CID:1676	phase II
BRD-K63126190	CNC[C@H](O)c1ccc(O)c(O)c1	CID:5816	phase II
BRD-K19761926	COC(=O)[C@@H]1CC2=CC(=O)CC[C@]2(C)[C@@]23O[C@@H]2C[C@@]2(C)[C@@H](CC[C@@]22CCC(=O)O2)[C@H]13	CID:443872	phase II
BRD-K57754230	Cc1cc(C)c(CNC(=O)c2cc(cc3n(ncc23)C2CCCC2)-c2ccc(CN3CCOCC3)cc2)c(=O)[nH]1	CID:60160561	phase II
BRD-K80608265	Oc1ccc(cc1)[C@@H]1Oc2ccc(O)cc2[C@@H]2CCC[C@H]12	CID:10286159	phase II
BRD-K82603084	OC(=O)CN(CCN(CC(O)=O)CC(O)=O)CC(O)=O	CID:6049	phase II
BRD-K16803204	O=C(Nc1nc2cccc(-c3ccc(CN4CCS(=O)(=O)CC4)cc3)n2n1)C1CC1	CID:49831257	phase II
BRD-K88025533	CCCCCCCCc1ccc(CCC(N)(CO)CO)cc1	CID:107970	phase II
BRD-K38852836	CC(C)c1cc(-c2n[nH]c(=O)n2-c2ccc3n(C)ccc3c2)c(O)cc1O	CID:135564985	phase II
BRD-K43002773	C[C@@H]1C[C@H](C2=C1C(=NC=N2)N3CCN(CC3)C(=O)[C@H](CNC(C)C)C4=CC=C(C=C4)Cl)O	CID:24788740	phase II
BRD-K71480163	CC(C)NC[C@@H](C(=O)N1CCN(CC1)c1ncnc2[C@@H](O)C[C@@H](C)c12)c1ccc(Cl)cc1	CID:59671085	phase II
BRD-K68938568	CN[C@@H](C)C(=O)N[C@@H](C1CCCCC1)C(=O)N1CCC[C@H]1C(=O)Nc1snnc1-c1ccccc1	CID:46940575	phase II
BRD-K23228615	C[C@H](O)C(=O)N1CCN(Cc2sc3c(nc(nc3c2C)-c2cnc(N)nc2)N2CCOCC2)CC1	CID:25254071	phase II
BRD-K99475619	CNCCn1c2c(cnc3cc4OCOc4cc23)c2cc(OC)c(OC)cc2c1=O	CID:10294813	phase II
BRD-K69001009	CN1CCN(CC1)C1CCN(CC1)C(=O)Nc1cc(Oc2ccc(NC(=O)C3(CC3)C(=O)Nc3ccc(F)cc3)c(F)c2)ccn1	CID:16118392	phase II
BRD-K49215523	Cc1nc2c(cc(cc2n1Cc1cccc(c1C)C(F)(F)F)N1CCOCC1)C(O)=O	CID:56949517	phase II
BRD-K01674964	NCCc1c[nH]cn1	CID:774	phase II
BRD-K51747290	NC(=O)NO	CID:3657	phase II
BRD-K36363294	COc1cc2c3n([C@H](C)c4ccccn4)c(=O)[nH]c3cnc2cc1-c1c(C)noc1C	CID:52912189	phase II
BRD-K08109215	CCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2cc(OC)ccc2-n2c(C)nnc12	CID:46943432	phase II
BRD-K31135544	CNC(=O)[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NCc3cccc(I)c3)ncnc12	CID:123683	phase II
BRD-K70301465	Nc1ncnc2n(nc(-c3ccc(Oc4ccccc4)cc3)c12)[C@@H]1CCCN(C1)C(=O)C=C	CID:24821094	phase II
BRD-K89208535	CCc1cc2CC(Cc2cc1CC)NC[C@H](O)c1ccc(O)c2[nH]c(=O)ccc12	CID:6918554	phase II
BRD-K93779381	C\C=C(\C)C(=O)O[C@H]1C(C)=C[C@@]23[C@H](C)C[C@@H]4[C@H]([C@H](C=C(CO)[C@@H](O)[C@]12O)C3=O)C4(C)C	CID:6918670	phase II
BRD-K52818472	CC(C)(C)c1cc(c(NC(=O)c2c[nH]c3ccccc3c2=O)cc1O)C(C)(C)C	CID:16220172	phase II
BRD-K54606188	Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)OC(C)(C)C)c1nnc(C)n-21)c1ccc(Cl)cc1	CID:46907787	phase II
BRD-K88506063	CC(C)NC(=O)COc1cccc(c1)-c1nc(Nc2ccc3[nH]ncc3c2)c2ccccc2n1	CID:11950170	phase II
BRD-K21718444	O=C(N1CCNCC1)c1ccc(cc1)\C=C\c1n[nH]c2ccccc12	CID:11427553	phase II
BRD-K68232650	COC[C@@H](NC(C)=O)C(=O)NCc1ccccc1	CID:219078	phase II
BRD-K48894757	CS(=O)(=O)c1cc(F)cc2c3CC[C@H](CC(O)=O)c3n(Cc3ccc(Cl)cc3)c12	CID:9867642	phase II
BRD-K08248804	CN[C@@H](C)C(=O)N[C@@H](C1CCCCC1)C(=O)N1CCC[C@H]1c1nc(cs1)C(=O)c1ccc(F)cc1	CID:24737642	phase II
BRD-K39974922	COc1cc2nccc(Oc3ccc(NC(=O)NC4CC4)c(Cl)c3)c2cc1C(N)=O	CID:9823820	phase II
BRD-K31812033	CC(C)(C)NC[C@H](O)COc1cccc2C(=O)CCCc12	CID:39468	phase II
BRD-K86118762	C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12	CID:11640390	phase II
BRD-K27955832	Nc1nc(OCc2cc(Br)cs2)c2[nH]cnc2n1	CID:3025944	phase II
BRD-K92213669	FC(F)(F)CNC(=O)C1(CCCCN2CCC(CC2)NC(=O)c2ccccc2-c2ccc(cc2)C(F)(F)F)c2ccccc2-c2ccccc12	CID:9853053	phase II
BRD-K41599323	NC(=O)N1CCC(CC(=O)N2CCC(CC2)[C@H]2c3ncc(Br)cc3CCc3cc(Cl)cc(Br)c23)CC1	CID:148195	phase II
BRD-K55013654	C[C@H]1CNCCc2ccc(Cl)cc12	CID:11658860	phase II
BRD-K56195681	Cc1c(F)cc(cc1-c1ccc(cn1)C(=O)NCC(C)(C)C)C(=O)NC1CC1	CID:11552706	phase II
BRD-K31309378	CNC(=O)c1cccc2cc(ccc12)Oc1ccnc2cc(OCC3(N)CC3)c(OC)cc12	CID:25031915	phase II
BRD-K54520417	Fc1ccc(cc1)-c1n(Cc2ccc(F)cc2Cl)nc2c(cccc12)C(F)(F)F	CID:16734800	phase II
BRD-K78055238	Fc1cc2CN(CCn3cc(C4=C(C(=O)NC4=O)c4cnc5ccccn45)c(c1)c23)C(=O)N1CCCCC1	CID:10029385	phase II
BRD-K78118466	Cc1cccc(n1)-c1nn2CCCc2c1-c1ccnc2ccc(cc12)C(N)=O	CID:10090485	phase II
BRD-K18961567	Cc1ccc(C(=O)Nc2ccc(Oc3cc4cnn(C)c4cc3-c3cn[nH]c3)c(F)c2)c(=O)n1-c1ccc(F)cc1	CID:44603533	phase II
BRD-K94534639	C[C@]1(CCSC(N)=N1)c1cc(c(F)cc1F)-c1cncnc1	CID:44251605	phase II
BRD-K17203476	C[C@@H](Oc1ccc2[nH]nc(\C=C\c3cnn(CCO)c3)c2c1)c1c(Cl)cncc1Cl	CID:46944259	phase II
BRD-K21396683	CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)[C@H](O)C(=O)NO)C(C)(C)C	CID:119031	phase II
BRD-K75844781	Clc1cccc(c1)N1CCNCC1	CID:1355	phase II
BRD-A82772293	CN1CCCC(CN2c3ccccc3Sc3ccccc23)C1	CID:6075	phase II
BRD-K09372874	COc1cc(NC(=O)Nc2cccc(CNC(=O)O[C@H]3CCOC3)c2)ccc1-c1cnco1	CID:153241	phase II
BRD-K27182532	Nc1nccc(Oc2ccc(NC(=O)c3c[nH]cc(-c4ccc(F)cc4)c3=O)cc2F)c1Cl	CID:44155856	phase II
BRD-K33251802	CCCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO	CID:51634	phase II
BRD-K56405753	CN(C[C@@H]1COCCO1)S(=O)(=O)Nc1ccc2ccc3ncc(cc3c(=O)c2c1)-c1cnn(C)c1	CID:44137946	phase II
BRD-K55512740	Cn1cc(cn1)-c1cnc2ccc3ccc(CS(=O)(=O)NCc4ccccn4)cc3c(=O)c2c1	CID:45142457	phase II
BRD-K08832567	Oc1ccc(cc1)[C@@H]1CC(=O)c2c(O)cc(O)cc2O1	CID:439246	phase II
BRD-K83699324	CN1CCN(CC1)c1ccc(OC(F)(F)F)c(Nc2ncc3CCc4c(nn(CCO)c4-c3n2)C(N)=O)c1	CID:49792852	phase II
BRD-K21025364	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)ncc1Cl	CID:9934347	phase II
BRD-K42805893	COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2ccccc12	CID:71496458	phase II
BRD-K53417444	CN(C)C[C@H]1CC[C@@H](CC1)Nc1c(cnc2ccc(nc12)-c1cc(Cl)c(O)c(Cl)c1)C(C)=O	CID:135398499	phase II
BRD-K26603252	COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OC	CID:4705	phase II
BRD-K37764012	CN(C)C[C@@H](NC(=O)N1Cc2c(Nc3nc(C)nc4ccsc34)n[nH]c2C1(C)C)c1ccccc1	CID:25227462	phase II
BRD-K86816506	FC(F)(F)c1ccc(Oc2cccc(C=C3CCN(CC3)C(=O)Nc3cccnn3)c2)nc1	CID:24771824	phase II
BRD-K07310275	COc1ccc(cn1)-c1cc2c(C)nc(N)nc2n([C@H]2CC[C@@H](CC2)OCCO)c1=O	CID:25033539	phase II
BRD-K79239947	CS(=O)(=O)c1cccc(CNc2nc(Nc3ccc4NC(=O)CCc4c3)ncc2C(F)(F)F)c1	CID:11612883	phase II
BRD-K13094524	COc1ccccc1S(=O)(=O)Nc1ccc2NC(=O)N(C)Cc2c1	CID:71271629	phase II
BRD-K95880107	CNC(=O)c1ccc(C)c(c1)-n1c(C)cc(OCc2ccc(F)cc2F)c(Br)c1=O	CID:22049997	phase II
BRD-K50000283	O=C1NCCc2[nH]c(cc12)-c1ccncc1	CID:11715767	phase II
BRD-K60997853	CNC(=O)c1nn(C)c-2c1C(C)(C)Cc1cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc-21	CID:16718576	phase II
BRD-K73381542	CNC[C@H](O)c1cccc(O)c1	CID:6041	phase II
BRD-K47642186	COc1ccc(cc1OC1CCCC1)C(=O)Nc1c(Cl)cncc1Cl	CID:154575	phase II
BRD-A28467416	O=C(Nc1ccncc1)Nc1ccc(cc1)-c1nc(nc(n1)N1CCOCC1)N1C2CCC1COC2	CID:46947264	phase II
BRD-K46290096	COCCOc1ccc(cc1)N1CCN(CCn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)CC1	CID:10117987	phase II
BRD-K14870255	Nc1nc(Nc2ccc3CC[C@@H](CCc3c2)N2CCCC2)nn1-c1cc2CCCc3ccccc3-c2nn1	CID:46215462	phase II
BRD-K52233191	COc1ccc(F)c(F)c1C(=O)c1cnc(NC2CCN(CC2)S(C)(=O)=O)nc1N	CID:6918852	phase II
BRD-K93123848	Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12	CID:11656518	phase II
BRD-K08586861	OC(=O)CCn1c2CC[C@H](Cc2c2ccccc12)NS(=O)(=O)c1ccc(F)cc1	CID:123879	phase II
BRD-K76694128	CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1	CID:25066467	phase II
BRD-K16730910	CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c(F)c2)ccn1	CID:11167602	phase II
BRD-K58486055	CC(C)Cc1ccc(cc1)[C@@H](C)C(=O)NS(C)(=O)=O	CID:9838712	phase II
BRD-K53814070	C[C@H]1CNCCCN1S(=O)(=O)c1cccc2cncc(F)c12	CID:9863672	phase II
BRD-K64538373	OCCONC(=O)c1cc(CN2OCCCC2=O)c(F)c(F)c1Nc1ccc(I)cc1F	CID:11548630	phase II
BRD-K33610132	COc1cc(ccc1Nc1ncc(c(Nc2cccc(NC(=O)C=C)c2)n1)C(F)(F)F)N1CCN(CC1)C(C)=O	CID:57335384	phase II
BRD-K03194791	FC(F)Oc1ccc(cc1OCC1CC1)C(=O)Nc1c(Cl)cncc1Cl	CID:449193	phase II
BRD-K20079257	NC(=O)c1cn(Cc2c(F)cccc2F)nn1	CID:129228	phase II
BRD-K98004573	Cc1cncc(CN2CCC(CC2)=C2c3ccc(Cl)cc3CCc3cccnc23)c1	CID:133017	phase II
BRD-K92613113	C[C@H](NCc1ccc(OCc2cccc(F)c2)cc1)C(N)=O	CID:131682	phase II
BRD-K19412355	COc1nccc(n1)-c1c(ncn1C1CCNCC1)-c1ccc(F)cc1	CID:9863367	phase II
BRD-K68532323	CC(C)[C@@H](N(CCCN)C(=O)c1ccc(C)cc1)c1oc2cc(Cl)ccc2c(=O)c1Cc1ccccc1	CID:9936388	phase II
BRD-K86797399	CCCCc1nc2cc(ccc2n1CCN(CC)CC)\C=C\C(=O)NO	CID:49855250	phase II
BRD-K21295289	NC(=O)C(c1ccccc1)(c1ccc(F)cc1)c1ccc(F)cc1	CID:216327	phase II
BRD-K80700417	CN1CCC(CNc2ccc3ncc(-c4cccc(OC(F)(F)F)c4)n3n2)CC1	CID:24795070	phase II
BRD-K89561498	CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(O)cc12	CID:104842	phase II
BRD-K71281111	CC1(C)Cc2c(c(nn2-c2ccc(C(N)=O)c(N[C@H]3CC[C@H](O)CC3)c2)C(F)(F)F)C(=O)C1	CID:24772860	phase II
BRD-K24723746	O=C(O[C@H]1CN2CCC1CC2)N1CCc2ccccc2[C@@H]1c1ccccc1	CID:154059	phase II
BRD-K16761703	CN1CCN(CC1)c1nc(C2=C(C(=O)NC2=O)c2c[nH]c3ccccc23)c2ccccc2n1	CID:10296883	phase II
BRD-K80343549	CC(C)(O)CC(=O)NCCn1ccc2ncnc(Nc3ccc(Oc4cccc(c4)C(F)(F)F)c(Cl)c3)c12	CID:11620908	phase II
BRD-K26667523	Cn1c2ncn(C[C@@H](O)CO)c(=O)c2c(Nc2ccc(I)cc2F)c(F)c1=O	CID:24963252	phase II
BRD-K58501140	Cc1cc(OCCCS(C)(=O)=O)cc(C)c1-c1cccc(COc2ccc3[C@H](CC(O)=O)COc3c2)c1	CID:24857286	phase II
BRD-K17555800	C[C@H]1CN([C@H](C)CN1Cc1ccc(F)cc1)C(=O)c1cc2c(cn(C)c2cc1Cl)C(=O)C(=O)N(C)C	CID:9871074	phase II
BRD-K74339692	CCOc1ccccc1OCCN[C@H](C)Cc1ccc(OC)c(c1)S(N)(=O)=O	CID:129211	phase II
BRD-K44844162	CC(C)n1nc(C)nc1-c1cn2CCOc3cc(ccc3-c2n1)-c1cnn(c1)C(C)(C)C(N)=O	CID:51001932	phase II
BRD-K84564571	CNC(=O)c1cc(COc2nnc(Nc3ccc(Cl)cc3)c3ccoc23)ccn1	CID:9808844	phase II
BRD-A93093700	CN1c2ccc(Cl)cc2C(=NC(O)C1=O)c1ccccc1	CID:5391	phase II
BRD-K48068743	Cc1cc(N2CCN(CC2)[C@@H]2CN[C@@H](C2)C(=O)N2CCSC2)n(n1)-c1ccccc1	CID:11949652	phase II
BRD-K15507868	CCO[C@@H](Cc1ccc(OCCc2ccc(OS(C)(=O)=O)cc2)cc1)C(O)=O	CID:208901	phase II
BRD-A86248581	OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)N1CCC(O)NC1=O	CID:29243	phase II
BRD-A16347691	OC(=O)CCCCC1CCSS1	CID:864	phase II
BRD-A92800748	COc1ccc2cc(ccc2c1)-c1nc([nH]c1-c1ccncc1)-c1ccc(cc1)S(C)=O	CID:23625762	phase II
BRD-K37111771	NCCNCCNCCN	CID:5565	phase II
BRD-K46692793	OC(c1ccccc1)(c1ccccc1)C12CC[N+](CCOCc3ccccc3)(CC1)CC2	CID:11519070	phase II
BRD-K86856088	CC(C)N1CCC(CC1)NC2=NC(=NC3=CC(=C(C=C32)OC)OCCCN4CCCC4)C5CCCCC5	CID:46224516	phase II
BRD-K88052444	NC(N)=O	CID:1176	phase II
BRD-K77625799	COc1cc2c(Nc3ccc(Br)cc3F)ncnc2cc1OCC1CCN(C)CC1	CID:3081361	phase II
BRD-K09711437	CCc1c(C(=O)C(N)=O)c2c(OCC(O)=O)cccc2n1Cc1ccccc1	CID:155815	phase II
BRD-K26756394	CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1	CID:51000408	phase II
BRD-K62391742	CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCC4CCOCC4)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1	CID:49846579	phase II
BRD-K44827188	Clc1cc(ccc1C(=O)Nc1ccc(Cl)c(c1)-c1ccccn1)S(C)(=O)=O	CID:24776445	phase II
BRD-K69776681	CC[C@H]1N(C(C)C)c2nc(Nc3ccc(cc3OC)C(=O)N[C@H]3CC[C@@H](CC3)N3CCN(CC4CC4)CC3)ncc2N(C)C1=O	CID:10461508	phase II
BRD-K53963539	Cc1ccc(Sc2ccccc2N2CCNCC2)c(C)c1	CID:9966051	phase II
BRD-K54640016	CC(C)OC(=O)C1=CN(CC(C)(C)c2c1[nH]c1ccccc21)C(=O)c1ccc(F)c(F)c1	CID:10026128	phase II
BRD-K87465484	COc1cc2c(NC3CCN(CC3)C3CCCCC3)nc(nc2cc1OCCCN1CCCCC1)N1CCCN(CC1)C(C)C	CID:53315882	phase II
